G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
LY2794193
CAS:2173037-97-1
LY2794193 is a highly effective and selective agonist of the mGlu3 receptor (hmGlu3 Ki=0.927 nM,EC50=0.47 …
Formula:
C16H18N2O6
Color and Shape:
Solid
Molecular weight:
334.32
Ref: TM-T15807
| 5mg | 490.00 € | ||
| 25mg | 1,679.00 € | ||
| 50mg | 2,209.00 € | ||
| 100mg | 3,061.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
IRL 2500
CAS:169545-27-1
IRL 2500 is an antagonist of Endothelin receptor with IC50s of 1.3 and 94 nM …
Formula:
C36H35N3O4
Purity:
98.29%
Color and Shape:
White Crystalline Solid
Molecular weight:
573.68
Ref: TM-T15596
| 1mg | 49.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 294.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 602.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
GLPG0974
CAS:1391076-61-1
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
Formula:
C25H25ClN2O4S
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
484.99
Ref: TM-T15388
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
Aclidinium
CAS:727649-81-2
Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, …
Formula:
C26H30NO4S2
Color and Shape:
Liquid
Molecular weight:
484.65
Ref: TM-T200043
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
SGL5213
CAS:1240305-17-2
SGL5213 is a potent oral SGLT1 inhibitor (IC50: 29 nM) with potential for treating type …
Formula:
C37H55N3O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
669.85
Ref: TM-T12892
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
Rolapitant hydrochloride
CAS:858102-79-1
Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki …
Formula:
C25H27ClF6N2O2
Purity:
98.35% - 99.79%
Color and Shape:
Solid
Molecular weight:
536.94
Ref: TM-T3724
| 1mg | 149.00 € | ||
| 5mg | 356.00 € | ||
| 10mg | 507.00 € | ||
| 25mg | 760.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,386.00 € | ||
| 200mg | 1,829.00 € | ||
| 1mL*10mM (DMSO) | 428.00 € |
Estimated delivery in United States, on Friday 21 Mar 2025
Cyclizine dihydrochloride
CAS:5897-18-7
Cyclizine dihydrochloride (Marzine hydrochloride) is a histamine H1 antagonist. It is given by mouth or …
Formula:
C18H24Cl2N2
Color and Shape:
Solid
Molecular weight:
339.3
Ref: TM-T3037
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Chlorcyclizine hydrochloride
CAS:14362-31-3
Chlorcyclizine hydrochloride is an antagonist of histamine H1.
Formula:
C18H22Cl2N2
Molecular weight:
337.29
Ref: TM-T10794
| 25mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Cyclobenzaprine hydrochloride
CAS:6202-23-9
Cyclobenzaprine hydrochloride (MK130 hydrochloride) , a centrally acting muscle relaxant with antidepressant activity, leads to …
Formula:
C20H22ClN
Purity:
99.98%
Color and Shape:
Crystalline Solid
Molecular weight:
311.86
Ref: TM-T1509
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Desmopressin
CAS:16679-58-6
Desmopressin (DDAVP)(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic …
Formula:
C46H64N14O12S2
Purity:
97.45%
Color and Shape:
Solid
Molecular weight:
1069.22
Ref: TM-T5019
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Naloxone hydrochloride
CAS:357-08-4
Naloxone hydrochloride (Naloxone HCl) is a specific opiate antagonist that has no agonist activity. It …
Formula:
C19H21NO4·HCl
Purity:
97.91%
Color and Shape:
White To Off-White/Powder
Molecular weight:
363.84
Ref: TM-T0102
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information |
Xylazine hydrochloride
CAS:23076-35-9
Xylazine hydrochloride (BAY 1470 hydrochloride) is an adrenergic alpha-2 agonist used as a sedative, analgesic …
Formula:
C12H16N2S·HCl
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
256.79
Ref: TM-T1500
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
(±)-Levomepromazine-d6
CAS:1189805-51-3
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and …
Formula:
C19H24N2OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
334.51
Ref: TM-T13470
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information |
Cyprodime
CAS:118111-54-9
Cyprodime is a selective μ-opioid receptor (MOR) antagonist with inhibitory effects on μ, δ, and …
Formula:
C22H29NO3
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
355.47
Ref: TM-T61273
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
6-Bromopravadoline
CAS:166599-63-9
6-Bromopravadoline (WIN 54461) (WIN 54461) is an antagonist of CB1. 6-Bromopravadoline acts as an inhibitor …
Formula:
C23H25BrN2O3
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
457.36
Ref: TM-T41350
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Pravadoline
CAS:92623-83-1
Pravadoline (WIN48098-6) is a cannabinoid receptor agonist. Pravadoline inhibited the PGs synthesis in mouse brain …
Formula:
C23H26N2O3
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
378.46
Ref: TM-T21380
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
Clocapramine dihydrochloride hydrate
CAS:60789-62-0
Clocapramine dihydrochloride hydrate (3-Chlorocarpipramine hydrochloride hydrate) is an antagonist of the 5-HT2A and D2 receptors.
Formula:
C28H41Cl3N4O2
Purity:
97.68%
Color and Shape:
Solid
Molecular weight:
572.01
Ref: TM-T10837
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
β-Casomorphin, bovine
CAS:72122-62-4
β-Casomorphin, bovine (β-Casomorphin, bovine(2TFA))(2TFA) is an opioid peptide isolated from casein peptone
Formula:
C41H55N7O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
789.92
Ref: TM-T7576
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information |
NTRC-844
CAS:1811503-67-9
NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity …
Formula:
C28H28FN3O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
489.54
Ref: TM-T28217
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
PrNMI
CAS:1541244-33-0
PrNMI is a highly effective and orally active agonist targeting the peripherally restricted cannabinoid 1 …
Formula:
C29H31NO
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
409.56
Ref: TM-T39024
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
