G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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OMDM-5
CAS:616884-66-3
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing …
Formula:
C26H44N2O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
432.64
Ref: TM-T12306
| 1mg | 94.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 436.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 835.00 € | ||
| 200mg | 1,089.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Vasopressin
CAS:11000-17-2
Vasopressin receptor agonist; antidiuretic
Formula:
C46H65N15O12S2
Purity:
Min. 95%
Color and Shape:
White Powder
Molecular weight:
1,084.23 g/mol
Ref: 3D-FV40959
| 1g | 1,348.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 451.00 € | ||
| 250mg | 716.00 € | ||
| 500mg | 1,003.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
LGD-6972
CAS:1207989-09-0
LGD-6972 is an antagonist of glucagon receptor.
Formula:
C43H46N2O5S
Purity:
98.8% - 99.33%
Color and Shape:
Solid
Molecular weight:
702.9
Ref: TM-T11845
| 1mg | 87.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 276.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
PSB 1115
CAS:152529-79-8
PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.
Formula:
C14H14N4O5S
Purity:
100% - 99.24%
Color and Shape:
Solid
Molecular weight:
350.35
Ref: TM-T23201
| 1mg | 66.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 29 Apr 2025
Lumateperone
CAS:313368-91-1
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).
Formula:
C24H28FN3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
393.5
Ref: TM-T21069
| 10mg | 39.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 115.00 € |
Estimated delivery in United States, on Tuesday 29 Apr 2025
AMG 837 calcium hydrate
CAS:1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.
Formula:
C52H44CaF6O8
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
950.97
Ref: TM-TQ0020
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 280.00 € | ||
| 100mg | 400.00 € | ||
| 200mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 29 Apr 2025
SR 142948
CAS:184162-64-9
SR 142948 is a neurotensin (NT) receptor antagonist.
Formula:
C39H51N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
685.85
Ref: TM-T23386
| 10mg | 878.00 € |
Estimated delivery in United States, on Tuesday 29 Apr 2025
SB-616234-A
CAS:908601-49-0
SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant …
Formula:
C32H36ClN5O3
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
574.11
Ref: TM-T12847
| 1mg | 103.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 358.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,007.00 € | ||
| 200mg | 1,358.00 € | ||
| 1mL*10mM (DMSO) | 313.00 € |
Estimated delivery in United States, on Tuesday 29 Apr 2025
BQ-788
CAS:173326-37-9
BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation …
Formula:
C34H51N5O7
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
641.8
Ref: TM-T10595
| 1mg | 134.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 467.00 € | ||
| 25mg | 746.00 € | ||
| 50mg | 1,006.00 € | ||
| 100mg | 1,363.00 € | ||
| 500mg | 2,674.00 € | ||
| 1mL*10mM (DMSO) | 358.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
Monlunabant
CAS:2712480-46-9
Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor …
Formula:
C26H22ClF3N6O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
591.00
Ref: TM-T79137
| 1mg | 352.00 € | ||
| 5mg | 876.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
GnRH-R antagonist 1
CAS:2826273-90-7
Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.
Formula:
C31H28F5N7O6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
721.65
Ref: TM-T72492
| 25mg | 2,245.00 € | ||
| 50mg | 2,972.00 € | ||
| 100mg | 4,019.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
15-keto-Prostaglandin E2
CAS:26441-05-4
15-keto-Prostaglandin E2, an endogenous metabolite, inhibits STAT3 activation through binding to Cys259 and regulates breast …
Formula:
C20H30O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
350.45
Ref: TM-T78582
| 1mg | 1,094.00 € | ||
| 5mg | 3,273.00 € | ||
| 10mg | 4,914.00 € | ||
| 25mg | 8,349.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.
Formula:
C24H33BrN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.44
Ref: TM-T10294
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
SB 243213 hydrochloride
CAS:200940-23-4
SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H20ClF3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
464.87
Ref: TM-T12859
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
Vofopitant
CAS:168266-90-8
Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for …
Formula:
C21H23F3N6O
Purity:
97.61%
Color and Shape:
Solid
Molecular weight:
432.44
Ref: TM-T13329
| 1mg | 97.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 342.00 € | ||
| 25mg | 554.00 € | ||
| 50mg | 802.00 € | ||
| 100mg | 1,079.00 € | ||
| 500mg | 2,157.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
SGLT inhibitor-1
CAS:2247314-23-2
SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s …
Formula:
C24H27FO8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
462.46
Ref: TM-T12893
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
SB-224289 hydrochloride
CAS:180084-26-8
SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
Formula:
C32H33ClN4O3
Purity:
97.82% - 98.09%
Color and Shape:
Solid
Molecular weight:
557.08
Ref: TM-T12841
| 5mg | 54.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
SCH 563705
CAS:473728-58-4
SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory …
Formula:
C23H27N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
425.48
Ref: TM-T16864
| 1mg | 309.00 € | ||
| 5mg | 738.00 € | ||
| 10mg | 1,154.00 € | ||
| 25mg | 1,716.00 € | ||
| 50mg | 2,326.00 € | ||
| 1mL*10mM (DMSO) | 828.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
CS-003 Free base
CAS:191672-52-3
CS-003: Triple neurokinin receptor antagonist; Ki=2.3 nM (NK1), 0.54 nM (NK2), 0.74 nM (NK3); treats …
Formula:
C34H38Cl2N2O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
673.65
Ref: TM-T10892
| 25mg | 2,384.00 € | ||
| 50mg | 3,159.00 € | ||
| 100mg | 4,299.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
Bzo-poxizid
CAS:1048973-64-3
Bzo-poxizid is a synthetic cannabinoid and a psychoactive substance.
Formula:
C20H21N3O2
Molecular weight:
335.40
Ref: TM-T200948
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
