G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ML314
CAS:1448895-09-7
ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased …
Formula:
C24H28N4O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
420.504
Ref: TM-TQ0075
| 1mg | 52.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SHA 68
CAS:847553-89-3
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with …
Formula:
C26H24FN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.49
Ref: TM-T12895
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Arotinolol
CAS:68377-92-4
Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency …
Formula:
C15H21N3O2S3
Color and Shape:
White Solid
Molecular weight:
371.54
Ref: TM-T10371
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
ML-290
CAS:1482500-76-4
ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. …
Formula:
C24H21F3N2O5S
Color and Shape:
Solid
Molecular weight:
506.49
Ref: TM-T16101
| 1mg | 91.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SB-399885 hydrochloride
CAS:402713-81-9
SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
Formula:
C18H22Cl3N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
482.81
Ref: TM-T12843
| 1mg | 44.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Protease-Activated Receptor-4
CAS:245443-52-1
Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
Formula:
C33H46N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
666.77
Ref: TM-T7380
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Pumosetrag Hydrochloride
CAS:194093-42-0
Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment …
Formula:
C15H18ClN3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
339.84
Ref: TM-T16683
| 1mg | 46.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Terazosin hydrochloride
CAS:63074-08-8
Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.
Formula:
C19H26ClN5O4
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
423.89
Ref: TM-T0197
| 50mg | 43.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 88.00 € | ||
| 500mg | 132.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Ritodrine hydrochloride
CAS:23239-51-2
Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing …
Formula:
C17H21NO3·HCl
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
323.82
Ref: TM-T1433
| 1g | 52.00 € | ||
| 200mg | 36.00 € | ||
| 500mg | 42.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Tolazoline hydrochloride
CAS:59-97-2
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of …
Formula:
C10H13ClN2
Purity:
100%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
196.68
Ref: TM-T1680
| 1g | 47.00 € | ||
| 5g | 89.00 € | ||
| 10g | 128.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 66.00 € | ||
| 500mg | 53.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Anandamide
CAS:94421-68-8
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but …
Formula:
C22H37NO2
Purity:
98.76%
Color and Shape:
Light Yellow Oil
Molecular weight:
347.53
Ref: TM-T14046
| 2mg | 72.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 426.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,333.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Naphazoline hydrochloride
CAS:550-99-2
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Formula:
C14H15ClN2
Purity:
97.6%
Color and Shape:
White Crystalline Powder White Crystalline Powder
Molecular weight:
246.74
Ref: TM-T0446
| 1g | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Trimipramine maleate
CAS:521-78-8
Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
Formula:
C24H30N2O4
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
410.51
Ref: TM-T1045
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 73.00 € | ||
| 500mg | 108.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Pericyazine
CAS:2622-26-6
Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.
Formula:
C21H23N3OS
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
365.49
Ref: TM-T16472
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 559.00 € | ||
| 500mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Carbazochrome sodium sulfonate
CAS:51460-26-5
Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
Formula:
C10H11N4NaO5S
Purity:
99.8%
Color and Shape:
Orange Yellow Crystalline Powder
Molecular weight:
322.03
Ref: TM-T0852
| 25mg | 35.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 94.00 € | ||
| 500mg | 217.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
SR59230A
CAS:174689-39-5
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s …
Formula:
C23H29NO6
Purity:
98.84%
Color and Shape:
Solid
Molecular weight:
415.48
Ref: TM-T13016
| 1mg | 52.00 € | ||
| 2mg | 75.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
CB1 antagonist 2
CAS:614726-85-1
CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with …
Formula:
C17H12Cl3N3O
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
380.66
Ref: TM-T14881
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 398.00 € | ||
| 500mg | 900.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Diphenhydramine hydrochloride
CAS:147-24-0
DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.
Formula:
C17H22ClNO
Purity:
99.89%
Color and Shape:
Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)
Molecular weight:
291.82
Ref: TM-T0330
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Oxolinic acid
CAS:14698-29-4
Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY …
Formula:
C13H11NO5
Purity:
98.15% - 98.39%
Color and Shape:
Crystals From Dimethylformamide White Crystalline Powder
Molecular weight:
261.23
Ref: TM-T1233
| 1g | 53.00 € | ||
| 250mg | 40.00 € | ||
| 500mg | 50.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
