G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ML-290
CAS:1482500-76-4
ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. …
Formula:
C24H21F3N2O5S
Color and Shape:
Solid
Molecular weight:
506.49
Ref: TM-T16101
| 1mg | 91.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
SUN B8155
CAS:345893-91-6
SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant …
Formula:
C14H15N3O3
Purity:
99.38% - 99.38%
Color and Shape:
Solid
Molecular weight:
273.29
Ref: TM-T23406
| 1mg | 51.00 € | ||
| 2mg | To inquire |
Estimated delivery in United States, on Monday 7 Apr 2025
Arotinolol
CAS:68377-92-4
Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency …
Formula:
C15H21N3O2S3
Color and Shape:
White Solid
Molecular weight:
371.54
Ref: TM-T10371
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Pumosetrag Hydrochloride
CAS:194093-42-0
Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment …
Formula:
C15H18ClN3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
339.84
Ref: TM-T16683
| 1mg | 46.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
SB-399885 hydrochloride
CAS:402713-81-9
SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
Formula:
C18H22Cl3N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
482.81
Ref: TM-T12843
| 1mg | 44.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
ML314
CAS:1448895-09-7
ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased …
Formula:
C24H28N4O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
420.504
Ref: TM-TQ0075
| 1mg | 52.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Protease-Activated Receptor-4
CAS:245443-52-1
Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
Formula:
C33H46N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
666.77
Ref: TM-T7380
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
SHA 68
CAS:847553-89-3
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with …
Formula:
C26H24FN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.49
Ref: TM-T12895
| 1mg | 41.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Clomipramine hydrochloride
CAS:17321-77-6
Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the …
Formula:
C19H23ClN2·HCl
Purity:
99.04% - 99.47%
Color and Shape:
White To Slightly Yellow Crystalline Powder
Molecular weight:
351.31
Ref: TM-T0255
| 1g | 62.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Timonacic
CAS:444-27-9
Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.
Formula:
C4H7NO2S
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
133.17
Ref: TM-T0221
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Salmeterol
CAS:89365-50-4
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
Formula:
C25H37NO4
Purity:
99.87% - 99.9%
Color and Shape:
Solid
Molecular weight:
415.57
Ref: TM-T12829
| 5mg | 55.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Lamotrigine
CAS:84057-84-1
Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
Formula:
C9H7Cl2N5
Purity:
99.76% - 99.95%
Color and Shape:
White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
Molecular weight:
256.09
Ref: TM-T0680
| 1g | 79.00 € | ||
| 5g | 258.00 € | ||
| 200mg | 37.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Tropisetron hydrochloride
CAS:105826-92-4
Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and …
Formula:
C17H21ClN2O2
Purity:
99.72% - 99.83%
Color and Shape:
Solid
Molecular weight:
320.82
Ref: TM-T1173
| 10mg | 52.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 106.00 € | ||
| 200mg | 159.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
EHP-101
CAS:1818428-24-8
EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related …
Formula:
C28H35NO3
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
433.58
Ref: TM-T13289
| 1mg | 107.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 620.00 € | ||
| 50mg | 868.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
BTRX-335140
CAS:2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic …
Formula:
C25H32FN5O2
Purity:
98% - 99.89%
Color and Shape:
Solid
Molecular weight:
453.55
Ref: TM-T14835
| 1mg | 105.00 € | ||
| 2mg | 155.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 406.00 € | ||
| 25mg | 840.00 € | ||
| 50mg | 1,378.00 € | ||
| 100mg | 1,882.00 € | ||
| 200mg | 2,632.00 € | ||
| 1mL*10mM (DMSO) | 283.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Quetiapine hemifumarate
CAS:111974-72-2
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, …
Formula:
C46H54N6O8S2
Purity:
100% - 99.59%
Color and Shape:
White Crystalline Solid
Molecular weight:
883.09
Ref: TM-T6241
| 1g | 52.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Clopidogrel
CAS:113665-84-2
Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.
Formula:
C16H16ClNO2S
Purity:
98.47%
Color and Shape:
White Powder
Molecular weight:
321.82
Ref: TM-T0182
| 100mg | 48.00 € | ||
| 200mg | 64.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Desipramine hydrochloride
CAS:58-28-6
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of …
Formula:
C18H23ClN2
Purity:
99.58% - 99.94%
Color and Shape:
White To Off-White Powder
Molecular weight:
302.842
Ref: TM-T0991
| 50mg | 42.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 66.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Mizolastine
CAS:108612-45-9
Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever …
Formula:
C24H25FN6O
Purity:
98% - 99.75%
Color and Shape:
Solid
Molecular weight:
432.49
Ref: TM-T0118
| 10mg | 42.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 177.00 € | ||
| 500mg | 298.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Xylometazoline hydrochloride
CAS:1218-35-5
Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.
Formula:
C16H24N2·HCl
Purity:
99.77% - 99.87%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
280.84
Ref: TM-T0042
| 1g | 35.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
