G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Protease-Activated Receptor-4
CAS:245443-52-1
Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
Formula:
C33H46N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
666.77
Ref: TM-T7380
| 1mg | 41.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
ML-290
CAS:1482500-76-4
ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. …
Formula:
C24H21F3N2O5S
Color and Shape:
Solid
Molecular weight:
506.49
Ref: TM-T16101
| 1mg | 91.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
SUN B8155
CAS:345893-91-6
SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant …
Formula:
C14H15N3O3
Purity:
99.38% - 99.38%
Color and Shape:
Solid
Molecular weight:
273.29
Ref: TM-T23406
| 1mg | 51.00 € | ||
| 2mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
SHA 68
CAS:847553-89-3
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with …
Formula:
C26H24FN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.49
Ref: TM-T12895
| 1mg | 41.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Pumosetrag Hydrochloride
CAS:194093-42-0
Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment …
Formula:
C15H18ClN3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
339.84
Ref: TM-T16683
| 1mg | 46.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Arotinolol
CAS:68377-92-4
Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency …
Formula:
C15H21N3O2S3
Color and Shape:
White Solid
Molecular weight:
371.54
Ref: TM-T10371
| 1mg | 41.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
ML314
CAS:1448895-09-7
ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased …
Formula:
C24H28N4O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
420.504
Ref: TM-TQ0075
| 1mg | 52.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
SB-399885 hydrochloride
CAS:402713-81-9
SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
Formula:
C18H22Cl3N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
482.81
Ref: TM-T12843
| 1mg | 44.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Carebastine
CAS:90729-42-3
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Formula:
C32H37NO4
Purity:
99.06%
Color and Shape:
Off-White Solid
Molecular weight:
499.64
Ref: TM-T10680
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 407.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Lamotrigine
CAS:84057-84-1
Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
Formula:
C9H7Cl2N5
Purity:
99.76% - 99.91%
Color and Shape:
White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
Molecular weight:
256.09
Ref: TM-T0680
| 1g | 83.00 € | ||
| 5g | 253.00 € | ||
| 200mg | 41.00 € | ||
| 500mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Maprotiline hydrochloride
CAS:10347-81-6
Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.
Formula:
C20H24ClN
Purity:
100% - 99.84%
Color and Shape:
White Powder
Molecular weight:
313.864
Ref: TM-T0172
| 50mg | 45.00 € | ||
| 100mg | 58.00 € | ||
| 200mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Pericyazine
CAS:2622-26-6
Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.
Formula:
C21H23N3OS
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
365.49
Ref: TM-T16472
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 559.00 € | ||
| 500mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
ML-109
CAS:1186649-91-1
ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
Formula:
C31H29N3O5
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
523.58
Ref: TM-T12073
| 1mg | 36.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 372.00 € | ||
| 100mg | 556.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Diphenhydramine hydrochloride
CAS:147-24-0
DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.
Formula:
C17H22ClNO
Purity:
99.89%
Color and Shape:
Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)
Molecular weight:
291.82
Ref: TM-T0330
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Mirtazapine
CAS:85650-52-8
Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked …
Formula:
C17H19N3
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T0137
| 5mg | 40.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 151.00 € | ||
| 200mg | 248.00 € | ||
| 500mg | 440.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
N6-Ethyladenosine
CAS:14357-08-5
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with …
Formula:
C12H17N5O4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
295.29
Ref: TM-T12161
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 205.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Ramatroban
CAS:116649-85-5
Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
Formula:
C21H21FN2O4S
Purity:
98.12% - 99.96%
Color and Shape:
Crystalline Solid
Molecular weight:
416.47
Ref: TM-T2396
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 347.00 € | ||
| 500mg | 587.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Alprenolol
CAS:13655-52-2
Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of …
Formula:
C15H23NO2
Purity:
99.73% - 99.78%
Color and Shape:
Solid
Molecular weight:
249.35
Ref: TM-T4560
| 50mg | 52.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Tegaserod maleate
CAS:189188-57-6
Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March …
Formula:
C20H27N5O5
Purity:
98% - 99.06%
Color and Shape:
White Powder
Molecular weight:
417.46
Ref: TM-T1551
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 194.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 497.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Deoxycholic acid
CAS:83-44-3
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.
Formula:
C24H40O4
Purity:
99.35%
Color and Shape:
Crystals From Alc Solid
Molecular weight:
392.57
Ref: TM-T2965
| 100mg | 57.00 € | ||
| 500mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
