G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
RU 24969 hemisuccinate
CAS:66611-27-6
RU 24969 is a selective agonist at the 5-HT1A and 5-HT1B receptors.
Formula:
C32H38N4O6
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
574.67
Ref: TM-T2289
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
5-Methoxytryptamine
CAS:608-07-1
5-Methoxytryptamine (3-(2-Aminoethyl)-5-methoxyindole) is a tryptamine derivative that acts as a full agonist at the 5-HT1, …
Formula:
C11H14N2O
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
190.24
Ref: TM-T5271
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
L-DOPA methyl ester (hydrochloride)
CAS:1421-65-4
L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formula:
C10H14ClNO4
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
247.675
Ref: TM-T7654
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Salvinorin A
CAS:83729-01-5
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
Formula:
C23H28O8
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
432.46
Ref: TM-T23306
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Lorcaserin HCl
CAS:846589-98-8
Lorcaserin is a selective serotonin agonist that has been recently approved as a weight loss …
Formula:
C11H14ClN·HCl
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
232.15
Ref: TM-T6572
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Octodrine hydrochloride
CAS:5984-59-8
Octodrine hydrochloride (1,5-Dimethylhexylamine) is a central nervous stimulant that increases the uptake of dopamine and …
Formula:
C8H20ClN
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
165.7
Ref: TM-T22389
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
β-Casomorphin, bovine TFA(72122-62-4(free base))
β-Casomorphin, bovine TFA is an opioid peptide isolated from casein peptone
Formula:
C43H56F3N7O11
Purity:
100%
Color and Shape:
Solid
Molecular weight:
903.95
Ref: TM-T7576L
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
SR17018
CAS:2134602-45-0
SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.
Formula:
C19H18Cl3N3O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
410.72
Ref: TM-T4407
| 1mL*10mM (DMSO) | Discontinued | Request information |
TC-O 9311 free base
CAS:444932-31-4
TC-O 9311 is a potent GPR139 agonist.
Formula:
C20H19N3O4
Purity:
99.24%
Color and Shape:
Soild
Molecular weight:
365.39
Ref: TM-T4626
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information | |
| 1mL*10mM (DMSO) | Discontinued | Request information |
Xylazine
CAS:7361-61-7
Xylazine (BAY 1470) is α2-adrenergic receptor agonist.
Formula:
C12H16N2S
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
220.33
Ref: TM-T7046
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Naltrindole hydrochloride
CAS:111469-81-9
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
Formula:
C26H27ClN2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
450.96
Ref: TM-T12169
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Clocapramine
CAS:47739-98-0
Clocapramine is a D2 and 5-HT2A receptors antagonist.
Formula:
C28H37ClN4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
481.07
Ref: TM-T10837L
| 5mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Naltriben
CAS:111555-58-9
Naltriben, a selective δ2-opioid receptor antagonist and TRPM7 activator, potentiates glioblastoma cell migration and invasion, …
Formula:
C26H25NO4
Purity:
98%
Molecular weight:
415.48
Ref: TM-T78615
| 5mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Levophacetoperane hydrochloride
CAS:23257-56-9
Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine …
Formula:
C14H20ClNO2
Purity:
98%
Molecular weight:
269.77
Ref: TM-T15744
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
(-)-WIN 55,212-3 mesylate
CAS:131543-25-4
(-)-WIN 55,212-3 mesylate is a low-activity enantiomer of WIN 55,212-2 mesylate with no neuroprotective activity …
Formula:
C28H30N2O6S
Color and Shape:
Solid
Molecular weight:
522.61
Ref: TM-T71963
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information |
ST1936 oxalate
CAS:1782228-83-4
ST1936 oxalate: selective 5-HT6 agonist, Ki=13 nM; also binds 5-HT7 (168 nM), 5-HT2B (245 nM).
Formula:
C15H19ClN2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
326.78
Ref: TM-T13007
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Naloxone benzoylhydrazone
CAS:119630-94-3
Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned …
Formula:
C26H27N3O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T12168
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
2-MNG
CAS:2101538-28-5
2-MNG (2-Mercaptonicotinoyl glycine) is a novel melanogenesis inhibitor. 2-MNG inhibits two mechanisms of UV-induced skin …
Formula:
C8H8N2O3S
Color and Shape:
Liquid
Molecular weight:
212.23
Ref: TM-T89029
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1mL*10mM (DMSO) | Discontinued | Request information |
(±)-Epibatidine
CAS:148152-66-3
(±)-Epibatidine is an agonist of nicotinic. (±)-Epibatidine is an agonist of neuronal nAChR.
Formula:
C11H13ClN2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
208.69
Ref: TM-T13468
| 5mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
