G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
AAZ-A 154 hydrobromide
CAS:2930845-96-6
AAZ-A 154 hydrobromide is a selective, competitive, non-hallucinogenic 5-HT2AR antagonist. It promotes neuronal growth in …
Formula:
C14H21BrN2O
Color and Shape:
Liquid
Molecular weight:
313.23
Ref: TM-T200446
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
Burapitant
CAS:537034-22-3
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke …
Formula:
C31H35Cl2F6N3O3
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
682.52
Ref: TM-T69140
| 1mg | 939.00 € | ||
| 5mg | 1,882.00 € | ||
| 25mg | 2,727.00 € | ||
| 50mg | 3,212.00 € | ||
| 100mg | 4,370.00 € |
Estimated delivery in United States, on Wednesday 25 Jun 2025
CB1/2 receptor-1
CAS:1260669-31-5
CB1/2 receptor-1 (compound 5.3) serves as an agonist for CB1/2 receptors and is utilized in …
Formula:
C33H48O2
Color and Shape:
Liquid
Molecular weight:
476.73
Ref: TM-T200966
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
SB-423562
CAS:351490-27-2
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
Formula:
C26H32N2O4
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
436.54
Ref: TM-T12846
| 1mg | 39.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 467.00 € | ||
| 200mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Wednesday 25 Jun 2025
AAZ-A 154
CAS:2481740-94-5
AAZ-A 154 is a selective, competitive, and non-hallucinogenic antagonist of the 5-HT2AR. It promotes neuronal …
Formula:
C14H20N2O
Color and Shape:
Liquid
Molecular weight:
232.32
Ref: TM-T200737
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
Fosrolapitant
CAS:2573694-38-7
Fosrolapitant is an antagonist of the neurokinin 1 (NK1) receptor.
Formula:
C27H29F6N2O8P
Color and Shape:
Liquid
Molecular weight:
654.49
Ref: TM-T201161
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
1'-Naphthoyl-2-methylindole
CAS:80749-33-3
1'-Naphthoyl-2-methylindole (Compound 88) acts as a cannabinoid mimic and an inhibitor of Win 55212-2, displaying …
Formula:
C20H15NO
Color and Shape:
Liquid
Molecular weight:
285.34
Ref: TM-T201477
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
FR-145715
CAS:149917-31-7
FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This …
Formula:
C16H21N5O2S
Color and Shape:
Liquid
Molecular weight:
347.44
Ref: TM-T201582
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
Remlifanserin
CAS:2289704-13-6
Remlifanserin is a potent inverse agonist of the serotonin receptor (5-HT2A).
Formula:
C24H29F2N3O2
Color and Shape:
Liquid
Molecular weight:
429.50
Ref: TM-T201055
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
CCX662
CAS:1226686-54-9
CCX662 is a CXCR7 antagonist. It inhibits the binding of 125I-CXCL12 to CXCR7 with an …
Formula:
C28H37N5O4S
Color and Shape:
Liquid
Molecular weight:
539.69
Ref: TM-T201863
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 25 Jun 2025
16,16-Dimethyl prostaglandin E2
CAS:39746-25-3
16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.
Formula:
C22H36O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
380.52
Ref: TM-T10046
| 1mg | 205.00 € | ||
| 5mg | 949.00 € | ||
| 10mg | 1,786.00 € |
Estimated delivery in United States, on Wednesday 25 Jun 2025
Apafant
CAS:105219-56-5
Apafant (WEB 2086) is a PAF antagonist that blocks eosinophil activation and can be used …
Formula:
C22H22ClN5O2S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
455.96
Ref: TM-T14300
| 1mg | 111.00 € | ||
| 5mg | 274.00 € | ||
| 10mg | 406.00 € | ||
| 25mg | 663.00 € |
Estimated delivery in United States, on Wednesday 25 Jun 2025
BQ-788
CAS:173326-37-9
BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation …
Formula:
C34H51N5O7
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
641.8
Ref: TM-T10595
| 1mg | 137.00 € | ||
| 2mg | 188.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 472.00 € | ||
| 25mg | 753.00 € | ||
| 50mg | 1,017.00 € | ||
| 100mg | 1,378.00 € | ||
| 500mg | 2,737.00 € | ||
| 1mL*10mM (DMSO) | 360.00 € |
Estimated delivery in United States, on Wednesday 25 Jun 2025
Rolapitant hydrochloride
CAS:858102-79-1
Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki …
Formula:
C25H27ClF6N2O2
Purity:
98.35% - 99.79%
Color and Shape:
Solid
Molecular weight:
536.94
Ref: TM-T3724
| 1mg | 153.00 € | ||
| 5mg | 365.00 € | ||
| 10mg | 520.00 € | ||
| 25mg | 780.00 € | ||
| 50mg | 1,054.00 € | ||
| 100mg | 1,425.00 € | ||
| 200mg | 1,882.00 € | ||
| 1mL*10mM (DMSO) | 439.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
Propiram fumarate HCl
CAS:945013-73-0
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study …
Formula:
C16H25N3O·xClH
Purity:
99.25%
Color and Shape:
Soild
Ref: TM-T28453L
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
LIT927
CAS:2172879-52-4
LIT927 (LIT-927) is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to …
Formula:
C17H13ClN2O3
Purity:
99.57% - 99.73%
Color and Shape:
Solid
Molecular weight:
328.75
Ref: TM-T5207
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information | |
| 1mL*10mM (DMSO) | Discontinued | Request information |
TC-O 9311 free base
CAS:444932-31-4
TC-O 9311 is a potent GPR139 agonist.
Formula:
C20H19N3O4
Purity:
99.24%
Color and Shape:
Soild
Molecular weight:
365.39
Ref: TM-T4626
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information | |
| 1mL*10mM (DMSO) | Discontinued | Request information |
SR17018
CAS:2134602-45-0
SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.
Formula:
C19H18Cl3N3O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
410.72
Ref: TM-T4407
| 1mL*10mM (DMSO) | Discontinued | Request information |
2-MNG
CAS:2101538-28-5
2-MNG (2-Mercaptonicotinoyl glycine) is a novel melanogenesis inhibitor. 2-MNG inhibits two mechanisms of UV-induced skin …
Formula:
C8H8N2O3S
Color and Shape:
Liquid
Molecular weight:
212.23
Ref: TM-T89029
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1mL*10mM (DMSO) | Discontinued | Request information |
