Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65624 products of "Quinazoline and Quinoline Derivatives"
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Deschloro-N-ethyl-ketamine Hydrochloride
CAS:Controlled Product<p>Applications Deschloro-N-ethyl-ketamine Hydrochloride is a derivative of Ketamine (K165300), an anesthetic agent and used as a depressant.<br>References Sass, W.C., et al.: Anal. Profiles Drug Subs., 6, 297 (1977), Reich, D.L., et al.: Can. J. Anaesth., 36, 186 (1989),<br></p>Formula:C14H19NO·HClColor and Shape:Off White SolidMolecular weight:253.80Celecoxib Carboxylic Acid
CAS:Controlled ProductFormula:C17H12F3N3O4SColor and Shape:Off WhiteMolecular weight:411.367-Hydroxy Loxapine
CAS:Controlled Product<p>Applications 7-Hydroxy Loxapine is a metabolite of Loxapine (L472750), a neuroleptic medication used to treat patients with schizophrenia and obsessive compulsive disorder.<br>References Kapur, S., et al.: Am. J. Psychiatry, 154, 1525 (1997); Rivers-Bulkeley, N. & Hollender, M.: Am. J. Psychiat., 139, 1345 (1982)<br></p>Formula:C18H18ClN3O2Color and Shape:NeatMolecular weight:343.81N-Deshydroxyethyl Dasatinib-d8
CAS:Controlled ProductFormula:C21D8H15ClN6OSColor and Shape:White SolidMolecular weight:451.013-acetyl-6-chloro-4-(4-ethoxyphenyl)quinolin-2(1H)-one
CAS:Purity:95.0%Molecular weight:341.7900085449219N,N-Dimethyl-4-hydroxymethoxy Clomiphene (~90%, contains ~10% Z-isomer)
CAS:Controlled ProductFormula:C25H26ClNO3Color and Shape:NeatMolecular weight:423.933-Methyl-1-{4-[4-(propan-2-yl)benzenesulfonyl]phenyl}-1H-pyrazol-5-amine
CAS:Purity:97%Molecular weight:355.4599914550781AMOZ-d5
CAS:Controlled Product<p>Applications A labelled metabolite of Nitrofuran.Environmental contaminants; Food contaminants; Heat processing contaminants<br>References Tribalat, L., et al.: Anal. Bioanal. Chem., 386, 2168 (2006), Chu, P., et al.: J. Agric. Food Chem., 55, 2129 (2007),<br></p>Formula:C82H5H10N3O3Color and Shape:NeatMolecular weight:206.254-(5-(3-Hydroxyphenyl)thiophen-2-yl)-2-methylphenol
CAS:Purity:95.0%Molecular weight:282.3599853515625N’-Cyano-N,N-dimethylguanidine
CAS:Controlled Product<p>Impurity Cimetidine EP Impurity G<br>Applications N-Cyano-N',N''-dimethylguanidine (Cimetidine EP Impurity G) is an impurity of Cimetidine (C441650), which acts as a competitive histamine H2-receptor antagonist which inhibits gastric acid secretion and reduces pepsin output (1).<br>References 1. Brimblecombe, R. et al.: J. Int. Med. Res. 1975 Mar:3(2) 86-92<br></p>Formula:C4H8N4Color and Shape:NeatMolecular weight:112.13Brivaracetam-d7
CAS:Controlled Product<p>Applications Brivaracetam-d7, is the labeled analogue of Brivaracetam (B677645), which is a 4-n-propyl analog of levetiracetam (L331500), and a racetam derivative with anticonvulsant properties.<br>References Rosenstiel, P., et al.:Neurotherapeutics, 4 (1), 84 (2007);<br></p>Formula:C11H13D7N2O2Color and Shape:Off White SolidMolecular weight:219.334-[4-[4-(Diphenylmethylene)-1-piperidinyl]-1-hydroxybutyl]-a,a-dimethyl-benzeneacetic Acid
CAS:<p>Applications 4-[4-[4-(Diphenylmethylene)-1-piperidinyl]-1-hydroxybutyl]-α,α-dimethyl-benzeneacetic acid is an impurity of fexofenadine (F322490), the active metabolite of Terfenadine (T114500), a H1-histamine receptor antagonist.<br>References Pratt, E., et al.: Diabet Med., 18, 515 (2001), Mizutani, N., et al.: J. Pharmacol. Sci., 93, 437 (2003), Scadding, G., et al.: Clin. Drug Invest., 25, 153 (2005), Asai, M., et al.: N. Engl. J. Med., 354, 307 (2006),<br></p>Formula:C32H37NO3Color and Shape:NeatMolecular weight:483.64(S)-Linagliptin
CAS:<p>Applications (S)-Linagliptin is a novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.<br>References Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011); Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011);<br></p>Formula:C25H28N8O2Color and Shape:NeatMolecular weight:472.545-Hydroxy Dantrolene
CAS:Controlled ProductFormula:C14H10N4O6Color and Shape:YellowMolecular weight:330.25N-Nitrosodesipramine
CAS:Formula:C18H21N3OColor and Shape:Yellow To Dark YellowMolecular weight:295.385-Morpholinopyridin-3-amine trihydrochloride
CAS:Color and Shape:SolidMolecular weight:288.6000061035156Tert-Butyl 2',6'-dichloro-5,6-dihydro-[4,4'-bipyridine]-1(2H)-carboxylate
CAS:Purity:97.0%Molecular weight:329.22000122070314'-Methylbiphenyl-2-carbonitrile
CAS:Controlled Product<p>Applications 4'-Methylbiphenyl-2-carbonitrile is an intermediate in the synthesis of glycogen synthase kinase-3 inhibitors with a selective sting for glycogen synthase kinase 3α.<br>References Lo Monte, F., et al.: J. Med. Chem., 55, 4407 (2012); Schaarschmidt, D., et al.: ACS. Catalysis., 1, 411 (2011);<br></p>Formula:C14H11NColor and Shape:NeatMolecular weight:193.241-(3-Chloropropyl)-1,3-dihydrobenzimidazol-2-one (>85%)
CAS:Controlled Product<p>Applications 1-(3-Chloropropyl)-1,3-dihydrobenzimidazol-2-one is a benzimidazole derivative used in the preparation of neuroleptic and antiallergic agents.<br>References Strupczewski, J. et al.: J. Med. Chem., 28, 761 (1985); Freter, K. et al.: Arzneim.-Forsch., 35, 272 (1985);<br></p>Formula:C10H11ClN2OPurity:~90%Color and Shape:White To BeigeMolecular weight:210.66N-[2-[[[[1-Methyl-5-[(triphenylmethyl)amino]-1H-pyrazol-4-yl]amino]carbonyl]amino]ethyl]carbamic acid tert-butyl ester
CAS:Purity:97%Molecular weight:540.6680297851562Ref: 10-F863727
1g16.00€5g45.00€10g87.00€1kg2,694.00€25g196.00€50g287.00€100g507.00€250g994.00€500g1,580.00€250mgTo inquireFingolimod
CAS:Controlled Product<p>Applications Fingolimod is a novel immune modulator that prolongs allograft transplant survival in numerous models by inhibiting lymphocyte emigration from lymphoid organs.<br>References Brinkmann, V., et al.: Transplantation, 72, 764 (2001), Brinkmann, et al.: J. Biol. Chem., 277, 24, 21453 (2002), Mtaloubian, M., et al.: Nature, 427, 355 (2004),<br></p>Formula:C19H33NO2Color and Shape:NeatMolecular weight:307.47N-Nitroso Duloxetine
CAS:Formula:C18H18N2O2SColor and Shape:Colourless To Light YellowMolecular weight:326.4132-(CHLOROMETHYL)-4-(2,2,3,3,4,4,4-HEPTAFLUOROBUTOXY)PYRIDINE
CAS:Purity:95.0%Molecular weight:325.6099853515625Quinoline Yellow (Technical Grade)
CAS:<p>Stability Hygroscopic<br>Applications Quinoline yellow, is a yellow powder used in lipstick, lotion, soap, shampoo, bubble bath, ingested drugs, and applied drugs applications.<br></p>Formula:C18H9NNa2O8S2Color and Shape:NeatMolecular weight:477.38Lisinopril Cyclohexyl Analogue
CAS:Controlled Product<p>Impurity Lisinopril EP Impurity F<br>Applications Lisinopril Cyclohexyl Analogue (Lisinopril EP Impurity F) is a Lisinopril (L468985) impurity.<br>References Paraskevas, G., et al.: J. Pharm. Biomed. Anal., 29, 865 (2002),<br></p>Formula:C21H37N3O5Color and Shape:NeatMolecular weight:411.544'-(Bromomethyl)-[1,1'-biphenyl]-2-carboxylic Acid
CAS:Controlled Product<p>Impurity Telmisartan Bromo Acid Impurity<br>Applications An impurity of Telmisartan (D294250). An intermediate in the preparation of antihypertensive agents.<br>References Sharma, M.C. et al.: Adv. Appl. Sci, Res., 1, 120 (2010); Sharma, M.C. et al.: Int. J. Adv. Pharmac. Sci., 1, 249 (2010);<br></p>Formula:C14H11BrO2Color and Shape:NeatMolecular weight:291.14O3-Desethyl Apremilast
CAS:Controlled ProductFormula:C20H20N2O7SColor and Shape:NeatMolecular weight:432.453-Phenyl-5-vinyl-1,2,4-oxadiazole
CAS:<p>Stability Light Sensitive<br>Applications 3-Phenyl-5-vinyl-1,2,4-oxadiazole is a chemical reagent used in the synthesis of pharmaceutically active motifs.<br>References Burns, A. et al.: Org. Biomol. Chem., 8, 2777 (2010); Catanese, B. et al.: Exp. Mol. Path. Supp., 2, 28 (1963);<br></p>Formula:C10H8N2OColor and Shape:NeatMolecular weight:172.1831-(4-Fluorophenyl)-3-thiophen-2-yl-1H-pyrazole-5-carboxylic acid
CAS:Purity:98.0%Color and Shape:Solid, Off-white powderMolecular weight:288.29998779296875Amisulpride-d5
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Labelled Amisulpride (A633250). Amisulpride is a neuroleptic agent, an analogue of Sulpiride (S689145). Amisulpride is used as an antipsychotic. Amisulpride is a dopamine receptor antagonist.<br>References Protais, P., et al.: Neuropharmacol., 24, 861 (1985), Perrault, G., et al.: J. Pharmacol. Exp. Ther., 280, 73 (1997),<br></p>Formula:C17D5H22N3O4SColor and Shape:Off White SolidMolecular weight:374.51N-Formyl Linagliptin
Controlled Product<p>Stability Hygroscopic<br>Applications N-Formyl Linagliptin is a derivative of Linagliptin (L465900), a novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.<br>References Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011); Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011);<br></p>Formula:C26H28N8O3Color and Shape:NeatMolecular weight:500.554-isopropyl-N-(pyridin-3-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Purity:95.0%Molecular weight:283.39001464843757-Hydroxy Quetiapine-d8
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A metabolite of Quetiapine, a Benzothiazepine with mixed serotonin and dopamine receptor antagonistic properties used as an antipsychotic.<br>References Newton, D., et al.: Drug Metab. Dispos., 23, 154 (1995), Tanaka, E., et al.: J. Clin. Pharm. Ther., 24, 7 (1999)<br></p>Formula:C21H17D8N3O3SColor and Shape:NeatMolecular weight:407.564-(Benzyloxy)picolinonitrile
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:210.235992431640622-Descyano-2-ethyl Formyl-tofacitinib
CAS:Controlled Product<p>Applications 2-Descyano-2-ethyl Formyl-tofacitinib is an impurity compound of Tofacitinib(C781351). Tofacitinib is a Janus kinase inhibitor for the treatment of rheumatoid arthritis.<br>References Sheiner, L., et al.: Clin. Pharmacol. Ther., 25, 358 (1979), Dayneka, N., et al.: J. Pharmacokin. Biopharm., 21, 457 (1993), Changelian, P., et al.: Science, 302, 875 (2003), Lee, H., et al.: Clin. Pharmacol. Ther., 73, 348 (2003), Hutmacher, M., et al.: J. Clin. Pharmacol., 47, 238 (2007),<br></p>Formula:C18H25N5O3Color and Shape:NeatMolecular weight:359.4232-(4-Methanesulfonyl-phenyl)-1-(6-methyl-pyridin-3-yl)-ethanone
CAS:<p>Applications This compound is an impurity in the synthesis of Etoricoxib (E934100), a specific inhibitor of COX-2 .<br>References McGeer, P.L., et al.: Exp. Gerontol., 37, 925 (2002), Chenevard, R., et al.: Circulation, 107, 405 (2003)<br></p>Formula:C15H15NO3SColor and Shape:BeigeMolecular weight:289.352-(4-Fluoro-phenyl)-quinoline-4-carboxylic acid
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:267.2590026855469Teflubenzuron
CAS:Controlled Product<p>Applications Teflubenzuron is an benzoylphenylurea chitin synthesis inhibitor used to control a wide range of insect pests and mites in fruit, vegetable, cereal and seed crops. Teflubenzuron is used in cannabis testing kits as a component of pesticide mixes (P698240).<br>References Carro, A.M., et al.: J. Separat. Sci., 35, 2866 (2012); Brock, T.C.M., et al.: Environ. Sci. Pollu. Res., 19, 3610 (2012);<br></p>Formula:C14H6Cl2F4N2O2Color and Shape:Off-WhiteMolecular weight:381.11rac-Mephenytoin
CAS:Controlled Product<p>Applications rac-Mephenytoin is an anticonvulsant agent.<br>References Shimada, et al.: Anal. Biochem., 147, 174 (1975), Dzhagatspanyan. IA., et al.: Pharm. Chem. J., 25, 181 (1991),<br></p>Formula:C12H14N2O2Color and Shape:White SolidMolecular weight:218.25
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