Benzodiazepine Derivatives
Benzodiazepines are organic compounds with a fused bicyclic benzodiazepine core, widely used in the development of drugs with anxiolytic, sedative, anticonvulsant, and muscle relaxant properties. Their derivatives include modified structures that enhance selectivity and pharmacokinetic profiles, enabling the creation of new molecules with advanced therapeutic applications. These compounds are used in the formulation of APIs for the treatment of sleep disorders, anxiety, epilepsy, and muscle spasms. Additionally, benzodiazepine derivatives are essential in the research of new psychotropic agents and in optimising neurological treatments.
At CymitQuimica, we offer high-purity benzodiazepine derivatives for applications in chemical synthesis, pharmaceutical development, and neuroscience.
Found 332 products of "Benzodiazepine Derivatives"
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4-Boc-8-Chloro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C14H19ClN2O2Purity:97.0%Molecular weight:282.777,8-Dimethoxy-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C11H16N2O2Purity:97.0%Molecular weight:208.2617-BROMO-2,3,4,5-TETRAHYDRO-1H-BENZO[E][1,4]DIAZEPINE HCL
CAS:Formula:C9H12BrClN2Purity:95.0%Molecular weight:263.568-Chloro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C9H11ClN2Purity:97.0%Color and Shape:SolidMolecular weight:182.652,3,4,5-Tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C9H12N2Purity:97.0%Color and Shape:White to yellow/orange crystalline powderMolecular weight:148.2098-Bromo-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one
CAS:Formula:C9H9BrN2OPurity:97.0%Molecular weight:241.0884-Boc-7,8-Dimethoxy-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C16H24N2O4Purity:97.0%Molecular weight:308.3787-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C10H14N2Purity:97.0%Color and Shape:SolidMolecular weight:162.2364-Boc-7-Hydroxy-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C14H20N2O3Purity:97.0%Molecular weight:264.3251,2,4,5-Tetrahydro-benzo[e][1,4]diazepin-3-one
CAS:Formula:C9H10N2OPurity:97.0%Color and Shape:SolidMolecular weight:162.1927-Fluoro-3,4-dihydro-4-methyl-1H-1,4-benzodiazepine-2,5-dione
CAS:Formula:C10H9FN2O2Purity:97%Molecular weight:208.1927-AMINO-4-BOC-4,5-DIHYDRO-1H-BENZO[E][1,4]DIAZEPIN-2(3H)-ONE
CAS:Formula:C14H19N3O3Purity:97.0%Molecular weight:277.3242-(2-Aminoacetamido)-5-nitro-2'-chlorobenzophenone Hydrochloride (Clonazepam Impurity)
CAS:Controlled ProductFormula:C15H12ClN3O4·ClHColor and Shape:WhiteMolecular weight:370.18743,3-Dimethyl Clobazam
Controlled ProductFormula:C18H17ClN2O2Color and Shape:NeatMolecular weight:328.79N,N-Dimethylformamide Diethyl Acetal
CAS:Controlled Product<p>Stability Moisture Sensitive<br>Applications N,N-Dimethylformamide Diethyl Acetal is used as a reagent in the design of EGF-R tyrosine kinase inhibitors. Also used in the synthesis of aminopyridine derivatives.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Traxler, P. et al.: J. Med. Chem., 40, 3601 (1997); Cheikh, N. et al.: Tetrahedron, 69, 1234 (2013);<br></p>Formula:C7H17NO2Color and Shape:NeatMolecular weight:147.223-Amino-4-(2-fluorophenyl)-1-methyl-6-nitroquinolin-2(1H)-one
CAS:Controlled ProductFormula:C16H12FN3O3Color and Shape:NeatMolecular weight:313.28N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide
CAS:Controlled Product<p>Applications N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formula:C14H10BrClN2O2Color and Shape:Light Yellow To BeigeMolecular weight:353.602-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide
CAS:Controlled Product<p>Applications 2-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formula:C14H10Br2N2O2Color and Shape:NeatMolecular weight:398.05Alprazolam 5,6-Epoxide
CAS:Controlled Product<p>Applications Alprazolam derivative.<br>References Hester, J. et al., J. of Med. Chem. 23, 643 (1980)<br></p>Formula:C17H13ClN4OColor and Shape:NeatMolecular weight:324.773-Amino-6-chloro-3,4-dihydro-2-methyl-4-phenyl-4-quinazolinol
CAS:Controlled ProductFormula:C15H14ClN3OColor and Shape:NeatMolecular weight:287.742-Amino-5-nitrobenzophenone
CAS:Controlled ProductFormula:C13H10N2O3Color and Shape:NeatMolecular weight:242.23Flumazenil Carboxylic Acid-D3
Controlled Product<p>Applications Flumazenil Carboxylic Acid-D3 is an isotope labelled form of Flumazenil Carboxylic Acid (F500455); a derivative of Flumazenil (F500455), a benzodiazepine antagonist that can prevent or abolish (at the receptor level) the effects of a benzodiazepine.<br>References Brogden, R. & Goa, K.: Drugs, 35, 448 (1988); Klotz, U. & Kanto, J.: Clin. Pharmacokinet., 14, 1 (1988)<br></p>Formula:C13H7D3FN3O3Color and Shape:NeatMolecular weight:278.257-Aminonorflunitrazepam
CAS:Controlled ProductFormula:C15H12FN3OColor and Shape:Light YellowMolecular weight:269.272-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine
CAS:Controlled Product<p>Applications 2-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine is an impurity of Alprazolam (A575650.<br>References Hester, J.B., et al.: J. Org. Chem., 44, 2688, (1979); Anjaneyulu, Y., et al.: Asian. J. Chem., 19, 3375 (2007);<br></p>Formula:C17H15ClN4OColor and Shape:White To Off-WhiteMolecular weight:326.783-Methyl Clobazam
CAS:Controlled Product<p>Applications 3-Methyl Clobazam is a metabolite of Clobazam (C582500), a benzodiazepine psychotherapeutic agent that has proven efficacy against multiple seizure types. An anxiolytic; anticonvulsant.<br>References Gastaut, H., et al.: Epilepsia, 20, 437 (1979); Guberman, A., et al.: Can J. Neurol. Sci., 17, 311 (1990); Munn, R., et al.: Pediatr. Neurol. 9, 465 (1993)<br></p>Formula:C17H15ClN2O2Color and Shape:NeatMolecular weight:314.77Clobazam CIV
CAS:Controlled Product<p>Clobazam (inn) and methyprylon (inn)</p>Formula:C16H13ClN2O2Color and Shape:White Crystalline PowderMolecular weight:300.066562-(2-Amino-5-bromobenzoyl)pyridine
CAS:<p>2-(2-Amino-5-bromobenzoyl)pyridine (2ABBP) is a chemical compound with the molecular formula C10H7BrN3. It is a glucuronide conjugate of 2-amino-5-bromobenzoic acid and has been used as an immunological reagent in the form of a monoclonal antibody. 2ABBP binds to dryopteris, which is a plant species that contains polyphenols called pteridines. 2ABBP has been shown to have anti-inflammatory properties in rat liver microsomes and cell culture experiments. The mechanism of action may involve inhibition of cyclooxygenase enzymes, which are involved in prostaglandin synthesis. 2ABBP also binds to human serum albumin and chaperones, proteins that bind other proteins or small molecules. The biological activity of 2ABBP may be due to its ability to form coval</p>Formula:C12H9BrN2OPurity:Min. 95%Molecular weight:277.12 g/molRef: 4Z-E-153009
Discontinued productRef: 4Z-A-231026
Discontinued product7-Amino Clonazepam-d4
CAS:Controlled Product<p>Applications A labelled major metabolite of Clonazepam (C587080).<br>References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),<br></p>Formula:C152H4H8ClN3OColor and Shape:NeatMolecular weight:289.75
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