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Angiogénesis

Angiogénesis

Los inhibidores de la angiogénesis son compuestos que interfieren con la formación de nuevos vasos sanguíneos, un proceso crucial en el crecimiento y la metástasis del cáncer. Al inhibir la angiogénesis, estos compuestos pueden restringir el suministro de sangre a los tumores, ralentizando o deteniendo su crecimiento. Los inhibidores de la angiogénesis son esenciales en la investigación del cáncer y en el desarrollo terapéutico, proporcionando información sobre los mecanismos de progresión tumoral y ofreciendo posibles tratamientos para el cáncer y otras enfermedades relacionadas con la angiogénesis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la angiogénesis de alta calidad para apoyar su investigación en oncología y biología vascular.

Subcategorías de "Angiogénesis"

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Se han encontrado 1483 productos de "Angiogénesis"

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  • Bleximenib oxalate

    CAS:
    <p>Bleximenib oxalate (Menin-MLL inhibitor 24 oxalate) is a menin-MLL inhibitor that blocks the binding of the menin-KMT2A complex to chromatin at gene promoters.</p>
    Fórmula:C34H52FN7O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:689.82
  • Poseltinib

    CAS:
    <p>Poseltinib is an oral, irreversible BTK inhibitor (IC50 1.95 nM) with higher selectivity over BMX, TEC, and TXK, blocking BCR, FcR, and TLR signaling.</p>
    Fórmula:C26H26N6O3
    Forma y color:Solid
    Peso molecular:470.52
  • Conteltinib tetrahydrochloride


    <p>Conteltinibtetrahydrochloride (CT-707 tetrahydrochloride) is the tetrahydrochloride form of Conteltinib. It acts as an inhibitor for FAK (IC50=1.6 nM), ALK, and Pyk2. When used in combination with Cabozantinib, Conteltinib tetrahydrochloride exhibits a synergistic antitumor effect.</p>
    Fórmula:C32H49Cl4N9O3S
    Forma y color:Solid
    Peso molecular:781.667
  • Afatinib D6

    CAS:
    <p>Afatinib D6 (BIBW 2992 D6) is a deuterium-labeled Afatinib. Afatinib is an irreversible EGFR family inhibitor.</p>
    Fórmula:C24H25ClFN5O3
    Forma y color:Solid
    Peso molecular:491.98
  • Aflibercept

    CAS:
    <p>Aflibercept has a wide range of applications in life science related research.</p>
    Forma y color:Liquid
  • Disitamab

    CAS:
    <p>Disitamab (RC48-0) is a humanized anti-HER2 monoclonal antibody used in ADC synthesis.</p>
    Pureza:95.00%
    Forma y color:Liquid
  • KG-548

    CAS:
    <p>KG-548 is a dual inhibitor of ARNT/TACC3 and HIF-1α, inhibiting lactate production, and can be used in cancer research.</p>
    Fórmula:C9H4F6N4
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:282.15
  • SM1-71

    CAS:
    <p>SM1-71 is a TAK1 inhibitor that inhibits MKNK2 and RSK2.SM1-71 acts as a kinase probe with anticancer activity.</p>
    Fórmula:C24H26ClN7O
    Pureza:96%
    Forma y color:Solid
    Peso molecular:463.96
  • EW-7195

    CAS:
    <p>EW-7195 inhibits ALK5/TGFβR1 (&gt;300x selective over p38α) with 4.83 nM IC50, blocking TGF-β1 signaling, EMT, and breast cancer lung metastasis.</p>
    Fórmula:C23H18N8
    Pureza:98.76%
    Forma y color:Solid
    Peso molecular:406.44
  • Momelotinib sulfate

    CAS:
    <p>Momelotinib sulfate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.</p>
    Fórmula:C23H26N6O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:610.62
  • Itacitinib adipate

    CAS:
    Itacitinib adipate: oral JAK1 inhibitor, tested in phase II myelofibrosis trial.
    Fórmula:C32H33F4N9O5
    Forma y color:Solid
    Peso molecular:699.66
  • BI-3663

    CAS:
    <p>BI-3663 is a selective PTK2/FAK PROTAC with cereblon ligands, degrading PTK2 (IC50: 18 nM), and shows anti-cancer properties.</p>
    Fórmula:C44H42F3N7O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:917.84
  • Regorafenib-d3

    CAS:
    <p>Regorafenib D3 is a deuterium labeled Regorafenib. Regorafenib is a multi-targeted receptor inhibitor of tyrosine kinase.</p>
    Fórmula:C21H15ClF4N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:485.83
  • Lestaurtinib

    CAS:
    <p>Lestaurtinib (CEP 701) is a FLT3 inhibitor that inhibits the phosphorylation of RPTKs and can be used to study leukemia.</p>
    Fórmula:C26H21N3O4
    Pureza:99.17%
    Forma y color:Off-White Solid
    Peso molecular:439.46
  • GMB-475

    CAS:
    <p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>
    Fórmula:C43H46F3N7O7S
    Pureza:98.78% - >99.99%
    Forma y color:Solid
    Peso molecular:861.93
  • Gefitinib-based PROTAC 3

    CAS:
    <p>Gefitinib-PROTAC 3 degrades EGFR in cancer cells; DC50s: 11.7 nM (HCC827) and 22.3 nM (H3255).</p>
    Fórmula:C47H57ClFN7O8S
    Pureza:97.29% - 98.25%
    Forma y color:Solid
    Peso molecular:934.51
  • N-piperidine Ibrutinib

    CAS:
    <p>N-piperidine Ibrutinib is a potent BTK inhibitor with IC50s of 51.0 for WT BTK and 30.7 nM for C481S BTK respectively.</p>
    Fórmula:C22H22N6O
    Pureza:96.65%
    Forma y color:Solid
    Peso molecular:386.45
  • Nastorazepide

    CAS:
    <p>Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity.</p>
    Fórmula:C29H36N4O5
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:520.62
  • Protein kinase inhibitor 6

    CAS:
    <p>Protein kinase inhibitor 6 is a protein kinase inhibitor.</p>
    Fórmula:C13H9FN2S
    Pureza:98.01%
    Forma y color:Solid
    Peso molecular:244.29
  • 2,4-DPD

    CAS:
    <p>2,4-DPD is competitive inhibitor of the oxygen-sensing enzyme HIF-α prolyl hydroxylase (HIF-PH)</p>
    Fórmula:C11H13NO4
    Pureza:99.74%
    Forma y color:Yellow Solid Crystalline
    Peso molecular:223.23