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Angiogénesis

Angiogénesis

Los inhibidores de la angiogénesis son compuestos que interfieren con la formación de nuevos vasos sanguíneos, un proceso crucial en el crecimiento y la metástasis del cáncer. Al inhibir la angiogénesis, estos compuestos pueden restringir el suministro de sangre a los tumores, ralentizando o deteniendo su crecimiento. Los inhibidores de la angiogénesis son esenciales en la investigación del cáncer y en el desarrollo terapéutico, proporcionando información sobre los mecanismos de progresión tumoral y ofreciendo posibles tratamientos para el cáncer y otras enfermedades relacionadas con la angiogénesis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la angiogénesis de alta calidad para apoyar su investigación en oncología y biología vascular.

Subcategorías de "Angiogénesis"

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Se han encontrado 1431 productos de "Angiogénesis"

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  • Regorafenib mesylate

    CAS:
    <p>Regorafenib mesylate is an oral multi-kinase inhibitor targeting VEGFR, PDGFRβ, Kit, RET, Raf-1 with strong anti-tumor and anti-angiogenic effects.</p>
    Fórmula:C22H19ClF4N4O6S
    Forma y color:Solid
    Peso molecular:578.92
  • Tropisetron

    CAS:
    <p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>
    Fórmula:C17H20N2O2
    Pureza:99.68%
    Forma y color:White Solid
    Peso molecular:284.35
  • SKLB4771

    CAS:
    <p>SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.</p>
    Fórmula:C25H27N7O3S2
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:537.66
  • 2-(1,8-naphthyridin-2-yl)phenol

    CAS:
    <p>2-NP is a STAT1 enhancer.</p>
    Fórmula:C14H10N2O
    Pureza:99.33% - 99.82%
    Forma y color:Solid
    Peso molecular:222.24
  • Radotinib

    CAS:
    <p>Radotinib (IY-5511), and sometimes referred to by its investigational name IY5511, is a drug for the treatment of different types of Y, most notably</p>
    Fórmula:C27H21F3N8O
    Pureza:99.13% - 99.97%
    Forma y color:Solid
    Peso molecular:530.5
  • BMS817378

    CAS:
    <p>BMS817378 is a potent and selective inhibitor of MET(IC50 : 1.7 nM).</p>
    Fórmula:C24H18ClF2N4O7P
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:578.85
  • SPHINX31

    CAS:
    <p>SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).</p>
    Fórmula:C27H24F3N5O2
    Pureza:98.81% - 99.3%
    Forma y color:Solid
    Peso molecular:507.51
  • Ibuprofen Lysine

    CAS:
    <p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>
    Fórmula:C19H32N2O4
    Pureza:99.26%
    Forma y color:Coa
    Peso molecular:352.47
  • Benidipine hydrochloride

    CAS:
    <p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>
    Fórmula:C28H32ClN3O6
    Pureza:99.80%
    Forma y color:Solid
    Peso molecular:542.03
  • Arnebin 1

    CAS:
    <p>(Rac)-Arnebin 1 (beta, beta-dimethylacrylshikonin) has anti-tumor, anti-inflammatory, anti-immune deficiency and protecting liver.</p>
    Fórmula:C21H22O6
    Pureza:98.76% - 99.81%
    Forma y color:Solid
    Peso molecular:370.396
  • Regorafenib monohydrate

    CAS:
    <p>Regorafenib Monohydrate is a novel oral multikinase inhibitor with IC50 values of 13, 4.2, 46, 22, 7, 1.5, 2.5, 28, 19 nM for VEGFR1, murine VEGFR2, murine</p>
    Fórmula:C21H17ClF4N4O4
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:500.83
  • AZD3759 hydrochloride

    CAS:
    <p>AZD3759 hydrochloride is an oral, CNS-penetrant EGFR inhibitor with IC50s of 0.2/0.3/0.2 nM.</p>
    Fórmula:C22H24Cl2FN5O3
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:496.36
  • Merestinib dihydrochloride

    CAS:
    <p>Merestinib dihydrochloride (LY2801653 dihydrochloride) is a kinase inhibitor with antitumor activity that inhibits MET and MKNK1/2.</p>
    Fórmula:C30H24Cl2F2N6O3
    Forma y color:Solid
    Peso molecular:625.45
  • CEP-28122 mesylate salt


    <p>CEP-28122 mesylate, a diaminopyrimidine, selectively inhibits ALK with IC50 of 1.9 nM and exhibits antitumor effects.</p>
    Fórmula:C29H39ClN6O6S
    Forma y color:Solid
    Peso molecular:635.17
  • JK-P3

    CAS:
    <p>JK-P3: a pyrazole inhibitor of VEGFR-2 (IC50: 7.8 μM), stalls FGFR 1/3 in vitro, halts HUVEC wound healing/tube formation, not cell growth.</p>
    Fórmula:C18H17N3O3
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:323.35
  • KX2-361

    CAS:
    <p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>
    Fórmula:C24H24FN3O2
    Pureza:99.64% - 99.68%
    Forma y color:Solid
    Peso molecular:405.46
  • Syk Inhibitor II dihydrochloride

    CAS:
    <p>Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.</p>
    Fórmula:C14H17Cl2F3N6O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:413.22
  • Blu-782

    CAS:
    <p>Blu-782 (ALK2-IN-1) is a activin receptor-like kinase-2 (ALK2) inhibitor ( IC50 of &lt;10 nM)</p>
    Fórmula:C31H42N6O4
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:562.7
  • Filgotinib

    CAS:
    <p>Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and TYK2 are 10 nM, 28 nM, 810 nM, and 116 nM, respectively.</p>
    Fórmula:C21H23N5O3S
    Pureza:98.03% - ≥95%
    Forma y color:Solid
    Peso molecular:425.5
  • CZC-8004

    CAS:
    <p>CZC-8004 (CZC-00008004) is a pan-kinase(ABL kinase) inhibitor and binds a range of tyrosine kinases.</p>
    Fórmula:C17H16FN5
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:309.34