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Angiogénesis

Angiogénesis

Los inhibidores de la angiogénesis son compuestos que interfieren con la formación de nuevos vasos sanguíneos, un proceso crucial en el crecimiento y la metástasis del cáncer. Al inhibir la angiogénesis, estos compuestos pueden restringir el suministro de sangre a los tumores, ralentizando o deteniendo su crecimiento. Los inhibidores de la angiogénesis son esenciales en la investigación del cáncer y en el desarrollo terapéutico, proporcionando información sobre los mecanismos de progresión tumoral y ofreciendo posibles tratamientos para el cáncer y otras enfermedades relacionadas con la angiogénesis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la angiogénesis de alta calidad para apoyar su investigación en oncología y biología vascular.

Subcategorías de "Angiogénesis"

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Se han encontrado 1522 productos de "Angiogénesis"

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  • Verteporfin

    CAS:
    <p>Verteporfin (BPD-MA) is a YAP inhibitor that inhibits YAP-TEAD interactions.</p>
    Fórmula:C41H42N4O8
    Pureza:95.37% - 99.82%
    Forma y color:Dark Green To Black Solid
    Peso molecular:718.79
  • Radotinib

    CAS:
    <p>Radotinib (IY-5511), and sometimes referred to by its investigational name IY5511, is a drug for the treatment of different types of Y, most notably</p>
    Fórmula:C27H21F3N8O
    Pureza:99.13% - 99.97%
    Forma y color:Solid
    Peso molecular:530.5
  • Vactosertib Hydrochloride

    CAS:
    Vactosertib Hydrochloride (EW-7197 Hydrochloride) is an ALK5 inhibitor, a TGF-β receptor I inhibitor with antimetastatic and anticancer effects.
    Fórmula:C22H19ClFN7
    Pureza:98.03%
    Forma y color:Solid
    Peso molecular:435.89
  • WS3

    CAS:
    WS3, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase pathway.
    Fórmula:C28H30F3N7O3
    Pureza:97.93% - 99.94%
    Forma y color:Solid
    Peso molecular:569.58
  • Endoxifen (Z-isomer)

    CAS:
    Endoxifen Z-isomer (EDX) is a key active metabolite of tamoxifen with higher affinity and specificity to estrogen receptors that inhibits aromatase activity.
    Fórmula:C25H27NO2
    Pureza:99.19% - 99.81%
    Forma y color:Solid
    Peso molecular:373.49
  • Protein kinase inhibitor 6

    CAS:
    <p>Protein kinase inhibitor 6 is a protein kinase inhibitor.</p>
    Fórmula:C13H9FN2S
    Pureza:98.01%
    Forma y color:Solid
    Peso molecular:244.29
  • PND-1186

    CAS:
    PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).
    Fórmula:C25H26F3N5O3
    Pureza:99.14% - 99.75%
    Forma y color:Solid
    Peso molecular:501.5
  • Ki20227

    CAS:
    Ki-20227 is a specific c-Fms tyrosine kinase(CSF1R) inhibitor (IC50: 2 nM).
    Fórmula:C24H24N4O5S
    Pureza:98.97% - 99.88%
    Forma y color:Solid
    Peso molecular:480.54
  • 2,4-DPD

    CAS:
    <p>2,4-DPD is competitive inhibitor of the oxygen-sensing enzyme HIF-α prolyl hydroxylase (HIF-PH)</p>
    Fórmula:C11H13NO4
    Pureza:99.74%
    Forma y color:Yellow Solid Crystalline
    Peso molecular:223.23
  • (Z)-Semaxinib

    CAS:
    (Z)-Semaxinib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor (IC50: 1.23 μM), 20-fold more selective for VEGFR over PDGFRβ, no inhibition for
    Fórmula:C15H14N2O
    Pureza:98.82% - ≥95%
    Forma y color:Solid
    Peso molecular:238.28
  • 2-(1,8-naphthyridin-2-yl)phenol

    CAS:
    <p>2-NP is a STAT1 enhancer.</p>
    Fórmula:C14H10N2O
    Pureza:99.33% - 99.82%
    Forma y color:Solid
    Peso molecular:222.24
  • Avitinib maleate

    CAS:
    Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
    Fórmula:C30H30FN7O6
    Pureza:98% - 99.74%
    Forma y color:Solid
    Peso molecular:603.61
  • AG-1557 hydrochloride (189290-58-2(free base))


    AG-1557 hydrochloride is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).
    Fórmula:C16H15ClIN3O2
    Pureza:98.64%
    Forma y color:Solid
    Peso molecular:443.66
  • Tropisetron

    CAS:
    Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.
    Fórmula:C17H20N2O2
    Pureza:99.68%
    Forma y color:White Solid
    Peso molecular:284.35
  • CCT241736

    CAS:
    CCT241736 is an orally bioavailable dual FLT3/Aurora kinase inhibitor that also inhibits clinically relevant FLT3-resistant mutants including FLT3-ITD and FLT3
    Fórmula:C22H23Cl2N7
    Pureza:96.2% - 99.81%
    Forma y color:Solid
    Peso molecular:456.37
  • Ripretinib

    CAS:
    Ripretinib (DCC-2618) is an orally bioavailable inhibitor of KIT and PDGFRA.
    Fórmula:C24H21BrFN5O2
    Pureza:99.07% - 99.62%
    Forma y color:Solid
    Peso molecular:510.36
  • Naluzotan

    CAS:
    <p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:450.64
  • ASP3026

    CAS:
    ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies,and Positive for Anaplastic Lymphoma Kinase.
    Fórmula:C29H40N8O3S
    Pureza:98.78% - 99.81%
    Forma y color:Solid
    Peso molecular:580.74
  • AG 1406

    CAS:
    <p>AG 1406 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2.</p>
    Fórmula:C16H18N2O
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:254.33
  • Bafetinib

    CAS:
    <p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>
    Fórmula:C30H31F3N8O
    Pureza:94.16% - 99.68%
    Forma y color:Solid
    Peso molecular:576.62