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Angiogénesis

Angiogénesis

Los inhibidores de la angiogénesis son compuestos que interfieren con la formación de nuevos vasos sanguíneos, un proceso crucial en el crecimiento y la metástasis del cáncer. Al inhibir la angiogénesis, estos compuestos pueden restringir el suministro de sangre a los tumores, ralentizando o deteniendo su crecimiento. Los inhibidores de la angiogénesis son esenciales en la investigación del cáncer y en el desarrollo terapéutico, proporcionando información sobre los mecanismos de progresión tumoral y ofreciendo posibles tratamientos para el cáncer y otras enfermedades relacionadas con la angiogénesis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la angiogénesis de alta calidad para apoyar su investigación en oncología y biología vascular.

Subcategorías de "Angiogénesis"

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Se han encontrado 1884 productos de "Angiogénesis"

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  • Tesevatinib

    CAS:
    Tesevatinib (XL-647) is an oral, multi-targeted tyrosine kinase inhibitor.Cost-effective and quality-assured.
    Fórmula:C24H25Cl2FN4O2
    Pureza:97.89% - 98.66%
    Forma y color:Solid
    Peso molecular:491.39
  • WZ-3146

    CAS:
    WZ3146: EGFR(L858R/E746_A750) inhibitor, IC50=2 nM, selective, doesn't block ERBB2(T798I).
    Fórmula:C24H25ClN6O2
    Pureza:97.15%
    Forma y color:Solid
    Peso molecular:464.95
  • CNX-2006

    CAS:
    CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM, with very weak inhibition at wild-type EGFR.
    Fórmula:C26H27F4N7O2
    Pureza:98.85% - 99.16%
    Forma y color:Solid
    Peso molecular:545.53
  • Arnebin 1

    CAS:
    <p>(Rac)-Arnebin 1 (beta, beta-dimethylacrylshikonin) has anti-tumor, anti-inflammatory, anti-immune deficiency and protecting liver.</p>
    Fórmula:C21H22O6
    Pureza:98.76% - 99.81%
    Forma y color:Solid
    Peso molecular:370.396
  • Merestinib dihydrochloride

    CAS:
    Merestinib dihydrochloride (LY2801653 dihydrochloride) is a kinase inhibitor with antitumor activity that inhibits MET and MKNK1/2.
    Fórmula:C30H24Cl2F2N6O3
    Forma y color:Solid
    Peso molecular:625.45
  • Syk Inhibitor II dihydrochloride

    CAS:
    Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.
    Fórmula:C14H17Cl2F3N6O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:413.22
  • GluR6 antagonist-1

    CAS:
    GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.
    Fórmula:C15H11ClN2OS
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:302.78
  • Adaphostin

    CAS:
    Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.
    Fórmula:C24H27NO4
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:393.48
  • Theliatinib tartrate

    CAS:
    Theliatinib: oral EGFR blocker, Ki 0.05 nM, IC50 3 nM (wild-type), 22 nM (T790M/L858R), >50x kinase selectivity.
    Fórmula:C29H32N6O8
    Forma y color:Solid
    Peso molecular:592.6
  • Trastuzumab

    CAS:
    Trastuzumab is a humanized monoclonal antibody for patients with invasive breast cancers that overexpress HER2.
    Pureza:97.1% (SDS-PAGE); 99.2% (SEC-HPLC) - SDS-PAGE: 97.1%;SEC-HPLC: 99.2%
    Forma y color:Liquid
    Peso molecular:Approximately 145.53 kDa
  • (Z)-SU4312

    CAS:
    <p>(Z)-SU4312 is a inhibitor of MAO-B and NOS(IC50 value of 0.2 μM, 19.0μM,respectively).</p>
    Fórmula:C17H16N2O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:264.32
  • Silymarin

    CAS:
    Silymarin, a liver-aiding polyphenolic flavonoid, is extracted from milk thistle seeds.
    Fórmula:C25H22O10
    Pureza:98%
    Forma y color:Yellow And Brown Powder
    Peso molecular:482.44
  • 1-Naphthyl PP1

    CAS:
    <p>1-Naphthyl PP1 (1-NA-PP 1) is a selective src inhibitor(v-Src and c-Fyn, c-Abl, CDK2 and CAMK II with IC50s of 1.0, 0.6, 0.6, 18 and 22 μM, respectively)</p>
    Fórmula:C19H19N5
    Pureza:99.85%
    Forma y color:White Cyrstalline Solid
    Peso molecular:317.39
  • Gefitinib dihydrochloride

    CAS:
    Gefitinib dihydrochloride: orally active, selective EGFR inhibitor (IC50: 33-54 nM), hinders tumor growth, induces autophagy and apoptosis in cancer research.
    Fórmula:C22H26Cl3FN4O3
    Forma y color:Solid
    Peso molecular:519.82
  • FGFR2-IN-3 hydrochloride

    CAS:
    FGFR2-IN-3 hydrochloride is a selective, orally active FGFR2 inhibitor.
    Fórmula:C28H25ClFN7O2
    Forma y color:Solid
    Peso molecular:546.0
  • Entrectinib

    CAS:
    Entrectinib (RXDX-101) is an orally Trk, ROS1, and ALK inhibitor. Entrectinib exhibits antitumor activity. Cost-effective and quality-assured.
    Fórmula:C31H34F2N6O2
    Pureza:98.03% - 99.61%
    Forma y color:Solid
    Peso molecular:560.64
  • Olmutinib hydrochloride

    CAS:
    Olmutinib is a third-gen EGFR inhibitor for T790M-positive lung cancer, blocking phosphorylation and tumor pathways. Approved in Korea (2016).
    Fórmula:C26H28Cl2N6O2S
    Forma y color:Solid
    Peso molecular:559.51
  • E-4031 dihydrochloride

    CAS:
    E-4031 dihydrochloride is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by blocking ERG K+ channels (IC50 = 29 nM)
    Fórmula:C21H29Cl2N3O3S
    Pureza:99.31% - 99.87%
    Forma y color:Solid
    Peso molecular:474.44
  • WS6

    CAS:
    WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase pathway.
    Fórmula:C29H31F3N6O3
    Pureza:97.65% - 99.95%
    Forma y color:Solid
    Peso molecular:568.59
  • Quizartinib HCl

    CAS:
    Quizartinib (AC220/AC010220) is an oral FLT3/STK1 inhibitor for treating AML, blocking kinase-driven cell proliferation and promoting apoptosis.
    Fórmula:C29H34Cl2N6O4S
    Forma y color:Solid
    Peso molecular:633.59