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Angiogénesis

Angiogénesis

Los inhibidores de la angiogénesis son compuestos que interfieren con la formación de nuevos vasos sanguíneos, un proceso crucial en el crecimiento y la metástasis del cáncer. Al inhibir la angiogénesis, estos compuestos pueden restringir el suministro de sangre a los tumores, ralentizando o deteniendo su crecimiento. Los inhibidores de la angiogénesis son esenciales en la investigación del cáncer y en el desarrollo terapéutico, proporcionando información sobre los mecanismos de progresión tumoral y ofreciendo posibles tratamientos para el cáncer y otras enfermedades relacionadas con la angiogénesis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la angiogénesis de alta calidad para apoyar su investigación en oncología y biología vascular.

Subcategorías de "Angiogénesis"

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Se han encontrado 2061 productos de "Angiogénesis"

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  • Blu-782

    CAS:
    <p>Blu-782 (ALK2-IN-1) is a activin receptor-like kinase-2 (ALK2) inhibitor ( IC50 of &lt;10 nM)</p>
    Fórmula:C31H42N6O4
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:562.7
  • Radotinib

    CAS:
    <p>Radotinib (IY-5511), and sometimes referred to by its investigational name IY5511, is a drug for the treatment of different types of Y, most notably</p>
    Fórmula:C27H21F3N8O
    Pureza:99.13% - 99.97%
    Forma y color:Solid
    Peso molecular:530.5
  • Masitinib

    CAS:
    Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in animals, specifically dogs.
    Fórmula:C28H30N6OS
    Pureza:97.56% - >99.99%
    Forma y color:Solid
    Peso molecular:498.64
  • Mubritinib

    CAS:
    Mubritinib (TAK-165) (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM.
    Fórmula:C25H23F3N4O2
    Pureza:98.61% - 99.85%
    Forma y color:Solid
    Peso molecular:468.47
  • MAZ51

    CAS:
    MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
    Fórmula:C21H18N2O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:314.38
  • Theliatinib tartrate

    CAS:
    Theliatinib: oral EGFR blocker, Ki 0.05 nM, IC50 3 nM (wild-type), 22 nM (T790M/L858R), >50x kinase selectivity.
    Fórmula:C29H32N6O8
    Forma y color:Solid
    Peso molecular:592.6
  • ZM323881

    CAS:
    ZM323881 is a potent and selective inhibitor of VEGFR2 with an IC 50 of less than 2 nM.
    Fórmula:C22H18FN3O2
    Forma y color:Solid
    Peso molecular:375.4
  • Saracatinib difumarate

    CAS:
    Saracatinib difumarate is an orally available dual-specific inhibitor of Src and Abl with anti-invasive and anti-tumor activities.
    Fórmula:C35H40ClN5O13
    Forma y color:Solid
    Peso molecular:774.18
  • SB1317 hydrochloride (1204918-72-8(free base))


    SB1317 hydrochloride (1204918-72-8(free base)) (TG-02 hydrochloride) is an effective inhibitor of CDK2/JAK2/FLT3 (IC50: 13/73/56 nM).
    Fórmula:C23H25ClN4O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:408.92
  • 4SC-203

    CAS:
    <p>4SC-203 is a multi-kinase inhibitor with potential anti-tumor activity.Cost-effective and quality-assured.</p>
    Fórmula:C33H38N8O4S
    Pureza:96.4% - 99.67%
    Forma y color:Solid
    Peso molecular:642.77
  • JK-P3

    CAS:
    JK-P3: a pyrazole inhibitor of VEGFR-2 (IC50: 7.8 μM), stalls FGFR 1/3 in vitro, halts HUVEC wound healing/tube formation, not cell growth.
    Fórmula:C18H17N3O3
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:323.35
  • Oglufanide

    CAS:
    <p>Oglufanide (H-Glu-Trp-OH) is a naturally occurring thymic immunomodulator,and inhibits vascular endothelial growth factor (VEGF).</p>
    Fórmula:C16H19N3O5
    Pureza:99.80%
    Forma y color:Solid
    Peso molecular:333.34
  • CHIR-124

    CAS:
    CHIR-124 is an effective Chk1 inhibitor (IC50: 0.3 nM). It has 2, 000-fold selectivity against Chk2, 500- to 5, 000-fold less activity against Cdc2 and CDK2/4.
    Fórmula:C23H22ClN5O
    Pureza:96.33% - 98.35%
    Forma y color:Solid
    Peso molecular:419.91
  • Vandetanib trifluoroacetate

    CAS:
    Vandetanib trifluoroacetate: oral VEGFR2/KDR inhibitor, IC50=40nM, also blocks VEGFR3/FLT4 (110nM) and EGFR/HER1 (500nM).
    Fórmula:C24H25BrF4N4O4
    Forma y color:Solid
    Peso molecular:589.386
  • 5-phenylthieno[2,3-d]pyrimidin-4-amine

    CAS:
    5-phenylthieno[2,3-d]pyrimidin-4-amine is a heterocycle that inhibits enzymes like kinases, may treat diseases.
    Fórmula:C12H9N3S
    Pureza:97%
    Forma y color:Solid
    Peso molecular:227.29
  • ZM-447439

    CAS:
    ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.
    Fórmula:C29H31N5O4
    Pureza:99.11% - 99.59%
    Forma y color:Pale Yellow Solid
    Peso molecular:513.59
  • Nintedanib esylate

    CAS:
    Nintedanib esylate (BIBF 1120 esylate) is a potent triple angiokinase inhibitor for VEGFR1/2/3, FGFR1/2/3 and PDGFRα/β
    Fórmula:C31H33N5O4·C2H6O3S
    Pureza:99.43% - 99.98%
    Forma y color:Solid
    Peso molecular:649.76
  • Vandetanib

    CAS:
    Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 and EGFR.
    Fórmula:C22H24BrFN4O2
    Pureza:99.7% - >99.99%
    Forma y color:White Solid
    Peso molecular:475.35
  • MNS

    CAS:
    MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.
    Fórmula:C9H7NO4
    Pureza:98.53%
    Forma y color:Yellow Powder
    Peso molecular:193.16
  • Almonertinib mesylate

    CAS:
    Almonertinib mesylate: EGFR tyrosine kinase inhibitor, targets EGFR-mutant non-small cell lung cancer.
    Fórmula:C31H39N7O5S
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:621.75