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Apoptosis

Apoptosis

Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.

Subcategorías de "Apoptosis"

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Se han encontrado 5600 productos de "Apoptosis"

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  • (S)-10-Hydroxycamptothecin

    CAS:
    <p>(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma.</p>
    Fórmula:C20H16N2O5
    Pureza:99.09% - 99.81%
    Forma y color:Solid
    Peso molecular:364.35
  • AZD0156

    CAS:
    <p>AZD0156 , an effective and specific inhibitors of ATM kinase, is potential antineoplastic activities and chemo-/radio-sensitizing.</p>
    Fórmula:C26H31N5O3
    Pureza:99.13% - 99.87%
    Forma y color:Solid
    Peso molecular:461.56
  • MGCD-265 analog

    CAS:
    <p>Glesatinib, an oral tyrosine kinase inhibitor, targets c-Met and VEGFR2 with IC50s of 29 nM and 10 nM, may treat cancer.</p>
    Fórmula:C26H20FN5O2S2
    Pureza:98.06% - 98.68%
    Forma y color:Solid
    Peso molecular:517.6
  • Boc-Asp(OMe)-fluoromethyl ketone

    CAS:
    <p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>
    Fórmula:C11H18FNO5
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:263.26
  • BMS-202

    CAS:
    <p>BMS-202 (PD1-PDL1 inhibitor 2) is an inhibitor of the PD-1 (Programmed death- 1) /PD-Ll (Programmed death-ligand 1) protein/protein interaction.</p>
    Fórmula:C25H29N3O3
    Pureza:97.92% - 99.66%
    Forma y color:Solid
    Peso molecular:419.52
  • SP2509

    CAS:
    <p>SP2509 is a specific histone demethylase LSD1 inhibitor(IC50 =13 nM).</p>
    Fórmula:C19H20ClN3O5S
    Pureza:98.82% - 99.53%
    Forma y color:Solid
    Peso molecular:437.9
  • PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Fórmula:C16H12N4S
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:292.36
  • Kaempferol

    CAS:
    <p>Kaempferol (Robigenin) is a natural flavonoid and an inverse agonist of ERRα and ERRγ.</p>
    Fórmula:C15H10O6
    Pureza:98% - 99.41%
    Forma y color:Yellow Needles From Alcohol And Water Solid
    Peso molecular:286.24
  • physalin F

    CAS:
    <p>Physalin F is a natural blocker of CaV2.3 (R-type) and CaV2.2 (N-type) voltage-gated calcium channels.Cost-effective and quality-assured.</p>
    Fórmula:C28H30O10
    Pureza:99.5% - 99.61%
    Forma y color:Solid
    Peso molecular:526.53
  • Apitolisib

    CAS:
    <p>Apitolisib (RG 7422) is a PI3K inhibitor, used in cancer trials, targeting PI3Kα, β, δ, γ (IC50= 5, 27, 7, 14 nM).</p>
    Fórmula:C23H30N8O3S
    Pureza:98.28% - 99.64%
    Forma y color:Solid
    Peso molecular:498.6
  • Kobe0065

    CAS:
    <p>Kobe0065: novel small-molecule, inhibits Ras–Raf, Ki=46±13 μM, blocks H-Ras·GTP/c-Raf-1 RBD binding.</p>
    Fórmula:C15H11ClF3N5O4S
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:449.79
  • SM-164

    CAS:
    <p>SM-164 binds to XIAP protein containing both the BIR2 and BIR3 domains (IC50: 1.39 nM). It acts as an extremely potent antagonist of XIAP.</p>
    Fórmula:C62H84N14O6
    Pureza:98.53% - 99.92%
    Forma y color:Solid
    Peso molecular:1121.42
  • FTI-277 hydrochloride

    CAS:
    <p>FTI-277 HCl: potent FTase inhibitor, IC50 500 pM, 100x more selective than GGTase I.</p>
    Fórmula:C22H30ClN3O3S2
    Pureza:97.57% - 97.61%
    Forma y color:Solid
    Peso molecular:484.07
  • Nutlin-3a

    CAS:
    <p>Nutlin-3a is the active enantiomer of Nutlin-3, an MDM2 antagonist that inhibits MDM2-p53 interaction. Nutlin-3a has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C30H30Cl2N4O4
    Pureza:95.62% - 99.71%
    Forma y color:Solid
    Peso molecular:581.49
  • Apoptozole

    CAS:
    <p>Apoptozole (Apoptosis Activator VII) is an inhibitor of the ATPase domain of Hsc70 and Hsp70, and can induce apoptosis.</p>
    Fórmula:C33H25F6N3O3
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:625.56
  • Quisinostat dihydrochloride

    CAS:
    <p>Quisinostat dihydrochloride (JNJ26854165(Quisinostat) 2HCl) 是一种有口服活性,高效的 pan-HDAC 抑制剂,具有广泛的抗肿瘤活性。它对 HDAC1、HDAC2、HDAC4、HDAC10和HDAC11 的IC50值分别为 0.11 nM、0.33 nM、0.64 nM、0.46 nM 和 0.37 nM。</p>
    Fórmula:C21H28Cl2N6O2
    Pureza:97.13%
    Forma y color:Solid
    Peso molecular:467.39
  • Atopaxar hydrochloride

    CAS:
    <p>Atopaxar hydrochloride is used in the Treatment of Cardiovascular Disorders.</p>
    Fórmula:C29H39ClFN3O5
    Forma y color:Solid
    Peso molecular:564.1
  • Y-27632

    CAS:
    <p>Y-27632 (Y-27632) is an orally potent, ATP-competitive inhibitor of ROCK-I and ROCK-II.</p>
    Fórmula:C14H21N3O
    Pureza:99.53% - 99.87%
    Forma y color:Solid
    Peso molecular:247.34
  • Calpeptin

    CAS:
    <p>Calpeptin is a potent, cell-permeable calpain inhibitor.</p>
    Fórmula:C20H30N2O4
    Pureza:97.06% - 98.33%
    Forma y color:White To Off-White Powder
    Peso molecular:362.46
  • 3-Bromopyruvic acid

    CAS:
    <p>3-Bromopyruvic acid (Hexokinase II Inhibitor II, 3-BP) is a hexokinase II inhibitor with Ki of 2.4 mM for glycolysis/hexokinase inhibition.</p>
    Fórmula:C3H3BrO3
    Pureza:95% - 99.644%
    Forma y color:White To Pale Yellow Crystalline Powder
    Peso molecular:166.96
  • Lexibulin

    CAS:
    <p>Lexibulin (CYT-997)(CYT-997) is a potent tubulin polymerization inhibitor (IC50: 10-100 nM, in Y cell lines).</p>
    Fórmula:C24H30N6O2
    Pureza:98.87%
    Forma y color:Solid
    Peso molecular:434.53
  • Cucurbitacin IIb

    CAS:
    <p>Cucurbitacin IIb is an active ingredient in Hemsleyadine, used to treat dysentery and other infections; it has anti-inflammatory effects.</p>
    Fórmula:C30H48O7
    Pureza:98.66% - >99.99%
    Forma y color:Solid
    Peso molecular:520.7
  • Ligustilide

    CAS:
    <p>3-Butylidene-4,5-dihydrophthalide is an effective constituent extracted from Angelica sinensis.</p>
    Fórmula:C12H14O2
    Pureza:96.03% - 98.14%
    Forma y color:Yellow Brown Powder
    Peso molecular:190.24
  • Dioscin

    CAS:
    <p>Dioscin (Collettiside III) is a saponin with antitumor activities.</p>
    Fórmula:C45H72O16
    Pureza:99.85% - 99.87%
    Forma y color:Solid
    Peso molecular:869.04
  • Tebufenozide

    CAS:
    <p>Tebufenozide is a novel nonsteroidal ecdysone agonist. It shows good efficacy and playing an increasingly important role in the control of Lepidopteran pests.</p>
    Fórmula:C22H28N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.47
  • Y-320

    CAS:
    <p>Y-320 is a new phenylpyrazoleanilide immunomodulator.</p>
    Fórmula:C27H29ClN6O2
    Pureza:98% - 99.64%
    Forma y color:Solid
    Peso molecular:505.01
  • PIK-75 hydrochloride

    CAS:
    <p>PIK-75 hydrochloride (PIK-75 HCl) is a p110α inhibitor, isoform-specific mutants at Ser773, and potently inhibits DNA-PK with IC50 of 2 nM in cell-free assay.</p>
    Fórmula:C16H14BrN5O4S·HCl
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:488.74
  • 5-Aminolevulinic acid hydrochloride

    CAS:
    <p>5-Aminolevulinic acid hydrochloride (5-ALA) serves as an intermediate in the body's heme biosynthesis and is the universal precursor of tetrapyrroles.</p>
    Fórmula:C5H10ClNO3
    Pureza:98% - 99.97%
    Forma y color:White To Pale Yellow Crystals Or
    Peso molecular:167.59
  • Fludarabine Phosphate

    CAS:
    <p>Fludarabine Phosphate (NSC 312887 Phosphate) is a fluorinated nucleotide antimetabolite analog of the antiviral agent vidarabine with antineoplastic activity.</p>
    Fórmula:C10H13FN5O7P
    Pureza:99.25% - 99.78%
    Forma y color:Solid
    Peso molecular:365.21
  • L-Theanine

    CAS:
    L-Theanine, a unique amino acid from Camellia sinensis tea, induces relaxation without drowsiness.
    Fórmula:C7H14N2O3
    Pureza:99.31% - 99.38%
    Forma y color:White Crystals From Ethanol + Water White Crystalline Solid
    Peso molecular:174.2
  • Glaucocalyxin A

    CAS:
    <p>Glaucocalyxin A improves drug delivery, activates apoptosis, inhibits cell growth, with potential as an antiplatelet agent.</p>
    Fórmula:C20H28O4
    Pureza:99.55% - 99.80%
    Forma y color:Solid
    Peso molecular:332.43
  • Phthalazinone pyrazole

    CAS:
    <p>Phthalazinone pyrazole: a potent, selective oral Aurora-A kinase inhibitor, overexpressed in tumors with oncogenic activity.</p>
    Fórmula:C18H15N5O
    Pureza:97.03%
    Forma y color:Solid
    Peso molecular:317.34
  • Pinoresinol

    CAS:
    <p>Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury</p>
    Fórmula:C20H22O6
    Pureza:98.67%
    Forma y color:Solid
    Peso molecular:358.39
  • 2-Deoxy-D-glucose

    CAS:
    <p>2-Deoxy-D-glucose (2-DG) is an analog of glucose, an inhibitor of glycolysis.</p>
    Fórmula:C6H12O5
    Pureza:99.31% - ≥98%
    Forma y color:White Powder
    Peso molecular:164.16
  • BX-912

    CAS:
    <p>BX-912 inhibits PDK1 with IC50 of 12 nM; over 10x more selective versus C-Kit, EGFR, PKA, PKC.</p>
    Fórmula:C20H23BrN8O
    Pureza:98.29% - 99.34%
    Forma y color:Solid
    Peso molecular:471.35
  • GDC-0152

    CAS:
    <p>GDC-0152 is a potent inhibitor of IAPs.</p>
    Fórmula:C25H34N6O3S
    Pureza:97.18% - 99.32%
    Forma y color:Solid
    Peso molecular:498.64
  • Lobaplatin

    CAS:
    <p>Lobaplatin (D-19466) (D-19466) is a diastereometric mixture of platinum(II) complexe.</p>
    Fórmula:C9H18N2O3Pt
    Pureza:98.00%
    Forma y color:Solid
    Peso molecular:397.33
  • L-Asparaginase

    CAS:
    <p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>
    Fórmula:NA
    Pureza:97%
    Forma y color:Solid
    Peso molecular:N/A
  • Elesclomol

    CAS:
    <p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>
    Fórmula:C19H20N4O2S2
    Pureza:97.17% - 99.51%
    Forma y color:Solid
    Peso molecular:400.52
  • Rilmenidine Phosphate

    CAS:
    <p>Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.</p>
    Fórmula:C10H19N2O5P
    Pureza:99.87% - ≥95%
    Forma y color:Solid
    Peso molecular:278.24
  • LRRK2-IN-1

    CAS:
    <p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>
    Fórmula:C31H38N8O3
    Pureza:98% - 98.82%
    Forma y color:Solid
    Peso molecular:570.69
  • NSC 95397

    CAS:
    <p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>
    Fórmula:C14H14O4S2
    Pureza:98.66%
    Forma y color:Solid
    Peso molecular:310.39
  • Diffractaic Acid

    CAS:
    <p>Diffractaic Acid (NSC 685595) can inhibit LTB4 biosynthesis in A-23187-stimulated bovine PMNL cells with activity value of 8 μM.</p>
    Fórmula:C20H22O7
    Pureza:99.81% - 99.87%
    Forma y color:Solid
    Peso molecular:374.38
  • SKI II

    CAS:
    <p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>
    Fórmula:C15H11ClN2OS
    Pureza:99.34% - 99.93%
    Forma y color:Solid
    Peso molecular:302.78
  • STF-118804

    CAS:
    <p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 &lt;10 nM.</p>
    Fórmula:C25H23N3O4S
    Pureza:98.66%
    Forma y color:Solid
    Peso molecular:461.53
  • GMB-475

    CAS:
    <p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>
    Fórmula:C43H46F3N7O7S
    Pureza:98.78% - >99.99%
    Forma y color:Solid
    Peso molecular:861.93
  • 2-Hydroxychalcone

    CAS:
    <p>2-Hydroxychalcone (2-(2-Hydroxybenzal)Acetophenone) can be used as antiparasitic hit compounds when Methoxylated. It inhibits invasion of breast cancer cells.</p>
    Fórmula:C15H12O2
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:224.25
  • Phellamurin

    CAS:
    <p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>
    Fórmula:C26H30O11
    Pureza:97.91%
    Forma y color:Solid
    Peso molecular:518.51
  • Nafamostat mesylate

    CAS:
    <p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>
    Fórmula:C19H17N5O2·2CH4O3S
    Pureza:97.36% - 99.76%
    Forma y color:Tan To Pale Orange Solid
    Peso molecular:539.58
  • KW-2449

    CAS:
    <p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>
    Fórmula:C20H20N4O
    Pureza:98.43% - 99.69%
    Forma y color:Solid
    Peso molecular:332.4
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Fórmula:C30H18O10
    Pureza:98.21% - 99.22%
    Forma y color:Odourless Whitish Solid
    Peso molecular:538.46
  • BAY 87-2243

    CAS:
    <p>BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).</p>
    Fórmula:C26H26F3N7O2
    Pureza:98% - 99.95%
    Forma y color:Solid
    Peso molecular:525.53
  • Niraparib tosylate monohyrate

    CAS:
    Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.
    Fórmula:C26H30N4O5S
    Pureza:97.7% - 98.41%
    Forma y color:Solid
    Peso molecular:510.61
  • SKI-178

    CAS:
    <p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>
    Fórmula:C21H22N4O4
    Pureza:97.09%
    Forma y color:Solid
    Peso molecular:394.42
  • Afatinib Dimaleate

    CAS:
    <p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>
    Fórmula:C32H33ClFN5O11
    Pureza:98.11% - 99.87%
    Forma y color:Solid
    Peso molecular:718.08
  • Psoralen

    CAS:
    <p>Psoralen (Ficusin) is a furocoumarin that intercalates with DNA, inhibiting DNA synthesis and cell division.</p>
    Fórmula:C11H6O3
    Pureza:99.3% - 99.87%
    Forma y color:Crystals From Ether Crystalline Solid
    Peso molecular:186.16
  • Isolongifolene

    CAS:
    <p>Isolongifolene ((-)-Isolongifolene), a tricyclic sesquiterpene isolated from Murraya koenigii, exhibits antioxidant, anti-inflammatory, anticancer, and</p>
    Fórmula:C15H24
    Pureza:90.13% - 99.46%
    Forma y color:Colorless Or Light Yellow Liquid
    Peso molecular:204.35
  • ERK1/2 inhibitor 2

    CAS:
    <p>ERK1/2 inhibitor 2 (ASTX029) is a selective and orally bioavailable ERK 1/2 inhibitor, with potential antineoplastic activity.</p>
    Fórmula:C29H31ClFN5O5
    Pureza:98.99%
    Forma y color:Solid
    Peso molecular:584.04
  • LY294002

    CAS:
    <p>LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).</p>
    Fórmula:C19H17NO3
    Pureza:98% - 99.96%
    Forma y color:Pale Yellow Solid
    Peso molecular:307.34
  • Bardoxolone

    CAS:
    <p>Bardoxolone (CDDO) inhibits iNOS, COX-2 in cells; IC50=0.4nM. Reduces ROS/RNS, DNA damage, &amp; cancer growth; triggers apoptosis &amp; boosts antioxidant genes.</p>
    Fórmula:C31H41NO4
    Pureza:97.9% - 98.97%
    Forma y color:Solid
    Peso molecular:491.66
  • Thalidomide-O-C4-NH2 hydrochloride

    CAS:
    <p>Thalidomide-linker 9: a cereblon ligand, E3 ligase conjugate for PROTAC tech.</p>
    Fórmula:C17H20ClN3O5
    Pureza:98.33%
    Forma y color:Solid
    Peso molecular:381.81
  • Laquinimod sodium

    CAS:
    <p>Laquinimod (ABR-215062) sodium is an oral agent for MS, halting neurodegeneration and inflammation.</p>
    Fórmula:C19H16ClN2NaO3
    Forma y color:Solid
    Peso molecular:378.79
  • PFI-1

    CAS:
    <p>PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 μM in a cell-free assay.</p>
    Fórmula:C16H17N3O4S
    Pureza:98.74% - 99.19%
    Forma y color:Solid
    Peso molecular:347.39
  • MCB-613

    CAS:
    <p>MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.</p>
    Fórmula:C20H20N2O
    Pureza:98.17% - 99.754%
    Forma y color:Solid
    Peso molecular:304.39
  • SKLB-163

    CAS:
    <p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>
    Fórmula:C18H16ClN3O2S2
    Pureza:99.23%
    Forma y color:Solid
    Peso molecular:405.92
  • Mitoxantrone diacetate

    CAS:
    <p>Mitoxantrone diacetate hinders topoisomerase II &amp; PKC, fights tumors &amp; orthopoxviruses (IC50: 8.5μM, EC50: 0.25-0.8μM).</p>
    Fórmula:C26H36N4O10
    Forma y color:Solid
    Peso molecular:564.592
  • Fedratinib

    CAS:
    Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.
    Fórmula:C27H36N6O3S
    Pureza:97.31% - 99.96%
    Forma y color:Solid
    Peso molecular:524.68
  • Chelerythrine

    CAS:
    <p>1.</p>
    Fórmula:C21H18NO4
    Pureza:98.36%
    Forma y color:Solid
    Peso molecular:348.37
  • Dimethyl malonate

    CAS:
    <p>Dimethyl Malonate is a Succinate Dehydrogenase inhibitor.</p>
    Fórmula:C5H8O4
    Pureza:≥95%
    Forma y color:Liquid
    Peso molecular:132.11
  • Itanapraced

    CAS:
    <p>Itanapraced (CHF5074), a γ-secretase modulator, reduces Aβ42/40 secretion (IC50: 3.6/18.4 μM).</p>
    Fórmula:C16H11Cl2FO2
    Pureza:98% - 99.79%
    Forma y color:Solid
    Peso molecular:325.16
  • Meloxicam sodium

    CAS:
    <p>Meloxicam sodium is a non-steroidal anti-inflammatory agent, inhibits COX activity, with IC 50 s of 0.49 μM and 36.6 μM for COX-2 and COX-1, respectively [1].</p>
    Fórmula:C14H12N3NaO4S2
    Forma y color:Solid
    Peso molecular:373.38
  • 3'-Hydroxypterostilbene

    CAS:
    <p>3'-Hydroxypterostilbene suppresses colon cancer cell growth (COLO 205, HCT-116, HT-29) by triggering apoptosis and autophagy, affecting key pathways.</p>
    Fórmula:C16H16O4
    Pureza:98.25% - 99.19%
    Forma y color:Solid
    Peso molecular:272.3
  • Benzoylpaeoniflorin

    CAS:
    <p>1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes.</p>
    Fórmula:C30H32O12
    Pureza:95.86% - 97.28%
    Forma y color:Solid
    Peso molecular:584.57
  • Cinchonine monohydrochloride hydrate

    CAS:
    <p>Cinchonine monohydrochloride hydrate: natural antimalarial, inhibits platelet aggregation &amp; cancer cell growth, blocks fat cell formation.</p>
    Fórmula:C19H25ClN2O2
    Forma y color:Solid
    Peso molecular:348.87
  • Ulinastatin

    CAS:
    <p>Ulinastatin is a multivalent Kunitz-type serine protease inhibitor with anti-inflammatory properties.</p>
    Fórmula:C13H16O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:220.10994
  • Droxinostat

    CAS:
    <p>Droxinostat (NS 41080) is a selective inhibitor of HDAC, mostly for HDACs 6 and 8 with IC50 of 2.47 μM and 1.46 μM, greater than 8-fold selective against HDAC3</p>
    Fórmula:C11H14ClNO3
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:243.69
  • RG7112

    CAS:
    <p>RG7112 (RO5045337) (RO5045337) is an orally bioavailable and selective p53-MDM2 inhibitor.</p>
    Fórmula:C38H48Cl2N4O4S
    Pureza:99.66% - 99.9%
    Forma y color:Solid
    Peso molecular:727.78
  • 8-Bromo-cAMP sodium salt

    CAS:
    <p>8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) is a long-acting derivative of cyclic AMP. 8-Bromo-cAMP is an activator of cyclic AMP-dependent protein kinase.</p>
    Fórmula:C10H10BrN5NaO6P
    Pureza:98% - 99.94%
    Forma y color:Off-White Powder
    Peso molecular:430.08
  • C5 Lenalidomide

    CAS:
    <p>C5 Lenalidomide is an chemical weith inconclusive biological activity.</p>
    Fórmula:C13H13N3O3
    Pureza:99.4%
    Forma y color:Solid
    Peso molecular:259.26
  • Kinetin riboside

    CAS:
    <p>Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)</p>
    Fórmula:C15H17N5O5
    Pureza:98.17%
    Forma y color:White Solid
    Peso molecular:347.33
  • Dacomitinib

    CAS:
    <p>Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.</p>
    Fórmula:C24H25ClFN5O2
    Pureza:99.4% - 99.72%
    Forma y color:Solid
    Peso molecular:469.94
  • Flupentixol dihydrochloride

    CAS:
    <p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.76% - >99.99%
    Forma y color:White Or Off-White Solid
    Peso molecular:507.43
  • Ricolinostat

    CAS:
    <p>Ricolinostat (Rocilinostat) is an orally bioavailable, specific inhibitor of histone deacetylase 6 (HDAC6) with potential antineoplastic activity.</p>
    Fórmula:C24H27N5O3
    Pureza:97.17% - 99.76%
    Forma y color:Solid
    Peso molecular:433.5
  • Sodium Demethylcantharidate

    CAS:
    <p>Sodium Demethylcantharidate (Sodium norcantharidin) is extracted from Mylabris phqlarata pallas and has potent antitumor activity.</p>
    Fórmula:C8H9O5·Na
    Pureza:99.66% - ≥98%
    Forma y color:Solid
    Peso molecular:208.14
  • Thalidomide-O-amido-C6-NH2 TFA

    CAS:
    <p>Thalidomide-O-amido-C6-NH2 TFA (Cereblon Ligand-Linker Conjugates 11 TFA), a synthesized E3 ligase ligand-linker conjugate containing a Thalidomide-based</p>
    Fórmula:C46H53F6N8O16
    Pureza:95.16%
    Forma y color:Solid
    Peso molecular:1087.95
  • ICCB280

    CAS:
    <p>ICCB280 was capable of inducing differentiation and apoptosis of ATRA-resistant patient blasts strongly signify that the activity of this compound can overcome</p>
    Fórmula:C23H18N2O4
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:386.4
  • NSC-87877 disodium

    CAS:
    <p>NSC-87877 disodium (NSC87877) is a cell-permeable inhibitor of both SHP-1 and SHP-2. NSC-87877 also inhibits EGF-induced Erk1/2 activation in HEK293 cells.</p>
    Fórmula:C19H13N3O7S2·2Na
    Pureza:97.89%
    Forma y color:Solid
    Peso molecular:503.42
  • Lenaldekar

    CAS:
    <p>Lenaldekar (LDK) inhibits T-cell expansion and autoimmune encephalomyelitis.</p>
    Fórmula:C18H14N4
    Pureza:97.73%
    Forma y color:Solid
    Peso molecular:286.33
  • Bicyclol

    CAS:
    <p>Bicyclol is an oral anti-hepatitis drug, decreasing ALT/AST levels by 50% and inhibiting HBV/HCV, boosting efficacy with interferon/lamivudine/adefovir.</p>
    Fórmula:C19H18O9
    Pureza:99.64% - 99.85%
    Forma y color:Solid
    Peso molecular:390.34
  • CBL0137 hydrochloride

    CAS:
    <p>CBL0137 hydrochloride (Curaxin-137 hydrochloride) is an inhibitor of the histone chaperone FACT, which also activates p53 and inhibits NF-κB.Cost-effective and quality-assured.</p>
    Fórmula:C21H25ClN2O2
    Pureza:99.35% - 99.86%
    Forma y color:Solid
    Peso molecular:372.88
  • Trametinib (DMSO solvate)

    CAS:
    <p>Trametinib (DMSO solvate) (GSK-1120212 (DMSO solvate)) is a Highly Potent and Selective MEK Inhibitor that specifically inhibits MEK1/2(IC50 :2 nM)</p>
    Fórmula:C28H29FIN5O5S
    Pureza:98.82% - 99.92%
    Forma y color:Solid
    Peso molecular:693.53
  • TCS PrP Inhibitor 13

    CAS:
    <p>TCS PrP Inhibitor 13 (5-(4-Nitrophenyl)-2-Phenyl-4H-Pyrazol-3-One) is an antiprion agent inhibiting protease-resistant prion protein (PrP-res) accumulation.</p>
    Fórmula:C15H11N3O3
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:281.27
  • Inauhzin

    CAS:
    <p>Inauhzin (INZ) reactivates p53, inhibits SIRT1, induces Y cell apoptosis without genotoxic stress (IC50=3 uM in A549).</p>
    Fórmula:C25H19N5OS2
    Pureza:98% - 99.36%
    Forma y color:Solid
    Peso molecular:469.58
  • Tenovin-6 Hydrochloride

    CAS:
    <p>Tenovin-6 HCl: Inhibits SIRT1 (21µM), SIRT2 (10µM), HDAC8; potent p53 activator.</p>
    Fórmula:C25H35ClN4O2S
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:491.09
  • Azoramide

    CAS:
    <p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>
    Fórmula:C15H17ClN2OS
    Pureza:99.08% - 99.85%
    Forma y color:Solid
    Peso molecular:308.83
  • Laquinimod

    CAS:
    <p>Laquinimod (LAQ) is an effective immunomodulator, which is currently under development in phase III trials for the treatment of multiple sclerosis as an oral</p>
    Fórmula:C19H17ClN2O3
    Pureza:98.42% - 98.84%
    Forma y color:Solid
    Peso molecular:356.8
  • A-419259

    CAS:
    <p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>
    Fórmula:C29H34N6O
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:482.62
  • PKD-IN-1 dihydrochloride (956121-30-5 free base)

    CAS:
    <p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>
    Fórmula:C18H21Cl3N4O
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:415.75
  • Tauroursodeoxycholate

    CAS:
    <p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>
    Fórmula:C26H45NO6S
    Pureza:98.77% - 99.93%
    Forma y color:White Solid
    Peso molecular:499.7
  • PEAQX

    CAS:
    <p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>
    Fórmula:C17H17BrN3O5P
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:454.21