
Apoptosis
Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.
Subcategorías de "Apoptosis"
- ASK(6 productos)
- BCL(11 productos)
- Caspasa(125 productos)
- FOXO1(3 productos)
- IAP(66 productos)
- Mdm2(12 productos)
- PD-1 / PD-L1(125 productos)
- PDK(9 productos)
- PERK(25 productos)
- Serina / treonina quinasa(15 productos)
- Survivin(13 productos)
- TNF(92 productos)
- c-RET(51 productos)
- p53(62 productos)
Mostrar 6 subcategorías más
Se han encontrado 5600 productos de "Apoptosis"
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Tauroursodeoxycholate
CAS:<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Fórmula:C26H45NO6SPureza:98.77% - 99.93%Forma y color:White SolidPeso molecular:499.7AR42
CAS:<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Fórmula:C18H20N2O3Pureza:98.46% - 98.96%Forma y color:SolidPeso molecular:312.36Sulforaphane
CAS:<p>Sulforaphane is a natural isothiocyanate that activates Nrf2. Sulforaphane has antitumor and anti-inflammatory activities. Cost-effective and quality-assured.</p>Fórmula:C6H11NOS2Pureza:95% - 99.79%Forma y color:Light Yellow LiquidPeso molecular:177.29Trolox
CAS:<p>Trolox is a vitamin E analogue, used in reducing oxidative stress or damage.</p>Fórmula:C14H18O4Pureza:98.90% - 99.90%Forma y color:White To Fainly Beige Crystalline PowderPeso molecular:250.29Thalidomide-NH-CH2-COOH
CAS:<p>Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a</p>Fórmula:C15H13N3O6Pureza:96.3800%Forma y color:SolidPeso molecular:331.28Apocynin
CAS:<p>Apocynin (NSC 2146) is a specific NADPH-oxidase inhibitor (IC50: 10 μM).</p>Fórmula:C9H10O3Pureza:99.71% - 99.98%Forma y color:Yellowish To Brown PowderPeso molecular:166.17Eltrombopag Olamine
CAS:<p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>Fórmula:C29H36N6O6Pureza:99.59% - 99.89%Forma y color:SolidPeso molecular:564.63HA15
CAS:<p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>Fórmula:C23H22N4O3S2Pureza:99.77% - 99.86%Forma y color:SolidPeso molecular:466.58CA-4948
CAS:<p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>Fórmula:C24H25N7O5Pureza:99.35% - 99.88%Forma y color:SolidPeso molecular:491.5Tenovin-6
CAS:<p>Tenovin-6 is a p53 transcriptional activity agonist.</p>Fórmula:C25H34N4O2SPureza:97.71% - >99.99%Forma y color:SolidPeso molecular:454.63FOXO4-DRI acetate
<p>FOXO4-DRI acetate is a bioactive chemical.</p>Fórmula:C36H64N14O14SPureza:99.10%Forma y color:SolidPeso molecular:5358.06Periplocin
CAS:<p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>Fórmula:C36H56O13Pureza:99.66% - 99.74%Forma y color:SolidPeso molecular:696.82Thalidomide-O-COOH
CAS:<p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>Fórmula:C15H12N2O7Pureza:98% - 98.29%Forma y color:SolidPeso molecular:332.27Thalidomide-4-OH
CAS:<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Fórmula:C13H10N2O5Pureza:99.59%Forma y color:SolidPeso molecular:274.23Thalidomide-NH-C4-NH-Boc
CAS:<p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>Fórmula:C22H28N4O6Pureza:98.87%Forma y color:SolidPeso molecular:444.48Methoxyamine HCl
CAS:<p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>Fórmula:CH6ClNOPureza:≥98%Forma y color:SolidPeso molecular:83.51Alogliptin Benzoate
CAS:<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Fórmula:C25H27N5O4Pureza:99.94% - >99.99%Forma y color:White PowderPeso molecular:461.51OICR-9429
CAS:<p>OICR-9429 blocks WDR5 binding to MLL/Histone 3, hindering acute myeloid leukemia cell growth in vitro.</p>Fórmula:C29H32F3N5O3Pureza:97.07% - 99.93%Forma y color:SolidPeso molecular:555.59Thalidomide-O-amido-PEG3-C2-NH2 TFA
CAS:<p>Synthetic E3 ligase ligand-linker, Thalidomide-O-amido-PEG3-C2-NH2 TFA, used in PROTAC with cereblon ligand and PEG.</p>Fórmula:C25H31F3N4O11Pureza:99.82%Forma y color:SolidPeso molecular:620.54Ketorolac hemicalcium
CAS:<p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation & pain, used in cancer research.</p>Fórmula:C30H24CaN2O6Forma y color:SolidPeso molecular:548.608Verteporfin
CAS:<p>Verteporfin (BPD-MA) is a YAP inhibitor that inhibits YAP-TEAD interactions.</p>Fórmula:C41H42N4O8Pureza:95.37% - 99.82%Forma y color:Dark Green To Black SolidPeso molecular:718.79Sulfaphenazole
CAS:<p>Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki: 63/29 μM for</p>Fórmula:C15H14N4O2SPureza:97.53% - 99.67%Forma y color:SolidPeso molecular:314.36PK11000
CAS:<p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>Fórmula:C6H5ClN2O4SPureza:99.70%Forma y color:SolidPeso molecular:236.63Abacavir monosulfate
CAS:<p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>Fórmula:C14H20N6O5SForma y color:SolidPeso molecular:384.41Benidipine hydrochloride
CAS:<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Fórmula:C28H32ClN3O6Pureza:99.80%Forma y color:SolidPeso molecular:542.03Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Fórmula:C23H27F3N4O10Pureza:95.74% - 99%Forma y color:SolidPeso molecular:576.48IMT1
CAS:<p>IMT1 (Propanamide, N,N-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2H-1-benzopyran-7-yl]oxy]-) has anticancer activity.</p>Fórmula:C21H21NO4Pureza:98.07% - 98.14%Forma y color:SolidPeso molecular:351.4Piperazine Erastin
CAS:<p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>Fórmula:C35H41ClN6O4Pureza:99.52%Forma y color:SolidPeso molecular:645.19MS7972
CAS:<p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>Fórmula:C14H13NO2Pureza:99.78%Forma y color:SolidPeso molecular:227.26KX2-361
CAS:<p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>Fórmula:C24H24FN3O2Pureza:99.64% - 99.68%Forma y color:SolidPeso molecular:405.46Ralimetinib dimesylate
CAS:<p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>Fórmula:C24H29FN6·2CH4O3SPureza:98% - 99.38%Forma y color:SolidPeso molecular:612.74Pomolic acid
CAS:<p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>Fórmula:C30H48O4Pureza:96.84% - 99.79%Forma y color:SolidPeso molecular:472.7Crebanine
CAS:<p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>Fórmula:C20H21NO4Pureza:99.17% - 99.77%Forma y color:SolidPeso molecular:339.39Cilengitide
CAS:<p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>Fórmula:C27H40N8O7Pureza:98% - 99.8%Forma y color:SolidPeso molecular:588.66Mitochonic acid 5
CAS:<p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>Fórmula:C18H13F2NO3Pureza:98.85%Forma y color:SolidPeso molecular:329.3Nutlin-3
CAS:<p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C30H30Cl2N4O4Pureza:98.13% - 99.89%Forma y color:SolidPeso molecular:581.49Avadomide HCl
CAS:<p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>Fórmula:C14H15ClN4O3Forma y color:SolidPeso molecular:322.75NAE-IN-M22
CAS:<p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>Fórmula:C20H24Cl2N2Pureza:97.65%Forma y color:SolidPeso molecular:363.32NSC622608
CAS:<p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>Fórmula:C9H12BrN3OS2Pureza:98.48%Forma y color:SolidPeso molecular:322.24Ibuprofen Lysine
CAS:<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Fórmula:C19H32N2O4Pureza:99.26%Forma y color:CoaPeso molecular:352.471-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Forma y color:SolidPeso molecular:248.75Bardoxolone Methyl
CAS:<p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>Fórmula:C32H43NO4Pureza:97.81% - 99.09%Forma y color:SolidPeso molecular:505.69RA375
CAS:<p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>Fórmula:C30H25ClN4O7Pureza:99.56%Forma y color:SolidPeso molecular:588.99SRT 2183
CAS:<p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>Fórmula:C27H24N4O2SPureza:97.86%Forma y color:SolidPeso molecular:468.572-Bromohexadecanoic acid
CAS:<p>2-Bromohexadecanoic acid (2-BP) is a PPARδ agonist, and a palmitoylation inhibitor, inhibiting DHHC-mediated palmitoylation. Cost-effective and quality-assured.</p>Fórmula:C16H31BrO2Pureza:97% - 98.3%Forma y color:White Crystalline PowderPeso molecular:335.32Vildagliptin dihydrate
CAS:<p>Vildagliptin dihydrate: potent, selective DPP-IV inhibitor with 3.5 nM IC50, high oral bioavailability, effective against hyperglycemia.</p>Fórmula:C17H29N3O4Forma y color:SolidPeso molecular:339.436Decursin
CAS:<p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>Fórmula:C19H20O5Pureza:97.22% - 99.84%Forma y color:SolidPeso molecular:328.36Deguelin
CAS:<p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>Fórmula:C23H22O6Pureza:96.39% - 99.29%Forma y color:SolidPeso molecular:394.42Thalidomide-O-amido-PEG-C2-NH2 hydrochloride
CAS:<p>Thalidomide-O-amido-PEG-C2-NH2 HCl is a cereblon ligand-linker for PROTAC synthesis.</p>Fórmula:C19H23ClN4O7Pureza:95%Forma y color:SolidPeso molecular:454.862Mirdametinib
CAS:<p>Mirdametinib (PD325901) is an MEK inhibitor (IC50=0.33 nM) with selective, non-ATP-competitive, and oral activity.</p>Fórmula:C16H14F3IN2O4Pureza:99.11% - 99.63%Forma y color:White PowderPeso molecular:482.19Darapladib
CAS:<p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>Fórmula:C36H38F4N4O2SPureza:99.82% - >99.99%Forma y color:SolidPeso molecular:666.77BTR-1
CAS:<p>5-Benzylidene-3-ethyl rhodanine(BTR-1 (5-Benzylidene-3-ethyl rhodanine)) is an active anti-cancer agent. BTR-1 activates apoptosis and induces cell death.</p>Fórmula:C12H11NOS2Pureza:98%Forma y color:SolidPeso molecular:249.35GDC-0623
CAS:<p>GDC-0623 (RG 7421) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1.</p>Fórmula:C16H14FIN4O3Pureza:98.95% - 99.02%Forma y color:SolidPeso molecular:456.21Devimistat
CAS:<p>Devimistat (6,8-Bis(benzylthio)octanoic acid) , a lipoate analog, inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase</p>Fórmula:C22H28O2S2Pureza:98.06% - 99.24%Forma y color:SolidPeso molecular:388.59Necroptosis-IN-1
CAS:<p>Necroptosis-IN-1 is a potent necroptosis inhibitor of RIPK1. It is an analog of Necrostatin-1.</p>Fórmula:C12H10ClN3O2Pureza:99.73% - 99.8%Forma y color:SolidPeso molecular:263.68Diallyl Trisulfide
CAS:<p>Diallyl Trisulfide is an organic polysulfide compound found in garlic that acts as an H2S donor.</p>Fórmula:C6H10S3Pureza:95% - ≥98%Forma y color:LiquidPeso molecular:178.34All-trans-retinal
CAS:<p>All-trans-retinal (Vitamin A aldehyde) is a one of the major vitamin A metabolites in the retina.</p>Fórmula:C20H28OPureza:98.56% - 98.70%Forma y color:SolidPeso molecular:284.44CBL0137
CAS:<p>CBL0137 (Curaxin 137), a metabolically stable curaxin, activates p53 (EC50: 0.37 μM) and inhibits NF-κB (EC50: 0.47 μM).</p>Fórmula:C21H24N2O2Pureza:99.57% - 99.68%Forma y color:SolidPeso molecular:336.43VLX600
CAS:<p>VLX600 is an iron-chelating oxidative phosphorylation (OXPHOS) inhibitor, is a cell-permeable anticancer agent.</p>Fórmula:C17H15N7Pureza:98.62%Forma y color:SolidPeso molecular:317.35Alemtuzumab
CAS:<p>Alemtuzumab is a humanized monoclonal antibody against CD52 an antigen found on the surface of normal and malignant lymphocytes.</p>Pureza:97.2% (SDS-PAGE); 96.7% (SEC-HPLC) - 98.00%Forma y color:LiquidPeso molecular:146.04 kDaChlorfenapyr
CAS:<p>Chlorfenapyr (AC 303630) is a pyrrole insecticide and converts active substances (insecticidal activity) in insects by a multifunctional oxidase</p>Fórmula:C15H11BrClF3N2OPureza:99.33% - 99.49%Forma y color:Off-White To Light Brown Powder With An Halide OdorPeso molecular:407.61Amifostine trihydrate
CAS:<p>Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.</p>Fórmula:C5H15N2O3PS·3H2OPureza:99.71% - 99.80%Forma y color:SolidPeso molecular:268.27Oxaprozin potassium
CAS:<p>Oxaprozin potassium is an oral COX inhibitor (IC50: 2.2 μM for COX-1, 36 μM for COX-2), induces apoptosis, and blocks NF-κB activation.</p>Fórmula:C18H14KNO3Forma y color:SolidPeso molecular:331.412Autophagy-IN-A9
CAS:<p>Autophagy-IN-A9 is a bioactive chemical.</p>Fórmula:C15H11ClFN3Pureza:99.72%Forma y color:SolidPeso molecular:287.72Ibuprofen sodium
CAS:<p>Ibuprofen sodium is a selective COX-1 inhibitor, anti-inflammatory, and NO donor, used in pain, swelling, and cancer research.</p>Fórmula:C13H17NaO2Forma y color:SolidPeso molecular:228.267Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Forma y color:SolidPeso molecular:336.38PAC-1
CAS:<p>PAC-1 (Procaspase activating compound 1) has been used in trials studying the treatment of Lymphoma, Melanoma, Solid Tumors, Breast Cancer and Thoracic Cancers.</p>Fórmula:C23H28N4O2Pureza:96.78% - 99.77%Forma y color:SolidPeso molecular:392.49Thalidomide 5-fluoride
CAS:<p>Thalidomide 5-fluoride (H-Isoindole-1,3(2H)-dione, 2-(2,6-dioxo-3-piperidinyl)-5-fluoro-) is a thalidomide-based Cereblon ligand that binds to the IRAK4 protein</p>Fórmula:C13H9FN2O4Pureza:98.62%Forma y color:SolidPeso molecular:276.22Stavudine sodium
CAS:<p>Stavudine sodium, an oral HIV-1/2 inhibitor, also hinders mtDNA replication, NLRP3 inflammasome, and Amyloid-β autophagy, prompting apoptosis.</p>Fórmula:C10H11N2NaO4Forma y color:SolidPeso molecular:246.198OTS964
CAS:<p>OTS964 is an oral TOPK inhibitor (IC50: 28nM), also targets CDK11, especially CDK11B (Kd: 40nM).</p>Fórmula:C23H24N2O2SForma y color:SolidPeso molecular:392.51Dauricine
CAS:<p>1.</p>Fórmula:C38H44N2O6Pureza:99.24% - 99.75%Forma y color:White PowderPeso molecular:624.77Etonogestrel
CAS:<p>Etonogestrel (Implanon) is a steroidal progestin used as hormonal contraceptives.</p>Fórmula:C22H28O2Pureza:99.59% - 99.59%Forma y color:SolidPeso molecular:324.46PRT062607 hydrochloride
CAS:<p>PRT062607 hydrochloride (P505-15 Hydrochloride) is a selective inhibitor of Syk. PRT062607 displays at least 80-fold selectivity for Syk over other kinases.</p>Fórmula:C19H23N9O·HClPureza:97.7% - 99.81%Forma y color:SolidPeso molecular:429.91Siramesine hydrochloride
CAS:<p>Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit</p>Fórmula:C30H32ClFN2OPureza:99.72% - >99.99%Forma y color:SolidPeso molecular:491.04Oxychlororaphine
CAS:<p>Oxychlororaphine (phenazine-1-carboxamide) inhibits strongly the growth of Streptomyces sp. 441.</p>Fórmula:C13H9N3OPureza:98.3%Forma y color:Green-Yellow SolidPeso molecular:223.23Pitavastatin sodium
CAS:<p>Pitavastatin sodium inhibits HMG-CoA reductase, enhances LDL-C receptors, and has various protective effects.</p>Fórmula:C25H23FNNaO4Forma y color:SolidPeso molecular:443.45L67
CAS:<p>L67 (DNA Ligase Inhibitor) is a competitive human DNA ligase inhibitor, inhibits DNA ligases I and III (IC50: 10 μM).</p>Fórmula:C16H14Br2N4O4Pureza:98.34% - 99.56%Forma y color:SolidPeso molecular:486.11CRT0066101 dihydrochloride
CAS:<p>CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).</p>Fórmula:C18H22N6O·2HClPureza:99.85%Forma y color:SolidPeso molecular:411.33Thalidomide-O-C6-NH2 hydrochloride
CAS:<p>Thalidomide-O-C6-NH2 hydrochloride (4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride) is a synthesized E3 ligase ligand-</p>Fórmula:C19H24ClN3O5Pureza:97.45%Forma y color:SolidPeso molecular:409.86Azathioprine Sodium
CAS:<p>Azathioprine Sodium is a pro-drug converted to 6-MP, inhibiting DNA/RNA synthesis, curbing cell proliferation, especially in lymphocytes.</p>Fórmula:C9H6N7NaO2SForma y color:SolidPeso molecular:299.24Asiatic acid
CAS:<p>Asiatic acid (Dammarolic acid) is the aglycone of asiaticoside used in wound healing with antioxidant, anti-inflammatory, and neuroprotective properties.</p>Fórmula:C30H48O5Pureza:98.01% - 99.52%Forma y color:Solid PowderPeso molecular:488.7NVP-TAE 684
CAS:<p>NVP-TAE 684 (TAE684) is a excellently effective and specific ALK inhibitor(IC50=3 nM).</p>Fórmula:C30H40ClN7O3SPureza:98% - 99.82%Forma y color:SolidPeso molecular:614.2Minodronic acid monohydrate
CAS:<p>Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。</p>Fórmula:C9H14N2O8P2Pureza:≥95%Forma y color:SolidPeso molecular:340.16Buprofezin
CAS:<p>Buprofezin (Applaud) is an insecticide used for control of insect pests such as mealybugs, leafhoppers and whitefly on vegetable crops.</p>Fórmula:C16H23N3OSPureza:99.02% - 99.34%Forma y color:White To Pale Yellow Crystalline PowderPeso molecular:305.44Quizartinib HCl
CAS:<p>Quizartinib (AC220/AC010220) is an oral FLT3/STK1 inhibitor for treating AML, blocking kinase-driven cell proliferation and promoting apoptosis.</p>Fórmula:C29H34Cl2N6O4SForma y color:SolidPeso molecular:633.59BML-277
CAS:<p>BML-277 (C 3742) is a selective checkpoint kinase 2 (Chk2) inhibitor.</p>Fórmula:C20H14ClN3O2Pureza:98.03% - ≥95%Forma y color:Tan SolidPeso molecular:363.8Brusatol
CAS:<p>Brusatol (NSC-172924) is a natural product isolated from the Brucea javanica plant. It inhibits Nrf2.</p>Fórmula:C26H32O11Pureza:99.35% - 99.95%Forma y color:SolidPeso molecular:520.53Gefitinib dihydrochloride
CAS:<p>Gefitinib dihydrochloride: orally active, selective EGFR inhibitor (IC50: 33-54 nM), hinders tumor growth, induces autophagy and apoptosis in cancer research.</p>Fórmula:C22H26Cl3FN4O3Forma y color:SolidPeso molecular:519.82Rafoxanide
CAS:<p>Rafoxanide as a dual CDK4/6 inhibitor for the treatment of skin cancer.</p>Fórmula:C19H11Cl2I2NO3Pureza:99.47%Forma y color:Slight Yellowish Brown Injectable Solution &White Oral SolutionPeso molecular:626.01Fenoldopam mesylate
CAS:<p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>Fórmula:C16H16ClNO3·CH4O3SPureza:99.19%Forma y color:SolidPeso molecular:401.86RRX-001
CAS:<p>RRx-001 is a potent inhibitor ofglucose 6-phosphate dehydrogenase(G6PD) and with potent antimalarial activity</p>Fórmula:C5H6BrN3O5Pureza:99.91% - ≥95%Forma y color:SolidPeso molecular:268.02HLCL-61 hydrochloride
CAS:<p>HLCL-61 hydrochloride (HLCL-61 HCL) is a potent and selective PRMT5 inhibitor for the treatment of acute myeloid leukemia.</p>Fórmula:C23H24N2O·ClHPureza:99.88% - 99.95%Forma y color:SolidPeso molecular:380.91Tylvalosin tartrate
CAS:<p>Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) is a macrolide antibiotic that can against Gram-positive bacteria.</p>Fórmula:C57H93NO25Pureza:99.25%Forma y color:SolidPeso molecular:1192.344'-bromo-Resveratrol
CAS:<p>4'-bromo-Resveratrolis a potent inhibitor of the deacetylases sirtuin 1 (SIRT1) and 3 (SIRT3)</p>Fórmula:C14H11BrO2Pureza:99.00%Forma y color:SolidPeso molecular:291.14Fraxetin
CAS:<p>Fraxetin (7,8-dihydroxy-6-methoxy coumarin) has dual-antioxidative ,hepatoprotective and antihyperglycemic functions, it shows potent protective effects against</p>Fórmula:C10H8O5Pureza:98% - 99.59%Forma y color:Light Yellow Crystalline FlakesPeso molecular:208.17Butein
CAS:<p>Butein is a cAMP-specific PDE inhibitor, protein tyrosine kinase inhibitor, and SIRT1 activator.Cost-effective and quality-assured.</p>Fórmula:C15H12O5Pureza:98.76% - >99.99%Forma y color:SolidPeso molecular:272.25Zoledronic acid disodium tetrahydrate
CAS:<p>Zoledronic Acid, a potent bisphosphonate, inhibits osteoclasts and has anti-cancer effects.</p>Fórmula:C5H16N2Na2O11P2Forma y color:SolidPeso molecular:388.113Topotecan hydrochloride hydrate
CAS:<p>Orally active Topotecan HCl hydrate inhibits Topoisomerase I, blocks G0/G1 & S phases, and induces apoptosis.</p>Fórmula:C23H26ClN3O6Forma y color:SolidPeso molecular:475.93YUM70
CAS:<p>YUM70 inhibits GRP78 (IC50: 1.5μM), inducing ER stress and apoptosis in pancreatic cancer.</p>Fórmula:C21H19ClN2O4Pureza:97.25%Forma y color:SolidPeso molecular:398.84Afimetoran
CAS:<p>Afimetoran (BMS-986256) is a toll-like receptor antagonist. Afimetoran can be used in the research of inflammatory and autoimmune diseases.</p>Fórmula:C26H32N6OPureza:99.81% - 99.94%Forma y color:SolidPeso molecular:444.57

