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Caspasa

Caspasa

Los inhibidores de caspasas son compuestos que bloquean la actividad de las caspasas, una familia de proteasas que son ejecutores centrales de la apoptosis. Las caspasas escinden sustratos específicos dentro de la célula para desencadenar el proceso apoptótico, lo que conduce a la muerte celular programada. Los inhibidores de caspasas se utilizan para estudiar los mecanismos de la apoptosis, así como para prevenir la muerte celular no deseada en varios modelos de investigación. Estos inhibidores también se exploran en contextos terapéuticos para proteger las células de la apoptosis en enfermedades como la neurodegeneración. En CymitQuimica, ofrecemos una amplia gama de inhibidores de caspasas de alta calidad para apoyar su investigación en apoptosis, muerte celular y campos relacionados.

Se han encontrado 125 productos de "Caspasa"

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  • Aspirin

    CAS:
    <p>Aspirin (Acetylsalicylic Acid) is a COX inhibitor. Aspirin has anti-inflammatory, antipyretic and analgesic activities. Cost-effective and quality-assured.</p>
    Fórmula:C9H8O4
    Pureza:99.78% - 99.91%
    Forma y color:White Solid Crystalline
    Peso molecular:180.16
  • Thiabendazole

    CAS:
    <p>Thiabendazole (2-(4-Thiazolyl)benzimidazole) is a benzimidazole derivative with anthelminthic property.</p>
    Fórmula:C10H7N3S
    Pureza:99.14%
    Forma y color:Light Yellow Powder
    Peso molecular:201.25
  • Diclofenac diethylamine

    CAS:
    <p>Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).</p>
    Fórmula:C18H22Cl2N2O2
    Pureza:99.81% - 99.87%
    Forma y color:Solid
    Peso molecular:369.29
  • Crustecdysone

    CAS:
    <p>Crustecdysone (Hydroxyecdysone) is a steroid hormone that regulates the processes of molting or ecdysis in insects.</p>
    Fórmula:C27H44O7
    Pureza:99.06% - 99.67%
    Forma y color:Canary Yellow Fine Powder
    Peso molecular:480.63
  • Diclofenac

    CAS:
    <p>Diclofenac: a nonsteroidal compound inhibiting COX-1 and COX-2, reducing pro-inflammatory prostaglandins.</p>
    Fórmula:C14H11Cl2NO2
    Pureza:99.69% - 99.97%
    Forma y color:Crystals From Ether-Petroleum Ether Solid
    Peso molecular:296.15
  • Lacidipine

    CAS:
    <p>Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.</p>
    Fórmula:C26H33NO6
    Pureza:99.98%
    Forma y color:White-To-Off-White Crystalline Solid
    Peso molecular:455.54
  • Ac-FLTD-CMK

    CAS:
    <p>Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.</p>
    Fórmula:C26H37ClN4O8
    Pureza:95.17%
    Forma y color:Solid
    Peso molecular:569.05
  • Ac-YVAD-CMK

    CAS:
    <p>Ac-YVAD-CMK: Irreversible Caspase-1 inhibitor; halts pyroptosis, IL-1β/IL-18; neuroprotective and anti-inflammatory.</p>
    Fórmula:C24H33ClN4O8
    Pureza:97.08% - 99.909%
    Forma y color:Solid
    Peso molecular:540.99
  • Oxidopamine hydrobromide

    CAS:
    <p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>
    Fórmula:C8H12BrNO3
    Pureza:98.22% - 99.88%
    Forma y color:Beige To Brown Fine Crystalline Powder
    Peso molecular:250.09
  • Q-VD-OPH

    CAS:
    <p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>
    Fórmula:C26H25F2N3O6
    Pureza:97.8% - 98.95%
    Forma y color:Solid
    Peso molecular:513.5
  • Diclofenac sodium

    CAS:
    <p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>
    Fórmula:C14H10Cl2NNaO2
    Pureza:98.21% - 99.73%
    Forma y color:White Or Off-White Powder
    Peso molecular:318.13
  • Fenbufen

    CAS:
    <p>Fenbufen (Lederfen) is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis.</p>
    Fórmula:C16H14O3
    Pureza:98.35% - 98.46%
    Forma y color:White Solid
    Peso molecular:254.28
  • Dehydrocorydaline chloride

    CAS:
    <p>Dehydrocorydaline chloride (13-Methylpalmatine chloride) is an alkaloid with anti-inflammatory and anti-cancer activity. Can improve the activation of p38 MAPK.</p>
    Fórmula:C22H24ClNO4
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:401.88
  • ML-9

    CAS:
    <p>ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively.</p>
    Fórmula:C15H18Cl2N2O2S
    Pureza:99.69%
    Forma y color:Crystalline Solid
    Peso molecular:361.29
  • Terfenadine

    CAS:
    <p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>
    Fórmula:C32H41NO2
    Pureza:98.76% - 99.75%
    Forma y color:Solid
    Peso molecular:471.67
  • Oxidopamine hydrochloride

    CAS:
    <p>Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.</p>
    Fórmula:C8H12ClNO3
    Pureza:98.34% - 99.85%
    Forma y color:Physical Description Beige Solid (Ntp 1992)
    Peso molecular:205.64
  • Ac-Trp-Glu-His-Asp-Aldehyde

    CAS:
    <p>Ac-Trp-Glu-His-Asp-Aldehyde is a powerful and selective inhibitor of caspase-1, demonstrating a K_i value of 56 pM [1] [2].</p>
    Fórmula:C28H33N7O9
    Forma y color:Solid
    Peso molecular:611.6
  • TNF-α-IN-11


    <p>TNF-α-IN-11 (Compound 10) is a TNF-α inhibitor exhibiting a dissociation constant (K D) of 12.06 μM.</p>
    Fórmula:C24H26N2O5
    Forma y color:Solid
    Peso molecular:422.47
  • IRF1-IN-2

    CAS:
    <p>IRF1-IN-2 is a small molecule IRF1 inhibitor that suppresses pyroptosis, protecting against radiation-induced skin damage.</p>
    Fórmula:C18H20N2O4S
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:360.43
  • TD1092


    <p>TD1092, a pan-IAP degrader, activates caspase 3/7, induces apoptosis in cancer cells, inhibits NF-κB, and is used in cancer research.</p>
    Fórmula:C55H70N8O9
    Forma y color:Solid
    Peso molecular:987.19