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RAAS

RAAS

Los inhibidores del sistema renina-angiotensina-aldosterona (RAAS) son compuestos que se dirigen a la vía del RAAS, conocida principalmente por su papel en la regulación de la presión arterial y el equilibrio de líquidos, pero que también influye en la angiogénesis. La vía del RAAS puede contribuir al desarrollo de nuevos vasos sanguíneos en los tumores, apoyando así su crecimiento. Inhibir los componentes del RAAS puede, por lo tanto, tener efectos antiangiogénicos, lo que convierte a estos inhibidores en herramientas valiosas en el tratamiento de ciertos cánceres y trastornos vasculares. En CymitQuimica, ofrecemos una gama de inhibidores de alta calidad del RAAS para apoyar su investigación en biología cardiovascular, oncología y angiogénesis.

Se han encontrado 87 productos de "RAAS"

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  • Telmisartan

    CAS:
    <p>Telmisartan (BIBR 277) is an Angiotensin 2 Receptor Blocker. The mechanism of action of telmisartan is as an Angiotensin 2 Receptor Antagonist.</p>
    Fórmula:C33H30N4O2
    Pureza:99.88% - 99.97%
    Forma y color:White Or Off White Crystalline Powder
    Peso molecular:514.62
  • Pomisartan 2HCl


    <p>Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.</p>
    Fórmula:C31H32Cl2N4O2
    Pureza:99.88%
    Forma y color:Soild
    Peso molecular:563.52
  • Losartan potassium

    CAS:
    <p>Losartan potassium (DuP-753 potassium) , an Angiotensin II Receptor Blocker, selectively and competitively blocks the binding of angiotensin II to the</p>
    Fórmula:C22H22ClKN6O
    Pureza:99.9% - >99.99%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:461.01
  • Losartan

    CAS:
    <p>Losartan (DuP-753) is an angiotensin II receptor antagonist.</p>
    Fórmula:C22H23ClN6O
    Pureza:99.48% - >99.99%
    Forma y color:Off White Solid Powder
    Peso molecular:422.91
  • Olmesartan Medoxomil

    CAS:
    <p>Olmesartan Medoxomil (Benicar) is an angiotensin II type 1 receptor blocker that is used to manage hypertension.</p>
    Fórmula:C29H30N6O6
    Pureza:99.89% - 99.9%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:558.59
  • Zansecimab

    CAS:
    <p>Zansecimab (LY-3127804) is a monoclonal antibody targeting angiopoietin 2 (Ang 2) for the study of cardiovascular and immune diseases.</p>
    Pureza:97.8% (SDS-PAGE); 99.7% (SEC-HPLC) - 97.8% (SDS-PAGE); 99.7% (SEC-HPLC)
    Forma y color:Liquid
  • Brain Natriuretic Peptide (1-32), rat

    CAS:
    <p>Rat Brain Natriuretic Peptide (1-32) is a 32-amino-acid peptide from heart, released when ventricles stretch excessively.</p>
    Fórmula:C146H239N47O44S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3452.94
  • Angiotensin amide

    CAS:
    <p>Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.</p>
    Fórmula:C49H70N14O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1031.17
  • Saralasin

    CAS:
    Competitive non-selective angiotensin II antagonist.
    Fórmula:C42H65N13O10
    Pureza:98%
    Forma y color:Powder
    Peso molecular:912
  • TRV055 acetate


    <p>TRV055 acetate is a ligand of angiotensin II type 1 receptor and stimulates cellular Gq-mediated signaling.</p>
    Fórmula:C44H61N9O11
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:892.01
  • Angiotensin II 5-valine

    CAS:
    <p>ngiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors.</p>
    Fórmula:C49H69N13O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:N/A
  • Alunacedase alfa

    CAS:
    <p>Alunacedase alfa (APN-01) is an angiotensin-converting enzyme 2 with antiviral activity.</p>
    Pureza:99.1% (SDS-PAGE); 99.9% (SEC-HPLC) - 99.1% (SDS-PAGE); 99.9% (SEC-HPLC)
    Forma y color:Liquid
  • Azilsartan Medoxomil Potassium

    CAS:
    <p>Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.</p>
    Fórmula:C30H23N4O8·K
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:606.62
  • Aliskiren D6 Hydrochloride

    CAS:
    <p>Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).</p>
    Fórmula:C30H54ClN3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:594.26
  • [Sar1, Ile8]-Angiotensin II

    CAS:
    <p>[Sar1, Ile8]-Angiotensin II(3TFA) is a peptide that has multiple effects on vascular smooth muscle.</p>
    Fórmula:C46H73N13O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:968.15
  • [Sar1, Ile8]-Angiotensin II acetate


    <p>'[Sar1, Ile8]-Angiotensin II acetate triggers oxidases and prompts superoxide in muscles; has varied vascular impacts.</p>
    Fórmula:C48H77N13O12
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:1028.2
  • [Sar1, Ile8]-Angiotensin II TFA


    <p>[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.</p>
    Fórmula:C48H74F3N13O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1082.18
  • Angiotensin II (1-4), human TFA


    <p>Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.</p>
    Fórmula:C26H38F3N7O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:665.62
  • Handle region peptide, rat

    CAS:
    <p>Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.</p>
    Fórmula:C54H101N15O12S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1184.54
  • Angiotensin II (5-8), human

    CAS:
    <p>Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II</p>
    Fórmula:C26H36N6O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:512.6