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Proteasas / Proteasoma

Proteasas / Proteasoma

Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.

Subcategorías de "Proteasas / Proteasoma"

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Se han encontrado 1044 productos de "Proteasas / Proteasoma"

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  • Zampilimab

    CAS:
    <p>Zampilimab (UCB-7858) is a humanised monoclonal antibody targeting TGM2, inhibits the cross-linking transamidase activity of TG2, renal fibrosis.</p>
    Pureza:95%
    Forma y color:Liquid
  • HCV-IN-30

    CAS:
    <p>HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).</p>
    Fórmula:C36H44N6O4
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:624.77
  • Carboxypeptidase G2 (CPG2) Inhibitor

    CAS:
    <p>Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.</p>
    Fórmula:C13H15NO6S
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:313.33
  • Cathepsin Inhibitor 1

    CAS:
    <p>Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.</p>
    Fórmula:C20H24ClN5O2
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:401.89
  • A-933548

    CAS:
    <p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>
    Fórmula:C25H21N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.47
  • Cysteine Protease inhibitor hydrochloride

    CAS:
    <p>Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.</p>
    Fórmula:C18H15ClN4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.79
  • Tec-IN-21

    CAS:
    <p>Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).</p>
    Fórmula:C16H15ClN4O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:362.83
  • Sheng Gelieting

    CAS:
    <p>CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.</p>
    Fórmula:C17H16F6N4O
    Forma y color:Solid
    Peso molecular:406.33
  • CP-471474

    CAS:
    <p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>
    Fórmula:C16H17FN2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:368.38
  • AGLME

    CAS:
    <p>AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.</p>
    Fórmula:C11H21N3O4
    Forma y color:Solid
    Peso molecular:259.3
  • SJA6017

    CAS:
    <p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>
    Fórmula:C17H25FN2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:372.45
  • SQ 32602

    CAS:
    <p>SQ 32602 is a cathepsin E inhibitor.</p>
    Fórmula:C32H52N3O7P
    Forma y color:Solid
    Peso molecular:621.74
  • Tyrosinase-IN-8


    <p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>
    Fórmula:C16H12O4
    Forma y color:Solid
    Peso molecular:268.26
  • DPP-4-IN-2

    CAS:
    <p>DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.</p>
    Fórmula:C18H18N6O
    Forma y color:Solid
    Peso molecular:334.38
  • Alvelestat tosylate

    CAS:
    Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.
    Fórmula:C32H30F3N5O7S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:717.73
  • Thrombin Inhibitor 2

    CAS:
    <p>Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.</p>
    Fórmula:C19H16ClF3N6O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:452.82
  • (Rac)-Tanomastat

    CAS:
    <p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>
    Fórmula:C23H19ClO3S
    Forma y color:Solid
    Peso molecular:410.91
  • PSI-7409 tetrasodium

    CAS:
    <p>PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.</p>
    Fórmula:C10H16FN2Na4O14P3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:592.117
  • Evogliptin HCl

    CAS:
    <p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>
    Fórmula:C19H27ClF3N3O3
    Forma y color:Solid
    Peso molecular:437.88
  • LY 806303

    CAS:
    <p>LY 806303 is a highly selective thrombin inhibitor.</p>
    Fórmula:C16H14O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:318.34
  • Nucleoside-Analog-2

    CAS:
    <p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>
    Fórmula:C9H11N5O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:285.21
  • BI-L 45XX

    CAS:
    <p>BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.</p>
    Fórmula:C10H9F3N2O2S
    Forma y color:Solid
    Peso molecular:278.25
  • Tyrphostin 47

    CAS:
    <p>Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.</p>
    Fórmula:C10H8N2O2S
    Forma y color:Solid
    Peso molecular:220.25
  • Levovirin valinate HCl

    CAS:
    <p>Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.</p>
    Fórmula:C13H22ClN5O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:379.8
  • Ici 186756

    CAS:
    <p>Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.</p>
    Fórmula:C33H49N5O9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:659.77
  • Chymase-IN-2

    CAS:
    <p>Chymase-IN-2 is a modulator of chymase.</p>
    Fórmula:C19H15ClF2NO3PS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:441.82
  • A-953227

    CAS:
    <p>A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.</p>
    Fórmula:C25H20FN5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:457.46
  • Duazomycin

    CAS:
    <p>Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.</p>
    Fórmula:C8H11N3O4
    Forma y color:Solid
    Peso molecular:213.19
  • Moxicoumone

    CAS:
    <p>Moxicoumone is an anticoagulant agent.</p>
    Fórmula:C22H30N2O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:418.48
  • GLS1 Inhibitor

    CAS:
    <p>GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.</p>
    Fórmula:C19H21N7O2S
    Forma y color:Solid
    Peso molecular:411.48
  • Tyrphostin A46

    CAS:
    <p>Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.</p>
    Fórmula:C10H8N2O3
    Pureza:98%
    Forma y color:Off-White Solid
    Peso molecular:204.18
  • NVP DPP 728 dihydrochloride

    CAS:
    <p>NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.</p>
    Fórmula:C15H18N6O
    Forma y color:Solid
    Peso molecular:298.34
  • MDK0734

    CAS:
    <p>MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>
    Fórmula:C15H17N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:271.31
  • Bz-D-Arg-pNA hydrochloride

    CAS:
    <p>Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.</p>
    Fórmula:C19H23ClN6O4
    Forma y color:Solid
    Peso molecular:434.88
  • FQ

    CAS:
    <p>FQ is a novel reversible inhibitor of mixed-type tyrosinase.</p>
    Fórmula:C14H9FN2O
    Forma y color:Solid
    Peso molecular:240.23
  • ND-336

    CAS:
    <p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>
    Fórmula:C16H18ClNO3S2
    Forma y color:Solid
    Peso molecular:371.9
  • ADAMTS-5 Inhibitor

    CAS:
    <p>ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.</p>
    Fórmula:C16H11ClF3N3OS3
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:449.92
  • DPP-IV-IN-1

    CAS:
    <p>DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).</p>
    Fórmula:C11H18FN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:243.28
  • TNIK-IN-1

    CAS:
    <p>TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).</p>
    Fórmula:C19H17N5O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:395.43
  • Diethyl pyimDC

    CAS:
    <p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>
    Fórmula:C14H15N3O4
    Forma y color:Solid
    Peso molecular:289.29
  • Aldumastat

    CAS:
    <p>Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.</p>
    Fórmula:C20H24F2N4O3
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:406.43
  • YM-53601

    CAS:
    <p>YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.</p>
    Fórmula:C21H22ClFN2O
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:372.86
  • MK-4882

    CAS:
    <p>MK-4882 is an effective inhibitor of HCV NS5A.</p>
    Fórmula:C42H50N8O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:778.9
  • Gosogliptin

    CAS:
    <p>Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.</p>
    Fórmula:C17H24F2N6O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:366.41
  • Nucleoside-Analog-1

    CAS:
    Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.
    Fórmula:C9H9N5O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:267.2
  • Sortin1

    CAS:
    <p>Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.</p>
    Fórmula:C26H19NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:441.43
  • MDK7677

    CAS:
    <p>MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>
    Fórmula:C12H10N4O3
    Forma y color:Solid
    Peso molecular:258.23
  • Furaprofen

    CAS:
    <p>Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.</p>
    Fórmula:C17H14O3
    Pureza:98.49% - 99.52%
    Forma y color:Solid
    Peso molecular:266.29
  • GEMSA

    CAS:
    <p>GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].</p>
    Fórmula:C7H13N3O4S
    Forma y color:Solid
    Peso molecular:235.26
  • WAY-151693

    CAS:
    <p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>
    Fórmula:C21H22ClN3O5S
    Forma y color:Solid
    Peso molecular:463.93
  • AK 275

    CAS:
    <p>AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.</p>
    Fórmula:C20H31N3O4
    Forma y color:Solid
    Peso molecular:377.48
  • AZD-9684

    CAS:
    <p>AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.</p>
    Fórmula:C10H14N2O2S
    Forma y color:Solid
    Peso molecular:226.3
  • ITX-4520

    CAS:
    <p>ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.</p>
    Fórmula:C24H23F2N3OS
    Forma y color:Solid
    Peso molecular:439.52
  • Epostatin

    CAS:
    <p>Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.</p>
    Fórmula:C23H33N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:431.53
  • L 722151

    CAS:
    <p>L 722151 is an FXIIIa inhibitor.</p>
    Fórmula:C8H9ClN2O5S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:344.82
  • Chymase-IN-1

    CAS:
    <p>Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).</p>
    Fórmula:C20H15ClNO4PS
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:431.83
  • GSK-2793660

    CAS:
    <p>GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.</p>
    Fórmula:C20H27N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:357.45
  • ADAMTS-5-IN-2

    CAS:
    <p>ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.</p>
    Fórmula:C17H15N3OS
    Forma y color:Solid
    Peso molecular:309.39
  • Safironil

    CAS:
    <p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>
    Fórmula:C15H23N3O4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:309.36
  • TNK2-IN-1

    CAS:
    <p>TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.</p>
    Fórmula:C23H24N6O2
    Forma y color:Solid
    Peso molecular:416.48
  • SP-Chymostatin B

    CAS:
    <p>SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.</p>
    Fórmula:C30H41N7O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:595.69
  • K 579

    CAS:
    <p>K 579 is a dipeptidyl peptidase IV inhibitor.</p>
    Fórmula:C17H24N6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:328.41
  • Antiviral agent 30

    CAS:
    <p>Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].</p>
    Fórmula:C21H32N2O3S
    Forma y color:Solid
    Peso molecular:392.56
  • PTIQ

    CAS:
    <p>MMP-3 expression inhibitor</p>
    Fórmula:C13H17NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:235.28
  • BAY-678 racemate

    CAS:
    <p>BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.</p>
    Fórmula:C20H15F3N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:400.35
  • WNK-IN-7

    CAS:
    <p>WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.</p>
    Fórmula:C26H29N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:399.53
  • ABT-770

    CAS:
    <p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>
    Fórmula:C22H22F3N3O6
    Forma y color:Solid
    Peso molecular:481.42
  • BR351 precursor

    CAS:
    <p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>
    Fórmula:C27H32N2O8S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:576.68
  • CA 074

    CAS:
    <p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>
    Fórmula:C18H29N3O6
    Pureza:97.80%
    Forma y color:Solid
    Peso molecular:383.44
  • XMU-MP-2

    CAS:
    <p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>
    Fórmula:C32H33F3N8O2
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:618.65
  • RS-104966

    CAS:
    <p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>
    Fórmula:C19H21NO6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:391.44
  • Ono-3307 mesylate

    CAS:
    <p>no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.</p>
    Fórmula:C15H18N4O7S2
    Pureza:97.60% - 98.16%
    Forma y color:Solid
    Peso molecular:430.46
  • Thrombin inhibitor 6

    CAS:
    <p>Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.</p>
    Fórmula:C18H19ClN4O2S
    Forma y color:Solid
    Peso molecular:390.89
  • 2',5-Difluoro-2'-deoxycytidine

    CAS:
    <p>2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.</p>
    Fórmula:C9H11F2N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:263.2
  • Gü1303

    CAS:
    <p>Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).</p>
    Fórmula:C20H22N4O3
    Forma y color:Solid
    Peso molecular:366.41
  • LY 135305

    CAS:
    <p>LY 135305 is a inhibition of spontaneous metastasis.</p>
    Fórmula:C19H20ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:297.82
  • Batimastat sodium salt

    CAS:
    <p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>
    Fórmula:C23H31N3NaO4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:500.63
  • HCV-IN-37

    CAS:
    <p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>
    Fórmula:C31H35F2N5
    Forma y color:Solid
    Peso molecular:515.64
  • BrBzGCp2

    CAS:
    <p>BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.</p>
    Fórmula:C27H38BrN3O6S
    Pureza:98.68% - 98.68%
    Forma y color:Solid
    Peso molecular:612.58
  • ACH-806

    CAS:
    <p>ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.</p>
    Fórmula:C19H20F3N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:411.44
  • Tyrosinase-IN-1

    CAS:
    <p>Tyrosinase-IN-1: potent inhibitor for skin-whitening &amp; food preservation with uses in cosmetics &amp; medicine.</p>
    Fórmula:C10H9N3O2S2
    Forma y color:Solid
    Peso molecular:267.33
  • KIN1400

    CAS:
    <p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>
    Fórmula:C24H17F2N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:449.47
  • MK-2048

    CAS:
    <p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>
    Fórmula:C21H21ClFN5O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:461.87
  • OM-189

    CAS:
    <p>OM-189 is a selective inhibitor of synthetic thrombin.</p>
    Fórmula:C24H36N6O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:488.65
  • Adafosbuvir PM

    CAS:
    <p>Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.</p>
    Fórmula:C10H13FN2O6
    Pureza:97.08%
    Forma y color:Solid
    Peso molecular:276.22
  • FK-448 Free base

    CAS:
    <p>FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.</p>
    Fórmula:C25H30N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:406.52
  • BMS-986094

    CAS:
    <p>INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.</p>
    Fórmula:C30H39N6O9P
    Forma y color:Solid
    Peso molecular:658.64
  • BR351

    CAS:
    <p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>
    Fórmula:C20H25FN2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:424.49
  • LB-30057

    CAS:
    <p>LB-30057 is used as an oral thrombin inhibitor.</p>
    Fórmula:C26H31N5O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:493.62
  • U 27391

    CAS:
    <p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>
    Fórmula:C23H36N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:448.56
  • MDL-101146, (S)-

    CAS:
    <p>MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.</p>
    Fórmula:C29H37F5N4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:632.62
  • Gemigliptin Tartrate(911637-19-9 free base)

    CAS:
    <p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>
    Fórmula:C22H25F8N5O8
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:639.45
  • Cysteine protease inhibitor-2

    CAS:
    <p>Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.</p>
    Fórmula:C13H5N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:247.21
  • ZD8321

    CAS:
    <p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>
    Fórmula:C18H28F3N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:423.43
  • Proteasome-IN-1

    CAS:
    <p>Proteasome-IN-1 is an inhibitor of proteasome.</p>
    Fórmula:C42H35N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:657.76
  • Tanomastat

    CAS:
    <p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>
    Fórmula:C23H19ClO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.91
  • IMB-26

    CAS:
    <p>IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.</p>
    Fórmula:C20H23BrN2O6
    Forma y color:Solid
    Peso molecular:467.31
  • TAPI-1

    CAS:
    <p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>
    Fórmula:C26H37N5O5
    Pureza:≥95%
    Forma y color:Solid
    Peso molecular:499.6
  • Desethyl KBT-3022

    CAS:
    <p>Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.</p>
    Fórmula:C23H20N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.48
  • ZYZ-488

    CAS:
    <p>ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.</p>
    Fórmula:C20H29N3O11
    Pureza:99.04%
    Forma y color:Solid
    Peso molecular:487.46
  • STOCK2S-26016

    CAS:
    <p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>
    Fórmula:C20H19N3O2
    Forma y color:Solid
    Peso molecular:333.38
  • Efegatran sulfate

    CAS:
    <p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>
    Fórmula:C21H34N6O7S
    Pureza:≥98% - ≥98%
    Forma y color:Solid
    Peso molecular:514.6
  • AA9 TG2 inhibitor

    CAS:
    <p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>
    Fórmula:C32H36N4O5
    Forma y color:Solid
    Peso molecular:556.65
  • Desirudin

    CAS:
    <p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>
    Forma y color:Solid
  • GS-9256

    CAS:
    <p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>
    Fórmula:C46H56ClF2N6O8PS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:957.46
  • Z-LLF-CHO

    CAS:
    <p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>
    Fórmula:C29H39N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:509.64
  • MMP13-IN-4

    CAS:
    <p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>
    Fórmula:C21H17BrN4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:485.29
  • Cyclophilin inhibitor 3

    CAS:
    <p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>
    Fórmula:C34H38N4O6
    Forma y color:Solid
    Peso molecular:598.69
  • ND-322 HCl

    CAS:
    <p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>
    Fórmula:C15H16ClNO3S2
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:357.88
  • DTS

    CAS:
    <p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>
    Fórmula:C14H14S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:278.46
  • Prodipine hydrochloride

    CAS:
    <p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>
    Fórmula:C20H26ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:315.88
  • SLK/STK10-IN-1

    CAS:
    <p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>
    Fórmula:C17H13ClN2O3
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:328.75
  • ZD-0892

    CAS:
    <p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>
    Fórmula:C24H32F3N3O5
    Pureza:95% - 99.53%
    Forma y color:Solid
    Peso molecular:499.52
  • Grazoprevir sodium salt

    CAS:
    <p>Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.</p>
    Fórmula:C38H50N6NaO9S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:789.9
  • Tyrosinase-IN-4

    CAS:
    <p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>
    Fórmula:C15H9ClO3
    Forma y color:Solid
    Peso molecular:272.68
  • JPM-OEt

    CAS:
    <p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>
    Fórmula:C20H28N2O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:392.45
  • N-Phenylthiourea

    CAS:
    <p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>
    Fórmula:C7H8N2S
    Pureza:99.71%
    Forma y color:Solid
    Peso molecular:152.22
  • (S)-BI-1001

    CAS:
    <p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>
    Fórmula:C19H15BrClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.68
  • p-Aminobenzamidine dihydrochloride

    CAS:
    <p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>
    Fórmula:C7H11Cl2N3
    Pureza:99.00% - 99.56%
    Forma y color:Solid
    Peso molecular:208.088
  • PF-00356231 hydrochloride

    CAS:
    <p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>
    Fórmula:C25H21ClN2O3S
    Pureza:98.39%
    Forma y color:Solid
    Peso molecular:464.96
  • Ro 09-1679

    CAS:
    <p>Ro 09-1679 is a thrombin inhibitor.</p>
    Fórmula:C22H39N9O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:525.6
  • Cathepsin L/S-IN-1


    <p>Cathepsin L/S-IN-1 inhibits Cathepsin L &amp; S (IC50: 4.10 &amp; 1.79 μM) and reduces metastasis in pancreatic cancer cells.</p>
    Fórmula:C29H33BrN4O4S
    Forma y color:Solid
    Peso molecular:613.57
  • NNGH

    CAS:
    <p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>
    Fórmula:C13H20N2O5S
    Pureza:98.41%
    Forma y color:Solid
    Peso molecular:316.37
  • Navuridine

    CAS:
    <p>Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.</p>
    Fórmula:C9H11N5O4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:253.22
  • ZM223 hydrochloride (2031177-48-5 free base)


    <p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>
    Fórmula:C23H18ClF3N4O2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:538.99
  • Diprotin B

    CAS:
    <p>Diprotin B is a dipeptidyl peptidase IV inhibitor.</p>
    Fórmula:C16H29N3O4
    Pureza:98%
    Forma y color:White Lyophilized Powder
    Peso molecular:327.42
  • HCV-IN-3

    CAS:
    <p>HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).</p>
    Fórmula:C13H11F2NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:235.23
  • Calpain Inhibitor XII

    CAS:
    <p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>
    Fórmula:C26H34N4O5
    Forma y color:Solid
    Peso molecular:482.57
  • Flovagatran

    CAS:
    <p>Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.</p>
    Fórmula:C27H36BN3O7
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:525.4
  • RO-9187

    CAS:
    <p>RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).</p>
    Fórmula:C9H12N6O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:284.23
  • Plasma kallikrein-IN-3

    CAS:
    <p>Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.</p>
    Fórmula:C20H23N5O2
    Forma y color:Solid
    Peso molecular:365.43
  • 2-MPPA

    CAS:
    <p>2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.</p>
    Fórmula:C8H14O4S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:206.26
  • Calpain-2-IN-1

    CAS:
    <p>Calpain-2-IN-1 is a selective calpain-2 inhibitor that prolongs ERK activation and thus enhances learning and memory.</p>
    Fórmula:C28H37N3O7
    Forma y color:Solid
    Peso molecular:527.61
  • Tyrosinase-IN-10

    CAS:
    <p>Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'</p>
    Fórmula:C16H12O4
    Forma y color:Solid
    Peso molecular:268.26
  • TAPI-0

    CAS:
    <p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>
    Fórmula:C24H32N4O5
    Forma y color:Solid
    Peso molecular:456.53
  • NAAA-IN-2

    CAS:
    <p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>
    Fórmula:C11H13N3O2S
    Forma y color:Solid
    Peso molecular:251.3
  • HCV-IN-35

    CAS:
    <p>HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.</p>
    Fórmula:C30H36ClN5
    Forma y color:Solid
    Peso molecular:502.09
  • MMP-1-IN-1


    <p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>
    Fórmula:C14H17ClN2O3
    Forma y color:Solid
    Peso molecular:296.75
  • Calpain Inhibitor XI

    CAS:
    <p>Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.</p>
    Fórmula:C26H40N4O6
    Forma y color:Solid
    Peso molecular:504.62
  • (3S,4S)-A2-32-01


    <p>(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .</p>
    Fórmula:C19H27NO2
    Forma y color:Solid
    Peso molecular:301.42
  • Azo-Resveratrol

    CAS:
    <p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>
    Fórmula:C12H10N2O3
    Forma y color:Solid
    Peso molecular:230.22
  • AM 4299 B

    CAS:
    <p>AM 4299 B is a novel inhibitor of a thiol protease.</p>
    Fórmula:C16H27N3O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:373.4
  • HCV-IN-34

    CAS:
    <p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>
    Fórmula:C31H36ClN5
    Forma y color:Solid
    Peso molecular:514.1
  • MDL 27399

    CAS:
    <p>MDL 27399 suppresses human neutrophil cathepsin G.</p>
    Fórmula:C26H36N4O8
    Forma y color:Solid
    Peso molecular:532.59
  • Tyrosinase-IN-7

    CAS:
    <p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>
    Fórmula:C15H10O5
    Pureza:99%
    Forma y color:Solid
    Peso molecular:270.24
  • CAA0225

    CAS:
    <p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>
    Fórmula:C28H29N3O5
    Forma y color:Solid
    Peso molecular:487.55
  • BC-05

    CAS:
    <p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>
    Fórmula:C21H29BN2O9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:464.27
  • RID-F

    CAS:
    <p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>
    Fórmula:C38H50N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:566.82
  • AL-9

    CAS:
    <p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>
    Fórmula:C23H22N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:402.45
  • Immunoproteasome inhibitor 1

    CAS:
    <p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>
    Fórmula:C20H26N2O4
    Forma y color:Solid
    Peso molecular:358.43
  • PMPA sodium

    CAS:
    <p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>
    Fórmula:C6H11Na4O7P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:318.08
  • JO146

    CAS:
    <p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。</p>
    Fórmula:C31H44N3O7P
    Forma y color:Solid
    Peso molecular:601.67
  • L-873724

    CAS:
    <p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>
    Fórmula:C23H26F3N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.53
  • (R)-ND-336

    CAS:
    <p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>
    Fórmula:C16H18ClNO3S2
    Forma y color:Solid
    Peso molecular:371.89
  • Tyrosinase-IN-11

    CAS:
    <p>Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.</p>
    Fórmula:C15H14O5
    Forma y color:Solid
    Peso molecular:274.27
  • Kallikrein 5-IN-2

    CAS:
    <p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation &amp; itching.</p>
    Fórmula:C23H22N6O
    Forma y color:Solid
    Peso molecular:398.46
  • VA4 TG2 inhibitor

    CAS:
    <p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>
    Fórmula:C33H41N5O6S
    Forma y color:Solid
    Peso molecular:635.77
  • AZD5248

    CAS:
    <p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>
    Fórmula:C22H22N4O2
    Forma y color:Solid
    Peso molecular:374.44
  • MMP-2/9-IN-1

    CAS:
    <p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>
    Fórmula:C14H16IN7S
    Forma y color:Solid
    Peso molecular:441.29
  • GLS1 Inhibitor-3

    CAS:
    <p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>
    Fórmula:C30H32N10O2S
    Forma y color:Solid
    Peso molecular:596.71
  • Elastase-IN-1

    CAS:
    <p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>
    Fórmula:C17H12N4O3
    Forma y color:Solid
    Peso molecular:320.3
  • HCV-IN-36

    CAS:
    <p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>
    Fórmula:C30H36ClN5
    Forma y color:Solid
    Peso molecular:502.09
  • BRD-8899

    CAS:
    <p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>
    Fórmula:C17H22N4O3S
    Forma y color:Solid
    Peso molecular:362.45
  • Tyrosinase-IN-5

    CAS:
    <p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>
    Fórmula:C18H13N3O6
    Forma y color:Solid
    Peso molecular:367.31
  • BMS-363131

    CAS:
    <p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of &lt;1.7 nM.</p>
    Fórmula:C28H40N6O5
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:540.65
  • α-Glucosidase-IN-5

    CAS:
    <p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>
    Fórmula:C15H13NO3
    Forma y color:Solid
    Peso molecular:255.27
  • SAP2-IN-1

    CAS:
    <p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>
    Fórmula:C34H29NO7
    Forma y color:Solid
    Peso molecular:563.6
  • Elasnin

    CAS:
    <p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>
    Fórmula:C24H40O4
    Forma y color:Solid
    Peso molecular:392.57
  • MMP2-IN-2

    CAS:
    <p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>
    Fórmula:C13H8N4O4
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:284.23
  • Glutaminase-IN-4

    CAS:
    <p>Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).</p>
    Fórmula:C23H22N6O2S2
    Forma y color:Solid
    Peso molecular:478.59
  • L 658758

    CAS:
    <p>L 658758 is an inhibitor of serine proteinase.</p>
    Fórmula:C16H20N2O9S
    Forma y color:Solid
    Peso molecular:416.4
  • ASPER-29

    CAS:
    <p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>
    Fórmula:C31H29BrN2O5S
    Forma y color:Solid
    Peso molecular:621.54
  • CAY10704

    CAS:
    <p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>
    Fórmula:C18H20Cl2N2
    Forma y color:Solid
    Peso molecular:335.27
  • DPP-4-IN-1

    CAS:
    <p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>
    Fórmula:C19H19ClN6
    Forma y color:Solid
    Peso molecular:366.85
  • AA10 TG2 inhibitor

    CAS:
    <p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>
    Fórmula:C32H36N4O5
    Forma y color:Solid
    Peso molecular:556.65
  • BAY8040

    CAS:
    <p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>
    Fórmula:C21H16F3N5O2
    Forma y color:Solid
    Peso molecular:427.38
  • PK44 phosphate

    CAS:
    <p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>
    Fórmula:C17H19F5N7O5P
    Forma y color:Solid
    Peso molecular:527.349
  • VEL-0230

    CAS:
    <p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>
    Fórmula:C14H24NNaO5
    Forma y color:Solid
    Peso molecular:309.33
  • Alicapistat

    CAS:
    <p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>
    Fórmula:C25H27N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:433.5
  • Tyrosinase-IN-6

    CAS:
    <p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>
    Fórmula:C24H31N3O2
    Forma y color:Solid
    Peso molecular:393.52
  • Cysteine Protease inhibitor

    CAS:
    <p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>
    Fórmula:C18H14N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.33
  • Anticancer agent 82

    CAS:
    <p>Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.</p>
    Fórmula:C19H18Cl2N4O
    Forma y color:Solid
    Peso molecular:389.28
  • Tyrosinase-IN-3

    CAS:
    <p>Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.</p>
    Fórmula:C21H23NO5
    Forma y color:Solid
    Peso molecular:369.41
  • BC-23

    CAS:
    <p>BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.</p>
    Fórmula:C21H14ClN3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.87
  • Gü2602

    CAS:
    <p>Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for mature</p>
    Fórmula:C16H22N4O3
    Forma y color:Solid
    Peso molecular:318.37
  • Cofrogliptin

    CAS:
    <p>Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).</p>
    Fórmula:C18H19F5N4O3S
    Forma y color:Solid
    Peso molecular:466.43
  • GSK2793660 HCl

    CAS:
    <p>GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.</p>
    Fórmula:C22H32ClN3O3
    Forma y color:Solid
    Peso molecular:421.96
  • HCV-IN-33

    CAS:
    <p>HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.</p>
    Fórmula:C31H36ClN5
    Forma y color:Solid
    Peso molecular:514.1
  • JNJ-10329670

    CAS:
    <p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>
    Fórmula:C30H34ClF3N6O3S
    Forma y color:Solid
    Peso molecular:651.14
  • Setrobuvir

    CAS:
    <p>Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension with</p>
    Fórmula:C25H25FN4O6S2
    Pureza:98.92% - >99.99%
    Forma y color:Solid
    Peso molecular:560.62
  • KM-023

    CAS:
    <p>KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.</p>
    Fórmula:C18H19N3O3
    Pureza:99.47% - >99.99%
    Forma y color:Solid
    Peso molecular:325.36
  • AGPS-IN-2i

    CAS:
    AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.
    Fórmula:C18H17F2N3O2
    Pureza:98.92%
    Forma y color:Solid
    Peso molecular:345.34
  • TS-021

    CAS:
    <p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>
    Fórmula:C17H24FN3O5S
    Pureza:>99.99% - >99.99%
    Forma y color:Solid
    Peso molecular:401.45
  • 20S Proteasome activator 1

    CAS:
    <p>20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.</p>
    Fórmula:C27H19ClF2N2OS
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:492.97
  • CPA inhibitor

    CAS:
    <p>CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.</p>
    Fórmula:C18H19NO4
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:313.35
  • Uprifosbuvir

    CAS:
    <p>Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.</p>
    Fórmula:C22H29ClN3O9P
    Pureza:99.73% - >99.99%
    Forma y color:Solid
    Peso molecular:545.91
  • Atevirdine

    CAS:
    <p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>
    Fórmula:C21H25N5O2
    Pureza:98.20%
    Forma y color:Solid
    Peso molecular:379.46
  • CZL55

    CAS:
    <p>CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).</p>
    Fórmula:C20H22N2O6
    Pureza:98.19%
    Forma y color:Solid
    Peso molecular:386.4
  • Granotapide

    CAS:
    <p>Granotapide is a microsomal triglyceride transfer protein (MTP) inhibitor that treats and rather prevents atherosclerosis, coronary artery disease, metabolic</p>
    Fórmula:C39H37F3N2O8
    Pureza:99.70% - 99.79%
    Forma y color:Solid
    Peso molecular:718.71
  • BAY-43-9695

    CAS:
    <p>BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.</p>
    Fórmula:C22H25N3O4S
    Pureza:99.50% - 99.65%
    Forma y color:Solid
    Peso molecular:427.52