Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(35 productos)
- Cisteína proteasa(96 productos)
- DPP-4(20 productos)
- Glutaminasa(40 productos)
- Proteasa del VIH(451 productos)
- PAI-1(25 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(53 productos)
- Proteasoma(94 productos)
- Serina proteasa(49 productos)
- p97(14 productos)
Mostrar 3 subcategorías más
Se han encontrado 1039 productos de "Proteasas / Proteasoma"
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TNK2-IN-1
CAS:<p>TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.</p>Fórmula:C23H24N6O2Forma y color:SolidPeso molecular:416.48Moxicoumone
CAS:<p>Moxicoumone is an anticoagulant agent.</p>Fórmula:C22H30N2O6Pureza:98%Forma y color:SolidPeso molecular:418.48K 579
CAS:<p>K 579 is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C17H24N6OPureza:98%Forma y color:SolidPeso molecular:328.41PTIQ
CAS:<p>MMP-3 expression inhibitor</p>Fórmula:C13H17NO3Pureza:98%Forma y color:SolidPeso molecular:235.28RO-9187
CAS:<p>RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).</p>Fórmula:C9H12N6O5Pureza:98%Forma y color:SolidPeso molecular:284.23Ro 09-1679
CAS:<p>Ro 09-1679 is a thrombin inhibitor.</p>Fórmula:C22H39N9O6Pureza:98%Forma y color:SolidPeso molecular:525.6N-Phenylthiourea
CAS:<p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>Fórmula:C7H8N2SPureza:99.71%Forma y color:SolidPeso molecular:152.22Tyrphostin A46
CAS:<p>Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.</p>Fórmula:C10H8N2O3Pureza:98%Forma y color:Off-White SolidPeso molecular:204.18JPM-OEt
CAS:<p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>Fórmula:C20H28N2O6Pureza:98%Forma y color:SolidPeso molecular:392.45KIN1400
CAS:<p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>Fórmula:C24H17F2N3O2SPureza:98%Forma y color:SolidPeso molecular:449.47Grazoprevir sodium salt
CAS:Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.Fórmula:C38H50N6NaO9SPureza:98%Forma y color:SolidPeso molecular:789.9Prodipine hydrochloride
CAS:<p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>Fórmula:C20H26ClNPureza:98%Forma y color:SolidPeso molecular:315.88ZM223 hydrochloride (2031177-48-5 free base)
<p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>Fórmula:C23H18ClF3N4O2S2Pureza:98%Forma y color:SolidPeso molecular:538.99FK-448 Free base
CAS:<p>FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.</p>Fórmula:C25H30N2O3Pureza:98%Forma y color:SolidPeso molecular:406.52(S)-BI-1001
CAS:<p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>Fórmula:C19H15BrClNO3Pureza:98%Forma y color:SolidPeso molecular:420.68BMS-986094
CAS:<p>INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.</p>Fórmula:C30H39N6O9PForma y color:SolidPeso molecular:658.64Navuridine
CAS:<p>Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.</p>Fórmula:C9H11N5O4Pureza:99.83%Forma y color:SolidPeso molecular:253.22p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Fórmula:C7H11Cl2N3Pureza:99.00% - 99.56%Forma y color:SolidPeso molecular:208.088LB-30057
CAS:<p>LB-30057 is used as an oral thrombin inhibitor.</p>Fórmula:C26H31N5O3SPureza:98%Forma y color:SolidPeso molecular:493.62U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Forma y color:SolidPeso molecular:448.56MDK0734
CAS:<p>MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Fórmula:C15H17N3O2Pureza:98%Forma y color:SolidPeso molecular:271.31MDL-101146, (S)-
CAS:<p>MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.</p>Fórmula:C29H37F5N4O6Pureza:98%Forma y color:SolidPeso molecular:632.62PMPA sodium
CAS:<p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>Fórmula:C6H11Na4O7PPureza:98%Forma y color:SolidPeso molecular:318.08IMB-26
CAS:<p>IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.</p>Fórmula:C20H23BrN2O6Forma y color:SolidPeso molecular:467.31Tyrosinase-IN-4
CAS:<p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>Fórmula:C15H9ClO3Forma y color:SolidPeso molecular:272.68Desethyl KBT-3022
CAS:<p>Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.</p>Fórmula:C23H20N2O4SPureza:98%Forma y color:SolidPeso molecular:420.48PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Forma y color:SolidPeso molecular:464.96DTS
CAS:<p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>Fórmula:C14H14S3Pureza:98%Forma y color:SolidPeso molecular:278.46Calpain Inhibitor XII
CAS:<p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>Fórmula:C26H34N4O5Forma y color:SolidPeso molecular:482.57STOCK2S-26016
CAS:<p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>Fórmula:C20H19N3O2Forma y color:SolidPeso molecular:333.38AL-9
CAS:<p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>Fórmula:C23H22N4O3Pureza:98%Forma y color:SolidPeso molecular:402.45NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Fórmula:C13H20N2O5SPureza:98.41%Forma y color:SolidPeso molecular:316.37AA9 TG2 inhibitor
CAS:<p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>Fórmula:C32H36N4O5Forma y color:SolidPeso molecular:556.65Desirudin
CAS:<p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>Forma y color:SolidCyclophilin inhibitor 3
CAS:<p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>Fórmula:C34H38N4O6Forma y color:SolidPeso molecular:598.69Diprotin B
CAS:<p>Diprotin B is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C16H29N3O4Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:327.42ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Fórmula:C24H32F3N3O5Pureza:95% - 99.53%Forma y color:SolidPeso molecular:499.52FQ
CAS:<p>FQ is a novel reversible inhibitor of mixed-type tyrosinase.</p>Fórmula:C14H9FN2OForma y color:SolidPeso molecular:240.23SLK/STK10-IN-1
CAS:<p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>Fórmula:C17H13ClN2O3Pureza:99.34%Forma y color:SolidPeso molecular:328.75RID-F
CAS:<p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>Fórmula:C38H50N2O2Pureza:98%Forma y color:SolidPeso molecular:566.82ADAMTS-5 Inhibitor
CAS:<p>ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.</p>Fórmula:C16H11ClF3N3OS3Pureza:99.66%Forma y color:SolidPeso molecular:449.92BC-05
CAS:<p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>Fórmula:C21H29BN2O9Pureza:98%Forma y color:SolidPeso molecular:464.27TNIK-IN-1
CAS:<p>TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).</p>Fórmula:C19H17N5O3SPureza:98%Forma y color:SolidPeso molecular:395.43Diethyl pyimDC
CAS:<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Fórmula:C14H15N3O4Forma y color:SolidPeso molecular:289.29Aldumastat
CAS:Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.Fórmula:C20H24F2N4O3Pureza:99.87%Forma y color:SolidPeso molecular:406.43Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Fórmula:C15H10O5Pureza:99%Forma y color:SolidPeso molecular:270.24MK-4882
CAS:<p>MK-4882 is an effective inhibitor of HCV NS5A.</p>Fórmula:C42H50N8O7Pureza:98%Forma y color:SolidPeso molecular:778.9Efegatran sulfate
CAS:<p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>Fórmula:C21H34N6O7SPureza:≥98% - ≥98%Forma y color:SolidPeso molecular:514.6HCV-IN-34
CAS:<p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>Fórmula:C31H36ClN5Forma y color:SolidPeso molecular:514.1Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Fórmula:C23H19ClO3SPureza:98%Forma y color:SolidPeso molecular:410.91
