
Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(20 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(506 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(95 productos)
- Serina proteasa(55 productos)
- p97(15 productos)
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Se han encontrado 1093 productos de "Proteasas / Proteasoma"
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Paritaprevir
CAS:<p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。</p>Fórmula:C40H43N7O7SPureza:99.72%Forma y color:SolidPeso molecular:765.88Grazoprevir
CAS:<p>Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.</p>Fórmula:C38H50N6O9SPureza:99.36% - >99.99%Forma y color:SolidPeso molecular:766.9Letermovir
CAS:Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.Fórmula:C29H28F4N4O4Pureza:99.85% - 99.87%Forma y color:SolidPeso molecular:572.55Ref: TM-T5396
1mg88,00€5mg170,00€10mg283,00€25mg497,00€50mg707,00€100mg1.008,00€200mg1.359,00€1mL*10mM (DMSO)216,00€Ivachtin
CAS:<p>Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining</p>Fórmula:C20H21N3O7SPureza:99.74%Forma y color:SolidPeso molecular:447.46CA-074 methyl ester
CAS:CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!Fórmula:C19H31N3O6Pureza:97.26% - 99.58%Forma y color:SolidPeso molecular:397.47Bemnifosbuvir
CAS:Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.Fórmula:C24H33FN7O7PPureza:99.35% - 99.54%Forma y color:SolidPeso molecular:581.53Ditiocarb sodium
CAS:Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improvesFórmula:C5H10NNaS2Pureza:98.04%Forma y color:White Solid CrystallinePeso molecular:171.26Coblopasvir dihydrochloride
CAS:Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.Fórmula:C41H52Cl2N8O8Pureza:99.33%Forma y color:SolidPeso molecular:855.81Ref: TM-T25268L
1mg87,00€5mg187,00€10mg305,00€25mg518,00€50mg742,00€100mg1.017,00€1mL*10mM (DMSO)298,00€Elvitegravir
CAS:Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.Fórmula:C23H23ClFNO5Pureza:98.43% - 99.57%Forma y color:SolidPeso molecular:447.88Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Fórmula:C19H21Cl2N3Pureza:>99.99%Forma y color:SolidPeso molecular:362.3Nelfinavir Mesylate
CAS:Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).Fórmula:C33H49N3O7S2Pureza:95.81% - 99.97%Forma y color:A White Or Almost White PowderPeso molecular:663.89Bemnifosbuvir hemisulfate
CAS:Bemnifosbuvir hemisulfate (AT-527) is a potent inhibitor of HCV virus replication.Fórmula:C48H68F2N14O18P2SPureza:99.98%Forma y color:SolidPeso molecular:1261.15PTACH
CAS:PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).Fórmula:C20H26N2O2S2Pureza:87.44% - 99.74%Forma y color:SolidPeso molecular:390.56TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Fórmula:C28H38F3N5O7Pureza:98.06%Forma y color:SolidPeso molecular:613.62Lusutrombopag
CAS:Lusutrombopag (Mulpleta) is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients withFórmula:C29H32Cl2N2O5SPureza:99.96%Forma y color:SolidPeso molecular:591.55Ref: TM-TQ0223
1mg64,00€2mg92,00€5mg137,00€10mg208,00€25mg416,00€50mg628,00€100mg938,00€200mg1.293,00€1mL*10mM (DMSO)170,00€Asunaprevir
CAS:Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.Fórmula:C35H46ClN5O9SPureza:99.34% - 99.8%Forma y color:SolidPeso molecular:748.29Ref: TM-T4474
1mg52,00€5mg111,00€10mg180,00€25mg354,00€50mg540,00€100mg778,00€500mg1.605,00€1mL*10mM (DMSO)173,00€Camostat free base
CAS:Camostat (FOY 305) inhibits serine protease, treats cancer, viral infections, fibrosis, and blocks SARS-CoV, Coronavirus, and SARS-CoV-2 in studies.Fórmula:C20H22N4O5Forma y color:SolidPeso molecular:398.41(S,S)-TAPI-1
CAS:"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."Fórmula:C26H37N5O5Forma y color:SolidPeso molecular:499.6PSI-6130
CAS:PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.Fórmula:C10H14FN3O4Pureza:98.63% - 99.79%Forma y color:SolidPeso molecular:259.23Ref: TM-T7607
1mg40,00€5mg89,00€10mg129,00€25mg224,00€50mg329,00€100mg482,00€200mg652,00€1mL*10mM (DMSO)78,00€Daclatasvir
CAS:Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.Fórmula:C40H50N8O6Pureza:99.81% - 99.99%Forma y color:SolidPeso molecular:738.88
