
Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(20 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(506 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(95 productos)
- Serina proteasa(55 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 1093 productos de "Proteasas / Proteasoma"
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ABT530
CAS:ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.Fórmula:C57H65F5N10O8Pureza:99.15% - 99.93%Forma y color:SolidPeso molecular:1113.184-Phenoxybenzylamine
CAS:4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against HCV NS3/4a .Fórmula:C13H13NOPureza:97.26%Forma y color:SolidPeso molecular:199.25TCH-165
CAS:TCH-165 boosts 20S proteasome levels, enhancing IDP breakdown.Fórmula:C39H37N3O3Pureza:98.2% - 98.75%Forma y color:SolidPeso molecular:595.73Ref: TM-T17011
1mg74,00€5mg160,00€10mg250,00€25mg455,00€50mg682,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)205,00€Boc-Asp(OMe)-fluoromethyl ketone
CAS:<p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>Fórmula:C11H18FNO5Pureza:≥98%Forma y color:SolidPeso molecular:263.26VCH-916
CAS:VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.Fórmula:C26H36KNO4SPureza:98%Forma y color:SolidPeso molecular:497.73LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Fórmula:C23H29ClN8OForma y color:SolidPeso molecular:468.98Daclatasvir dihydrochloride
CAS:Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.Fórmula:C40H52Cl2N8O6Pureza:99.67%Forma y color:SolidPeso molecular:811.8Ref: TM-T1786
1g244,00€5mg42,00€10mg50,00€25mg60,00€50mg71,00€100mg81,00€500mg170,00€1mL*10mM (DMSO)52,00€Paritaprevir
CAS:<p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。</p>Fórmula:C40H43N7O7SPureza:99.72%Forma y color:SolidPeso molecular:765.88Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Fórmula:C27H37N3O7SPureza:99.67% - 99.76%Forma y color:White Amorphous SolidPeso molecular:547.667-Amino-4-methylcoumarin-3-acetic acid
CAS:7-Amino-4-methylcoumarin-3-acetic acid (7-Amino-4-methylcoumarin) is more suitable as a substrate for enteropeptidase than GD(4)K-NA.Fórmula:C12H11NO4Pureza:98.38%Forma y color:SolidPeso molecular:233.22GSK-A1
CAS:GSK-A1 is a specific inhibitor of PI4KA, also inhibited calcium-driven PRL secretion without affecting calcium signaling and Prl expression.Fórmula:C29H27FN6O4SPureza:97.97% - 98.97%Forma y color:SolidPeso molecular:574.63Ixazomib citrate
CAS:Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).Fórmula:C20H23BCl2N2O9Pureza:98.37% - >99.99%Forma y color:SolidPeso molecular:517.12MMP-9-IN-1
CAS:MMP-9-IN-1 is an inhibitor of specific matrix metalloproteinase-9 (MMP-9).Fórmula:C16H17F2N3O3SPureza:99.21% - 99.86%Forma y color:SolidPeso molecular:369.39Ref: TM-T8310
2mg74,00€5mg111,00€10mg170,00€25mg344,00€50mg525,00€100mg747,00€200mg1.017,00€1mL*10mM (DMSO)124,00€Tegobuvir
CAS:Tegobuvir (GS 333126) is a specific and covalent HCV NS5B polymerase inhibitor.Fórmula:C25H14F7N5Pureza:99.21%Forma y color:SolidPeso molecular:517.4Ref: TM-T17029
1mg88,00€5mg187,00€10mg311,00€25mg532,00€50mg750,00€100mg1.035,00€1mL*10mM (DMSO)213,00€Ac-DEVD-AMC
CAS:<p>Ac-DEVD-AMC (AC-ASP-MET-GLN-ASP-7-AMINO-4-METHYLCOUMARIN) is the substrate of Caspase-3 .</p>Fórmula:C30H37N5O13Pureza:98.20%Forma y color:White PowderPeso molecular:675.64Marimastat
CAS:<p>Marimastat (BB2516) (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C15H29N3O5Pureza:97.46% - 98.11%Forma y color:SolidPeso molecular:331.414-Butylresorcinol
CAS:4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.Fórmula:C10H14O2Pureza:99.48% - ≥95%Forma y color:Light Beige Solid PowderPeso molecular:166.22BMS-707035
CAS:BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.Fórmula:C17H19FN4O5SPureza:99.78%Forma y color:SolidPeso molecular:410.42Bortezomib-pinanediol
CAS:Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.Fórmula:C29H39BN4O4Pureza:97.5%Forma y color:Yellow SolidPeso molecular:518.46LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Fórmula:C25H29FN4O5Pureza:97.83% - 99.54%Forma y color:SolidPeso molecular:484.52Ref: TM-TQ0116
1mg96,00€2mg137,00€5mg210,00€10mg278,00€25mg487,00€50mg708,00€100mg998,00€1mL*10mM (DMSO)220,00€
