Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(20 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(506 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(95 productos)
- Serina proteasa(55 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 1093 productos de "Proteasas / Proteasoma"
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Bemnifosbuvir hemisulfate
CAS:Bemnifosbuvir hemisulfate (AT-527) is a potent inhibitor of HCV virus replication.Fórmula:C48H68F2N14O18P2SPureza:99.98%Forma y color:SolidPeso molecular:1261.15Batimastat
CAS:Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.Fórmula:C23H31N3O4S2Pureza:98.15% - 99.5%Forma y color:SolidPeso molecular:477.64Lusutrombopag
CAS:Lusutrombopag (Mulpleta) is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients withFórmula:C29H32Cl2N2O5SPureza:99.96%Forma y color:SolidPeso molecular:591.55Ref: TM-TQ0223
1mg64,00€2mg92,00€5mg137,00€10mg208,00€25mg416,00€50mg628,00€100mg938,00€200mg1.293,00€1mL*10mM (DMSO)170,00€LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Fórmula:C25H29FN4O5Pureza:97.83% - 99.54%Forma y color:SolidPeso molecular:484.52Ref: TM-TQ0116
1mg96,00€2mg137,00€5mg210,00€10mg278,00€25mg487,00€50mg708,00€100mg998,00€1mL*10mM (DMSO)220,00€(S,S)-TAPI-1
CAS:"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."Fórmula:C26H37N5O5Forma y color:SolidPeso molecular:499.6Bemnifosbuvir
CAS:Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.Fórmula:C24H33FN7O7PPureza:99.35% - 99.54%Forma y color:SolidPeso molecular:581.53STK16-IN-1
CAS:STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).Fórmula:C17H12FN3OPureza:99.52%Forma y color:SolidPeso molecular:293.3Ilomastat
CAS:<p>Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C20H28N4O4Pureza:97.04% - 99.51%Forma y color:SolidPeso molecular:388.46CA-074 methyl ester
CAS:CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!Fórmula:C19H31N3O6Pureza:97.26% - 99.58%Forma y color:SolidPeso molecular:397.47Voxilaprevir
CAS:Voxilaprevir is an inhibitor of hepatitis C virus (HCV) nonstructural (NS) protein 3/4A protease.Fórmula:C40H52F4N6O9SPureza:99.83% - 99.98%Forma y color:SolidPeso molecular:868.93Ref: TM-T19862
1mg80,00€5mg311,00€10mg445,00€25mg747,00€50mg1.008,00€100mg1.359,00€200mg1.833,00€1mL*10mM (DMSO)415,00€Etravirine
CAS:Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.Fórmula:C20H15BrN6OPureza:97.61% - 99.74%Forma y color:White To Off-White SolidPeso molecular:435.28Ref: TM-T2551
2mg35,00€5mg52,00€10mg80,00€25mg149,00€50mg216,00€100mg329,00€200mg485,00€1mL*10mM (DMSO)52,00€HZ-1157
CAS:HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.Fórmula:C12H16N4OPureza:98.23%Forma y color:SolidPeso molecular:232.284-Phenoxybenzylamine
CAS:4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against HCV NS3/4a .Fórmula:C13H13NOPureza:97.26%Forma y color:SolidPeso molecular:199.25(Arg)9 TFA (143413-47-2 free base)
CAS:(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.Fórmula:C56H111F3N36O12Pureza:>99.99%Forma y color:SolidPeso molecular:1537.71Letermovir
CAS:Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.Fórmula:C29H28F4N4O4Pureza:99.85% - 99.87%Forma y color:SolidPeso molecular:572.55Ref: TM-T5396
1mg88,00€5mg170,00€10mg283,00€25mg497,00€50mg707,00€100mg1.008,00€200mg1.359,00€1mL*10mM (DMSO)216,00€Vesnarinone
CAS:Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFórmula:C22H25N3O4Pureza:96.69% - 98.13%Forma y color:SolidPeso molecular:395.45Ref: TM-T3465
2mg35,00€5mg52,00€10mg80,00€25mg117,00€100mg313,00€200mg452,00€1mL*5mM (DMSO)49,00€50mg*5mM (DMSO)210,00€Boceprevir
CAS:Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.Fórmula:C27H45N5O5Pureza:95% - 99.16%Forma y color:SolidPeso molecular:519.68Ref: TM-T4988
1mg35,00€5mg70,00€10mg96,00€25mg144,00€50mg187,00€100mg274,00€200mg378,00€1mL*10mM (DMSO)80,00€Daclatasvir
CAS:Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.Fórmula:C40H50N8O6Pureza:99.81% - 99.99%Forma y color:SolidPeso molecular:738.88ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Fórmula:C22H19N3O2SPureza:99.12% - 99.87%Forma y color:SolidPeso molecular:389.47Ref: TM-T3423
1mg35,00€5mg80,00€10mg97,00€25mg188,00€50mg311,00€100mg500,00€500mg1.093,00€1mL*10mM (DMSO)88,00€Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Fórmula:C27H37N3O7SPureza:99.67% - 99.76%Forma y color:White Amorphous SolidPeso molecular:547.66
