Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(23 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(495 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(88 productos)
- Serina proteasa(51 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 993 productos de "Proteasas / Proteasoma"
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Lenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Fórmula:C39H32ClF10N7O5S2Pureza:99.61% - 99.87%Forma y color:SolidPeso molecular:968.28Ref: TM-T11465
1mg187,00€5mg376,00€10mg565,00€25mg998,00€50mg1.388,00€100mg1.882,00€200mg2.622,00€1mL*10mM (DMSO)615,00€BDCRB
BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.Fórmula:C12H11BrCl2N2O4Pureza:99.41% - 99.85%Forma y color:SoildPeso molecular:398.04BILB-1941
CAS:BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.Fórmula:C34H34N4O4Pureza:99.51% - 99.65%Forma y color:SolidPeso molecular:562.66Ref: TM-T26815
1mg296,00€5mg718,00€10mg982,00€25mg1.485,00€50mg2.008,00€100mg2.637,00€1mL*10mM (DMSO)1.044,00€DB04760
CAS:DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.Fórmula:C22H20F2N4O2Pureza:99.93% - 99.99%Forma y color:SolidPeso molecular:410.42Ref: TM-T15055
1mg84,00€5mg205,00€10mg309,00€25mg522,00€50mg747,00€100mg1.035,00€500mg2.052,00€1mL*10mM (DMSO)178,00€JNJ-10311795
CAS:JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.Fórmula:C40H35N2O6PPureza:97.43%Forma y color:SolidPeso molecular:670.69Setrobuvir
CAS:Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension withFórmula:C25H25FN4O6S2Pureza:99.95% - 99.97%Forma y color:SolidPeso molecular:560.62Ref: TM-T28762
1mg229,00€5mg570,00€10mg812,00€25mg1.216,00€50mg1.663,00€100mg2.242,00€500mg4.494,00€1mL*10mM (DMSO)737,00€Sovaprevir
CAS:Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Fórmula:C43H53N5O8SPureza:99.89%Forma y color:SolidPeso molecular:799.97Ref: TM-T28830
1mg253,00€5mg620,00€10mg884,00€25mg1.314,00€50mg1.773,00€100mg2.385,00€1mL*10mM (DMSO)982,00€Melagatran
CAS:Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.Fórmula:C22H31N5O4Pureza:98.29% - >99.99%Forma y color:SolidPeso molecular:429.51Ref: TM-T11994
1mg487,00€5mg1.134,00€10mg1.468,00€25mg2.215,00€50mg2.962,00€100mg4.024,00€1mL*10mM (DMSO)1.071,00€Opaviraline
CAS:Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.Fórmula:C14H17FN2O3Pureza:99.94%Forma y color:SolidPeso molecular:280.29Ref: TM-T28255
1mg378,00€5mg922,00€10mg1.225,00€25mg1.853,00€50mg2.490,00€100mg3.353,00€1mL*10mM (DMSO)823,00€MMP2-IN-3
CAS:MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Fórmula:C23H21N3OPureza:99.38%Forma y color:SolidPeso molecular:355.43Ref: TM-T61271
1mg64,00€5mg132,00€10mg195,00€25mg315,00€50mg439,00€100mg590,00€200mg793,00€1mL*10mM (DMSO)140,00€Sirpiglenastat
CAS:Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Fórmula:C22H27N5O5Pureza:98.01% - 98.37%Forma y color:SolidPeso molecular:441.48Isatoribine
CAS:Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.Fórmula:C10H12N4O6SPureza:98.99% - 99.75%Forma y color:SolidPeso molecular:316.29AGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Fórmula:C18H17F2N3O2Pureza:98.92%Forma y color:SolidPeso molecular:345.34Ref: TM-T69685
1mg74,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€1mL*10mM (DMSO)154,00€HIV-1 integrase inhibitor 8
CAS:HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].
Fórmula:C21H24O2Pureza:98.91%Forma y color:SolidPeso molecular:308.41MMP-2/MMP-9 Inhibitor I
CAS:MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.Fórmula:C21H19NO4SPureza:99.98%Forma y color:SolidPeso molecular:381.44Ref: TM-T21512
1mg56,00€5mg119,00€10mg177,00€25mg356,00€50mg590,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)133,00€MK-8325
CAS:MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailabilityFórmula:C43H54Cl2F2N8O6SiPureza:99.61%Forma y color:SolidPeso molecular:915.93BAY-43-9695
CAS:BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.Fórmula:C22H25N3O4SPureza:99.50% - 99.98%Forma y color:SolidPeso molecular:427.52BMS-929075
CAS:BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokineticFórmula:C31H24F2N4O3Pureza:99.81% - 99.94%Forma y color:SolidPeso molecular:538.54Ref: TM-T26863
1mg172,00€5mg432,00€10mg618,00€25mg973,00€50mg1.333,00€100mg1.791,00€500mg3.529,00€1mL*10mM (DMSO)538,00€(2RS)-FPMPA
CAS:(2RS)-FPMPA（FPMPA） has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).Fórmula:C9H13FN5O4PPureza:99.9% - >99.99%Forma y color:SolidPeso molecular:305.2P32/98 hemifumarate
CAS:P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.Fórmula:C22H40N4O6S2Pureza:99.46%Forma y color:SolidPeso molecular:520.71
