Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(23 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(495 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(88 productos)
- Serina proteasa(51 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 993 productos de "Proteasas / Proteasoma"
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Thrombin Inhibitor 2
CAS:Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.Fórmula:C19H16ClF3N6O2Pureza:98%Forma y color:SolidPeso molecular:452.82Flovagatran
CAS:Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.Fórmula:C27H36BN3O7Pureza:99.56%Forma y color:SolidPeso molecular:525.4Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Fórmula:C32H30F3N5O7S2Pureza:98%Forma y color:SolidPeso molecular:717.73MDK0734
CAS:MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.Fórmula:C15H17N3O2Pureza:98%Forma y color:SolidPeso molecular:271.31DPP-4-IN-2
CAS:DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.Fórmula:C18H18N6OForma y color:SolidPeso molecular:334.38Tyrosinase-IN-8
Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity whileFórmula:C16H12O4Forma y color:SolidPeso molecular:268.26Atevirdine
CAS:Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).
Fórmula:C21H25N5O2Pureza:98.20%Forma y color:SolidPeso molecular:379.46Tyrosinase-IN-2
CAS:Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Fórmula:C8H8N4O2SPureza:99.78%Forma y color:SolidPeso molecular:224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€PG-116800
CAS:PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Fórmula:C24H27N3O7SPureza:98.03% - 99.66%Forma y color:SolidPeso molecular:501.55TG-2-IN-1
CAS:TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].Fórmula:C8H13ClN2OSPureza:98.43%Forma y color:SolidPeso molecular:220.72Cathepsin X-IN-1
CAS:Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].
Fórmula:C15H13N3O3SPureza:99.34%Forma y color:SolidPeso molecular:315.35CPA inhibitor
CAS:CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.Fórmula:C18H19NO4Pureza:99.94%Forma y color:SolidPeso molecular:313.35Ref: TM-T10876
1mg57,00€5mg125,00€10mg163,00€25mg278,00€50mg405,00€100mgA consultar1mL*10mM (DMSO)138,00€TG2-IN-3h
CAS:TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFórmula:C21H26N4O4SPureza:99.34% - 99.76%Forma y color:SolidPeso molecular:430.522'-C-Methyladenosine
CAS:2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.Fórmula:C11H15N5O4Pureza:99.85%Forma y color:SolidPeso molecular:281.2720S Proteasome activator 1
CAS:20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Fórmula:C27H19ClF2N2OSPureza:99.82%Forma y color:SolidPeso molecular:492.97Gemigliptin
CAS:Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)Fórmula:C18H19F8N5O2Pureza:99.72%Forma y color:SolidPeso molecular:489.36Ref: TM-T7369
2mg38,00€5mg57,00€10mg93,00€25mg148,00€50mg245,00€100mg385,00€500mg873,00€1mL*10mM (DMSO)84,00€TY-51469
CAS:TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).Fórmula:C20H15FN2O6S4Pureza:99.65%Forma y color:SolidPeso molecular:526.6VRK-IN-1
CAS:VRK-IN-1 is a potent and selective inhibitor of cowpox-associated kinase 1 (VRK1), which can be used in the study of neurological disorders.Fórmula:C18H11F4NO2Pureza:99.18% - 99.25%Forma y color:SolidPeso molecular:349.28Ref: TM-T35863
1mg103,00€5mg236,00€10mg379,00€25mg750,00€50mg1.130,00€100mg1.510,00€200mg2.062,00€1mL*10mM (DMSO)259,00€UK-396082
CAS:UK-396082 is a TAFI inhibitor that inhibits Carboxypeptidase B and can be used in the study of thrombosis, atherosclerosis, cancer and fibrotic conditions.Fórmula:C12H21N3O2Pureza:99.89%Forma y color:SolidPeso molecular:239.31UPGL00004
CAS:UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Fórmula:C25H26N8O2S2Pureza:97.93%Forma y color:SolidPeso molecular:534.66
