Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(24 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(495 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(87 productos)
- Serina proteasa(51 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 992 productos de "Proteasas / Proteasoma"
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SQ 32056
CAS:SQ 32056 is a cathepsin E inhibitor.Fórmula:C37H56N4O5Pureza:98%Forma y color:SolidPeso molecular:636.86BMS-189664 HCl
CAS:BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Fórmula:C22H35ClN6O4SPureza:98%Forma y color:SolidPeso molecular:515.07LONP1-IN-2
CAS:LONP1-IN-2: Potent LONP1 inhibitor, IC50=0.187μM; weak on 20S proteasome (>10μM); for cancer research.Fórmula:C16H27BN4O4Forma y color:SolidPeso molecular:350.22Z-LVG
CAS:Z-LVG, an irreversible cysteine protease inhibitor and a tripeptide derivative of cystatin C, serves as an inhibitor of viral replication and is utilized inFórmula:C21H31N3O6Forma y color:SolidPeso molecular:421.49MMP-9 Inhibitor I
CAS:MMP-9 inhibitor I is an inhibitor of matrix metalloproteinase-9 (MMP-9) that is selective over MMP-1 and MMP-13 (IC50s = 5, 1,050, and 113 nM, respectively).Fórmula:C27H33N3O5SForma y color:SolidPeso molecular:511.63HCV-IN-44
CAS:HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].Fórmula:C24H26FN3O5SForma y color:SolidPeso molecular:487.54(1R,4S)-Yimitasvir diphosphate
CAS:Yimitasvir diphosphate, also known as Emitasvir, is an orally-administered inhibitor of the hepatitis C virus (HCV) nonstructural protein 5A (NS5A).Fórmula:C49H64N8O14P2Forma y color:SolidPeso molecular:1051.03MeOSuc-AAPV-CMK
CAS:MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediatedFórmula:C22H35ClN4O7Forma y color:SolidPeso molecular:502.99Ecallantide
CAS:Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.Fórmula:C305H448N88O91S8Forma y color:SolidPeso molecular:7059.88ABP 25
CAS:ABP 25 is a highly potent and selective activity-based probe (ABP) for cathepsin K imaging.Fórmula:C55H66ClN5O3Forma y color:SolidPeso molecular:880.6Ravidasvir HCl
CAS:Ravidasvir, also known as PPI-668 and ASC16, is a second-generation, orally active, potent and selective HCV NS5A protein inhibitor.Fórmula:C42H52Cl2N8O6Forma y color:SolidPeso molecular:835.828Cathepsin Inhibitor 2
CAS:Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).Fórmula:C19H21F6N3OPureza:98%Forma y color:SolidPeso molecular:421.38JW 480
CAS:JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.Fórmula:C22H23NO2Pureza:99.72%Forma y color:SolidPeso molecular:333.42Ref: TM-T22883
2mg35,00€5mg49,00€10mg79,00€25mg160,00€50mg259,00€100mg416,00€200mg587,00€1mL*10mM (DMSO)57,00€Z-DEVD-CMK
CAS:Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].Fórmula:C27H35ClN4O12Forma y color:SolidPeso molecular:643.04AA74-1
CAS:AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].Fórmula:C16H28N4O2Pureza:98%Forma y color:SolidPeso molecular:308.42DCLK1-IN-2
CAS:DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cellFórmula:C26H32N8O3SForma y color:SolidPeso molecular:536.65Atecegatran metoxil
CAS:Atecegatran Metoxil (AZD0837), an oral thrombin inhibitor in development for stroke prevention in atrial fibrillation, is well-tolerated with favorable PK.Fórmula:C22H23ClF2N4O5Forma y color:SolidPeso molecular:496.89Cyclotheonellazole A
CAS:Cyclotheonellazole A inhibits elastase (IC50=0.034nM) & chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.Fórmula:C44H54N9NaO14S2Forma y color:SolidPeso molecular:1020.07Tyropeptin A-4
CAS:Tyropeptin A-4 is used as a proteasome inhibitor.Fórmula:C31H41N3O6Pureza:98%Forma y color:SolidPeso molecular:551.67Inogatran
CAS:Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.Fórmula:C21H38N6O4Pureza:98%Forma y color:SolidPeso molecular:438.56
