
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.787 productos)
- Ciclo celular / Checkpoint(4.446 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.824 productos)
- Endocrinología / Hormonas(3.500 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.317 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.200 productos)
- Transportador de membrana / canal de iones(2.787 productos)
- Metabolismo(9.416 productos)
- Microbiología / Virología(6.968 productos)
- Neurociencia(9.919 productos)
- Otros inhibidores(37.928 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.649 productos)
Mostrar 16 subcategorías más
Se han encontrado 66626 productos de "Inhibidores"
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Ponesimod
CAS:<p>Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.</p>Fórmula:C23H25ClN2O4SPureza:99.42% - 99.96%Forma y color:SolidPeso molecular:460.97β-Ionone
CAS:<p>β-Ionone (β-lonone) is an end-ring analog of β-carotenoids which widely distributed in fruit and vegetables,with anti-proliferative, anti-metastatic</p>Fórmula:C13H20OPureza:98.52%Forma y color:Colourless Liquid OilyPeso molecular:192.33-methyl-1,2-dihydroquinolin-2-one
CAS:<p>3-methyl-1,2-dihydroquinolin-2-one is the first known micromolar inhibitors of the ATAD2 bromodomain.</p>Fórmula:C10H9NOPureza:99.62%Forma y color:SolidPeso molecular:159.18DHQ
CAS:<p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>Fórmula:C8H6N2O2Pureza:99.89%Forma y color:SolidPeso molecular:162.15Oxyphenisatin acetate
CAS:<p>Oxyphenisatin acetate inhibits the growth of the breast cancer cell lines MCF7, T47D, HS578T, and MDA-MB-468.</p>Fórmula:C24H19NO5Pureza:98% - 99.35%Forma y color:SolidPeso molecular:401.41Bosentan
CAS:<p>Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.</p>Fórmula:C27H29N5O6SPureza:99.74% - 99.84%Forma y color:Pale Yellow To Off-White SolidPeso molecular:551.614Hexapeptide-10 Acetate
<p>Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) is a synthetic peptide.</p>Fórmula:C30H57N7O10Pureza:98.84%Forma y color:SolidPeso molecular:675.81FEMA 4774
CAS:<p>FEMA 4774 (S9632) is a positive allosteric modulator of T1R2/T1R3. FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests</p>Fórmula:C19H25N3O4Pureza:99.97%Forma y color:SolidPeso molecular:359.424-Hydroxyisoleucine
CAS:<p>4-Hydroxyisoleucine (4-Hydroxy-L-isoleucine) has antidepressant-like, antidyslipidemic, and antihyperglycemic effects. It displays an insulinotropic activity.</p>Fórmula:C6H13NO3Pureza:99.83%Forma y color:SolidPeso molecular:147.17TBMP
CAS:<p>TBMP (butylated hydroxyanisole) is the viral envelope protein hemagglutinin (HA)-mediated entry novel inhibitor.</p>Fórmula:C11H16O2Pureza:99.42%Forma y color:SolidPeso molecular:180.24Epithalon TFA (307297-39-8 free base)
<p>Epithalon TFA (307297-39-8 free base) (Epithalon TFA) is an anti-aging agent and telomerase activator.</p>Fórmula:C16H23F3N4O11Pureza:≥95%Forma y color:SolidPeso molecular:504.37SCH54292
CAS:<p>SCH-54292 is a GDP exchange inhibitor.</p>Fórmula:C24H28N2O9SPureza:95.65%Forma y color:SolidPeso molecular:520.55D-(+)-Xylose
CAS:<p>D-(+)-Xylose (Wood sugar) is an aldopentose. Xylose is also found in mucopolysaccharides of connective tissue and sometimes in the urine.</p>Fórmula:C5H10O5Pureza:99.85%Forma y color:White Solid Crystalline PowderPeso molecular:150.13Fmoc-Asp-NH2
CAS:<p>Fmoc-Asp-NH2 is a cleavable ADC linker. Fmoc-Asp-NH2 can be used in the synthesis of antibody-drug conjugates (ADCs).</p>Fórmula:C19H18N2O5Pureza:98.41%Forma y color:SolidPeso molecular:354.36Fedratinib
CAS:Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.Fórmula:C27H36N6O3SPureza:97.31% - 99.96%Forma y color:SolidPeso molecular:524.68Raphin1
CAS:<p>Raphin1 is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B).</p>Fórmula:C8H8Cl2N4Pureza:99.39%Forma y color:SolidPeso molecular:231.08Kv2-IN-A1
CAS:<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Fórmula:C20H17ClN4OSPureza:98.83%Forma y color:SolidPeso molecular:396.89Anti-Inflammatory Peptide 1 Acetate
<p>Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.</p>Fórmula:C47H86N12O16S2Pureza:98.95%Forma y color:SolidPeso molecular:1139.39Menthone
CAS:<p>Menthone has anti-inflammary activity,, it can suppress the lipopolysaccharide (LPS)-induced proinflammatory cytokines, interleukin-1beta (IL-1beta) and tumor</p>Fórmula:C10H18OPureza:97.02% - ≥95%Forma y color:Colorless Oily Mobile Liq LiquidPeso molecular:154.25Berbamine dihydrochloride
CAS:<p>Berbamine dihydrochloride (Berbamine), a natural compound derived from the Berberis amurensis plant, has been shown to exhibit antitumor activity in several Ys.</p>Fórmula:C37H42Cl2N2O6Pureza:95% - 99.99%Forma y color:SolidPeso molecular:681.65Ginsenoside Rf
CAS:<p>Ginsenoside Rf (Panaxoside Rf) is a trace component of ginseng root. Ginsenoside Rf inhibits N-type Ca2+ channel.</p>Fórmula:C42H72O14Pureza:99.82%Forma y color:SolidPeso molecular:801.01GluR6 antagonist-1
CAS:<p>GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.</p>Fórmula:C15H11ClN2OSPureza:99.89%Forma y color:SolidPeso molecular:302.78CNX-2006
CAS:<p>CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM, with very weak inhibition at wild-type EGFR.</p>Fórmula:C26H27F4N7O2Pureza:98.85% - 99.16%Forma y color:SolidPeso molecular:545.53(±)-Ibipinabant
CAS:<p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>Fórmula:C23H20Cl2N4O2SPureza:99.28% - 99.83%Forma y color:SolidPeso molecular:487.4Molibresib besylate
CAS:<p>Molibresib besylate (GSK 525762C) is a BET protein family inhibitor used in the study of refractory hematologic malignant diseases.</p>Fórmula:C28H28ClN5O5SPureza:99.64% - 99.64%Forma y color:SolidPeso molecular:582.07AZ9482
CAS:<p>AZ9482, a potent PARP inhibitor with 2-piperazinyl-3-cyano-pyridine linkage, causes centrosome declustering in HeLa cells with an EC50 < 18 nM.</p>Fórmula:C26H22N6O2Pureza:99.18% - 99.86%Forma y color:SolidPeso molecular:450.49Suberic acid
CAS:<p>Suberic acid in urine indicates fatty acid oxidation issues, often linked to MCAD or carnitine deficiencies.</p>Fórmula:C8H14O4Pureza:99.80%Forma y color:White CrystalsPeso molecular:174.19BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Forma y color:SolidPeso molecular:479.872-Amino-3-hydroxypyridine
CAS:<p>2-Amino-3-hydroxypyridine as a chromogenic reagent for the spectrophotometric determination of osmium.</p>Fórmula:C5H6N2OPureza:99.98%Forma y color:Light Beige Solid PowderPeso molecular:110.11BIX02189
CAS:<p>BIX02189 is a potent and selective inhibitor of MEK5 and ERK5(IC50 : 1.5 nM and 59 nM).</p>Fórmula:C27H28N4O2Pureza:97.84%Forma y color:SolidPeso molecular:440.54Co 101244 hydrochloride
CAS:<p>Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.</p>Fórmula:C21H28ClNO3Pureza:99.76%Forma y color:SolidPeso molecular:377.9Tomatine
CAS:<p>Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.</p>Fórmula:C50H83NO21Pureza:98.42% - 99.94%Forma y color:White To Light YellowPeso molecular:1034.19(+)-Peusedanol
CAS:<p>(+)-Peusedanol is a natural product isolated from Peucedanumjaponicum.</p>Fórmula:C14H16O5Pureza:99.37%Forma y color:SolidPeso molecular:264.27Licorice-saponin H2
CAS:<p>Licorice-saponin H2 (Licoricesaponin H2) is a natural product</p>Fórmula:C42H62O16Pureza:99.58% - 99.76%Forma y color:SolidPeso molecular:822.93Ethoxyacetic acid
CAS:<p>Ethoxyacetic acid is an endogenous metabolite of ethylene glycol monoethyl ether acetate.</p>Fórmula:C4H8O3Pureza:≥98%Forma y color:Physical Description Liquid (Ntp 1992)Peso molecular:104.1Fumaric acid
CAS:<p>Fumaric acid reduces eotaxin-1 in TNF-α-activated fibroblasts via p38 MAPK/NF-κB. It's an oncometabolite found in high levels in tumors.</p>Fórmula:C4H4O4Pureza:98.77% - 98.80%Forma y color:Colorless Needles Monoclinic Prisms Or Leaflets From Water Solid CrystallinePeso molecular:116.07Hemiphloin
CAS:<p>Hemiphloin: natural flavonoid with anti-inflammatory properties, potential skin disease therapy.</p>Fórmula:C21H22O10Pureza:99.26%Forma y color:SolidPeso molecular:434.39Crizotinib
CAS:<p>Crizotinib (PF-02341066) is an ATP-competitive small-molecule tyrosine kinases inhibitor of c-MET (IC50: 8 nM) and ALK (IC50: 20 nM) receptor.</p>Fórmula:C21H22Cl2FN5OPureza:99% - 99.87%Forma y color:SolidPeso molecular:450.34TTA-A2
CAS:<p>TTA-A2: T-type calcium channel blocker; anticonvulsant targeting Cav3.1, Cav3.2; IC50 of 89/92 nM; potential for treating neurological conditions.</p>Fórmula:C20H21F3N2O2Pureza:99.5% - 99.9%Forma y color:SolidPeso molecular:378.39MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Forma y color:SolidPeso molecular:470.513-Methoxyphenylethylamine
CAS:<p>3-Methoxyphenylethylamine 是一种生物活性化学品。</p>Fórmula:C9H13NOPureza:97.07%Forma y color:Less Liquid Colorless LiquidPeso molecular:151.21RP-54745
CAS:<p>RP-54745, a potential antirheumatic compound. Inhibitor of macrophage stimulation and interleukin-1 production.</p>Fórmula:C13H12ClNOS2Pureza:99.06%Forma y color:SolidPeso molecular:297.82Cichoric Acid
CAS:<p>Cichoric Acid (Dicaffeoyltartaric acid) is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues.</p>Fórmula:C22H18O12Pureza:97.87% - 98.77%Forma y color:SolidPeso molecular:474.37Dihydroxyacetone phosphate hemimagnesium hydrate
<p>Dihydroxyacetone phosphate hemimagnesium salt hydrate is a glycerone phosphate metabolite and a primary alpha-hydroxy ketone.</p>Fórmula:C3H7O6PMg·xH2OPureza:99.97%Forma y color:SolidPeso molecular:362.4BI-187004
CAS:<p>BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.</p>Fórmula:C21H18N4OPureza:98.63%Forma y color:SolidPeso molecular:342.39N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide
CAS:<p>N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide inhibits RecBCD and AddAB enzyme families.</p>Fórmula:C14H12N4OSPureza:99.8%Forma y color:SolidPeso molecular:284.34Atractylenolide II
CAS:<p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>Fórmula:C15H20O2Pureza:99.89% - 99.93%Forma y color:SolidPeso molecular:232.32SU9516
CAS:<p>SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also has inhibitory effects on CDK1 and CDK4, with IC50s of 40 nM and 200 nM, respectively.</p>Fórmula:C13H11N3O2Pureza:99.34% - 99.87%Forma y color:SolidPeso molecular:241.25Methylsticin
CAS:<p>Methysticin, a kavalactone from kava roots, inhibits osteoclasts, NF-χB, stimulates Nrf2, reduces Na+ channel peaks, and hinders fungal growth.</p>Fórmula:C15H14O5Pureza:99.27% - 99.37%Forma y color:White PowderPeso molecular:274.27Ladostigil hydrochloride
CAS:<p>Ladostigil hydrochloride: oral dual cholinesterase and MAO-B/AChE inhibitor; IC50s: 37.1 & 31.8 μM; potential for depression and Alzheimer's research.</p>Fórmula:C16H21ClN2O2Forma y color:SolidPeso molecular:308.8Hosenkoside C
CAS:<p>Hosenkoside C is a baccharane glycoside found in the seeds of Impatiens balsamina.</p>Fórmula:C48H82O20Pureza:99.49% - 99.54%Forma y color:SolidPeso molecular:979.15Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Fórmula:C34H60N14O12SPureza:96.79% - 99.65%Forma y color:White PowderPeso molecular:888.99Azumolene
CAS:<p>Azumolene (EU4093 free base)</p>Fórmula:C13H9BrN4O3Pureza:98.1% - 98.35%Forma y color:SolidPeso molecular:349.14CNQX disodium
CAS:<p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>Fórmula:C9H2N4Na2O4Pureza:97.77%Forma y color:SolidPeso molecular:276.12Theaflavin 3,3′-digallate
CAS:<p>Theaflavin 3,3'-digallate, a major polyphenol found in black tea, is an inducer of oxidative stress which has anti-inflammatory and cancer</p>Fórmula:C43H32O20Pureza:98.71% - 99.86%Forma y color:SolidPeso molecular:868.7Magnesium glycinate
CAS:<p>Magnesium glycinate supplement enhances body's magnesium for muscle, nerve function, and bone health.</p>Fórmula:C4H8MgN2O4Pureza:≥95%Forma y color:CoaPeso molecular:172.42Praeruptorin C
CAS:<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Fórmula:C24H28O7Pureza:99.6% - 99.92%Forma y color:SolidPeso molecular:428.47CS-0047390
CAS:<p>CS-0047390 ((S)-Di-tert-butyl 2-(3-((S)-6-amino-1-(tert-butoxy)-1-oxohexan-2-yl)ureido)pentanedioate), also known as tert-Butyl-DCL, is a PSMA inhibitor and a</p>Fórmula:C24H45N3O7Pureza:≥98%Forma y color:SolidPeso molecular:487.63Aloeresin D
CAS:<p>Aloeresin D, a natural chromone glycoside, inhibits β-Secretase (BACE1) activity (IC50: 39 μM).</p>Fórmula:C29H32O11Pureza:98.11% - 99.57%Forma y color:SolidPeso molecular:556.56Tyrosyltyrosine acetate
<p>Tyrosyltyrosine acetate is a peptide.</p>Fórmula:C20H24N2O7Pureza:99.88%Forma y color:SolidPeso molecular:404.414-Pyridoxic Acid
CAS:<p>4-Pyridoxic Acid (4-Pyridoxinsaeure), a water-soluble catabolite of vitamin B6, secreted from the urine.</p>Fórmula:C8H9NO4Pureza:99.42% - 99.82%Forma y color:SolidPeso molecular:183.16DS-1971a
CAS:<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Fórmula:C20H21ClFN5O3SPureza:99.66%Forma y color:SolidPeso molecular:465.934,5-Dicaffeoylquinic acid
CAS:<p>1.</p>Fórmula:C25H24O12Pureza:98.86% - ≥95%Forma y color:SolidPeso molecular:516.45Visomitin
CAS:<p>Visomitin (SKQ1) is a mitochondria-targeted antioxidant that decreases transmembrane potential and production of reactive oxygen species (ROS).</p>Fórmula:C36H42BrO2PPureza:95.44% - 99.54%Forma y color:Highly Hydroscopic Solid)Peso molecular:617.61Hyperoside
CAS:<p>Hyperoside (Hyperin) is a naturally occuring flavonoid compound which shows multiple bioactivities, including myocardial protection, anti-redox, and anti-</p>Fórmula:C21H20O12Pureza:98% - 99.82%Forma y color:SolidPeso molecular:464.38Simeprevir sodium
CAS:<p>Simeprevir is a drug for the treatment and cure of hepatitis C.</p>Fórmula:C38H46N5NaO7S2Pureza:98%Forma y color:SolidPeso molecular:771.92Deacetylasperulosidic Acid
CAS:<p>Deacetylasperulosidic Acid is a natural compound of Morinda citrifolia fruit. It has antioxidant activity by increasing superoxide dismutase activity.</p>Fórmula:C16H22O11Pureza:99.37%Forma y color:SolidPeso molecular:390.346-FAM
CAS:<p>6-Carboxyfluorescein (6-FAM) contains a carboxylic acid functional group, facilitating reactions with primary amines through carbodiimide activation.</p>Fórmula:C21H12O7Pureza:97.23% - 98.73%Forma y color:Orange SolidPeso molecular:376.32Spirostan-3-ol
CAS:<p>Spirostan-3-ol, a saponin isolate with potential anti-cancer properties, is a Sarsasapogenin stereoisomer.</p>Fórmula:C27H44O3Pureza:99.92%Forma y color:White Or Off-Withe PowderPeso molecular:416.64D-Luciferin potassium
CAS:<p>D-Luciferin potassium (D-Luciferin K Salt) is a popular bioluminescent substrate of luciferase in the presence of ATP.</p>Fórmula:C11H7KN2O3S2Pureza:98.00% - >99.99%Forma y color:SolidPeso molecular:318.415-Bromoindole
CAS:<p>5-bromoindole is a potential inhibitor of glycogen synthase kinase 3 (GSK-3)and an important pharmaceutical chemical intermediate</p>Fórmula:C8H6BrNPureza:99.99%Forma y color:White To Beige Crystalline PowderPeso molecular:196.043-Hydroxyanthranilic acid
CAS:<p>3-Hydroxyanthranilic acid (3-HYDROXY-2-AMINOBENZOIC ACID), also known as 2-amino-3-hydroxy-benzoate or 3-ohaa, belongs to the class of organic compounds known</p>Fórmula:C7H7NO3Pureza:98.69% - 99.45%Forma y color:Leaflets In Water SolidPeso molecular:153.142-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid
CAS:<p>2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0^2,7^.0^9,14^.0^15,19^]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid - a synthesis precursor.</p>Fórmula:C25H16ClNO4Pureza:99.6% - 99.87%Forma y color:SolidPeso molecular:429.85LY2334737
CAS:<p>LY2334737 is an orally available prodrug of gemcitabine with antineoplastic activity.</p>Fórmula:C17H25F2N3O5Pureza:98.82%Forma y color:SolidPeso molecular:389.39GSK467
CAS:<p>GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).</p>Fórmula:C17H13N5O2Pureza:99.55%Forma y color:SolidPeso molecular:319.32Maropitant
CAS:<p>Maropitant is a selective neurokinin (NK1) receptor antagonist.</p>Fórmula:C32H40N2OPureza:97.35% - 99.75%Forma y color:SolidPeso molecular:468.67Cisapride tartrate
CAS:<p>Cisapride tartrate is chemically related to metoclopramide, but unlike metoclopramide, it does not cross the blood-brain barrier or have antidopaminergic</p>Fórmula:C27H35ClFN3O10Forma y color:SolidPeso molecular:616.04JNJ-42153605
CAS:<p>JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).</p>Fórmula:C22H23F3N4Pureza:97.25% - 98.57%Forma y color:SolidPeso molecular:400.44Fumagillin
CAS:<p>Fumagillin (Amebacilin) is a selective and potent irreversible inhibitor of Methionine aminopeptidase 2 (MetAP2), used as an antibiotic to treat</p>Fórmula:C26H34O7Pureza:95% - ≥98%Forma y color:Light Yellow SolidPeso molecular:458.543-Amino-4-methylpentanoic acid
CAS:<p>DL-Homovaline, a beta-amino acid with an amino group at position 3 and a methyl at 4.</p>Fórmula:C6H13NO2Pureza:99.82%Forma y color:White Fine Crystalline PowderPeso molecular:131.17GLPG0187
CAS:<p>GLPG0187, a broad spectrum integrin receptor antagonist, inhibits αvβ1-integrin (IC50: 1.3 nM).</p>Fórmula:C29H37N7O5SPureza:99.4% - 99.70%Forma y color:SolidPeso molecular:595.71BIX01294 (hydrochloride hydrate)
CAS:<p>BIX01294 inhibits G9a HMTase (IC50=1.7μM), less effective on GLP, and aids in induced pluripotent stem cell generation.</p>Fórmula:C28H43Cl3N6O3Forma y color:SolidPeso molecular:618.04Glutaminase C-IN-1
CAS:<p>Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.</p>Fórmula:C27H27BrN2OPureza:99.68% - >99.99%Forma y color:SolidPeso molecular:475.42Carfilzomib
CAS:<p>Carfilzomib (PR-171) is a proteasome inhibitor that irreversibly binds to the chymotrypsin of the 20S proteasome.</p>Fórmula:C40H57N5O7Pureza:99.6% - 99.84%Forma y color:SolidPeso molecular:719.91AM095
CAS:<p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>Fórmula:C27H23N2NaO5Pureza:98.87%Forma y color:SolidPeso molecular:478.47Milnacipran ((1S-cis) hydrochloride)
CAS:<p>Milnacipran (1S-cis) hydrochloride (Levomilnacipran Hydrochloride) is a serotonin-norepinephrine reuptake inhibitor (SNRI), treatment of fibromyalgia.</p>Fórmula:C15H23ClN2OPureza:99.81%Forma y color:SolidPeso molecular:282.81Menthyl acetate
CAS:<p>(1R)-(-)-Menthyl acetate (L-Menthyl acetate) is a derivative of L-menthol.</p>Fórmula:C12H22O2Pureza:97.8% - ≥95%Forma y color:SolidPeso molecular:198.3AZ 11645373
CAS:<p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>Fórmula:C24H21N3O5SPureza:99.47%Forma y color:SolidPeso molecular:463.51Apiin
CAS:<p>Apiin (Apioside) reduces and stabilizes, inhibits iNOS and nitrite in J774.A1 cells pre-LPS.</p>Fórmula:C26H28O14Pureza:99.77% - ≥95%Forma y color:WhitePeso molecular:564.49γ-1-MSH, amide acetate (72629-65-3 free base)
<p>γ-1-MSH, amide acetate (72629-65-3 free base), a putative hormone in the N-terminal region of the ACTH/beta- endorphin (beta-EP) precursor protein, was studied</p>Fórmula:C74H101N21O16SPureza:>99.99%Forma y color:SolidPeso molecular:1572.81Phellamurin
CAS:<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Fórmula:C26H30O11Pureza:97.91%Forma y color:SolidPeso molecular:518.513-hydroxy-3-phenylpentanamide
CAS:<p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>Fórmula:C11H15NO2Pureza:98.42%Forma y color:SolidPeso molecular:193.24HIV-1 Nef-IN-1
CAS:<p>HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).</p>Fórmula:C18H16O2Pureza:99.90%Forma y color:SolidPeso molecular:264.32Guaiazulene
CAS:<p>Guaiazulene (azulon) belongs to the class of organic compounds known as guaianes.</p>Fórmula:C15H18Pureza:99.35%Forma y color:Dark Blue Semi-SolidPeso molecular:198.3AZ960
CAS:<p>AZ960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).</p>Fórmula:C18H16F2N6Pureza:96.02% - 98.51%Forma y color:SolidPeso molecular:354.36SMER3
CAS:<p>SMER3 is an inhibitor of the Skp1-Cullin-F-box (SCF)(Met30) ubiquitin ligase, a member of the SCF E3-ligase family, which regulates diverse cellular processes</p>Fórmula:C11H4N4O2Pureza:98.35%Forma y color:SolidPeso molecular:224.18Temsirolimus
CAS:<p>Temsirolimus (CCI-779) is a specific mTOR inhibitor ( IC50: 1.76 μM), used in the treatment of advanced renal cell cancer.</p>Fórmula:C56H87NO16Pureza:97.76% - >99.99%Forma y color:White Crystalline PowderPeso molecular:1030.29Lofemizole
CAS:<p>Lofemizole is an antagonist of CYP1A2.</p>Fórmula:C10H9ClN2Pureza:97.11%Forma y color:SolidPeso molecular:192.64Sal003
CAS:<p>Sal003, an effective cell-permeable analog, inhibitis the eIF2α phosphatase.</p>Fórmula:C18H15Cl4N3OSPureza:99.17% - 99.77%Forma y color:SolidPeso molecular:463.21Thiacetazone
CAS:<p>Thiacetazone (Diazam) is a thiosemicarbazone that thioacetazone treatment of pulmonary tuberculosis</p>Fórmula:C10H12N4OSPureza:99.07%Forma y color:SolidPeso molecular:236.29
