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Inhibidores

Inhibidores

Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.

Subcategorías de "Inhibidores"

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Se han encontrado 66641 productos de "Inhibidores"

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  • L-Carnitine

    CAS:
    <p>L-Carnitine aids fatty acid oxidation in mitochondria for energy, excluding the brain.</p>
    Fórmula:C7H15NO3
    Pureza:99.29% - 99.94%
    Forma y color:White Crystalline Hygroscopic Powder Solid
    Peso molecular:161.20
  • Clobetasone butyrate

    CAS:
    <p>Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such as</p>
    Fórmula:C26H32ClFO5
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:478.98
  • Bendamustine hydrochloride

    CAS:
    <p>Bendamustine hydrochloride (EP-3101) (IC50 of 50 μM) is an alkylating agent associated with DNA damage.</p>
    Fórmula:C16H21Cl2N3O2·HCl
    Pureza:97.71%
    Forma y color:Solid
    Peso molecular:394.72
  • Primaquine diphosphate

    CAS:
    <p>Primaquine diphosphate is the phosphate salt form of primaquine, a synthetic, 8-aminoquinoline derivative with antimalarial properties.</p>
    Fórmula:C15H21N3O·2H3PO4
    Pureza:98.06% - 99.73%
    Forma y color:Orange Powder
    Peso molecular:455.34
  • Nevanimibe hydrochloride

    CAS:
    <p>Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50</p>
    Fórmula:C27H40ClN3O
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:458.08
  • Vabicaserin hydrochloride

    CAS:
    <p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>
    Fórmula:C15H21ClN2
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:264.79
  • AZD7624

    CAS:
    <p>AZD7624 is an p38 inhibitor. It has potent anti-inflammatory activity.</p>
    Fórmula:C27H30FN5O3
    Pureza:98.82%
    Forma y color:Solid
    Peso molecular:491.56
  • Homatropine Methylbromide

    CAS:
    <p>Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.</p>
    Fórmula:C17H24BrNO3
    Pureza:98.97%
    Forma y color:Solid
    Peso molecular:370.29
  • 5-hydroxytryptophan

    CAS:
    <p>5-hydroxytryptophan (NSC-92523) is the immediate precursor in the biosynthesis of SEROTONIN from tryptophan. It is used as an antiepileptic and antidepressant.</p>
    Fórmula:C11H12N2O3
    Pureza:99.52%
    Forma y color:Minute Rods Or Needles From Ethanol White Solid
    Peso molecular:220.22
  • Ciliobrevin D

    CAS:
    <p>Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.</p>
    Fórmula:C17H8Cl3N3O2
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:392.62
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:348.87
  • Enarodustat

    CAS:
    <p>Enarodustat (JTZ-951) is an orally active factor inhibitor of prolyl hydroxylase (EC50: 0.22 μM) and has the potential for renal anemia treatment.</p>
    Fórmula:C17H16N4O4
    Pureza:99.73% - 99.75%
    Forma y color:Solid
    Peso molecular:340.33
  • Danthron

    CAS:
    <p>Danthron (Antrapurol) is a natural product, regulates glucose, and lipid metabolism by activating AMPK.</p>
    Fórmula:C14H8O4
    Pureza:99.51% - 99.97%
    Forma y color:Red Or Red-Yellow Needles Or Leaves (From Alcohol) Physical Description Orange Crystalline Powder Almost Odorless And Tasteless (Ntp 1992)
    Peso molecular:240.21
  • LCKLSL hydrochloride


    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Fórmula:C30H58ClN7O8S
    Pureza:98.02% - 99.31%
    Forma y color:Solid
    Peso molecular:712.34
  • Mizoribine

    CAS:
    <p>Mizoribine (NSC-289637) belongs to the family of 1-Ribosyl-imidazolecarboxamides. Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.</p>
    Fórmula:C9H13N3O6
    Pureza:98.38% - 99.95%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:259.22
  • Acedoben

    CAS:
    <p>Acedoben (4-acetamidobenzoic acid) is the acetyl derivative of para-aminobenzoic acid (PABA).</p>
    Fórmula:C9H9NO3
    Pureza:99.91%
    Forma y color:Physical Description Needles Or Off-White Powder (Ntp 1992)
    Peso molecular:179.17
  • Desbenzyl Donepezil Hydrochloride

    CAS:
    <p>Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.</p>
    Fórmula:C17H24ClNO3
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:325.83
  • Tioconazole

    CAS:
    <p>Tioconazole (Vagistat) is a synthetic imidazole derivative, inhibits cell wall synthesis by inhibiting the biosynthesis of ergosterol or other sterols.</p>
    Fórmula:C16H13Cl3N2OS
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:387.71
  • Zileuton

    CAS:
    <p>Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.</p>
    Fórmula:C11H12N2O2S
    Pureza:98.72% - 99.43%
    Forma y color:Crystalline Solid
    Peso molecular:236.29
  • 4'-Demethylepipodophyllotoxin

    CAS:
    <p>4'-Demethylepipodophyllotoxin (DMEP) is a potent inhibitor of microtubule assembly.</p>
    Fórmula:C21H20O8
    Pureza:98.49% - 99.72%
    Forma y color:White Crystalline Powder
    Peso molecular:400.38
  • Ascorbyl palmitate

    CAS:
    <p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>
    Fórmula:C22H38O7
    Pureza:99.52%
    Forma y color:White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like Odour
    Peso molecular:414.53
  • MOG peptide (35-55), mouse, rat acetate


    <p>Mouse, rat MOG peptide (35-55) acetate, part of myelin glycoprotein, for immune disease research.</p>
    Pureza:97.88%
    Forma y color:Soild
  • Linaclotide

    CAS:
    <p>Linaclotide treats IBS-C &amp; chronic constipation; it's a selective guanylate cyclase C agonist.</p>
    Fórmula:C59H79N15O21S6
    Pureza:97.93% - 98.71%
    Forma y color:Solid
    Peso molecular:1526.74
  • RA190

    CAS:
    <p>RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.</p>
    Fórmula:C28H23Cl5N2O2
    Pureza:97.7%
    Forma y color:Solid
    Peso molecular:596.76
  • Procurcumadiol

    CAS:
    <p>Procurcumadiol (5-Hydroxyprocurcumenol) is a natural product found in Curcuma longa and Curcuma phaeocaulis.</p>
    Fórmula:C15H22O3
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:250.33
  • Acetylleucine

    CAS:
    <p>Acetylleucine (N-Acetyl-DL-leucine) is an agent used in the treatment of vertigo.</p>
    Fórmula:C8H15NO3
    Pureza:99.77%
    Forma y color:White Powder
    Peso molecular:173.21
  • Kira8

    CAS:
    <p>Kira8 (AMG-18) is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity (IC50: 5.9 nM).</p>
    Fórmula:C31H29ClN6O3S
    Pureza:98.07%
    Forma y color:Solid
    Peso molecular:601.12
  • DCZ0415

    CAS:
    <p>DCZ0415: Potent TRIP13 inhibitor; combats myeloma in vitro, in vivo, and in drug-resistant patients; hinders DNA repair and NF-κB activity.</p>
    Fórmula:C23H20N2O2
    Pureza:99.34% - 99.95%
    Forma y color:Solid
    Peso molecular:356.42
  • Oxybutynin chloride

    CAS:
    <p>Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.</p>
    Fórmula:C22H32ClNO3
    Pureza:99.27% - >99.99%
    Forma y color:White Powder
    Peso molecular:393.96
  • 2',5'-Dideoxyadenosine

    CAS:
    <p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>
    Fórmula:C10H13N5O2
    Pureza:99.55%
    Forma y color:White Solid
    Peso molecular:235.24
  • SNDX-5613

    CAS:
    <p>Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.</p>
    Fórmula:C32H47FN6O4S
    Pureza:99.12% - 99.74%
    Forma y color:Solid
    Peso molecular:630.82
  • MRT-83

    CAS:
    <p>MRT-83 is a potent Smo antagonist.</p>
    Fórmula:C31H30N4O5
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:538.59
  • Atropine methyl bromide

    CAS:
    <p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>
    Fórmula:C18H26BrNO3
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:384.308
  • (3S,4R,5S)-1,3,4,5,6-Pentahydroxyhexan-2-one

    CAS:
    <p>(3S,4R,5S)-1,3,4,5,6-Pentahydroxyhexan-2-one (L(-)-Sorbopyranose) is a ketose belonging to the group of sugars known as monosaccharides.</p>
    Fórmula:C6H12O6
    Pureza:99.97%
    Forma y color:Rhombohedral Crystals From Ethanol White To Off-White Crystalline Powder
    Peso molecular:180.16
  • NE 10790

    CAS:
    <p>NE 10790, similar to risedronate, is a mild bone resorption inhibitor but poorly blocks FPP synthase.</p>
    Fórmula:C8H10NO6P
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:247.14
  • Unesbulin

    CAS:
    <p>Unesbulin (PTC596) is an orally active and selective inhibitor of B-cell-specific Moloney murine leukemia virus integration site 1 (BMI-1).</p>
    Fórmula:C19H13F5N6
    Pureza:98.71%
    Forma y color:Solid
    Peso molecular:420.34
  • Trospium chloride

    CAS:
    <p>Trospium chloride treats urinary incontinence without causing liver damage.</p>
    Fórmula:C25H30ClNO3
    Pureza:99.84% - >99.99%
    Forma y color:White To Off-White Powder
    Peso molecular:427.964
  • Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Fórmula:C9H10O4
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:182.17
  • Dibenzosuberone

    CAS:
    <p>Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline.</p>
    Fórmula:C15H12O
    Pureza:99.83%
    Forma y color:Clear To Yellow Liquid
    Peso molecular:208.26
  • DSP Crosslinker

    CAS:
    <p>DSP Crosslinker is a cleavable ADC linker, used in antibody-drug conjugates (ADCs) synthesis[1].</p>
    Fórmula:C14H16N2O8S2
    Pureza:97.89% - 99.94%
    Forma y color:Powder
    Peso molecular:404.42
  • Diphenylacetonitrile

    CAS:
    <p>Diphenylacetonitrile (Dipan) is used as herbicide and industrial intermediate.</p>
    Fórmula:C14H11N
    Pureza:98.56%
    Forma y color:White Crystal
    Peso molecular:193.24
  • Lanraplenib

    CAS:
    <p>Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.</p>
    Fórmula:C23H25N9O
    Pureza:98.35%
    Forma y color:Solid
    Peso molecular:443.5
  • Aliskiren hemifumarate

    CAS:
    <p>Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.</p>
    Fórmula:C30H53N3O6C4H4O4
    Pureza:96.18% - 99.21%
    Forma y color:Solid
    Peso molecular:1219.6
  • PF-3450074

    CAS:
    <p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>
    Fórmula:C27H27N3O2
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:425.52
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Forma y color:Solid
    Peso molecular:529.53
  • Sodium Nitroprusside

    CAS:
    <p>Sodium Nitroprusside (Ro 21-2498) is a potent vasodilator, releasing in blood with no spontaneously.</p>
    Fórmula:Na2Fe(CN)5NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:261.92
  • D-Glucuronic acid lactone

    CAS:
    <p>D-Glucuronic acid lactone (Dicurone) is a naturally occurring chemical that is an important structural component of nearly all connective tissues.</p>
    Fórmula:C6H8O6
    Pureza:98.59% - 99.15%
    Forma y color:Solid
    Peso molecular:176.12
  • Tigecycline

    CAS:
    <p>Tigecycline (GAR-936), a broad-spectrum glycylcycline, disrupts protein synthesis by binding the 30S ribosomal subunit.</p>
    Fórmula:C29H39N5O8
    Pureza:98.81% - >99.99%
    Forma y color:Powder
    Peso molecular:585.65
  • Arjungenin

    CAS:
    <p>Arjungenin, a triterpene derived from Terminalia arjuna, exhibits insect feeding-deterrent and growth inhibitory properties.</p>
    Fórmula:C30H48O6
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:504.7
  • Chloroxine

    CAS:
    <p>Chloroxine (Capitrol) is a quinoline derivative with antibacterial activity. Topical administration of chloroxine diminishes mitotic activity in the epidermis.</p>
    Fórmula:C9H5Cl2NO
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:214.05