
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.834 productos)
- Apoptosis(6.315 productos)
- Ciclo celular / Checkpoint(4.875 productos)
- Cromatina / Epigenética(2.613 productos)
- Señalización citoesquelética(1.567 productos)
- Daño al ADN / Reparación del ADN(2.872 productos)
- Endocrinología / Hormonas(3.754 productos)
- Enzima(3.672 productos)
- GPCR / proteína G(9.015 productos)
- Inmunología e inflamación(3.904 productos)
- Virus de la gripe(300 productos)
- Señalización JAK / STAT(415 productos)
- Señalización MAPK(1.257 productos)
- Transportador de membrana / canal de iones(3.155 productos)
- Metabolismo(10.137 productos)
- Microbiología / Virología(7.620 productos)
- Neurociencia(10.442 productos)
- Otros inhibidores(35.847 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.429 productos)
- Proteasas / Proteasoma(1.691 productos)
- Células madre y Derivados(732 productos)
- Tirosina quinasa / adaptadores(1.982 productos)
- Ubiquitinación(1.726 productos)
Mostrar 16 subcategorías más
Se han encontrado 66515 productos de "Inhibidores"
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NB-360
CAS:NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.Fórmula:C21H19F4N5O2Pureza:99.72%Forma y color:SolidPeso molecular:449.4Ref: TM-T12188
1mg104,00€5mg215,00€10mg318,00€25mg510,00€50mg692,00€100mg888,00€500mg1.783,00€1mL*10mM (DMSO)235,00€Tuvusertib
CAS:Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.Fórmula:C16H12F2N8OPureza:98.44% - 99.66%Forma y color:SolidPeso molecular:370.32Ref: TM-T10406
1mg58,00€5mg124,00€10mg187,00€25mg363,00€50mg505,00€100mg717,00€1mL*10mM (DMSO)142,00€BCL6-IN-3
CAS:BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Fórmula:C24H31ClF2N6O2Pureza:98.17%Forma y color:SolidPeso molecular:508.99Ref: TM-T10487
1mg109,00€5mg241,00€10mg355,00€25mg532,00€50mg745,00€100mg1.018,00€500mgA consultar1mL*10mM (DMSO)370,00€DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Fórmula:C22H24FN3O3Pureza:98.22% - 99.74%Forma y color:SolidPeso molecular:397.44KU-60019
CAS:KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).
Fórmula:C30H33N3O5SPureza:98.05% - 98.50%Forma y color:SolidPeso molecular:547.67NRX-252114
CAS:NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Fórmula:C22H12Cl2F3N3O2SPureza:99.70%Forma y color:SolidPeso molecular:510.32Enbezotinib
CAS:Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Fórmula:C21H21FN6O3Pureza:99.84%Forma y color:SolidPeso molecular:424.43Ref: TM-T62285
1mg77,00€5mg166,00€10mg253,00€25mg414,00€50mg567,00€100mg745,00€1mL*10mM (DMSO)182,00€Simmitecan hydrochloride
CAS:Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.Fórmula:C34H39ClN4O6Pureza:98.20% - 98.93%Forma y color:SolidPeso molecular:635.15Evixapodlin
CAS:Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.Fórmula:C34H36Cl2N8O4Pureza:97.02%Forma y color:SolidPeso molecular:691.61Ref: TM-T36487
1mg111,00€5mg264,00€10mg424,00€25mg747,00€50mg1.008,00€100mg1.359,00€200mg1.833,00€1mL*10mM (DMSO)405,00€NDI-034858
CAS:NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseasesFórmula:C23H24N8O3Pureza:>99.99%Forma y color:SolidPeso molecular:460.49HRO761
CAS:HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.Fórmula:C31H31ClF3N9O5Pureza:98.74% - 99.62%Forma y color:SolidPeso molecular:702.08Ref: TM-T72107
1mg57,00€5mg118,00€10mg167,00€25mg280,00€50mg475,00€100mg708,00€1mL*10mM (DMSO)778,00€AChE/BChE-IN-10
CAS:AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.
Fórmula:C26H30N2O2Pureza:99.55% - 99.88%Forma y color:SoildPeso molecular:402.53Glycosyltransferase-IN-1
Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.Fórmula:C19H21N5OPureza:99.76%Forma y color:SolidPeso molecular:335.4DRB18
CAS:DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.Fórmula:C22H23ClN2O2Pureza:99.54%Forma y color:SolidPeso molecular:382.88Ref: TM-T22317
1mg89,00€5mg215,00€10mg340,00€25mg687,00€50mg1.108,00€100mg1.485,00€500mg2.962,00€1mL*10mM (DMSO)236,00€Tigemonam
CAS:Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.Fórmula:C12H15N5O9S2Pureza:97.71% - >99.99%Forma y color:SolidPeso molecular:437.41INCB054329
CAS:INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.Fórmula:C19H16N4O3Pureza:99.52%Forma y color:SolidPeso molecular:348.36SY-5609
CAS:SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.Fórmula:C23H26F3N6OPPureza:99.34% - >99.99%Forma y color:SolidPeso molecular:490.46Ref: TM-T36038
1mg139,00€2mg200,00€5mg343,00€10mg553,00€25mgA consultar50mgA consultar1mL*10mM (DMSO)373,00€AZD-5672
CAS:AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.Fórmula:C32H38F2N2O5S2Pureza:98.1%Forma y color:SolidPeso molecular:632.78Ref: TM-T30260
1mg192,00€5mg434,00€10mg610,00€25mg888,00€50mg1.243,00€100mg1.693,00€1mL*10mM (DMSO)530,00€WAY-213613 hydrochloride
CAS:WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.Fórmula:C16H13BrF2N2O4Pureza:99.14% - 99.37%Forma y color:SoildPeso molecular:415.19Ref: TM-T13330
1mg35,00€5mg80,00€10mg92,00€25mg215,00€50mg359,00€100mg610,00€200mg827,00€1mL*10mM (DMSO)89,00€KI696
CAS:KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.Fórmula:C28H30N4O6SPureza:99.74%Forma y color:SolidPeso molecular:550.63Ref: TM-T11758L
1mg137,00€5mg281,00€10mg423,00€25mg707,00€50mg1.018,00€100mg1.468,00€200mg1.963,00€1mL*10mM (DMSO)341,00€
