
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.834 productos)
- Apoptosis(6.315 productos)
- Ciclo celular / Checkpoint(4.875 productos)
- Cromatina / Epigenética(2.613 productos)
- Señalización citoesquelética(1.566 productos)
- Daño al ADN / Reparación del ADN(2.872 productos)
- Endocrinología / Hormonas(3.754 productos)
- Enzima(3.672 productos)
- GPCR / proteína G(9.015 productos)
- Inmunología e inflamación(3.904 productos)
- Virus de la gripe(300 productos)
- Señalización JAK / STAT(415 productos)
- Señalización MAPK(1.257 productos)
- Transportador de membrana / canal de iones(3.154 productos)
- Metabolismo(10.137 productos)
- Microbiología / Virología(7.620 productos)
- Neurociencia(10.423 productos)
- Otros inhibidores(35.848 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.429 productos)
- Proteasas / Proteasoma(1.691 productos)
- Células madre y Derivados(732 productos)
- Tirosina quinasa / adaptadores(1.982 productos)
- Ubiquitinación(1.726 productos)
Mostrar 16 subcategorías más
Se han encontrado 66516 productos de "Inhibidores"
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FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Fórmula:C28H27FN2O3Pureza:97.45%Forma y color:SolidPeso molecular:458.52ZD 7155 hydrochloride
CAS:ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.Fórmula:C26H27ClN6OPureza:99.8%Forma y color:SolidPeso molecular:474.98Ref: TM-T13390
1mg42,00€5mg88,00€10mg135,00€25mg235,00€50mg396,00€100mg635,00€200mg887,00€1mL*10mM (DMSO)90,00€Aleglitazar
CAS:Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.Fórmula:C24H23NO5SPureza:99.03%Forma y color:SolidPeso molecular:437.51Ref: TM-T14176
1mg233,00€5mg532,00€10mg718,00€25mg1.099,00€50mg1.485,00€100mg1.998,00€1mL*10mM (DMSO)538,00€Gemcitabine elaidate hydrochloride
CAS:CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.
Fórmula:C27H44ClF2N3O5Pureza:98.50% - 99.6%Forma y color:SolidPeso molecular:564.11XMD-17-51 Trifluoroacetate
CAS:XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.Fórmula:C23H25F3N8O3Pureza:99.65%Forma y color:SolidPeso molecular:518.49FGI-106 tetrahydrochloride
CAS:FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFórmula:C28H42Cl4N6Pureza:99.68%Forma y color:SolidPeso molecular:604.48Ref: TM-T11281L
1mg82,00€5mg161,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€1mL*10mM (DMSO)207,00€Sinefungin
CAS:Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFórmula:C15H23N7O5Pureza:98% - 98.12%Forma y color:SolidPeso molecular:381.39LY3143921 hydrate
CAS:LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].Fórmula:C16H14FN5O2Pureza:98.43%Forma y color:SolidPeso molecular:327.31ARN19702
CAS:ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.Fórmula:C21H22FN3O3S2Pureza:99.86%Forma y color:SolidPeso molecular:447.55Ref: TM-T9528
1mg52,00€5mg113,00€10mg177,00€25mg350,00€50mg560,00€100mg880,00€200mg1.189,00€500mg1.765,00€1mL*10mM (DMSO)124,00€Rineterkib
CAS:Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Fórmula:C26H27BrF3N5O2Pureza:99.73%Forma y color:SolidPeso molecular:578.42Ref: TM-T11224
1mg87,00€5mg170,00€10mg318,00€25mg538,00€50mg765,00€100mg1.035,00€1mL*10mM (DMSO)224,00€Rolapitant hydrochloride
CAS:Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Fórmula:C25H27ClF6N2O2Pureza:98.35% - 99.79%Forma y color:SolidPeso molecular:536.94Ref: TM-T3724
1mg153,00€5mg365,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€200mg1.882,00€1mL*10mM (DMSO)439,00€CK2 inhibitor 2
CAS:CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Fórmula:C21H17ClN4O2Pureza:99.02%Forma y color:SolidPeso molecular:392.84Ref: TM-T35557
1mg62,00€5mg138,00€10mg215,00€25mg425,00€50mg637,00€100mg853,00€200mg1.153,00€1mL*10mM (DMSO)152,00€10-Methoxycamptothecin
CAS:10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Fórmula:C21H18N2O5Pureza:98.36%Forma y color:SolidPeso molecular:378.38TGFβRI-IN-3
CAS:TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.Fórmula:C28H23N3O2SPureza:99.85%Forma y color:SoildPeso molecular:465.57Ref: TM-T9523
1mg84,00€5mg177,00€10mg281,00€25mg552,00€50mg859,00€100mg1.234,00€500mg2.457,00€1mL*10mM (DMSO)177,00€BRD0639
CAS:BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Fórmula:C21H22ClN5O4SPureza:99.85%Forma y color:SolidPeso molecular:475.95JAK2-IN-7
CAS:JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.Fórmula:C26H33N7OPureza:99.54%Forma y color:SolidPeso molecular:459.59Ref: TM-T35900
1mg138,00€5mg334,00€10mg597,00€25mg1.234,00€50mg1.648,00€100mg2.232,00€1mL*10mM (DMSO)339,00€BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFórmula:C21H17F2N5OPureza:99.53%Forma y color:SolidPeso molecular:393.39Ref: TM-T9498
1mg80,00€5mg147,00€10mg215,00€25mg439,00€50mg750,00€100mg1.009,00€1mL*10mM (DMSO)161,00€(E/Z)-GSK5182
CAS:GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Fórmula:C27H31NO3Pureza:97.58%Forma y color:SolidPeso molecular:417.54Ref: TM-T7709
1mg77,00€5mg167,00€10mg260,00€25mg477,00€50mg707,00€100mg1.063,00€1mL*10mM (DMSO)177,00€PD 151746
CAS:PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Fórmula:C11H8FNO2SPureza:98.63% - ≥95%Forma y color:SolidPeso molecular:237.25Durlobactam sodium salt
CAS:Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Fórmula:C8H10N3NaO6SPureza:97.01% - 99.03%Forma y color:SolidPeso molecular:299.23
