Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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Tubeimoside I
CAS :<p>Tubeimoside I (Tubeimoside-1)(Lobatoside-H) is an extract from Chinese herbal medicine Bolbostemma paniculatum (MAXIM).</p>Formule :C63H98O29Degré de pureté :98.89% - 99.94%Couleur et forme :SolidMasse moléculaire :1319.43Britannin
CAS :<p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>Formule :C19H26O7Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :366.41SC99
CAS :<p>SC99 inhibits JAK2-STAT3, reducing STAT3 genes, platelet activity, and has anti-myeloma, anti-thrombotic effects.</p>Formule :C15H8Cl2FN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :336.15Thalidomide-NH-C6-NH2 hydrochloride
CAS :<p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>Formule :C19H25ClN4O4Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :408.88Piperazine Erastin
CAS :<p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>Formule :C35H41ClN6O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :645.19Psoralen
CAS :<p>Psoralen (Ficusin) is a furocoumarin that intercalates with DNA, inhibiting DNA synthesis and cell division.</p>Formule :C11H6O3Degré de pureté :99.3% - 99.87%Couleur et forme :Crystals From Ether Crystalline SolidMasse moléculaire :186.16Thalidomide-propargyl
CAS :<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Formule :C16H12N2O5Degré de pureté :95.14%Couleur et forme :SolidMasse moléculaire :312.28Sodium Oxamate
CAS :<p>Sodium Oxamate (Oxamic acid sodium salt) is an LDH inhibitor that specifically inhibits LDHA.</p>Formule :C2H2NNaO3Degré de pureté :99.23% - ≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :111.03Ketorolac hemicalcium
CAS :<p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation & pain, used in cancer research.</p>Formule :C30H24CaN2O6Couleur et forme :SolidMasse moléculaire :548.608Mocetinostat
CAS :<p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>Formule :C23H20N6ODegré de pureté :99% - 99.21%Couleur et forme :SolidMasse moléculaire :396.443,4 Dichloroisocoumarin
CAS :<p>3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitor</p>Formule :C9H4Cl2O2Degré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :215.03Perhexiline
CAS :<p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>Formule :C19H35NCouleur et forme :SolidMasse moléculaire :277.49KRCA-0008
CAS :<p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>Formule :C30H37ClN8O4Degré de pureté :96.19%Couleur et forme :SolidMasse moléculaire :609.12Carnosic acid
CAS :<p>Carnosic acid is a lipid absorption inhibitor, endowed with antioxidative, antimicrobial, photoprotective potential, and antiproliferative properties.</p>Formule :C20H28O4Degré de pureté :98.31% - 99.5%Couleur et forme :Yellow PowderMasse moléculaire :332.43Bigelovin
CAS :<p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>Formule :C17H20O5Degré de pureté :99.61% - 99.72%Couleur et forme :SolidMasse moléculaire :304.34Thalidomide-O-amido-PEG3-C2-NH2 TFA
CAS :<p>Synthetic E3 ligase ligand-linker, Thalidomide-O-amido-PEG3-C2-NH2 TFA, used in PROTAC with cereblon ligand and PEG.</p>Formule :C25H31F3N4O11Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :620.54OICR-9429
CAS :<p>OICR-9429 blocks WDR5 binding to MLL/Histone 3, hindering acute myeloid leukemia cell growth in vitro.</p>Formule :C29H32F3N5O3Degré de pureté :97.07% - 99.93%Couleur et forme :SolidMasse moléculaire :555.59Quizartinib
CAS :<p>Quizartinib (AC220) is an inhibitor of FLT3 (Kd: 1.6 nM) and demonstrates high selectivity for FLT3 when tested against a panel of 227 additional kinases.</p>Formule :C29H32N6O4SDegré de pureté :98% - 99.42%Couleur et forme :SolidMasse moléculaire :560.67Sepantronium bromide
CAS :<p>Sepantronium bromide (YM155) is a small-molecule proapoptotic agent with potential antineoplastic activity.</p>Formule :C20H19BrN4O3Degré de pureté :99.68% - 99.85%Couleur et forme :SolidMasse moléculaire :443.26PF-573228
CAS :<p>PF-573228 is an ATP-competitive FAK inhibitor. In a cell-free assay, the IC50 of FAK is 4 nM.</p>Formule :C22H20F3N5O3SDegré de pureté :96.58% - 99.51%Couleur et forme :SolidMasse moléculaire :491.49Staurosporine
CAS :<p>Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-Fgr</p>Formule :C28H26N4O3Degré de pureté :99.24% - 99.82%Couleur et forme :Off-White PowderMasse moléculaire :466.53NSC 3852
CAS :<p>NSC 3852 is a potent inhibitor of histone deacetylase.</p>Formule :C9H6N2O2Degré de pureté :99.64%Couleur et forme :Slightly Yellow To Yellow-Green PowderMasse moléculaire :174.16Etretinate
CAS :<p>Etretinate (Ro 10-9359), an oral retinoid, treats psoriasis by promoting cell differentiation and reducing cell growth and inflammation.</p>Formule :C23H30O3Degré de pureté :97.89%Couleur et forme :Crystals Crystalline SolidMasse moléculaire :354.48α-Lipoic Acid sodium
CAS :<p>α-Lipoic Acid (Thioctic acid) sodium, an essential cofactor for mitochondrial enzyme complexes, serves as an antioxidant.</p>Formule :C8H13NaO2S2Couleur et forme :SolidMasse moléculaire :228.31Afatinib Dimaleate
CAS :<p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>Formule :C32H33ClFN5O11Degré de pureté :98.11% - 99.87%Couleur et forme :SolidMasse moléculaire :718.08SKI-178
CAS :<p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>Formule :C21H22N4O4Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :394.42Pinosylvin
CAS :<p>Pinosylvin (5-Styrylresorcinol) induces autophagy via AMPK activation. Pinosylvin is likely to act as a pro-angiogenic factor.</p>Formule :C14H12O2Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :212.24D-Saccharic acid 1,4-lactone hydrate
CAS :<p>D-Saccharic acid 1,4-lactone hydrate inhibits β-glucuronidase (IC50=48.4 μM); has anticarcinogenic, detoxifying, antioxidant traits.</p>Formule :C17H20ClN3ODegré de pureté :99.49% - ≥98%Couleur et forme :SolidMasse moléculaire :317.81Sacubitril/Valsartan
CAS :<p>Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for treatment of hypertension and heart failure.</p>Formule :C48H55N6O8Na3·5H2ODegré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :957.99LCL161
CAS :<p>LCL161 is a SMAC mimetic, an IAP antagonist with oral activity that inhibits XIAP and cIAP1. LCL161 has potential antitumor activity. Cost-effective and quality-assured.</p>Formule :C26H33FN4O3SDegré de pureté :99.13% - 99.87%Couleur et forme :SolidMasse moléculaire :500.63Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86Thalidomide-NH-CH2-COOH TFA
CAS :<p>2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) is mainly used in compounds Synthesis.</p>Formule :C17H14F3N3O8Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :445.3036Z-VAD-FMK
CAS :<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formule :C21H28FN3O7Degré de pureté :98.24% - 99.79%Couleur et forme :SolidMasse moléculaire :453.46Alogliptin Benzoate
CAS :<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Formule :C25H27N5O4Degré de pureté :99.94% - >99.99%Couleur et forme :White PowderMasse moléculaire :461.51Niraparib tosylate monohyrate
CAS :<p>Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.</p>Formule :C26H30N4O5SDegré de pureté :97.7% - 98.41%Couleur et forme :SolidMasse moléculaire :510.61GSK621
CAS :<p>GSK621 is a specific and potent AMPK activator.</p>Formule :C26H20ClN3O5Degré de pureté :97.02% - 97.05%Couleur et forme :SolidMasse moléculaire :489.91DD1
CAS :<p>DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.</p>Formule :C16H14N2O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :282.29BAY 87-2243
CAS :<p>BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).</p>Formule :C26H26F3N7O2Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :525.53Rosmarinic acid
CAS :<p>Rosmarinic acid (Labiatenic acid) is widely found in plants and has antioxidant, anti-inflammatory, and antibacterial activities.</p>Formule :C18H16O8Degré de pureté :98.88% - 99.73%Couleur et forme :Brown Fine PowderMasse moléculaire :360.31NSC59984
CAS :<p>NSC59984, a p53 pathway activator, induces mutant p53 protein degradation and p73 activation.</p>Formule :C12H15N3O4Degré de pureté :99.33% - 99.59%Couleur et forme :SolidMasse moléculaire :265.27BAY 61-3606
CAS :<p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>Formule :C20H18N6O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :390.4Chloropyramine
CAS :<p>Chloropyramine: H1 antagonist for allergies like conjunctivitis, asthma; has anti-breast cancer properties.</p>Formule :C16H20ClN3Couleur et forme :SolidMasse moléculaire :289.8SB 202190
CAS :<p>SB 202190 (FHPI) is a p38 MAPK inhibitor that inhibits p38α and p38β2 (IC50=50/100 nM) selectively and cell-permeably.</p>Formule :C20H14FN3ODegré de pureté :98% - 99.84%Couleur et forme :Pale YellowMasse moléculaire :331.3420(R)-Ginsenoside Rh2
CAS :<p>20(R)-Ginsenoside Rh2 (Ginsenoside Rh2) is a minor stereoisomer of ginsenoside Rh2, possesses matrix metalloproteinase inhibitory.</p>Formule :C36H62O8Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :622.87Amentoflavone
CAS :<p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>Formule :C30H18O10Degré de pureté :98.21% - 99.22%Couleur et forme :Odourless Whitish SolidMasse moléculaire :538.46WYC-209
CAS :<p>WYC-209 inhibits proliferation of malignant murine melanoma tumor-repopulating cells (TRCs, IC50: 0.19 uM). It targets the retinoic acid receptor (RAR).</p>Formule :C20H20N2O3SDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :368.452-tert-Butyl-1,4-benzoquinone
CAS :<p>TBQ, a BHA metabolite, activates Nrf2 and S-arylates Keap1 in RAW264.7 cells.</p>Formule :C10H12O2Degré de pureté :97.19%Couleur et forme :SolidMasse moléculaire :164.2Methoxyamine HCl
CAS :<p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>Formule :CH6ClNODegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :83.51KW-2449
CAS :<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Formule :C20H20N4ODegré de pureté :98.43% - 99.69%Couleur et forme :SolidMasse moléculaire :332.4SRS11-92
CAS :<p>SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1</p>Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.47Nafamostat mesylate
CAS :<p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>Formule :C19H17N5O2·2CH4O3SDegré de pureté :97.36% - 99.76%Couleur et forme :Tan To Pale Orange SolidMasse moléculaire :539.58Benidipine
CAS :<p>Benidipine: potent oral calcium blocker, boosts nitric oxide synthase, enhances coronary flow, protects heart cells post-ischemia.</p>Formule :C28H31N3O6Couleur et forme :SolidMasse moléculaire :505.56Etidronic acid
CAS :<p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>Formule :C2H8O7P2Degré de pureté :99.93% - ≥95%Couleur et forme :Liquid SyrupMasse moléculaire :206.03TCS7010
CAS :<p>TCS7010 (Aurora A Inhibitor I) is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay.</p>Formule :C31H31ClFN7O2Degré de pureté :98.49% - 99.62%Couleur et forme :SolidMasse moléculaire :588.07Luminespib
CAS :<p>Luminespib (VER-52296) is an HSP90 inhibitor that inhibits HSP90α and HSP90β. Luminespib has antitumor activity. Cost-effective and quality-assured.</p>Formule :C26H31N3O5Degré de pureté :98% - 99.25%Couleur et forme :SolidMasse moléculaire :465.54Difurazon hydrochloride
CAS :<p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>Formule :C14H13ClN6O6Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :396.74dBET6
CAS :<p>dBET6 is a selective and cell-permeable degrader of BET based on PROTAC (IC50: 14 nM). It has antitumor activity.</p>Formule :C42H45ClN8O7SDegré de pureté :97.57% - 99.12%Couleur et forme :SolidMasse moléculaire :841.37Thalidomide-NH-C4-NH-Boc
CAS :<p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>Formule :C22H28N4O6Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :444.48Thalidomide-4-OH
CAS :<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Formule :C13H10N2O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :274.23Dinaciclib
CAS :<p>Dinaciclib (SCH 727965) is a CDK inhibitor that selectively inhibits CDK1, CDK2, CDK5, and CDK9 (IC50 = 3/1/1/4 nM).</p>Formule :C21H28N6O2Degré de pureté :98.21% - 99.75%Couleur et forme :SolidMasse moléculaire :396.49GSK778 hydrochloride
CAS :<p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>Formule :C30H34ClN5O3Degré de pureté :97.26% - 98.35%Couleur et forme :SolidMasse moléculaire :548.08Astragalin
CAS :<p>Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid.</p>Formule :C21H20O11Degré de pureté :98.8% - ≥95%Couleur et forme :SolidMasse moléculaire :448.38PRLX-93936
CAS :<p>PRLX-93936 is a selective Ras pathway protein inhibitor that modulates RAS/JNK pathway-associated protein phosphorylation, anticancer activity.</p>Formule :C21H24N4O2Couleur et forme :SolidMasse moléculaire :364.44Desciclovir
CAS :<p>Desciclovir (DCV), a prodrug of the antiherpetic agent acyclovir (ACV), is converted in humans to ACV, presumably by xanthine oxidase.</p>Formule :C8H11N5O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :209.21Phellamurin
CAS :<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Formule :C26H30O11Degré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :518.51PNU-74654
CAS :<p>PNU 74654 blocks β-catenin/Tcf4, disrupting Wnt signaling (Kd = 450 nM).</p>Formule :C19H16N2O3Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :320.34Pracinostat
CAS :<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Formule :C20H30N4O2Degré de pureté :99.15% - 99.67%Couleur et forme :SolidMasse moléculaire :358.482-Hydroxychalcone
CAS :<p>2-Hydroxychalcone (2-(2-Hydroxybenzal)Acetophenone) can be used as antiparasitic hit compounds when Methoxylated. It inhibits invasion of breast cancer cells.</p>Formule :C15H12O2Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :224.25UC2288
CAS :<p>UC2288, a Sorafenib-based p21 attenuator, reduces p21 levels without affecting its stability.</p>Formule :C20H18ClF6N3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :481.82Brassinolide
CAS :<p>Brassinolide (Brassin lactone) is a plant hormone isolated from rapeseed (Brassica napus) promoting stem elongation and cell division.</p>Formule :C28H48O6Degré de pureté :98% - 99.189%Couleur et forme :Off-White SolidMasse moléculaire :480.682-HBA
CAS :<p>2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.</p>Formule :C17H14O3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :266.29GMB-475
CAS :<p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>Formule :C43H46F3N7O7SDegré de pureté :98.78% - >99.99%Couleur et forme :SolidMasse moléculaire :861.93Ginkgetin
CAS :<p>Ginkgetin: antiviral, antifungal, anti-inflammatory; COX-2 reducer; STAT3 inhibitor; pro-apoptotic in cancer; neuroprotective in Parkinson's.</p>Formule :C32H22O10Degré de pureté :98.63% - 99.94%Couleur et forme :SolidMasse moléculaire :566.51Indirubin
CAS :<p>Indirubin (Couroupitine B) is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 5 uM and 0.6 uM.</p>Formule :C16H10N2O2Degré de pureté :97.21% - 99.74%Couleur et forme :Reddish-Violet PowderMasse moléculaire :262.26Liproxstatin-1 hydrochloride
CAS :<p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>Formule :C19H22Cl2N4Couleur et forme :SolidMasse moléculaire :377.31Valproic Acid
CAS :<p>Valproic Acid (2-Propylpentanoic Acid) is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels.</p>Formule :C8H16O2Degré de pureté :97.78% - 99%Couleur et forme :Colourless To Pale Yellow Liquid ViscousMasse moléculaire :144.21MK-2206
CAS :<p>MK-2206: selective Akt inhibitor, oral, targets Akt1, Akt2, Akt3; effective in breast cancer, PIK3CA mutants, PTEN-deficient cells.</p>Formule :C25H22ClN5OCouleur et forme :SolidMasse moléculaire :443.94GSK1059615
CAS :<p>GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.</p>Formule :C18H11N3O2SDegré de pureté :99.3% - ≥95%Couleur et forme :SolidMasse moléculaire :333.36Millepachine
CAS :<p>Millepachine is a natural product found in the Chinese herbal medicine with strong antitumor effects against numerous human cancer cells.</p>Formule :C22H22O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :350.41Eltrombopag
CAS :<p>Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the platelet</p>Formule :C25H22N4O4Degré de pureté :99.27%Couleur et forme :Orange To Red SolidMasse moléculaire :442.47Milademetan free base
CAS :<p>Milademetan (DS-3032b) is a potent MDM2 inhibitor, potentially blocking cancer growth by targeting p53 protein.</p>Formule :C37H42Cl2FN5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :790.73STF-118804
CAS :<p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 <10 nM.</p>Formule :C25H23N3O4SDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :461.53Methoxychlor
CAS :<p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>Formule :C16H15Cl3O2Degré de pureté :98.82% - ≥95%Couleur et forme :Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment IfMasse moléculaire :345.65[6]-Gingerol
CAS :<p>[6]-Gingerol ((S)-(+)-[6]Gingerol), an antioxidant, protects HL-60 cells from oxidative stress. It has protective effects for tumors.</p>Formule :C17H26O4Degré de pureté :98% - 99.66%Couleur et forme :Light Yellow OilinessMasse moléculaire :294.39DIM-C-pPhCO2Me
CAS :<p>DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist.</p>Formule :C25H20N2O2Degré de pureté :99.55% - 99.86%Couleur et forme :SolidMasse moléculaire :380.44Epoxiconazole
CAS :<p>Epoxiconazole (BAS-480F) is a 14-α demethylase inhibitor. It inhibits ergosterol synthesis and fungal cell wall formation.</p>Formule :C17H13ClFN3ODegré de pureté :98.57%Couleur et forme :Solid PowderMasse moléculaire :329.76SKI II
CAS :<p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>Formule :C15H11ClN2OSDegré de pureté :99.34% - 99.93%Couleur et forme :SolidMasse moléculaire :302.78Diffractaic Acid
CAS :<p>Diffractaic Acid (NSC 685595) can inhibit LTB4 biosynthesis in A-23187-stimulated bovine PMNL cells with activity value of 8 μM.</p>Formule :C20H22O7Degré de pureté :99.81% - 99.87%Couleur et forme :SolidMasse moléculaire :374.38NSC 95397
CAS :<p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>Formule :C14H14O4S2Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :310.39Glyphosate
CAS :<p>Glyphosate (Atila) is an herbicide. It also is a possible carcinogen to humans.</p>Formule :C3H8NO5PDegré de pureté :99.12% - 99.91%Couleur et forme :White Crystals (Darkens) Ph (1% Solution In Water) 2 5 (Ntp 1992)Masse moléculaire :169.07S-trityl-L-Cysteine
CAS :<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Formule :C22H21NO2SDegré de pureté :97.02%Couleur et forme :Almost White To Light Yellow Granular PowderMasse moléculaire :363.47Daphnetin
CAS :<p>Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),</p>Formule :C9H6O4Degré de pureté :97.47% - 99.8%Couleur et forme :SolidMasse moléculaire :178.14SR-4835
CAS :<p>SR-4835 is a highly selective dual inhibitor of CDK12 and CDK13(CDK12: IC50=99 nM, Kd=98 nM; CDK13: Kd=4.9 nM), which disables triple-negative breast cancer (</p>Formule :C21H20Cl2N10ODegré de pureté :98.09% - >99.99%Couleur et forme :SolidMasse moléculaire :499.36kauran-16,17-diol
CAS :<p>Kauran-16,17-diol, a natural diterpenoid product, exhibits anti-tumoral and apoptosis-inducing activities by inhibiting NO production in LPS-induced RAW 264.7</p>Formule :C20H34O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :306.48Tanespimycin
CAS :<p>Tanespimycin (KOS 953) is an Hsp90 inhibitor (IC50=5 nM) and is selective. Tanespimycin depletes intracellular STK38/NDR1. High-Quality, Low-Cost!</p>Formule :C31H43N3O8Degré de pureté :99.07% - 99.83%Couleur et forme :Dark Purple SolidMasse moléculaire :585.69LRRK2-IN-1
CAS :<p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>Formule :C31H38N8O3Degré de pureté :98% - 98.82%Couleur et forme :SolidMasse moléculaire :570.69HO-3867
CAS :<p>HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.</p>Formule :C28H30F2N2O2Degré de pureté :91.18% - 99.21%Couleur et forme :SolidMasse moléculaire :464.55BAM7
CAS :<p>BAM 7 is a direct and specific activator of proapoptotic Bax (EC50: 3.3 μM).</p>Formule :C21H19N5O2SDegré de pureté :98.51% - 98.68%Couleur et forme :SolidMasse moléculaire :405.47Carfilzomib
CAS :<p>Carfilzomib (PR-171) is a proteasome inhibitor that irreversibly binds to the chymotrypsin of the 20S proteasome.</p>Formule :C40H57N5O7Degré de pureté :99.6% - 99.84%Couleur et forme :SolidMasse moléculaire :719.91TW-37
CAS :<p>TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).</p>Formule :C33H35NO6SDegré de pureté :97.06% - ≥95%Couleur et forme :SolidMasse moléculaire :573.7
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