
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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Topotecan
CAS :<p>Topotecan (NSC-609669) is a Topoisomerase I inhibitor,and is an antineoplastic agent used to treat ovarian cancer that works by inhibiting DNA topoisomerases.</p>Formule :C23H23N3O5Degré de pureté :96.14% - 98.23%Couleur et forme :Light Yellow Needle Crystal Or Crystalline PowderMasse moléculaire :421.45DRB
CAS :<p>DRB is a nucleoside analog that inhibits several carboxyl-terminal domain (CTD) kinases including casein kinase II (IC50 range of 4-10 μM)</p>Formule :C12H12Cl2N2O4Degré de pureté :99.46% - 99.83%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :319.14Inauhzin
CAS :<p>Inauhzin (INZ) reactivates p53, inhibits SIRT1, induces Y cell apoptosis without genotoxic stress (IC50=3 uM in A549).</p>Formule :C25H19N5OS2Degré de pureté :98% - 99.36%Couleur et forme :SolidMasse moléculaire :469.58Tenovin-6 Hydrochloride
CAS :<p>Tenovin-6 HCl: Inhibits SIRT1 (21µM), SIRT2 (10µM), HDAC8; potent p53 activator.</p>Formule :C25H35ClN4O2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :491.09S-(5'-Adenosyl)-L-methionine tosylate
CAS :<p>S-(5'-Adenosyl)-L-methionine tosylate (SAMe) is a ubiquitous methyl donor involved in a wide variety of biological reactions, including those mediated by DNA</p>Formule :C22H30N6O8S2Degré de pureté :80% - 98.18%Couleur et forme :SolidMasse moléculaire :570.64Azoramide
CAS :<p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>Formule :C15H17ClN2OSDegré de pureté :99.08% - 99.85%Couleur et forme :SolidMasse moléculaire :308.83Thalidomide-5-methyl
CAS :<p>Thalidomide-5-methyl is the Thalidomide-based cereblon (CRBN) ligand. Thalidomide-5-methyl is used in the recruitment of CRBN protein.</p>Formule :C14H12N2O4Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :272.26AZD3759 hydrochloride
CAS :<p>AZD3759 hydrochloride is an oral, CNS-penetrant EGFR inhibitor with IC50s of 0.2/0.3/0.2 nM.</p>Formule :C22H24Cl2FN5O3Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :496.36Ciprofloxacin hydrochloride monohydrate
CAS :<p>Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) is a fluoroquinolone antibiotic with potent antibacterial activity.</p>Formule :C17H21ClFN3O4Degré de pureté :99.23% - 99.85%Couleur et forme :White Or Yellowish Crystalline PowderMasse moléculaire :385.82Laquinimod
CAS :<p>Laquinimod (LAQ) is an effective immunomodulator, which is currently under development in phase III trials for the treatment of multiple sclerosis as an oral</p>Formule :C19H17ClN2O3Degré de pureté :98.42% - 98.84%Couleur et forme :SolidMasse moléculaire :356.8Tenovin-3
CAS :<p>Tenovin-3 acts as a p53 activator.</p>Formule :C18H21N3OSDegré de pureté :99.72% - ≥95%Couleur et forme :SolidMasse moléculaire :327.44Demethoxycurcumin
CAS :<p>Demethoxycurcumin: antioxidant, anti-inflammatory, anti-proliferative, anti-acanthamoebic, enhances chemo for resistant cancers, inhibits cancer pathways.</p>Formule :C20H18O5Degré de pureté :94.54% - 99.86%Couleur et forme :SolidMasse moléculaire :338.35A-419259
CAS :<p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>Formule :C29H34N6ODegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :482.62Ro-3306
CAS :<p>RO-3306: ATP-competitive CDK1 inhibitor, Ki 20 nM, >15x more selective than other human kinases.</p>Formule :C18H13N3OS2Degré de pureté :97.67% - 99.79%Couleur et forme :SolidMasse moléculaire :351.45PKD-IN-1 dihydrochloride (956121-30-5 free base)
CAS :<p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>Formule :C18H21Cl3N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :415.75Tauroursodeoxycholate
CAS :<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Formule :C26H45NO6SDegré de pureté :98.77% - 99.93%Couleur et forme :White SolidMasse moléculaire :499.7PEAQX
CAS :<p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>Formule :C17H17BrN3O5PDegré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :454.21AR42
CAS :<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Formule :C18H20N2O3Degré de pureté :98.46% - 98.96%Couleur et forme :SolidMasse moléculaire :312.36Emricasan
CAS :<p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>Formule :C26H27F4N3O7Degré de pureté :98.13% - 99%Couleur et forme :SolidMasse moléculaire :569.5Aloperine
CAS :<p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>Formule :C15H24N2Degré de pureté :98% - 99.88%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :232.361400W dihydrochloride
CAS :<p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>Formule :C10H17Cl2N3Degré de pureté :98% - 99.94%Couleur et forme :SolidMasse moléculaire :250.17Bilobalide
CAS :<p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>Formule :C15H18O8Degré de pureté :98.81% - 99.92%Couleur et forme :White SolidMasse moléculaire :326.3Ipatasertib
CAS :<p>Ipatasertib (GDC-0068) is a selective, ATP-competitive pan-Akt inhibitor that can lead to p53-independent PUMA activation.Cost-effective and quality-assured.</p>Formule :C24H32ClN5O2Degré de pureté :98.28% - 99.21%Couleur et forme :SolidMasse moléculaire :458Sulforaphane
CAS :<p>Sulforaphane is a natural isothiocyanate that activates Nrf2. Sulforaphane has antitumor and anti-inflammatory activities. Cost-effective and quality-assured.</p>Formule :C6H11NOS2Degré de pureté :95% - 99.79%Couleur et forme :Light Yellow LiquidMasse moléculaire :177.29Nω-Hydroxy-nor-L-Arginine Dihydrochloride
CAS :<p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>Formule :C5H14Cl2N4O3Degré de pureté :99.12% - 99.84%Couleur et forme :SolidMasse moléculaire :249.10ZZW-115 hydrochloride
CAS :<p>ZZW-115 hydrochloride inhibits the activity of NUPR1.</p>Formule :C24H34Cl3F3N4SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :573.97Chromium picolinate
CAS :<p>Chromium picolinate causes DNA damage and mutation. It is an activator of p38.</p>Formule :C18H12CrN3O6Degré de pureté :99.64%Couleur et forme :Violet-Red Crystalline PowderMasse moléculaire :418.30Thalidomide-NH-PEG1-NH2 hydrochloride
CAS :<p>Thalidomide-NH-PEG1-NH2 hydrochloride (4-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione HCl) is a synthetic E3 ligase ligand-</p>Formule :C17H21ClN4O5Degré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :396.83Trolox
CAS :<p>Trolox is a vitamin E analogue, used in reducing oxidative stress or damage.</p>Formule :C14H18O4Degré de pureté :98.90% - 99.90%Couleur et forme :White To Fainly Beige Crystalline PowderMasse moléculaire :250.29Thalidomide-NH-CH2-COOH
CAS :<p>Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a</p>Formule :C15H13N3O6Degré de pureté :96.3800%Couleur et forme :SolidMasse moléculaire :331.28Tetrahydroxyquinone monohydrate
CAS :<p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>Formule :C6H6O7Couleur et forme :SolidMasse moléculaire :190.11Apocynin
CAS :<p>Apocynin (NSC 2146) is a specific NADPH-oxidase inhibitor (IC50: 10 μM).</p>Formule :C9H10O3Degré de pureté :99.71% - 99.98%Couleur et forme :Yellowish To Brown PowderMasse moléculaire :166.17Alda-1
CAS :<p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>Formule :C15H11Cl2NO3Degré de pureté :98.5% - 99.63%Couleur et forme :SolidMasse moléculaire :324.16Metamizole magnesium
CAS :<p>Metamizole magnesium (Metamizolemagnesiumsalt) is a pain reliever, which can antispasmodic.</p>Formule :C26H32MgN6O8S2Degré de pureté :93.51%Couleur et forme :SolidMasse moléculaire :645.01ARRY 520 hydrochloride
CAS :<p>'ARRY 520 hydrochloride: a KSP inhibitor causing apoptosis and strong anti-proliferative effects.'</p>Formule :C20H23ClF2N4O2SDegré de pureté :98.06% - 99.62%Couleur et forme :SolidMasse moléculaire :456.94Eltrombopag Olamine
CAS :<p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>Formule :C29H36N6O6Degré de pureté :99.59% - 99.89%Couleur et forme :SolidMasse moléculaire :564.63HA15
CAS :<p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>Formule :C23H22N4O3S2Degré de pureté :99.77% - 99.86%Couleur et forme :SolidMasse moléculaire :466.58ISRIB (trans-isomer)
CAS :<p>ISRIB (trans-isomer) is a potent inhibitor of PERK that rescues protein translation and prevents SG formation in the presence of P-eIF2α. Cost effective and quality assured.</p>Formule :C22H24Cl2N2O4Degré de pureté :97.86% - 99.27%Couleur et forme :SolidMasse moléculaire :451.34Thalidomide 4-fluoride
CAS :<p>Thalidomide 4-fluoride (E3 ligase Ligand 4) (Cereblon ligand 4) is the Thalidomide-based Cereblon ligand.</p>Formule :C13H9FN2O4Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :276.22Thalidomide-O-amido-C6-NH2 hydrochloride
CAS :<p>Thalidomide-O-amido-C6-NH2 HCl, a cereblon ligand-linker for PROTAC synthesis.</p>Formule :C21H27ClN4O6Degré de pureté :97.33%Couleur et forme :SolidMasse moléculaire :466.915CA-4948
CAS :<p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>Formule :C24H25N7O5Degré de pureté :99.35% - 99.88%Couleur et forme :SolidMasse moléculaire :491.5Tenovin-6
CAS :<p>Tenovin-6 is a p53 transcriptional activity agonist.</p>Formule :C25H34N4O2SDegré de pureté :97.71% - >99.99%Couleur et forme :SolidMasse moléculaire :454.63Dacarbazine citrate
CAS :<p>Dacarbazine citrate treats lymphatic cancers, malignant melanoma, islet cell carcinoma, and soft tissue sarcoma.</p>Formule :C12H18N6O8Couleur et forme :SolidMasse moléculaire :374.31FOXO4-DRI acetate
<p>FOXO4-DRI acetate is a bioactive chemical.</p>Formule :C36H64N14O14SDegré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :5358.06Periplocin
CAS :<p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>Formule :C36H56O13Degré de pureté :99.66% - 99.74%Couleur et forme :SolidMasse moléculaire :696.82TrxR1-IN-B19
CAS :<p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>Formule :C21H22O5Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :354.4Thalidomide-O-amido-C3-NH2 TFA
CAS :<p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>Formule :C20H21F3N4O8Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :502.4Thalidomide-O-COOH
CAS :<p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>Formule :C15H12N2O7Degré de pureté :98% - 98.29%Couleur et forme :SolidMasse moléculaire :332.27Methoxychlor
CAS :<p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>Formule :C16H15Cl3O2Degré de pureté :98.82% - ≥95%Couleur et forme :Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment IfMasse moléculaire :345.65Liproxstatin-1 hydrochloride
CAS :<p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>Formule :C19H22Cl2N4Couleur et forme :SolidMasse moléculaire :377.31GSK778 hydrochloride
CAS :<p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>Formule :C30H34ClN5O3Degré de pureté :97.26% - 98.35%Couleur et forme :SolidMasse moléculaire :548.08Thalidomide-4-OH
CAS :<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Formule :C13H10N2O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :274.23Thalidomide-NH-C4-NH-Boc
CAS :<p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>Formule :C22H28N4O6Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :444.48Difurazon hydrochloride
CAS :<p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>Formule :C14H13ClN6O6Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :396.74Methoxyamine HCl
CAS :<p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>Formule :CH6ClNODegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :83.51Alogliptin Benzoate
CAS :<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Formule :C25H27N5O4Degré de pureté :99.94% - >99.99%Couleur et forme :White PowderMasse moléculaire :461.51OICR-9429
CAS :<p>OICR-9429 blocks WDR5 binding to MLL/Histone 3, hindering acute myeloid leukemia cell growth in vitro.</p>Formule :C29H32F3N5O3Degré de pureté :97.07% - 99.93%Couleur et forme :SolidMasse moléculaire :555.59Thalidomide-O-amido-PEG3-C2-NH2 TFA
CAS :<p>Synthetic E3 ligase ligand-linker, Thalidomide-O-amido-PEG3-C2-NH2 TFA, used in PROTAC with cereblon ligand and PEG.</p>Formule :C25H31F3N4O11Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :620.54Bigelovin
CAS :<p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>Formule :C17H20O5Degré de pureté :99.61% - 99.72%Couleur et forme :SolidMasse moléculaire :304.34KRCA-0008
CAS :<p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>Formule :C30H37ClN8O4Degré de pureté :96.19%Couleur et forme :SolidMasse moléculaire :609.12Perhexiline
CAS :<p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>Formule :C19H35NCouleur et forme :SolidMasse moléculaire :277.49Ketorolac hemicalcium
CAS :<p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation & pain, used in cancer research.</p>Formule :C30H24CaN2O6Couleur et forme :SolidMasse moléculaire :548.608Thalidomide-propargyl
CAS :<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Formule :C16H12N2O5Degré de pureté :95.14%Couleur et forme :SolidMasse moléculaire :312.28Thalidomide-NH-C6-NH2 hydrochloride
CAS :<p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>Formule :C19H25ClN4O4Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :408.88Britannin
CAS :<p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>Formule :C19H26O7Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :366.41Verteporfin
CAS :<p>Verteporfin (BPD-MA) is a YAP inhibitor that inhibits YAP-TEAD interactions.</p>Formule :C41H42N4O8Degré de pureté :95.37% - 99.82%Couleur et forme :Dark Green To Black SolidMasse moléculaire :718.79Sulfaphenazole
CAS :<p>Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki: 63/29 μM for</p>Formule :C15H14N4O2SDegré de pureté :97.53% - 99.67%Couleur et forme :SolidMasse moléculaire :314.36PK11000
CAS :<p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>Formule :C6H5ClN2O4SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :236.63Abacavir monosulfate
CAS :<p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>Formule :C14H20N6O5SCouleur et forme :SolidMasse moléculaire :384.41Benidipine hydrochloride
CAS :<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Formule :C28H32ClN3O6Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :542.03(ZE)-SU9516
CAS :<p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>Formule :C13H11N3O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :241.25Diclofenac Potassium
CAS :<p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>Formule :C14H10Cl2KNO2Degré de pureté :99.51%Couleur et forme :White To Yellowish Crystalline PowderMasse moléculaire :334.24Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS :<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Formule :C23H27F3N4O10Degré de pureté :95.74% - 99%Couleur et forme :SolidMasse moléculaire :576.48IMT1
CAS :<p>IMT1 (Propanamide, N,N-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2H-1-benzopyran-7-yl]oxy]-) has anticancer activity.</p>Formule :C21H21NO4Degré de pureté :98.07% - 98.14%Couleur et forme :SolidMasse moléculaire :351.4Cystamine dihydrochloride
CAS :<p>Cystamine dihydrochloride is a radiation-protective agent. It also protects against carbon tetrachloride liver damage.</p>Formule :C4H14Cl2N2S2Degré de pureté :98.91% - 99.81%Couleur et forme :White PowderMasse moléculaire :225.19MS7972
CAS :<p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>Formule :C14H13NO2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :227.26KX2-361
CAS :<p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>Formule :C24H24FN3O2Degré de pureté :99.64% - 99.68%Couleur et forme :SolidMasse moléculaire :405.46Fipronil
CAS :<p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>Formule :C12H4Cl2F6N4OSDegré de pureté :97.21%Couleur et forme :Solid PowderMasse moléculaire :437.15Ralimetinib dimesylate
CAS :<p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>Formule :C24H29FN6·2CH4O3SDegré de pureté :98% - 99.38%Couleur et forme :SolidMasse moléculaire :612.74Pomolic acid
CAS :<p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>Formule :C30H48O4Degré de pureté :96.84% - 99.79%Couleur et forme :SolidMasse moléculaire :472.7Crebanine
CAS :<p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>Formule :C20H21NO4Degré de pureté :99.17% - 99.77%Couleur et forme :SolidMasse moléculaire :339.39DEL-22379
CAS :<p>DEL-22379 is a water-soluble ERK dimerization inhibitor with IC50 of ~0.5 μM.</p>Formule :C26H28N4O3Degré de pureté :99.3% - 99.53%Couleur et forme :SolidMasse moléculaire :444.53Cilengitide
CAS :<p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>Formule :C27H40N8O7Degré de pureté :98% - 99.8%Couleur et forme :SolidMasse moléculaire :588.66Rabeprazole sodium
CAS :<p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>Formule :C18H20N3NaO3SDegré de pureté :98% - 99.912%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :381.42Deltamethrin
CAS :<p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>Formule :C22H19Br2NO3Degré de pureté :99.25% - 99.85%Couleur et forme :White To Off-White Crystals Or PowderMasse moléculaire :505.20Mitochonic acid 5
CAS :<p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>Formule :C18H13F2NO3Degré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :329.3Nutlin-3
CAS :<p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C30H30Cl2N4O4Degré de pureté :98.13% - 99.89%Couleur et forme :SolidMasse moléculaire :581.49Desmorpholinyl Navitoclax-NH-Me
CAS :<p>Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a</p>Formule :C44H51ClF3N5O5S3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :918.55Avadomide HCl
CAS :<p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>Formule :C14H15ClN4O3Couleur et forme :SolidMasse moléculaire :322.75NAE-IN-M22
CAS :<p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>Formule :C20H24Cl2N2Degré de pureté :97.65%Couleur et forme :SolidMasse moléculaire :363.32Anagrelide hydrochloride
CAS :<p>Anagrelide hydrochloride (BL4162A) serves as a treatment for essential thrombocytosis.</p>Formule :C10H7Cl2N3O·HClDegré de pureté :99.58%Couleur et forme :Off-White PowderMasse moléculaire :292.55NSC622608
CAS :<p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>Formule :C9H12BrN3OS2Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :322.24Lercanidipine hydrochloride
CAS :<p>Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.</p>Formule :C36H41N3O6·HClDegré de pureté :99.86% - 99.91%Couleur et forme :Pale-Yellow PowderMasse moléculaire :648.194-Oxofenretinide
CAS :<p>4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.</p>Formule :C26H31NO3Degré de pureté :96.89%Couleur et forme :SolidMasse moléculaire :405.53Ibuprofen Lysine
CAS :<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Formule :C19H32N2O4Degré de pureté :99.26%Couleur et forme :CoaMasse moléculaire :352.471-(1-Naphthyl) piperazine hydrochloride
CAS :<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Formule :C14H17ClN2Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :248.75Bardoxolone Methyl
CAS :<p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>Formule :C32H43NO4Degré de pureté :97.81% - 99.09%Couleur et forme :SolidMasse moléculaire :505.69RA375
CAS :<p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>Formule :C30H25ClN4O7Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :588.99SRT 2183
CAS :<p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>Formule :C27H24N4O2SDegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :468.572-Bromohexadecanoic acid
CAS :<p>2-Bromohexadecanoic acid (2-BP) is a PPARδ agonist, and a palmitoylation inhibitor, inhibiting DHHC-mediated palmitoylation. Cost-effective and quality-assured.</p>Formule :C16H31BrO2Degré de pureté :97% - 98.3%Couleur et forme :White Crystalline PowderMasse moléculaire :335.32
