
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(9 produits)
- BCL(1 produits)
- Caspase(154 produits)
- FOXO1(2 produits)
- IAP(67 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(127 produits)
- PDK(9 produits)
- PERK(23 produits)
- Sérine/thréonine kinase(17 produits)
- Survivant(14 produits)
- TNF(90 produits)
- c-RET(61 produits)
- p53(63 produits)
Affichez 6 plus de sous-catégories
6170 produits trouvés pour "Apoptose"
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Hexylresorcinol
CAS :Hexylresorcinol (4-Hexylresorcinol) is a substituted dihydroxybenzene used topically as an antiseptic for the treatment of minor skin infections.Formule :C12H18O2Degré de pureté :99.26% - 99.51%Couleur et forme :Solid Solid Particulate/PowderMasse moléculaire :194.27Umbelliferone
CAS :Umbelliferone, aka 7-Hydroxycoumarin, in anise and many plants, is a phytoalexin with antioxidant effects.Formule :C9H6O3Degré de pureté :98.65% - 99.64%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :162.14Lexatumumab
CAS :Lexatumumab (GHS-ETR2), a human antibody, targets TRAILR2 for anticancer effects and apoptosis in mesothelioma.
Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :143.48 kDaTafasitamab
CAS :Tafasitamab (XmAb5574) is an FC-modified humanized monoclonal antibody targeting the human B-cell surface antigen CD19 for the study of diffuse large B-cell
Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:99.3%Couleur et forme :LiquidMasse moléculaire :147.41 kDaSorafenib tosylate
CAS :Sorafenib tosylate (Bay 43-9006) is a potent multikinase inhibitor (IC50s: 6/20/22 nM for Raf-1/VEGFR-3/B-Raf).Formule :C21H16ClF3N4O3·C7H8O3SDegré de pureté :99.24% - 99.94%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :637.03Ecabet Sodium
CAS :Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.Formule :C20H27NaO5SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :402.48Conatumumab
CAS :Conatumumab (AMG 655) targets DR5 to induce apoptosis in tumors, with Kd of 1 nM (long DR5) and 0.8 nM (short DR5).Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145.44 kDaPropafenone
CAS :Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.Formule :C21H27NO3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :341.44Hydralazine hydrochloride
CAS :Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.Formule :C8H9ClN4Degré de pureté :99.85% - 99.86%Couleur et forme :Yellow Crystals White Crystalline SolidMasse moléculaire :196.64Dabuzalgron
CAS :Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence.Formule :C12H16ClN3O3SDegré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :317.79Ref: TM-T10952
1mg35,00€5mg79,00€10mg128,00€25mg200,00€50mg299,00€100mg432,00€200mg602,00€1mL*10mM (DMSO)86,00€Mitotane
CAS :Mitotane (NCI-C04933) is a derivative of the insecticide dichlorodiphenyldichloroethane that specifically inhibits cells of the adrenal cortex.
Formule :C14H10Cl4Degré de pureté :99.89% - ≥95%Couleur et forme :Less Powder (Ntp 1992) Physical Description Colorless Powder (Ntp 1992)Masse moléculaire :320.04APTO-253
CAS :APTO-253 (LOR-253) inhibits c-Myc expression, stabilizes G-quadruplex DNA, and induces cell cycle arrest and apoptosis in acute myeloid leukemia cells.Formule :C22H14FN5Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :367.38Ref: TM-T10352
1mg40,00€2mg52,00€5mg75,00€10mg96,00€25mg170,00€50mg255,00€100mg371,00€1mL*10mM (DMSO)84,00€GPI-1046
CAS :GPI-1046: immunophilin ligand, no antibiotic effect, reduces ethanol intake by boosting GLT1 in PFC and NAc-core.
Formule :C20H28N2O4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :360.45Vildagliptin
CAS :Vildagliptin (LAF237), an oral DPP-4 inhibitor with hypoglycemic effects, is metabolized and excreted in urine.Formule :C17H25N3O2Degré de pureté :97.81% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :303.40ACHP
CAS :ACHP (IKK-2 Inhibitor VIII) is a novel selective and potent IKK inhibitor with inhibitory effects on IKK-α and IKK-β.Formule :C21H24N4O2Degré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :364.44Ref: TM-T22021
1mg50,00€5mg101,00€10mg150,00€25mg241,00€50mg353,00€100mg602,00€200mg982,00€500mg1.963,00€Levonorgestrel
CAS :Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device.Formule :C21H28O2Degré de pureté :99.42% - 99.44%Couleur et forme :Crystals From Methanol SolidMasse moléculaire :312.45UCB-9260
CAS :UCB-9260 inhibits TNF signaling by stabilizing an asymmetric form of the trimer.Formule :C26H25N5ODegré de pureté :98.39% - 99.24%Couleur et forme :SolidMasse moléculaire :423.51Ref: TM-T13951
1mg92,00€2mg133,00€5mg219,00€10mg353,00€25mg602,00€50mg802,00€100mg1.108,00€200mg1.485,00€1mL*10mM (DMSO)245,00€Daunorubicin hydrochloride
CAS :Daunorubicin hydrochloride (Rubidomycin hydrochloride), an anthracycline aminoglycoside antineoplastic, inhibits DNA replication and repair and RNA and proteinFormule :C27H29NO10·HClDegré de pureté :96.21% - 99.53%Couleur et forme :Cancer DrugMasse moléculaire :563.99Ref: TM-T1511
5mg34,00€10mg52,00€25mg87,00€50mg113,00€100mg177,00€200mg281,00€500mg442,00€1mL*10mM (DMSO)59,00€Cemiplimab
CAS :Cemiplimab, a human antibody, blocks PD-1 to inhibit T-cell suppression in metastatic and skin cancer studies.
Degré de pureté :SDS-PAGE:97.2%;SEC-HPLC:95.2%Couleur et forme :LiquidMasse moléculaire :143.81 kDaiFSP1
CAS :iFSP1, a potent, selective, and glutathione-independent ferroptosis suppressor protein 1 (FSP1) (AIFM2) inhibitor with an EC50 of 103 nM, sensitizes diverseFormule :C20H13N5Degré de pureté :98.74% - 99.74%Couleur et forme :SolidMasse moléculaire :323.35Lidocaine Hydrochloride hydrate
CAS :Lidocaine Hydrochloride hydrate is an amide local anesthetic, has anti-inflammatory property.Formule :C14H22N2O·HCl·H2ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :288.82Lornoxicam
CAS :Lornoxicam (Chlortenoxicam) (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory, andFormule :C13H10ClN3O4S2Degré de pureté :98.74% - 99.28%Couleur et forme :Crystalline SolidMasse moléculaire :371.82Sophocarpine monohydrate
CAS :Sophocarpine monohydrate, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.Formule :C15H22N2ODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :246.35L-SelenoMethionine
CAS :L-Selenomethionine is a natural amino acid boosting cell growth and antioxidant enzyme levels.Formule :C5H11NO2SeDegré de pureté :99.5% - 99.67%Couleur et forme :White To Off-WhitepowderMasse moléculaire :196.11Idebenone
CAS :Idebenone (CV-2619) is a synthetic analogue of ubiquinone (Coenzyme Q10), a vital cell antioxidant and essential component of the Electron Transport Chain (ETCFormule :C19H30O5Degré de pureté :99.52%Couleur et forme :Yellow-Orange Crystalline PowderMasse moléculaire :338.44Meclizine dihydrochloride
CAS :Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiationFormule :C25H27ClN2·2HClDegré de pureté :98.05% - 99.79%Couleur et forme :White Slightly Yellowish Crystalline PowderMasse moléculaire :463.87Dacarbazine
CAS :Dacarbazine (DTIC-Dome) is an antineoplastic agent. It has significant activity against melanomas.Formule :C6H10N6ODegré de pureté :99.78% - 99.87%Couleur et forme :Ivory Microcrystaline Substance Physical Description White To Ivory Microcrystals Or Off-White Crystalline Solid (Ntp 1992)Masse moléculaire :182.18Nortriptyline
CAS :Nortriptyline is an antidepressant compound used for smoking cessation.Formule :C19H21NDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :263.38Sodium salicylate
CAS :Sodium salicylate (2-Hydroxybenzoic acid sodium salt), a metabolite of acetylsalicylic acid, can inhibit NF-kB and reduce oxidative stress.Formule :C7H5NaO3Degré de pureté :99.36% - 99.92%Couleur et forme :White Solid AmorphousMasse moléculaire :160.11MD-224
CAS :MD-224 is a highly potent and efficacious MDM2 degrader based on the proteolysistargeting chimera (PROTAC) concept,and as a new class of anticancer agent.Formule :C48H43Cl2FN6O6Degré de pureté :99.07% - >99.99%Couleur et forme :SolidMasse moléculaire :889.8Ref: TM-T11980
1mg66,00€5mg144,00€10mg224,00€25mg358,00€50mg512,00€100mg707,00€200mg982,00€1mL*10mM (DMSO)158,00€Theophylline monohydrate
CAS :Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Proadifen hydrochloride
CAS :Proadifen hydrochloride (RP-5171) is an inhibitor of drug metabolism and cytochrome P-450 enzyme system activity.Formule :C23H32ClNO2Degré de pureté :99.84% - >99.99%Couleur et forme :SolidMasse moléculaire :389.96Emeramide
CAS :Emeramide (BDTH2) is a thiol-redox antioxidant. It is also a heavy metal chelator.Formule :C12H16N2O2S2Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :284.4Flurbiprofen
CAS :Flurbiprofen is an anti-inflammatory, analgesic, antipyretic that reduces bone resorption by inhibiting carbonic anhydrase.Formule :C15H13FO2Degré de pureté :99.78% - 99.96%Couleur et forme :SolidMasse moléculaire :244.2609Sodium etidronate
CAS :Sodium etidronate (Didronel), a bisphosphonate, resists degradation, inhibits osteoclasts, and may boost bone formation.Formule :C2H6Na2O7P2Degré de pureté :99.5% - 99.75%Couleur et forme :LiquidMasse moléculaire :249.99Temozolomide
CAS :Temozolomide (TMZ) is a DNA alkylating agent with blood-brain barrier permeability and oral activity.Formule :C6H6N6O2Degré de pureté :98% - 99.87%Couleur et forme :Off-White To Light-Pink Crystalline SolidMasse moléculaire :194.15Ref: TM-T1178
1g225,00€10mg47,00€25mg71,00€50mg85,00€100mg90,00€200mg120,00€500mg158,00€1mL*10mM (DMSO)56,00€Cinchonine
CAS :Cinchonine (LA40221), a potent amide local anesthetic for surface use, is toxic and limited to spinal anesthesia.Formule :C19H22N2ODegré de pureté :99.45%Couleur et forme :White Or Almost White Solid PowderMasse moléculaire :294.39(E)-Cardamonin
CAS :(E)-Cardamonin (Alpinetin chalcone) is a chalconoid that has been isolated from several plants including Alpinia katsumadai and Alpinia conchigera.Formule :C16H14O4Degré de pureté :99.07% - 99.84%Couleur et forme :SolidMasse moléculaire :270.28HPPH
CAS :HPPH (Photochlor) (Photochlor) is a second-generation photosensitizer. It is used as photodynamic therapy (PDT) agent.Formule :C39H48N4O4Degré de pureté :99.72%Couleur et forme :Black Solid PowderMasse moléculaire :636.82Ref: TM-T15501
1mg63,00€2mg92,00€5mg137,00€10mg236,00€25mg409,00€50mgÀ demander1mL*10mM (DMSO)177,00€Epirubicin hydrochloride
CAS :Epirubicin hydrochloride (Pharmorubicin) is a Topo and Foxp3 inhibitor. Epirubicin hydrochloride has antitumor activity. Cost-effective and quality-assured.Formule :C27H30ClNO11Degré de pureté :98.13% - 99.79%Couleur et forme :Orange-Red At Neutral Phs And Violet Blue Over Ph 9 (Ntp 1992)Masse moléculaire :579.98Ref: TM-T0125
2mg37,00€5mg52,00€10mg84,00€25mg142,00€50mg226,00€100mg308,00€500mg745,00€1mL*10mM (DMSO)70,00€Sinomenine hydrochloride
CAS :Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Formule :C19H24ClNO4Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :365.85Benzbromarone
CAS :Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.Formule :C17H12Br2O3Degré de pureté :99.37% - 99.73%Couleur et forme :SolidMasse moléculaire :424.08Xanthone
CAS :Xanthone (Xanthenone) is currently used as ovicide for codling moth eggs and as a larvicide.Formule :C13H8O2Degré de pureté :99.44% - 99.86%Couleur et forme :Off-White PowderMasse moléculaire :196.2Genistin
CAS :Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-Formule :C21H20O10Degré de pureté :97.65% - 97.85%Couleur et forme :Colorless CrystalsMasse moléculaire :432.38Octocrylene
CAS :Octocrylene, found in sunscreens and cosmetics, penetrates skin, acting as a photosensitizer to increase free radicals when exposed to light.Formule :C24H27NO2Degré de pureté :99.21%Couleur et forme :Physical Description Yellow Viscous Liquid Insoluble In Water (Ntp 1992)Masse moléculaire :361.48C16 Ceramide
CAS :C16 Ceramide (Palmitoyl Ceramide) is a naturally occurring small molecule that activates p53 by directly and selectively binding to it.Formule :C34H67NO3Degré de pureté :99% - 99.92%Couleur et forme :White Crystalline SolidMasse moléculaire :537.90STL127705
CAS :STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.Formule :C22H20FN5O4Degré de pureté :99.53% - 99.81%Couleur et forme :SolidMasse moléculaire :437.42Ref: TM-T13017
1mg70,00€5mg150,00€10mg219,00€25mg369,00€50mg550,00€100mg722,00€1mL*10mM (DMSO)170,00€PI-273
CAS :PI-273, a Substrate-Competitive, Specific Small-Molecule Inhibitor of PI4KIIα, Inhibits the Growth of Breast Cancer CellsFormule :C16H16ClN3O2S2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :381.9Butylated hydroxytoluene
CAS :Butylated hydroxytoluene (BHT FCC/NF) is an organic chemical composed of 4-methylphenol modified with tert-butyl groups at positions 2 and 6.Formule :C15H24ODegré de pureté :99.72%Couleur et forme :Colourless Solid PowderMasse moléculaire :220.35Lomefloxacin hydrochloride
CAS :Lomefloxacin hydrochloride (Okacyn) is a fluoroquinolone that inhibits DNA replication in bacteria, causing cell death.Formule :C17H20ClF2N3O3Degré de pureté :99.43% - 99.75%Couleur et forme :White PowderMasse moléculaire :387.81

