
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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Amifostine
CAS :<p>Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.</p>Formule :C5H15N2O3PSDegré de pureté :99.88%Couleur et forme :White SolidMasse moléculaire :214.22Lonidamine
CAS :<p>Lonidamine (Diclondazolic Acid) is an indazole carboxylic acid derivative, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-</p>Formule :C15H10Cl2N2O2Degré de pureté :97.90%Couleur et forme :White To Light Yellow CrystalMasse moléculaire :321.16Genistin
CAS :<p>Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-</p>Formule :C21H20O10Degré de pureté :97.65% - 97.85%Couleur et forme :Colorless CrystalsMasse moléculaire :432.38Abacavir
CAS :<p>Abacavir (Ziagen) is a nucleoside reverse transcriptase inhibitor analog of guanosine.</p>Formule :C14H18N6ODegré de pureté :99.36% - 99.81%Couleur et forme :White PowderMasse moléculaire :286.33Hexamethonium Bromide
CAS :<p>Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.</p>Formule :C12H30Br2N2Degré de pureté :99.76%Couleur et forme :White Crystalline Powder And AgglomeratesMasse moléculaire :362.19Semapimod tetrahydrochloride
CAS :<p>Semapimod tetrahydrochloride (CPSI-2364 tetrahydrochloride) is a mitogen-activated protein kinase blocker and pro-inflammatory cytokine production inhibitor.</p>Formule :C34H56Cl4N18O2Degré de pureté :97.21% - 99.8%Couleur et forme :SolidMasse moléculaire :890.74Sodium salicylate
CAS :<p>Sodium salicylate (2-Hydroxybenzoic acid sodium salt), a metabolite of acetylsalicylic acid, can inhibit NF-kB and reduce oxidative stress.</p>Formule :C7H5NaO3Degré de pureté :99.36% - 99.92%Couleur et forme :White Solid AmorphousMasse moléculaire :160.11Duvakitug
CAS :<p>Duvakitug (SAR-447189) is a humanized IgG1-λ2 monoclonal antibody targeting TNFSF15/TL1A, which can be used to study ulcerative colitis and Crohn's disease.</p>Degré de pureté :SDS-PAGE:>95%;SEC-HPLC:96.17%Couleur et forme :LiquidMasse moléculaire :143.64 kDaSodium etidronate
CAS :<p>Sodium etidronate (Didronel), a bisphosphonate, resists degradation, inhibits osteoclasts, and may boost bone formation.</p>Formule :C2H6Na2O7P2Degré de pureté :99.5% - 99.75%Couleur et forme :LiquidMasse moléculaire :249.99Batabulin
CAS :<p>Batabulin (T138067), an antitumor agent, binds selectively to β-tubulin, halts microtubule formation, and induces apoptosis.</p>Formule :C13H7F6NO3SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :371.26Benzbromarone
CAS :<p>Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.</p>Formule :C17H12Br2O3Degré de pureté :99.37% - 99.73%Couleur et forme :SolidMasse moléculaire :424.08(E)-Cardamonin
CAS :<p>(E)-Cardamonin (Alpinetin chalcone) is a chalconoid that has been isolated from several plants including Alpinia katsumadai and Alpinia conchigera.</p>Formule :C16H14O4Degré de pureté :99.07% - 99.84%Couleur et forme :SolidMasse moléculaire :270.28Lomustine
CAS :<p>Lomustine (NSC-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.</p>Formule :C9H16ClN3O2Degré de pureté :98.36% - 99.44%Couleur et forme :Solid SolidMasse moléculaire :233.7Ecabet Sodium
CAS :<p>Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.</p>Formule :C20H27NaO5SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :402.48Cytarabine
CAS :<p>Cytarabine (Ara-C) is a nucleoside analog, an inhibitor of DNA synthesis (IC50=16 nM).</p>Formule :C9H13N3O5Degré de pureté :99.83% - 99.93%Couleur et forme :Fine Off-White Crystalline PowderMasse moléculaire :243.22Vorinostat
CAS :<p>Vorinostat (SAHA) is a pan-histone deacetylase (HDAC) inhibitor (IC50=10 nM) with inhibitory activity against HDAC1/2/3/6/7/11.</p>Formule :C14H20N2O3Degré de pureté :99.47% - 99.65%Couleur et forme :White Crystalline SolidMasse moléculaire :264.32Emamectin Benzoate
CAS :<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Formule :C56H81NO15Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :1008.256Metamizole sodium hydrate
CAS :<p>Metamizole sodium hydrate (Analgin) is a potent analgesic drug that has been demonstrated to inhibit cyclooxygenase (COX).</p>Formule :C13H18N3NaO5SDegré de pureté :99.69% - 99.89%Couleur et forme :White Or Light Yellow Crystalline Powder Odorless Tiny BitterMasse moléculaire :351.36Sodium 4-phenylbutyrate
CAS :<p>Sodium 4-phenylbutyrate (TriButyrate), a transcriptional regulator, reversibly inhibits class I and II HDACs resulting in a global increase in gene expression.</p>Formule :C10H11NaO2Degré de pureté :99.02% - >99.99%Couleur et forme :SolidMasse moléculaire :186.18Niacin
CAS :<p>Niacin is a water-soluble B vitamin with antihyperlipidemic effects, found in food and converted to niacinamide for coenzyme activity.</p>Formule :C6H5NO2Degré de pureté :99.05% - 99.72%Couleur et forme :White Solid PowderMasse moléculaire :123.11Propafenone
CAS :<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Formule :C21H27NO3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :341.44Mycophenolic acid
CAS :<p>Mycophenolic acid (Mycophenolate) is an inosine monophosphate dehydrogenase(IMPDH) inhibitor with anti-proliferative activity.</p>Formule :C17H20O6Degré de pureté :98.79% - 99.77%Couleur et forme :SolidMasse moléculaire :320.34Piceatannol
CAS :<p>Piceatannol (Astringenin) is a synthetic anti-inflammatory that blocks p56lck, syk kinases, and NF-κB, made from resveratrol.</p>Formule :C14H12O4Degré de pureté :98.66% - 99.73%Couleur et forme :Light Tan To Yellow PowderMasse moléculaire :244.24STL127705
CAS :<p>STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.</p>Formule :C22H20FN5O4Degré de pureté :99.53% - 99.81%Couleur et forme :SolidMasse moléculaire :437.42Butylated hydroxytoluene
CAS :<p>Butylated hydroxytoluene (BHT FCC/NF) is an organic chemical composed of 4-methylphenol modified with tert-butyl groups at positions 2 and 6.</p>Formule :C15H24ODegré de pureté :99.72%Couleur et forme :Colourless Solid PowderMasse moléculaire :220.35Bithionol
CAS :<p>Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential to</p>Formule :C12H6Cl4O2SDegré de pureté :99.04%Couleur et forme :White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)Masse moléculaire :356.059-cis-Retinoic Acid
CAS :<p>9-cis-Retinoic Acid (Alitretinoin) is a derivative of vitamin A. It is a RAR/RXR agonist and can be used to study advanced tumors.</p>Formule :C20H28O2Degré de pureté :98.32% - 99.34%Couleur et forme :SolidMasse moléculaire :300.44Olanzapine
CAS :<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Formule :C17H20N4SDegré de pureté :99.86% - ≥95%Couleur et forme :Yellowish Crystalline PowderMasse moléculaire :312.43Tirabrutinib hydrochloride
CAS :<p>Tirabrutinib hydrochloride is a potent, highly selective, irreversible oral BTK inhibitor.Cost-effective and quality-assured.</p>Formule :C25H23ClN6O3Degré de pureté :99.04% - 99.27%Couleur et forme :SolidMasse moléculaire :490.94Nebivolol hydrochloride
CAS :<p>Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.</p>Formule :C22H25F2NO4·HClDegré de pureté :99.77% - >99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :441.90Dostarlimab
CAS :<p>Dostarlimab (TSR-042) is an immune checkpoint inhibitor targeting PD-1, blocking its interaction with its ligands PD-L1 and PD-L2.</p>Degré de pureté :>95%Couleur et forme :LiquidNimbolide
CAS :<p>Nimbolide, from neem, inhibits CDK4/6, NF-κB, Wnt, PI3K-Akt, MAPK, JAK-STAT pathways and induces apoptosis.</p>Formule :C27H30O7Degré de pureté :95.84% - 99.4%Couleur et forme :SolidMasse moléculaire :466.52Ruplizumab
CAS :<p>PF-03732010 is a humanized antibody targeting P-calmodulin with antitumor and antimetastatic activity.</p>Degré de pureté :98.5% (SDS-PAGE); 98.7% (SEC-HPLC) - 98.5% (SDS-PAGE); 98.7% (SEC-HPLC)Couleur et forme :LiquidDocetaxel
CAS :<p>Docetaxel (RP-56976) is a semi-synthetic analog of paclitaxel, a microtubule depolymerization inhibitor (IC50=0.2 μM).</p>Formule :C43H53NO14Degré de pureté :98.6% - 99.29%Couleur et forme :Off-White CrystMasse moléculaire :807.88Penpulimab
CAS :<p>Penpulimab is a monoclonal antibody targeting PD-1 with antitumor activity, used in studies of pancreatic cancer.</p>Degré de pureté :96.8% (SEC-HPLC) - 96.8% (SEC-HPLC)Couleur et forme :LiquidFlumethasone
CAS :<p>Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.</p>Formule :C22H28F2O5Degré de pureté :99.38% - 99.96%Couleur et forme :White Crystalline PowderMasse moléculaire :410.45Lomefloxacin hydrochloride
CAS :<p>Lomefloxacin hydrochloride (Okacyn) is a fluoroquinolone that inhibits DNA replication in bacteria, causing cell death.</p>Formule :C17H20ClF2N3O3Degré de pureté :99.43% - 99.75%Couleur et forme :White PowderMasse moléculaire :387.81Pioglitazone hydrochloride
CAS :<p>Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties and potential antineoplastic</p>Formule :C19H20N2O3S·HClDegré de pureté :99.64% - >99.99%Couleur et forme :White Crystals Or Crystalline PowderMasse moléculaire :392.90Cl-amidine hydrochloride
CAS :<p>Cl-amidine hydrochloride is an orally available PAD inhibitor that blocks histone 3 deimination.Cost-effective and quality-assured.</p>Formule :C14H20Cl2N4O2Degré de pureté :92.34% - 98.14%Couleur et forme :SolidMasse moléculaire :347.24Sodium metatungstate
CAS :<p>Sodium metatungstate (Sodium polyoxotungstate) is a potent inhibitor of ecto-nucleoside triphosphate diphosphohydrolase (NTPDase)(Ki values of 2.58 μM, 3.26 μM</p>Formule :H2Na6O40W12Degré de pureté :80%Couleur et forme :White - GreyMasse moléculaire :2985.99Hydralazine hydrochloride
CAS :<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Formule :C8H9ClN4Degré de pureté :99.85% - 99.86%Couleur et forme :Yellow Crystals White Crystalline SolidMasse moléculaire :196.64Adarotene
CAS :<p>Adarotene (ST1926) induces apoptosis, causes DNA damage, and has strong antiproliferative effects on human tumors.</p>Formule :C25H26O3Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :374.47Desonide
CAS :<p>Desonide is a synthetic topical steroid that reduces inflammation by inhibiting key inflammatory mediators.</p>Formule :C24H32O6Degré de pureté :99.5% - 99.74%Couleur et forme :SolidMasse moléculaire :416.51Simvastatin
CAS :<p>Simvastatin (MK 733) is an HMG-CoA reductase inhibitor (Ki=0.2 nM) with oral activity.</p>Formule :C25H38O5Degré de pureté :98.54% - 99.13%Couleur et forme :SolidMasse moléculaire :418.57Lidocaine
CAS :<p>Lidocaine, an amide local anesthetic, reduces pain and inflammation by dampening ICAM-1, cytokines, and neutrophil influx.</p>Formule :C14H22N2ODegré de pureté :99.95% - >99.99%Couleur et forme :Needles From Benzene Or Alcohol SolidMasse moléculaire :234.34GPI-1046
CAS :<p>GPI-1046: immunophilin ligand, no antibiotic effect, reduces ethanol intake by boosting GLT1 in PFC and NAc-core.</p>Formule :C20H28N2O4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :360.45(E)-Methyl 4-coumarate
CAS :<p>(E)-Methyl 4-coumarate (OMpCA) is a predicted metabolite generated by BioTransformer1 that is produced by the metabolism of methyl 3-phenylprop-2-enoate.</p>Formule :C10H10O3Degré de pureté :99.68% - 99.97%Couleur et forme :White Crystal PowderMasse moléculaire :178.18CDDO-dhTFEA
CAS :<p>CDDO-dhTFEA, a synthetic oleanane triterpenoid, effectively activates Nrf2 while inhibiting the NF-κB pro-inflammatory transcription factor.</p>Formule :C33H45F3N2O3Degré de pureté :95.61% - 99.59%Couleur et forme :SolidMasse moléculaire :574.72Amitriptyline hydrochloride
CAS :<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Formule :C20H24ClNDegré de pureté :97% - 99.94%Couleur et forme :Crystals White To Off-White PowderMasse moléculaire :313.86Deferasirox
CAS :<p>Deferasirox (CGP-72670) is an oral iron chelating agent used to treat chronic iron overload.</p>Formule :C21H15N3O4Degré de pureté :98.79% - 99.4%Couleur et forme :SolidMasse moléculaire :373.36

