Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(94 produits)
- CDK(500 produits)
- Arrêt du cycle cellulaire(4 produits)
- Chk(42 produits)
- DYRK(48 produits)
- Dynamine(23 produits)
- Ferroptose(215 produits)
- HSP(169 produits)
- Intégrine(224 produits)
- Kinésine(66 produits)
- LIM Kinase(19 produits)
- Microtubules associés(261 produits)
- PKC(102 produits)
- PLK(28 produits)
- ROCK(70 produits)
- Rho(2 produits)
- Wee1(15 produits)
- c-Myc(69 produits)
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3477 produits trouvés pour "Cycle cellulaire/point de contrôle"
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Abemaciclib methanesulfonate
CAS :<p>Abemaciclib methanesulfonate (LY2835219) is a specific and effective inhibitor of CDK4(IC50=2 nM) and CDK6(IC50=10 nM).</p>Formule :C27H32F2N8·CH4O3SDegré de pureté :98.69% - 99.44%Couleur et forme :SolidMasse moléculaire :602.7BUR1
CAS :<p>BUR1 is a Saccharomyces cerevisiae cyclin-dependent kinase (CDK) and is homologous to mammalian Cdk9, which functions in transcriptional elongation.</p>Formule :C16H17N5Degré de pureté :90%Couleur et forme :SolidMasse moléculaire :279.34NSC23005 Sodium
CAS :<p>NSC23005 sodium is a novel and effective p18 inhibitor (ED50=5.21 nM) in promoting Hematopoietic stem cells (HSCs) expansion in both murine and human models.</p>Formule :C13H16NNaO4SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :305.32Monastrol
CAS :<p>Monastrol ((±)-Monastrol) is a potent and cell-permeable inhibitor of the mitotic kinesin Eg5.</p>Formule :C14H16N2O3SDegré de pureté :98.02% - 98.59%Couleur et forme :SolidMasse moléculaire :292.35AUZ 454
CAS :<p>AUZ 454 (K03861) is a type II CDK2 inhibitor with Kd of 50/18.6/15.4/9.7 nM for CDK2(WT), CDK2(C118L), CDK2(A144C), and CDK2(C118L/A144C), respectlvely.</p>Formule :C24H26F3N7O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :501.5CX-5461
CAS :<p>CX5461 is an orally rRNA synthesis inhibitor that inhibits Pol I-driven rRNA transcription. CX5461 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C27H27N7O2SDegré de pureté :95.44% - 99.25%Couleur et forme :SolidMasse moléculaire :513.61Pipobroman
CAS :<p>Pipobroman (Vercyte) is an alkylating anti-cancer drug effective in PV and ET with low toxicity and thrombosis risk.</p>Formule :C10H16Br2N2O2Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :356.05BVDV-IN-1
CAS :<p>BVDV-IN-1 is a non-nucleoside inhibitor (NNI) of bovine viral diarrhea virus (BVDV), with an EC50 of 1.8 μM.</p>Formule :C20H22N4ODegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :334.41PND-1186
CAS :<p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>Formule :C25H26F3N5O3Degré de pureté :99.14% - 99.75%Couleur et forme :SolidMasse moléculaire :501.52-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi
CAS :<p>2-Amino-4-hydroxypyrrolo[2,3-d]pyrimidine serves as an intermediate.</p>Formule :C6H6N4ODegré de pureté :99.21% - 99.42%Couleur et forme :SolidMasse moléculaire :150.14Myoseverin
CAS :<p>Myoseverin triggers myotube fission into single cells, influencing genes for growth, immunity, matrix remodeling, and stress, aiding healing and regeneration.</p>Formule :C24H28N6O2Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :432.52OSU-T315
CAS :<p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>Formule :C30H30F3N5ODegré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :533.59HMN-176
CAS :<p>HMN-176 is a stilbene derivative which inhibits mitosis, interfering with polo-like kinase-1 (plk1).</p>Formule :C20H18N2O4SDegré de pureté :98.92% - 98.99%Couleur et forme :SolidMasse moléculaire :382.43PTC-209
CAS :<p>PTC-209 is a potent and selective BMI-1 inhibitor.</p>Formule :C17H13Br2N5OSDegré de pureté :99.43% - 99.887%Couleur et forme :SolidMasse moléculaire :495.19Antitumor agent-152
CAS :<p>Organic compound, potential dCK inhibitor, with 2-ethyl-3-methoxyphenyl-1,3-thiazole and pyrimidine units.</p>Formule :C17H19N5O2S2Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :389.5TC-E 5003
CAS :<p>TC-E 5003 (NSC-30176) is a selective inhibitor of PRMT1 with IC50 of 1.5 μM.</p>Formule :C16H14Cl2N2O4SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :401.26PHA-680632
CAS :<p>PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, respectively.</p>Formule :C28H35N7O2Degré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :501.62MK-8745
CAS :<p>MK-8745 is a potent and selective Aurora A inhibitor.</p>Formule :C20H19ClFN5OSDegré de pureté :99.09% - 99.79%Couleur et forme :SolidMasse moléculaire :431.91Purvalanol B
CAS :<p>Purvalanol B (NG 95) is a CDK inhibitor that inhibits Cdk2/cyclin A, Cdk2/cyclin E, Cdk5/p35, and Cdk2/cyclin B (IC50s = 6, 9, 6, and 6 nM, respectively)</p>Formule :C20H25ClN6O3Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :432.9C/EBPα inducer 1
CAS :<p>C/EBPα inducer 1 (4(3H)-Quinazolinone, 6-fluoro-2-[(1E)-2-(5-nitro-2-furanyl)ethenyl]-3-phenyl-) is a potential inducer of myeloid differentiation via</p>Formule :C20H12FN3O4Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :377.33VPC-80051 racemate
CAS :<p>VPC-80051 is the first small molecule inhibitor of hnRNP A1 splicing activity by using a computer-aided drug discovery approach.</p>Formule :C16H13F2N3ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :301.29HALOFUGINONE LACTATE
CAS :<p>HALOFUGINONE LACTATE is a halogenated derivative of febrifugine, a natural quinazolinone-containing compound found in the Chinese herb D.</p>Formule :C19H23BrClN3O6Degré de pureté :99.70% - 99.96%Couleur et forme :SolidMasse moléculaire :504.8WEE1-IN-3
CAS :<p>WEE1-IN-3 (JUN76288) is a potent Wee1 kinase inhibitor with an IC50 of <10 nM. It treatment of cancer and other proliferative diseases.</p>Formule :C28H31N7O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :497.59CB-6644
CAS :<p>CB-6644 is a small molecule inhibitor of the ATPase activity of the RUVBL1/2 complex.Cost-effective and quality-assured.</p>Formule :C29H34ClFN4O5Degré de pureté :96.33% - 99.85%Couleur et forme :SolidMasse moléculaire :573.062-Chloropyrazine
CAS :<p>2-Chloropyrazine is used in chemical industry.</p>Formule :C4H3ClN2Degré de pureté :98.98% - 99.89%Couleur et forme :Clear Colorless To Yellowish LiquidMasse moléculaire :114.53ARQ 621
CAS :<p>ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. Phase 1.</p>Formule :C28H24Cl2FN5O2Degré de pureté :97.01% - 98.38%Couleur et forme :SolidMasse moléculaire :552.43Bredinin aglycone
CAS :<p>Bredinin aglycone (SM-108) is a purine nucleotide analog.</p>Formule :C4H5N3O2Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :127.1Palbociclib monohydrochloride
CAS :<p>Palbociclib monohydrochloride (PD 0332991 hydrochloride) is a selective inhibitor of CDK4/6, with no inhibition against a panel of 36 additional protein kinases</p>Formule :C24H29N7O2·HClDegré de pureté :99.73% - >99.99%Couleur et forme :SolidMasse moléculaire :483.99Nolatrexed
CAS :<p>Nolatrexed is a thymidylate synthase inhibitor with potential anticancer activity.</p>Formule :C14H12N4OSDegré de pureté :97.53%Couleur et forme :SolidMasse moléculaire :284.34Rac1 Inhibitor W56 acetate(1095179-01-3 free base)
<p>Rac1 Inhibitor W56 acetate(1095179-01-3 free base) is a peptide comprising residues 45-60 of the guanine nucleotide exchange factor (GEF) recognition/activation</p>Formule :C76H121N19O25SDegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :1732.95Eptifibatide acetate (148031-34-9 free base)
CAS :<p>Eptifibatide acetate (148031-34-9), a cyclic heptapeptide GP IIb/IIIa inhibitor antiplatelet drug.</p>Formule :C35H49N11O9S2·xC2H4O2Degré de pureté :99.7% - 99.87%Couleur et forme :SolidMasse moléculaire :831.96 (free base)roxifiban
CAS :<p>Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.</p>Formule :C21H29N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.48PTC-209 hydrobromide
CAS :<p>PTC-209 hydrobromide (PTC-209 HBr) is the hydrobromide salt of PTC-209, which is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM, and results in</p>Formule :C17H13Br2N5OS·HBrDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :576.1CVT-313
CAS :<p>CVT-313 (NG-26) is a potent, selective, reversible, and ATP-competitive inhibitor.</p>Formule :C20H28N6O3Degré de pureté :97.46% - 97.97%Couleur et forme :SolidMasse moléculaire :400.47YKL-5-124
CAS :<p>YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7/Mat1/CycH, CDK2 and CDK9 respectively, displays</p>Formule :C28H33N7O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :515.61GW779439X
CAS :<p>GW779439X is an inhibitor of CDK.</p>Formule :C22H21F3N8Degré de pureté :97.87%Couleur et forme :SolidMasse moléculaire :454.45KB-0742 dihydrochloride
CAS :<p>KB-0742 dihydrochloride is a potent, selective and orally inhibitor of CDK9.</p>Formule :C16H27Cl2N5Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :360.33Besifloxacin Hydrochloride
CAS :<p>Besifloxacin Hydrochloride (BOL-303224-A) is a fourth-generation fluoroquinolone antibiotic.</p>Formule :C19H21ClFN3O3·HClDegré de pureté :99.20%Couleur et forme :Pale Yellow SolidMasse moléculaire :430.3TH588
CAS :<p>TH588 is nudix hydrolase family inhibitor that effectively and selectively engages and inhibits the MTH1(IC50: 5 nM) in cells.</p>Formule :C13H12Cl2N4Degré de pureté :96.05% - 99.82%Couleur et forme :SolidMasse moléculaire :295.17LP-935509
CAS :<p>LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1).Cost-effective and quality-assured.</p>Formule :C20H24N6O3Degré de pureté :98.78% - 99.64%Couleur et forme :SolidMasse moléculaire :396.44Raltitrexed
CAS :<p>Raltitrexed (D1694)(IC50 of 9 nM), a thymidylate synthase inhibitor, is used for the inhibition of L1210 cell growth.</p>Formule :C21H22N4O6SDegré de pureté :98.99% - 99.29%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :458.49AMG 900
CAS :<p>AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM.</p>Formule :C28H21N7OSDegré de pureté :98.4% - 99.51%Couleur et forme :SolidMasse moléculaire :503.58MKC3946
CAS :<p>MKC3946 is an effective and soluble IRE1α inhibitor which triggered modest growth inhibition in multiple myeloma cell lines.</p>Formule :C21H20N2O3SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :380.462′-O-Methylcytidine
CAS :<p>2′-O-Methylcytidine inhibits NS5B-catalyzed RNA synthesis in vitro, in a manner that is competitive with substrate nucleoside triphosphate.</p>Formule :C10H15N3O5Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :257.24Palbociclib Isethionate
CAS :<p>Palbociclib Isethionate (PD 0332991 isethionate) 是一种高选择性的CDK4/6抑制剂，IC50为11 nM 和16 nM。它对一组 36 种额外的蛋白激酶没有抑制作用。</p>Formule :C24H29N7O2·C2H6O4SDegré de pureté :99.01% - 99.27%Couleur et forme :SolidMasse moléculaire :573.66Arginine-glycine-aspartic acid
CAS :<p>RGD (RGD (Arg-Gly-Asp) Peptides) (Arg-Gly-Asp) Peptides is a cell adhesion motif which can mimic cell adhesion proteins and bind to integrins.</p>Formule :C12H22N6O6Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :346.34Natalizumab
CAS :<p>Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.</p>Degré de pureté :98.00%Couleur et forme :LiquidMasse moléculaire :N/AFUBP1-IN-1
CAS :<p>FUBP1-in-1: Potent FUBP1 inhibitor with 11.0 M IC50, disrupts FUBP1-DNA binding.</p>Formule :C19H14F3N3O2SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :405.39BMS-265246
CAS :<p>BMS-265246 is a potent and selective CDK1/2 inhibitor.</p>Formule :C18H17F2N3O2Degré de pureté :99.25% - 99.57%Couleur et forme :SolidMasse moléculaire :345.34ML264
CAS :<p>ML264 (CID-51003603) is a selective kruppel-like factor 5 (KLF5) inhibitor, which potently Inhibits growth of Colorectal Cancer.</p>Formule :C17H21ClN2O4SDegré de pureté :99.33% - 99.45%Couleur et forme :SolidMasse moléculaire :384.88XMD8-92
CAS :<p>XMD8-92 is an effective and specific BMK1/ERK5 inhibitor (Kd: 80 nM).</p>Formule :C26H30N6O3Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :474.55Verosudil hydrochloride
CAS :<p>Verosudil (AR-12286) is a selective Rho kinase inhibitor, reducing IOP in XFS & OHT/XFG, offering a new treatment option.</p>Formule :C17H18ClN3O2SCouleur et forme :SolidMasse moléculaire :363.86CCT241736
CAS :<p>CCT241736 is an orally bioavailable dual FLT3/Aurora kinase inhibitor that also inhibits clinically relevant FLT3-resistant mutants including FLT3-ITD and FLT3</p>Formule :C22H23Cl2N7Degré de pureté :96.2% - 99.81%Couleur et forme :SolidMasse moléculaire :456.37NY2267
CAS :<p>NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl</p>Formule :C38H43N3O6Degré de pureté :99.16% - 99.27%Couleur et forme :SolidMasse moléculaire :637.7610058-F4
CAS :<p>10058-F4 inhibits c-Myc-Max, blocking c-Myc target gene activation, causing cell-cycle arrest & apoptosis.</p>Formule :C12H11NOS2Degré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :249.35BTB-1
CAS :<p>BTB-1 (NSC156750) is a novel small molecule inhibitor of the mitotic motor protein Kif18A.</p>Formule :C12H8ClNO4SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :297.71Alisertib
CAS :<p>Alisertib (MLN 8237) is a specific Aurora A inhibitor (IC50: 1.2 nM). The selectivity of Alisertib(MLN 8237) is >200-fold higher for Aurora A than Aurora B.</p>Formule :C27H20ClFN4O4Degré de pureté :98.31% - >99.99%Couleur et forme :SolidMasse moléculaire :518.92SNS-314
CAS :<p>SNS-314 inhibits Aurora kinases A and B, blocking cell division in AK-overexpressing tumors.</p>Formule :C18H15ClN6OS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.93LDN-192960 hydrochloride
CAS :<p>LDN-192960 hydrochloride is an inhibitor of Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) and Haspin with IC50s of 48 nM and 10 nM, respectively.</p>Formule :C18H22Cl2N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.35Abemaciclib
CAS :<p>Abemaciclib (LY2835219) is a dual inhibitor of CDK4/6 (IC50=2/10 nM) with selectivity and specificity.</p>Formule :C27H32F2N8Degré de pureté :99.43% - 99.87%Couleur et forme :SolidMasse moléculaire :506.59Silver sulfadiazine
CAS :<p>Silver sulfadiazine (Dermazin) is a sulfonamide-based topical agent with antibacterial and antifungal activity.</p>Formule :C10H9AgN4O2SDegré de pureté :99.04% - 99.58%Couleur et forme :SolidMasse moléculaire :357.14Camostat mesylate
CAS :<p>Camostat mesylate (FOY-S980) is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.</p>Formule :C21H26N4O8SDegré de pureté :99.31% - 99.85%Couleur et forme :Crystalline SolidMasse moléculaire :494.52Tipiracil
CAS :<p>Tipiracil inhibits thymidine phosphorylase, enhancing trifluridine bioavailability, and is studied in colorectal and gastric cancer treatment.</p>Formule :C9H11ClN4O2Degré de pureté :99.815%Couleur et forme :SolidMasse moléculaire :242.66H-Gly-Arg-Gly-Asp-Asn-Pro-OH
CAS :<p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>Formule :C23H38N10O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :614.61Adefovir dipivoxil
CAS :<p>Adefovir dipivoxil (GS 0840) is a dipivoxil formulation of adefovir, a nucleoside reverse transcriptase inhibitor analog of adenosine with activity against</p>Formule :C20H32N5O8PDegré de pureté :98% - 99.80%Couleur et forme :It Has Broad-Spectrum Antiviral ActivityMasse moléculaire :501.47Ilorasertib
CAS :<p>Ilorasertib (ABT-348) inhibits Aurora kinases A/B/C & RET, PDGFRβ, Flt1 (IC50: 1-120 nM).</p>Formule :C25H21FN6O2SDegré de pureté :96.17% - 97.49%Couleur et forme :SolidMasse moléculaire :488.545-Fluorocytidine
CAS :<p>5-Fluorocytidine with antiviral activity</p>Formule :C9H12FN3O5Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :261.21JNJ-7706621
CAS :<p>JNJ-7706621 is a potent aurora kinase inhibitor, and also inhibits CDK1 and CDK2.</p>Formule :C15H12F2N6O3SDegré de pureté :99.1% - 99.85%Couleur et forme :SolidMasse moléculaire :394.36KW-2449
CAS :<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Formule :C20H20N4ODegré de pureté :98.43% - 99.69%Couleur et forme :SolidMasse moléculaire :332.46-Bromo-2-hydroxy-3-methoxybenzaldehyde
CAS :<p>6-Bromo-2-hydroxy-3-methoxybenzaldehyde (NSC-95682) is an inhibitor of IRE-1α (IC50 : 0.08 μM).</p>Formule :C8H7BrO3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :231.04Ara-G
CAS :<p>Ara-G, a deoxyguanosine analog, inhibits DNA synthesis, targeting T cell leukemia by converting to araGTP.</p>Formule :C10H13N5O5Degré de pureté :98.74%Couleur et forme :Slightly Off White To White PowderMasse moléculaire :283.24Empesertib
CAS :<p>Empesertib (BAY 1161909) is an orally bioavailable and selective inhibitor Mps1(IC50 < 1 nM), with potential antineoplastic activity.</p>Formule :C29H26FN5O4SDegré de pureté :97.45% - 99.4%Couleur et forme :SolidMasse moléculaire :559.61Longdaysin
CAS :<p>Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).</p>Formule :C16H16F3N5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :335.33Danusertib
CAS :<p>Danusertib (PHA-739358) is a small-molecule 3-aminopyrazole derivative with potential antineoplastic activity.</p>Formule :C26H30N6O3Degré de pureté :97.88% - 98.79%Couleur et forme :White PowderMasse moléculaire :474.55CCG-100602
CAS :<p>CCG-100602 inhibits RhoA/C-mediated, SRF-driven luciferase expression in PC-3 prostate cancer cells (IC50 :9.8 μM).</p>Formule :C21H17ClF6N2O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :478.824μ8C
CAS :<p>4μ8C (IRE1 Inhibitor III)(IC50=76 nM) is an effective and specific IRE1 Rnase inhibitor.</p>Formule :C11H8O4Degré de pureté :97.48% - 98.45%Couleur et forme :SolidMasse moléculaire :204.18Didox
CAS :<p>Didox (NSC-324360), a synthetic RR inhibitor, lowers oxidative injury markers in HIV-related dementia.</p>Formule :C7H7NO4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :169.13T56-LIMKi
CAS :<p>T56-LIMKi (T5601640) is a selective inhibitor of LIMK2.</p>Formule :C19H14F3N3O3Degré de pureté :98.39% - 99.57%Couleur et forme :SolidMasse moléculaire :389.33BAY-1816032
CAS :<p>BAY-1816032 is a benzimidazole budding inhibition relieved homolog protein 1 kinase (BUB1) inhibitor.Cost-effective and quality-assured.</p>Formule :C27H24F2N6O4Degré de pureté :98.02% - 99.81%Couleur et forme :SolidMasse moléculaire :534.51Mycro 3
CAS :<p>Mycro 3 is potent and selective for c-Myc in whole cell assays.</p>Formule :C24H17ClF2N6O4Degré de pureté :99.51% - 99.61%Couleur et forme :SolidMasse moléculaire :526.88ZCL278
CAS :<p>ZCL278 is a selective Cdc42 GTPase inhibitor.</p>Formule :C21H19BrClN5O4S2Degré de pureté :96.29% - 99.72%Couleur et forme :SolidMasse moléculaire :584.89BRD32048
CAS :<p>BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.</p>Formule :C16H22N6ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :314.39Tirapazamine
CAS :<p>Tirapazamine (Win59075) triggers apoptosis in hypoxic cells by damaging DNA and enhances effects of radiation and cisplatin.</p>Formule :C7H6N4O2Degré de pureté :96.65% - 99.87%Couleur et forme :Orange-Red Crystalline PowderMasse moléculaire :178.15GAK inhibitor 49 hydrochloride
<p>Potent GAK inhibitor 49 hydrochloride: ATP-competitive, highly selective, Ki=0.54 nM, IC50=56 nM, binds to RIPK2.</p>Formule :C20H23ClN2O5Couleur et forme :SolidMasse moléculaire :406.86PfDHODH-IN-1
CAS :<p>PfDHODH-IN-1 is an inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase(PfDHODH) which catalyzes the rate-limiting step for DNA and RNA biosynthesis.</p>Formule :C14H11F3N2O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :296.24TP-353
CAS :<p>TP-353 (EOS-61973) is a CDK7 inhibitor.</p>Formule :C35H30FNO3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :531.62ENMD-2076
CAS :<p>ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.</p>Formule :C21H25N7Degré de pureté :97.63% - ≥95%Couleur et forme :SolidMasse moléculaire :375.47Isoindigotin
CAS :<p>Isoindigotin is used in the therapy of Y.</p>Formule :C16H10N2O2Degré de pureté :98.14% - ≥95%Couleur et forme :SolidMasse moléculaire :262.26Cyclo(RGDyK) trifluoroacetate
CAS :<p>Cyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with IC50 of 20 nM.</p>Formule :C31H43F6N9O12Degré de pureté :95.28% - ≥95%Couleur et forme :SolidMasse moléculaire :847.72IXA4
CAS :<p>IXA4 is a highly selective, nontoxic activator of IRE1/XBP1s and reduces APP secretion by activating IRE1.</p>Formule :C24H28N4O4Degré de pureté :99.8% - 99.85%Couleur et forme :SolidMasse moléculaire :436.5Alovudine
CAS :<p>3'-Fluoro-3'-deoxythymidine (3'-Deoxy-3'-fluorothymidine) is a marker of DNA synthesis,which is less susceptible to inflammatory changes than FDG.</p>Formule :C10H13FN2O4Degré de pureté :99.41%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.22STF-083010
CAS :<p>STF-083010 is a selective inhibitor of the IRE1α endonuclease.</p>Formule :C15H11NO3S2Degré de pureté :98.09% - 99.45%Couleur et forme :SolidMasse moléculaire :317.381,4-Anthraquinone
CAS :<p>1,4-Anthraquinone: anticancer, hinders nucleoside transport, inhibits synthesis, fragments DNA, curbs L1210 cell growth; aids HPLC analysis of NAC, CAP.</p>Formule :C14H8O2Degré de pureté :95.96% - 97.01%Couleur et forme :Orange Brown SolidMasse moléculaire :208.21BI-1347
CAS :<p>BI-1347 is a potent, selective inhibitor of CDK8/cyclinC (IC50: 1 nM). It shows tumor growth inhibition in an in vivo xenograft model.</p>Formule :C22H20N4ODegré de pureté :96.7% - 99.63%Couleur et forme :SolidMasse moléculaire :356.42COH29
CAS :<p>COH29 is an oral RNR-blocking thiazole that may reduce DNA synthesis and promote apoptosis, with potential cancer-treating properties.</p>Formule :C22H16N2O5SDegré de pureté :97.04% - 98.92%Couleur et forme :SolidMasse moléculaire :420.44Pyridostatin Trihydrochloride
CAS :<p>Pyridostatin Trihydrochloride (RR-82 Trihydrochloride) is a G-quadruplexe stabilizer, with a Kd of 490 nM.</p>Formule :C31H35Cl3N8O5Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :706.02Fialuridine
CAS :<p>Fialuridine (DRG-0098), a DNA polymerase inhibitor, shows strong anti-HBV effects both in vitro and in vivo.</p>Formule :C9H10FIN2O5Degré de pureté :99.71% - 99.88%Couleur et forme :Less Crystals Colourless CrystalsMasse moléculaire :372.09Simeprevir sodium
CAS :<p>Simeprevir is a drug for the treatment and cure of hepatitis C.</p>Formule :C38H46N5NaO7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :771.92Dasabuvir
CAS :<p>Dasabuvir (ABT-333) blocks HCV replication by inhibiting the essential NS5B RNA polymerase.</p>Formule :C26H27N3O5SDegré de pureté :99.54% - 99.62%Couleur et forme :SolidMasse moléculaire :493.57EG1
CAS :<p>EG1, a novel specific inhibitor of Pax2 transcription activation, targets the DNA binding domain and inhibits embryonic kidney development.</p>Formule :C22H18N2O5Degré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :390.39
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