
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(116 produits)
- CDK(547 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(46 produits)
- Dynamine(27 produits)
- Ferroptose(227 produits)
- HSP(180 produits)
- Intégrine(276 produits)
- Kinésine(87 produits)
- LIM Kinase(21 produits)
- Microtubules associés(273 produits)
- PKC(127 produits)
- PLK(25 produits)
- ROCK(61 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(77 produits)
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3923 produits trouvés pour "Cycle cellulaire/point de contrôle"
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Levoleucovorin Calcium
CAS :Levoleucovorin Calcium (CL307782), a calcium salt of the folinic acid, is used in cancer chemotherapy as an adjuvant.Formule :C20H21N7O7·CaDegré de pureté :99.07% - ≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :511.55-Chloro-2'-deoxyuridine
CAS :5-Chloro-2'-deoxyuridine (5-Chlorodeoxyuridine) is a thymine analog.Formule :C9H11ClN2O5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :262.65Mps1-IN-3 hydrochloride
Mps1-IN-3 HCl: potent Mps1 inhibitor (IC50: 50 nM), hampers glioblastoma growth, enhances vincristine efficacy in vivo.Formule :C26H32ClN7O4SCouleur et forme :SolidMasse moléculaire :574.09CRT0044876
CAS :CRT0044876 (7-NO2-ICA) is a potent and selective APE1 inhibitor with IC50 of ~3 μM.Formule :C9H6N2O4Degré de pureté :98.27% - 98.98%Couleur et forme :Brown PowderMasse moléculaire :206.15EG1
CAS :EG1, a novel specific inhibitor of Pax2 transcription activation, targets the DNA binding domain and inhibits embryonic kidney development.Formule :C22H18N2O5Degré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :390.39Ref: TM-T27246
1mL*10mM (DMSO)33,00€2mg34,00€5mg54,00€10mg86,00€25mg130,00€50mg187,00€100mg260,00€200mg370,00€Fanotaprim
CAS :Fanotaprim is a dihydrofolate reductase (DHFR) inhibitor.Formule :C19H22N8ODegré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :378.43Ref: TM-T36692
1mg50,00€2mg71,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg170,00€25mg318,00€50mg442,00€100mg627,00€200mg845,00€Tegafur-Uracil
CAS :Tegafur-Uracil, an oral anticancer agent for solid tumor research, inhibits thymidylate synthase.Formule :C12H13FN4O5Couleur et forme :SolidMasse moléculaire :312.257AT9283
CAS :AT9283 (J-504568) is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora B and Abl(T315I).Formule :C19H23N7O2Degré de pureté :99.83% - 99.98%Couleur et forme :SolidMasse moléculaire :381.43Ref: TM-T3068
2mg39,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg111,00€25mg231,00€50mg371,00€100mg595,00€200mg833,00€GDC-0575
CAS :GDC-0575 (ARRY-575) is a highly-selective oral small-molecule Chk1 inhibitor(IC50 of 1.2 nM).Formule :C16H20BrN5ODegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :378.27N1-Methylpseudouridine
CAS :N1-Methylpseudouridine (1-Methylpseudouridine) is a methylpseudouridine and enhances translation through eIF2α-dependent and independent mechanisms byFormule :C10H14N2O6Degré de pureté :98.95% - 99.88%Couleur et forme :SolidMasse moléculaire :258.23Fadraciclib
CAS :Fadraciclib (CYC065) is an orally available, second-generation ATP-competitive inhibitor of CDK2/CDK9 kinases (IC50s: 5/26 nM).Formule :C21H31N7ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :397.52Ref: TM-TQ0053
1mg42,00€2mg55,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg145,00€25mg260,00€50mg414,00€100mg583,00€HA-100
CAS :HA-100 is an inhibitor of protein kinaseFormule :C13H15N3O2SDegré de pureté :99.44%Couleur et forme :Pale Yellow Crystalline SolidMasse moléculaire :277.34TCS7010
CAS :TCS7010 (Aurora A Inhibitor I) is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay.Formule :C31H31ClFN7O2Degré de pureté :98.49% - 99.62%Couleur et forme :SolidMasse moléculaire :588.07IMM-H007
CAS :IMM-H007 is a novel lipid-lowering agent, increasing abca1 protein expressionFormule :C22H23N5O8Degré de pureté :97.73%Couleur et forme :SolidMasse moléculaire :485.45Ref: TM-T9010
1mg38,00€5mg92,00€1mL*10mM (DMSO)124,00€10mg128,00€25mg215,00€50mg304,00€100mg411,00€200mg570,00€BAY-1816032
CAS :BAY-1816032 is a benzimidazole budding inhibition relieved homolog protein 1 kinase (BUB1) inhibitor.Cost-effective and quality-assured.Formule :C27H24F2N6O4Degré de pureté :98.02% - 99.81%Couleur et forme :SolidMasse moléculaire :534.51Ref: TM-T10467
1mg35,00€5mg80,00€1mL*10mM (DMSO)95,00€10mg119,00€25mg230,00€50mg339,00€100mg485,00€200mg665,00€MSC2530818
CAS :MSC2530818 is an effective, selective and orally available CDK8 inhibitor (IC50: 2.6 nM).Formule :C18H17ClN4ODegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :340.81Ref: TM-TQ0266
1mg63,00€5mg137,00€1mL*10mM (DMSO)150,00€10mg215,00€25mg462,00€50mg692,00€100mg964,00€Longdaysin
CAS :Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).Formule :C16H16F3N5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :335.33ML216
CAS :ML216 (CID-49852229) inhibits BLM helicase (IC50: 1.8 μM), 28-fold selective over RECQ1, RECQ5, and UvrD (IC50s > 50 μM).Formule :C15H9F4N5OSDegré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :383.325-Fluorocytidine
CAS :5-Fluorocytidine with antiviral activityFormule :C9H12FN3O5Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :261.21CRT0066854
CAS :CRT-0066854 is a PKCι and PKCζ inhibitor. CRT0066854 was able to restore polarized morphogenesis in the dysplastic H-Ras spheroids.Formule :C24H25N5SCouleur et forme :SolidMasse moléculaire :415.55Adefovir dipivoxil
CAS :Adefovir dipivoxil (GS 0840) is a dipivoxil formulation of adefovir, a nucleoside reverse transcriptase inhibitor analog of adenosine with activity againstFormule :C20H32N5O8PDegré de pureté :98% - 99.80%Couleur et forme :It Has Broad-Spectrum Antiviral ActivityMasse moléculaire :501.47SL327
CAS :SL327 is a selective inhibitor for MEK1/2 with IC50 of 0.18 μM/0.22 μM; able to transport through the blood-brain barrier.Formule :C16H12F3N3SDegré de pureté :97.98% - >99.99%Couleur et forme :SolidMasse moléculaire :335.35Talotrexin
CAS :Talotrexin (PT523), a nonpolyglutamatable antifolate analog of Aminopterin, inhibits DHFR and RFC, targeting tumor growth.Formule :C27H27N9O6Couleur et forme :SolidMasse moléculaire :573.56BTB-1
CAS :BTB-1 (NSC156750) is a novel small molecule inhibitor of the mitotic motor protein Kif18A.Formule :C12H8ClNO4SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :297.716-Thio-2'-Deoxyguanosine
CAS :6-Thio-2'-Deoxyguanosine (β-TGdR) is a nucleoside analog and telomerase substrate.Formule :C10H13N5O3SDegré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :283.31BTYNB
CAS :BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1. MDK6620 downregulates β-TrCP1 mRNA and reduces activation of NF-κB.Formule :C12H9BrN2OSDegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :309.185-Fluoroorotic acid
CAS :5-Fluoroorotic acid is an inhibitor of thymidylate synthase.Formule :C5H3FN2O4Degré de pureté :99.7% - >99.99%Couleur et forme :White To Pale Yellow PowderMasse moléculaire :174.09IMP-1088
CAS :IMP-1088 is a potent inhibitor of human N-myristoyltransferases NMT1 and NMT2 dual.Formule :C25H29F2N5ODegré de pureté :98.48% - 99.52%Couleur et forme :SolidMasse moléculaire :453.53Ref: TM-T9350
1mg137,00€2mg178,00€5mg268,00€1mL*10mM (DMSO)294,00€10mg444,00€25mg790,00€50mg1.063,00€XMD8-92
CAS :XMD8-92 is an effective and specific BMK1/ERK5 inhibitor (Kd: 80 nM).Formule :C26H30N6O3Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :474.55FUBP1-IN-1
CAS :FUBP1-in-1: Potent FUBP1 inhibitor with 11.0 M IC50, disrupts FUBP1-DNA binding.Formule :C19H14F3N3O2SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :405.39Ref: TM-T11332
1mg72,00€1mL*10mM (DMSO)144,00€5mg160,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€Palbociclib
CAS :Palbociclib is an oral CDK4/6 inhibitor, halts Rb phosphorylation, arrests cell cycle, and curbs tumor growth.Formule :C24H29N7O2Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :447.53A-674563 2HCl(552325-73-2(fb-2hcl))
A-674563 2HCl is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.Formule :C22H24Cl2N4ODegré de pureté :94.66%Couleur et forme :SolidMasse moléculaire :431.36Ref: TM-T6139L
1mg81,00€5mg131,00€1mL*10mM (DMSO)161,00€10mg178,00€25mg318,00€50mg479,00€100mg692,00€Besifloxacin Hydrochloride
CAS :Besifloxacin Hydrochloride (BOL-303224-A) is a fourth-generation fluoroquinolone antibiotic.Formule :C19H21ClFN3O3·HClDegré de pureté :99.20%Couleur et forme :Pale Yellow SolidMasse moléculaire :430.3Ref: TM-T6406
5mg38,00€1mL*10mM (DMSO)52,00€10mg57,00€25mg97,00€50mg172,00€100mg319,00€200mg470,00€500mg750,00€roxifiban
CAS :Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.
Formule :C21H29N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.48CCG-222740
CAS :CCG-222740 is an inhibitor of Rho/MRTF pathwayFormule :C23H19ClF2N2O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :444.86Ref: TM-T7764
2mg39,00€5mg62,00€1mL*10mM (DMSO)66,00€10mg94,00€25mg172,00€50mg260,00€100mg371,00€200mg530,00€GSK-25
CAS :GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K, and a dramatically improved P450 profile.Formule :C24H16Cl2F2N6ODegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :513.33Ref: TM-T4488
1mg44,00€2mg56,00€5mg87,00€1mL*10mM (DMSO)89,00€10mg111,00€25mg168,00€50mg258,00€100mg430,00€PNU112455A hydrochloride
CAS :PNU112455A hydrochloride is an ATP site competetive inhibitor of CDK2 and CDK5,binds to the ATP site of CDK2 and CDK5 with Kms of 3.6 and 3.2 μM, respectively.Formule :C10H12ClN5O2SDegré de pureté :98.58% - 99.22%Couleur et forme :SolidMasse moléculaire :301.75Ref: TM-T8230
2mg44,00€5mg71,00€1mL*10mM (DMSO)79,00€10mg100,00€25mg172,00€50mg266,00€100mg434,00€500mg964,00€Eptifibatide acetate (148031-34-9 free base)
CAS :Eptifibatide acetate (148031-34-9), a cyclic heptapeptide GP IIb/IIIa inhibitor antiplatelet drug.Formule :C35H49N11O9S2·xC2H4O2Degré de pureté :99.7% - 99.87%Couleur et forme :SolidMasse moléculaire :891.012-Chloropyrazine
CAS :2-Chloropyrazine is used in chemical industry.Formule :C4H3ClN2Degré de pureté :98.98% - 99.89%Couleur et forme :Clear Colorless To Yellowish LiquidMasse moléculaire :114.53CB-6644
CAS :CB-6644 is a small molecule inhibitor of the ATPase activity of the RUVBL1/2 complex.Cost-effective and quality-assured.Formule :C29H34ClFN4O5Degré de pureté :96.33% - 99.85%Couleur et forme :SolidMasse moléculaire :573.06Ref: TM-T10693
1mg205,00€5mg416,00€1mL*10mM (DMSO)525,00€10mg533,00€25mg748,00€50mg973,00€100mg1.260,00€ML367
CAS :ML367 inhibits ATAD5 stabilization with low micromolar activity, serving as a probe molecule.Formule :C19H12F2N4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :334.326-Bromo-2-hydroxy-3-methoxybenzaldehyde
CAS :6-Bromo-2-hydroxy-3-methoxybenzaldehyde (NSC-95682) is an inhibitor of IRE-1α (IC50 : 0.08 μM).Formule :C8H7BrO3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :231.04APTO-253 HCl
CAS :APTO-253 (LOR-253/LT-253) is a small-molecule MTF-1 inhibitor with antitumor properties, reducing cyclin D1, hypoxia, and angiogenesis gene expression.Formule :C22H15ClFN5Couleur et forme :SolidMasse moléculaire :403.84RI-2
CAS :RI-2, a potent RAD51 inhibitor, has a 44.17 μM IC50 and selectively blocks human HR repair.Formule :C21H18Cl2N2O4Degré de pureté :99.63% - 99.86%Couleur et forme :SolidMasse moléculaire :433.28Ref: TM-T2628
1mg70,00€2mg92,00€5mg152,00€1mL*10mM (DMSO)166,00€10mg266,00€25mg413,00€50mg605,00€100mg863,00€Ribociclib succinate hydrate
CAS :Ribociclib succinate hydrate is a highly specific CDK4/6 inhibitor (IC50s: 10 nM and 39 nM, respectively).Formule :C27H38N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :570.651VPC-80051 racemate
CAS :VPC-80051 is the first small molecule inhibitor of hnRNP A1 splicing activity by using a computer-aided drug discovery approach.Formule :C16H13F2N3ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :301.29C/EBPα inducer 1
CAS :C/EBPα inducer 1 (4(3H)-Quinazolinone, 6-fluoro-2-[(1E)-2-(5-nitro-2-furanyl)ethenyl]-3-phenyl-) is a potential inducer of myeloid differentiation viaFormule :C20H12FN3O4Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :377.33MK-8745
CAS :MK-8745 is a potent and selective Aurora A inhibitor.Formule :C20H19ClFN5OSDegré de pureté :99.09% - 99.79%Couleur et forme :SolidMasse moléculaire :431.91TC-E 5003
CAS :TC-E 5003 (NSC-30176) is a selective inhibitor of PRMT1 with IC50 of 1.5 μM.Formule :C16H14Cl2N2O4SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :401.26CAN508
CAS :CAN508: potent CDK9/T1 inhibitor; IC50 0.35 μM, Cdk2/E; Ki 13.3 μM, IC50 20 μM; 38x selective; antitumor.Formule :C9H10N6ODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :218.22TAK-632
CAS :TAK-632 is a potent pan-Raf inhibitor.Formule :C27H18F4N4O3SDegré de pureté :98% - 99.5%Couleur et forme :SolidMasse moléculaire :554.52NU6027
CAS :NU6027 is a potent ATR/CDK inhibitor, inhibits CDK1/2, ATR and DNA-PK with Ki of 2.5 μM/1.3 μM, 0.4 μM and 2.2 μM, enter cells more readily than the 6-Formule :C11H17N5O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :251.29M2I-1
CAS :M2I-1 inhibits Mad2 binding to Cdc20, disrupting SAC-related PPI and Mad2 dynamics, blocks Mad2-F-Mbp1 in FP assays.Formule :C19H24N4O4SDegré de pureté :99.02% - >99.99%Couleur et forme :SolidMasse moléculaire :404.48Poloxin
CAS :Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).Formule :C18H19NO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :297.35Antitumor agent-152
CAS :Organic compound, potential dCK inhibitor, with 2-ethyl-3-methoxyphenyl-1,3-thiazole and pyrimidine units.Formule :C17H19N5O2S2Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :389.5Ref: TM-T50079
1mg85,00€5mg170,00€1mL*10mM (DMSO)185,00€10mg253,00€25mg414,00€50mg583,00€100mg783,00€200mg1.054,00€Cdk5 Substrate acetate
Cdk5, a serine/threonine kinase active in neurons, phosphorylates proteins like histone H1; its synthetic substrate has a Km of 5 µM.Formule :C55H103N15O14Degré de pureté :96.21%Couleur et forme :SolidMasse moléculaire :1198.5Palmatine
CAS :Palmatine, also known as Burasaine, inhibits dopamine production and may treat flavivirus, jaundice, dysentery, hypertension, and liver issues.Formule :C21H22NO4Degré de pureté :96.28% - 99.49%Couleur et forme :SolidMasse moléculaire :352.4Preq1-Dihydrochloride
CAS :Preq1-Dihydrochloride, a queuosine pathway intermediate, binds strongly to PreQ1 riboswitch aptamer, suppressing protein expression.Formule :C7H11Cl2N5ODegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :252.1Myoseverin
CAS :Myoseverin triggers myotube fission into single cells, influencing genes for growth, immunity, matrix remodeling, and stress, aiding healing and regeneration.
Formule :C24H28N6O2Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :432.52PF 477736
CAS :PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (Formule :C22H25N7O2Degré de pureté :97.58% - 99.94%Couleur et forme :SolidMasse moléculaire :419.48SPHINX
CAS :SPHINX is a new generation inhibitor of SPRK1Formule :C17H17F3N2O3Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :354.322-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi
CAS :2-Amino-4-hydroxypyrrolo[2,3-d]pyrimidine serves as an intermediate.Formule :C6H6N4ODegré de pureté :99.21% - 99.42%Couleur et forme :SolidMasse moléculaire :150.141,7-Diaminoheptane
CAS :1,7-Diaminoheptane, an aliphatic amine, is used in peptide synthesis and as a substrate, ligand, or reagent.Formule :C7H18N2Degré de pureté :99.97%Couleur et forme :White To Light Yellow Crystalline ChunksMasse moléculaire :130.23Pipobroman
CAS :Pipobroman (Vercyte) is an alkylating anti-cancer drug effective in PV and ET with low toxicity and thrombosis risk.Formule :C10H16Br2N2O2Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :356.05BS194
CAS :BS194 is as a potent cyclin-dependent protein kinases (CDKs) inhibitor.Formule :C20H27N5O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :385.46Fasudil dihydrochloride
CAS :Fasudil dihydrochloride inhibits ROCK1/2, PKA, PKC, PKG, and acts as a Ca²⁺ channel blocker and vasodilator, supporting vascular, cardiovascular, and signaling research.Formule :C14H19Cl2N3O2SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :364.29AZ3146
CAS :AZ3146 is a selective Mps1 inhibitor with IC50 of ~35 nM.Formule :C24H32N6O3Degré de pureté :97.84% - >99.99%Couleur et forme :SolidMasse moléculaire :452.55A-286982
CAS :A 286982 blocks the LFA-1 and ICAM-1 integrin-ligand interaction.Formule :C24H27N3O4SDegré de pureté :97.81%Couleur et forme :SolidMasse moléculaire :453.55Ref: TM-T21781
1mg34,00€2mg48,00€5mg71,00€1mL*10mM (DMSO)77,00€10mg102,00€25mg200,00€50mg333,00€100mg495,00€9-Ethylguanine
CAS :9-Ethylguanine is a model nucleobase commonly used in the studies of DNA interactions with organometallic complexes.Formule :C7H9N5ODegré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :179.18CWHM-12
CAS :CWHM-12 is a potent inhibitor of αV integrins (IC50s of 0.2/0.8/1.5/1.8 nM for αvβ8/αvβ3/αvβ6/αvβ1).Formule :C26H32BrN5O6Degré de pureté :98.05% - 99.83%Couleur et forme :SolidMasse moléculaire :590.47Ref: TM-TQ0250
1mg40,00€2mg52,00€5mg88,00€1mL*10mM (DMSO)96,00€10mg126,00€25mg221,00€50mg369,00€100mg550,00€Spermine tetrahydrochloride
CAS :Spermine tetrahydrochloride, a polyamine in all eukaryotic cells, protects DNA from free radicals.Formule :C10H26N4·4HClDegré de pureté :99.75% - 99.82%Couleur et forme :SolidMasse moléculaire :348.18GJ103 sodium salt
CAS :GJ103 sodium salt, a GJ072 analog, lowers surface tension, viscosity, and pH in aqueous solutions, aiding molecular movement.Formule :C16H13N4NaO3SDegré de pureté :99.70% - 99.91%Couleur et forme :SolidMasse moléculaire :364.36Sovilnesib
CAS :Sovilnesib is a kinesin-like protein KIF18A inhibitor. Sovilnesib can be used for the cancer research.Formule :C26H34F2N6O4SDegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :564.65Ref: TM-T39994
1mg96,00€5mg235,00€1mL*10mM (DMSO)259,00€10mg376,00€25mg630,00€50mg898,00€100mg1.216,00€Gadodiamide
CAS :Gadodiamide is an MRI contrast agent, used in MR imaging procedures to assist in the visualization of blood vessels.Formule :C16H26GdN5O8Degré de pureté :99.86% - 99.93%Couleur et forme :SolidMasse moléculaire :573.66GS-441524 HCl
CAS :GS-441524: Inhibits FIP virus, EC50 at 0.78 μM, precursor to active triphosphate, non-toxic up to 100 μM, works at ≥1 μM, metabolite of Remdesivir.Formule :C12H14ClN5O4Couleur et forme :SolidMasse moléculaire :327.722,2'-Anhydrouridine
CAS :2,2'-Anhydrouridine (2,2'-Cyclouridine) is a research tool for antiviral and anticancer studies.Formule :C9H10N2O5Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :226.19Bohemine
CAS :Bohemine is a cyclin-dependent kinase inhibitor.Formule :C18H24N6ODegré de pureté :99.09% - 99.53%Couleur et forme :SolidMasse moléculaire :340.42Nemorubicin HCL
CAS :Nemorubicin HCL, a PNU152243A salt, acts on resistant tumors via topoisomerase I inhibition and targets NER pathway upregulated cells.Formule :C32H38ClNO13Couleur et forme :SolidMasse moléculaire :680.1PRT4165
CAS :PRT4165 (NSC600157) is a potent PRC1-mediated H2A ubiquitylation inhibitor.Formule :C15H9NO2Degré de pureté :98.91% - 99.6%Couleur et forme :SolidMasse moléculaire :235.24Ref: TM-T3110
5mg43,00€10mg49,00€1mL*10mM (DMSO)50,00€25mg88,00€50mg112,00€100mg182,00€200mg254,00€500mg427,00€KIRA6
CAS :KIRA6 is an effective inhibitor of IRE1α RNase kinase (IC50: 0.6 μM). It can trigger an apoptotic response.
Formule :C28H25F3N6ODegré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :518.53M2N12
CAS :M2N12 selectively inhibits Cdc25C (IC50=0.09μM) and has anti-tumor properties, affecting Cdc25A and B as well.Formule :C20H16ClN5O2Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :393.83Ref: TM-T11929
1mg84,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg236,00€25mg447,00€50mg670,00€100mg982,00€N2-Methylguanosine
CAS :N2-methylguanosine is a modified nucleoside of tRNA that occurs at several specific locations in many tRNA's
Formule :C11H15N5O5Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :297.27Triciribine
CAS :Triciribine (NSC-154020) is a DNA synthesis inhibitor, and it also inhibits Akt and HIV-1/2.Formule :C13H16N6O4Degré de pureté :99.01% - 99.87%Couleur et forme :SolidMasse moléculaire :320.3Ref: TM-T6065
1mg38,00€2mg49,00€5mg80,00€1mL*10mM (DMSO)88,00€10mg116,00€25mg207,00€50mg329,00€100mg512,00€200mg727,00€Rg3039
CAS :Rg3039 (PF-06687859) is a potent DcpS inhibitor. DcpS is a therapeutic target for spinal muscular atrophy (SMA). RG3039 improves motor function in SMA mice.Formule :C21H23Cl2N5ODegré de pureté :98.24% - 99.58%Couleur et forme :SolidMasse moléculaire :432.35ML-7 hydrochloride
CAS :ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM);Formule :C15H18ClIN2O2SDegré de pureté :99% - 99.26%Couleur et forme :White PowderMasse moléculaire :452.74Ref: TM-T3050
2mg34,00€5mg47,00€1mL*10mM (DMSO)52,00€10mg71,00€25mg141,00€50mg230,00€100mg334,00€200mg434,00€Hu7691
CAS :Hu7691 is an Akt inhibitor that inhibits Akt1, Akt2, and Akt3, suppresses neuroblastoma cell proliferation, and induces differentiation of neuroblastoma cells.Formule :C22H22ClF3N4ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :450.88Ganciclovir sodium
CAS :Ganciclovir sodium, a sodium salt with anti-CMV and HSV-1 antiviral properties.Formule :C9H13N5NaO4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :278.227BIO
CAS :7BIO triggers nonapoptotic death, blocks FLT3, DYRK1A/2, Aurora B/C kinases.
Formule :C16H10BrN3O2Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :356.17Lurbinectedin
CAS :Lurbinectedin (PM01183) is a DNA minor groove covalent binder. Lurbinectedin also shows effective anti-tumor activity.Formule :C41H44N4O10SDegré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :784.87MTOB
CAS :MTOB, a CtBP substrate, inhibits CtBP-linked cancer activity in cells/mice and regulates TCF-4, affecting CSC proliferation.Formule :C5H7NaO3SDegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :170.16VX-11e
CAS :VX-11e (TCS ERK 11e) is a potent, selective, and orally bioavailable ERK(Extracellular Signal-Regulated Kinase) inhibitor; antitumor agent.Formule :C24H20Cl2FN5O2Degré de pureté :98.92% - ≥98%Couleur et forme :SolidMasse moléculaire :500.35Piritrexim isethionate
CAS :Piritrexim isethionate, a fat-soluble DHFR inhibitor, shows efficacy in metastatic urothelial cancer with a 5-day oral regimen.Formule :C19H25N5O6SCouleur et forme :SolidMasse moléculaire :451.49HA-100 hydrochloride
CAS :HA-100 hydrochloride inhibits protein kinases PKG, PKA, PKC, MLC-kinase (IC50: 4-240 μM) and ROCK.Formule :C13H16ClN3O2SCouleur et forme :SolidMasse moléculaire :313.8Tirofiban hydrochloride monohydrate
CAS :Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.Formule :C22H39ClN2O6SDegré de pureté :98.81% - >99.99%Couleur et forme :White SolidMasse moléculaire :495.07GSK-923295
CAS :GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).Formule :C32H38ClN5O4Degré de pureté :96.22% - 98.02%Couleur et forme :SolidMasse moléculaire :592.13Ref: TM-T2039
1mg49,00€5mg97,00€1mL*10mM (DMSO)136,00€10mg168,00€25mg283,00€50mg432,00€100mg605,00€200mg852,00€ON-013100
CAS :ON-013100 is an antineoplastic drug. ON-013100 also acts as a mitotic inhibitor that could inhibit Cyclin D1 expression.Formule :C19H22O7SDegré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :394.44Ref: TM-T16391
1mg48,00€1mL*10mM (DMSO)60,00€5mg71,00€10mg100,00€25mg172,00€50mg268,00€100mg404,00€200mg570,00€Voruciclib
CAS :Voruciclib: oral, selective CDK inhibitor (Ki: 0.626-9.1 nM), reduces MCL-1, targets CDK9 in diffuse large B-cell lymphoma.Formule :C22H19ClF3NO5Degré de pureté :99.89% - 99.99%Couleur et forme :SolidMasse moléculaire :469.84MLN8054 sodium
CAS :MLN8054 sodium is an Aurora A inhibitor.Formule :C25H14ClF2N4NaO2Couleur et forme :SolidMasse moléculaire :498.84PHA-767491
CAS :PHA-767491 (CAY10572) is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and 34 nM, respectively.Formule :C12H11N3ODegré de pureté :99.49% - >99.99%Couleur et forme :SolidMasse moléculaire :213.24Ref: TM-T6206
2mg34,00€5mg49,00€1mL*10mM (DMSO)50,00€10mg64,00€25mg92,00€50mg138,00€100mg197,00€200mg295,00€SBC-115337
CAS :SBC-115337 is a PCSK9 inhibitor.Formule :C29H19N3O4Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :473.48

