
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(94 produits)
- CDK(500 produits)
- Arrêt du cycle cellulaire(4 produits)
- Chk(42 produits)
- DYRK(48 produits)
- Dynamine(23 produits)
- Ferroptose(215 produits)
- HSP(169 produits)
- Intégrine(224 produits)
- Kinésine(66 produits)
- LIM Kinase(19 produits)
- Microtubules associés(261 produits)
- PKC(102 produits)
- PLK(28 produits)
- ROCK(70 produits)
- Rho(2 produits)
- Wee1(15 produits)
- c-Myc(69 produits)
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3477 produits trouvés pour "Cycle cellulaire/point de contrôle"
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D-Xylofuranose, 1,2,3,5-tetraacetate
CAS :<p>1,2,3,5-Tetra-O-acetyl-D-xylofuranose is a starting material for the synthesis of nucleosides.</p>Formule :C13H18O9Couleur et forme :SolidMasse moléculaire :318.28Myt1-IN-1
CAS :<p>Myt1-IN-1 has anticancer effects that is a potent inhibitor of Myt1 with an IC 50 of <10 nM [1].</p>Formule :C16H15ClN4O2Couleur et forme :SolidMasse moléculaire :330.77AM-TS23
CAS :<p>AM-TS23 is used as a DNA polymerase lambda and beta inhibitor.</p>Formule :C17H12N2O3S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.48ML366
CAS :<p>ML366 is a Vibrio cholerae Quorum Sensing inhibitor Acting via the LuxO response regulator.</p>Formule :C17H19N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.35HBX28258
CAS :<p>HBX28258, a human USP7 inhibitor, binds covalently and selectively deactivates USP7 in colon cancer and kidney cells.</p>Formule :C26H30ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :435.99JNJ-9676
CAS :<p>JNJ-9676 is an orally active inhibitor of the coronavirus membrane protein, thereby blocking viral assembly and release.coronavirus and SARS-CoV.</p>Formule :C28H21F2N5O2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :497.5DHODH-IN-3
CAS :<p>DHODH-IN-3: Human DHODH inhibitor with IC50 of 261 nM, Kiapp 32 nM, potential anti-malaria drug.</p>Formule :C17H13ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.75OXA-06 Dihydrochloride
CAS :<p>OXA-06 Dihydrochloride is a PANC-1 cell migration and MYPT1 phosphorylation inhibitor.</p>Formule :C21H18FN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.39Lysine-methotrexate
CAS :<p>Lysine-methotrexate is an anticancer drug. It is an inhibitor of dihydrofolate reductase.</p>Formule :C21H27N9O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.5Type II topoisomerase inhibitor 1
CAS :<p>Potent E. coli DNA gyrase inhibitor (IC50: 1.7 nM), targets Asp73; weak topoisomerase IV inhibitor (IC50: 0.98 μM).</p>Formule :C18H15N3O4Couleur et forme :SolidMasse moléculaire :337.33Ulecaciclib
CAS :<p>Ulecaciclib: oral, BBB-permeable CDK inhibitor; favorable pharmacokinetics; ki: 0.62 μM (CDK2/A), 3 nM (CDK6/D3), 0.2 nM (CDK4/D1), 0.63 μM (CDK7/H).</p>Formule :C25H33FN8SCouleur et forme :SolidMasse moléculaire :496.65LY 207702
CAS :<p>LY 207702, a difluorinated purine nucleoside, exhibits antitumor activity in preclinical models.</p>Formule :C10H12F2N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.24Codon readthrough inducer 1
CAS :<p>Codon readthrough inducer 1 contains pyrimidine bases and shows good readthrough activity.</p>Formule :C15H11N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.26MS0017509
CAS :<p>MS0017509 is a DNA damage repair inhibitor.</p>Formule :C11H10N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :198.22Cdc7-IN-13
CAS :<p>Cdc7-IN-13 (compound 84) is a highly potent CDC7 inhibitor, exhibiting an IC50 value of <1 nM. This compound holds promise for cancer research [1].</p>Formule :C18H20N4O2SCouleur et forme :SolidMasse moléculaire :356.44AZD7762 HCl
CAS :<p>AZD7762 HCl is a checkpoint kinase inhibitor, driving checkpoint abrogation and enhancing DNA-targeted treatment.</p>Formule :C17H20ClFN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.882'-Fluorothymidine
CAS :<p>2'-Fluorothymidine is a selective substrate for TK2, related to thymidine and methyluridine.</p>Formule :C10H13FN2O5Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :260.22GR 144053 trihydrochloride
CAS :<p>platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonist</p>Formule :C18H30Cl3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.82VPC-70619
CAS :<p>VPC-70619: Oral, selective N-Myc inhibitor; blocks cancer growth by hindering N-Myc-Max/DNA binding; well-absorbed.</p>Formule :C16H8ClF3N4OCouleur et forme :SolidMasse moléculaire :364.71Tetrahydrouridine
CAS :<p>Tetrahydrouridine (NSC-112907; THU) is a multidrug resistance modulator.</p>Formule :C9H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :248.23Cdc7-IN-9
CAS :<p>Cdc7-IN-9 can be used for the research of cancer which is a potent inhibitor of Cdc7 [1].</p>Formule :C15H17N5OSCouleur et forme :SolidMasse moléculaire :315.39CID 5951923
CAS :<p>CID 5951923 is an inhibitor of KLF5 transcription factor with an IC50 of 603 nM.</p>Formule :C16H18N2O7SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :382.39DAP-81
CAS :<p>DAP-81, a diaminopyrimidine, inhibits Plk1 (IC50: 0.9 nM), disrupts microtubules, causes monopolar spindles; in preclinical studies.</p>Formule :C25H20N6O4Couleur et forme :SolidMasse moléculaire :468.46CDK4/6-IN-9
CAS :<p>CDK4/6-IN-9 selectively inhibits CDK4/6 (IC50: 905 nM); potential for MM research.</p>Formule :C22H23FN8Couleur et forme :SolidMasse moléculaire :418.47HBV-IN-16
CAS :<p>HBV-IN-16, a quinoline derivative, inhibits HBV cccDNA, key for viral replication (from patent WO2019121357A1).</p>Formule :C22H20ClNO4Couleur et forme :SolidMasse moléculaire :397.85CDK7-IN-12
CAS :<p>CDK7-IN-12 inhibits CDK7 to control transcription and cell cycle, halting tumor growth in vitro/vivo with cancer research potential.</p>Formule :C20H19F3N6Couleur et forme :SolidMasse moléculaire :400.4Phelorphan
CAS :<p>Phelorphan is an inhibitor of enkephalinase.</p>Formule :C20H22N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.46Crisnatol mesylate
CAS :<p>Crisnatol, a potent and selective DNA intercalator, has potential anticancer activity.</p>Formule :C24H27NO5SCouleur et forme :SolidMasse moléculaire :441.54BAY-958
CAS :<p>BAY-958 is a potent and selective inhibitor of PTEFb/CDK9.</p>Formule :C17H16FN5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.4Werner syndrome RecQ helicase-IN-3
CAS :<p>Potent WRN inhibitor, Werner syndrome RecQ helicase-IN-3, is orally active with 0.06 µM IC50; exhibits antiproliferative and anticancer effects.</p>Formule :C31H30ClF3N8O5Couleur et forme :SolidMasse moléculaire :687.07CFM-1
CAS :<p>CFM-1 is an antagonist of the anaphase-promoting complex (APC)-2. It also is a cell cycle and apoptosis regulatory protein (CARP)-1 interaction antagonist.</p>Formule :C12H7BrN2O2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.23Mps-BAY2b
CAS :<p>Mps-BAY2b is a novel MPS1 inhibitor.</p>Formule :C20H23N5OCouleur et forme :SolidMasse moléculaire :349.43Indirubin-5-sulfonate
CAS :<p>Indirubin-5-sulfonate inhibits GSK-3β & CDKs with IC50: 55/35/150/300/65 nM for CDK1/B, 2/A&E, 4/D1, 5/p35.</p>Formule :C16H10N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :342.33RUC-1
CAS :<p>RUC-1 is an αIIbβ3-selective ADP-induced platelet aggregation inhibitor.</p>Formule :C11H15N5OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.33Homocarbonyltopsentin
CAS :<p>Homocarbonyltopsentin: Small molecule, binds TSL2 pentaloops, enhances SMN2 E7 splicing, EC50 16 μM.</p>Formule :C21H14N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :370.36Guanoctine hydrochloride
CAS :<p>Guanoctine hydrochloride has antihypertensive activity.</p>Formule :C9H22ClN3Couleur et forme :SolidMasse moléculaire :207.74NSC 109555 ditosylate
CAS :<p>Chk2 inhibitor,ATP-competitive</p>Formule :C26H32N10O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :580.6614α-Demethylase/DNA Gyrase-IN-2
CAS :<p>14α-Demethylase/DNA Gyrase-IN-2 (Compound 6a) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.</p>Formule :C24H22N4O4Couleur et forme :SolidMasse moléculaire :430.46BDM44768
CAS :<p>BDM44768 is an insulin-degrading enzyme (IDE) inhibitor that acts by inducing glucose intolerance.</p>Formule :C24H22FN5O3Couleur et forme :SolidMasse moléculaire :447.46IRE1α kinase-IN-3
CAS :<p>IRE1α kinase-IN-3 is a potent, ATP-competitive inhibitor of IRE1α (Ki: 480 nM).</p>Formule :C29H32N6O3SCouleur et forme :SolidMasse moléculaire :544.67Mps1-IN-4
CAS :<p>Mps1-IN-4 is a compound that selectively inhibits Monopolar spindle 1 (Mps1), exhibiting antiproliferative properties useful in cancer research.</p>Formule :C26H31F3N6O2Couleur et forme :SolidMasse moléculaire :516.56CDK7-IN-8
CAS :<p>CDK7-IN-8 is a potent inhibitor of CDK7 (IC50: 54.29 nM) and exhibits inhibitory activity against several cancer cells and in vivo tumor models.</p>Formule :C25H38N8O3Couleur et forme :SolidMasse moléculaire :498.62Nucleoside-Analog-2
CAS :<p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>Formule :C9H11N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.212'-Deoxy-L-guanosine
CAS :<p>2'-Deoxy-L-guanosine is a nucleoside that shows antibiotic properties by inhibiting protein synthesis, leading to cell death.</p>Formule :C10H13N5O4Couleur et forme :SolidMasse moléculaire :267.24VE-465
CAS :<p>VE-465 is an inhibitor of Aurora kinase, which involves in multiple mitotic events.</p>Formule :C22H28N8OSCouleur et forme :SolidMasse moléculaire :452.58Antitumor agent-85
<p>Antitumor agent-85 stabilizes G4-DNA with potent anti-tumor effects.</p>Formule :C24H33N7Couleur et forme :SolidMasse moléculaire :419.57XU1
CAS :<p>XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Formule :C12H8N2ODegré de pureté :98.58% - 99.59%Couleur et forme :SolidMasse moléculaire :196.2HBV-IN-15
CAS :<p>HBV-IN-15, a flavone derivative, is a potent cccDNA inhibitor, potentially aiding HBV research.</p>Formule :C24H23ClO6Couleur et forme :SolidMasse moléculaire :442.89PD-1-IN-22
CAS :<p>PD-1-IN-22 is a potent programmed cell death-1 (PD-1)/programmed cell death-ligand 1 (PD-L1) interaction inhibitor(IC50 of 92.3 nM).</p>Formule :C25H25N5O4Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :459.5TC-Mps1-12
CAS :<p>TC-Mps1-12 is an effective and selective inhibitor of monopolar spindle 1 (IC50: 6.4 nM) .</p>Formule :C17H20N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.38CB 3717
CAS :<p>CB 3717 is an enzyme inhibitor, antineoplastic agent, folic acid antagonist.</p>Formule :C24H23N5O6Couleur et forme :SolidMasse moléculaire :477.47Pyrazofurin
CAS :<p>Pyrazofurin, a pyrimidine analogue, blocks cell growth and DNA synthesis by targeting UMP synthase & orotate-phosphoribosyltransferase (IC50: 0.06-0.37 μM).</p>Formule :C9H13N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :259.22IPR-803
CAS :<p>IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity.</p>Formule :C27H23N3O4Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :453.49Datelliptium chloride
CAS :<p>Datelliptium chloride is a DNA-intercalating agent derived from ellipticine. Datelliptium chloride shows anti-tumor activities.</p>Formule :C23H28ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.94Sibrafiban
CAS :<p>Sibrafiban (RO 48-3657), an oral, nonpeptide prodrug, inhibits platelet aggregation as a selective IIb/IIIa antagonist.</p>Formule :C20H28N4O6Couleur et forme :SolidMasse moléculaire :420.46CFI-400437
CAS :<p>CFI-400437 is an ATP-competitive PLK4 inhibitor (IC50: 0.6 nM) and is an indolequinone derivative.</p>Formule :C29H28N6O2Couleur et forme :SolidMasse moléculaire :492.57IACS-4759
CAS :<p>IACS-4759 is a novel potent and selective MTH1 inhibitor with excellent cell permeability and good metabolic stability in microsomes.</p>Formule :C10H17N3O2Couleur et forme :SolidMasse moléculaire :211.26FINDY
CAS :<p>FINDY selectively inhibits DYRK1A at 35 μM IC50, blocking Ser97 autophosphorylation, useful for neurological disorder research.</p>Formule :C16H17NO2S2SiCouleur et forme :SolidMasse moléculaire :347.53CDK-IN-10
CAS :<p>CDK-IN-10 is a cell cycle protein-dependent kinase (CDK) inhibitor with potential anticancer activity for cancer research.</p>Formule :C18H18N4O2Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :322.36SR7826
CAS :<p>SR7826 is a selective LIMK inhibitor.</p>Formule :C22H21N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.43MtTMPK-IN-6
CAS :<p>MtTMPK-IN-6 inhibits M. tuberculosis thymidylate kinase with IC50 of 29 μM, promising for TB research.</p>Formule :C23H25N3O3Couleur et forme :SolidMasse moléculaire :391.46ERCC1-XPF-IN-1
CAS :<p>ERCC1-XPF-IN-1: potent ERCC1-XPF inhibitor (IC50: 0.49 μM), hampers CPD removal, boosts UV toxicity, hinders DNA repair.</p>Formule :C28H32ClN5O2Couleur et forme :SolidMasse moléculaire :506.04CLT-28643
CAS :<p>CLT-28643 is a specific α5β1-Integrin inhibitor that prevents fibrosis in GFS, inhibits tumor growth and angiogenesis, suppresses fibrosis and inflammation.</p>Formule :C19H17N3O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :351.36ML372
CAS :<p>ML372 is a potent and selective SMN Modulator (EC50 = 12 nM, 325% increase inSMN2) with good potency, pharmacokinetics, tolerance, and CNS penetration.</p>Formule :C18H20N2O4SCouleur et forme :SolidMasse moléculaire :360.43BMS-587101
CAS :<p>BMS-587101 is a small molecule antagonist of LFA-1, which can reduce inflammation and joint destruction in the mouse model of arthritis.</p>Formule :C26H20Cl2N4O4SCouleur et forme :SolidMasse moléculaire :555.43PFM03
CAS :<p>PFM03 is a endonuclease inhibitor that specifically blocks Mre11,reduce MRN endonuclease activity, blocking hMRN-mediated endonucleotomy and nuclear exocytosis.</p>Formule :C14H15NO2S2Degré de pureté :99.81% - 99.98%Couleur et forme :SolidMasse moléculaire :293.4c-Myc inhibitor 9
CAS :<p>c-Myc inhibitor 9 (compound 332) with logEC50 ≥6, suppresses tumors in mice, useful for cancer research.</p>Formule :C27H31N5OSCouleur et forme :SolidMasse moléculaire :473.63CDK7-IN-20
<p>CDK7-IN-20: potent, irreversible CDK7 inhibitor, IC50 of 4nM, 206x selectivity vs. other CDKs, potential for ADPKD study.</p>Formule :C30H26N6O3Couleur et forme :SolidMasse moléculaire :518.57Integrin modulator 1
CAS :<p>Integrin modulator 1 is a selective α4β1 integrin agonist (IC50 9.8 nM) that enhances adhesion with EC50 12.9 nM, aiding integrin-dependent studies.</p>Formule :C13H14N2O4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :262.26EMD534085
CAS :<p>EMD534085 is an effective and selective mitotic kinesin-5 inhibitor (IC50: 8 nM).</p>Formule :C25H31F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :476.53Chrysotobibenzyl
CAS :<p>Chrysotobibenzyl from Dendrobium pulchellum stems may trigger cell death in detached cells and hinder lung cancer growth.</p>Formule :C19H24O5Couleur et forme :SolidMasse moléculaire :332.39XMD-17-51
CAS :<p>XMD-17-51 has DCLK1 kinase inhibitory activity, inhibits DCLK1 and cell proliferation, and can be used in lung cancer research.</p>Formule :C21H24N8ODegré de pureté :99.04%Couleur et forme :SoildMasse moléculaire :404.478RK64
CAS :<p>8RK64 is a covalent UCHL1 inhibitor ( IC 50 : 0.32 μM) .</p>Formule :C14H16N8O2SCouleur et forme :SolidMasse moléculaire :360.45,10-Dideazafolic acid
CAS :<p>5,10-Dideazafolic acid is an antileukemic drug.</p>Formule :C21H21N5O6Couleur et forme :SolidMasse moléculaire :439.42CDK7-IN-13
CAS :<p>CDK7-IN-13: A potent pyrimidine-based CDK7 inhibitor, potential for various cancers. See CN114249712A.</p>Formule :C20H23F3N6OSDegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :452.5Indirubin-3'-monoxime-5-sulphonic acid
CAS :<p>Indirubin-3'-monoxime-5-sulphonic acid is a potent and selective inhibitor of GSK-3β, CDK5, and CDK1 with IC50s of 80nM,5 nM, and 7 nM, respectively.</p>Formule :C16H11N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.3410-Deazaaminopterin
CAS :<p>10-Deazaaminopterin is a poly-gamma-glutamyl metabolite of the experimental anticancer drug, a folic acid antagonist, antineoplastic agent enzyme inhibitor.</p>Formule :C20H21N7O5Couleur et forme :SolidMasse moléculaire :439.42Antibacterial agent 89
CAS :<p>Antibacterial agent 89 blocks bacterial transcription and clostridial cytotoxins, inhibiting β'CH-σ interactions.</p>Formule :C21H10Cl2F3NO5SCouleur et forme :SolidMasse moléculaire :516.27P1788
CAS :<p>P1788 is a dihydroorotate dehydrogenase (DHODH) inhibitor that can induce DNA damage [1].</p>Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3Cdc7-IN-7c
CAS :<p>Cdc7-IN-7c (Cdc7 inhibitor-7c) has antitumor activity and has inhibitory effect on liver cancer, lung cancer, kidney cancer, brain cancer and cervical cancer.</p>Formule :C15H17N5OSDegré de pureté :98.19% - 99.22%Couleur et forme :SolidMasse moléculaire :315.39AS-0141
CAS :<p>AS-0141 (Cdc7-IN-6) 是一种有效的 Cdc7 激酶抑制剂 (IC50=4 nM),具有抗肿瘤活性。Cdc7 是一种丝氨酸苏氨酸蛋白激酶酶,在细胞周期中对 DNA 复制的启动至关重要。</p>Formule :C21H22F3N5O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :465.43Anticancer agent 73
CAS :<p>Anticancer agent 73 inhibits TRBP, disrupting TRBP-Dicer, and hinders HCC growth and spread by altering HCC miRNA and protein expression.</p>Formule :C14H15NO4Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :261.27AzddMeC
CAS :<p>AzddMeC (Az-Dcme) is an HIV-1 reverse transcriptase and HIV-1 replication inhibitor with antiretroviral activity.AzddMeC is used in the study of HIV-1 infection</p>Formule :C10H14N6O3Degré de pureté :97.14% - 99.62%Couleur et forme :SolidMasse moléculaire :266.26ITX3
CAS :<p>ITX3 is a specific, non-toxic, active and selective TrioN RhoGEF inhibitor with IC50 of 76 μM.</p>Formule :C22H17N3OSDegré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :371.45Firategrast
CAS :<p>Firategrast (SB 683699) is an orally active and specific α4β1/α4β7 integrin antagonist.Firategrast reduces the transport of lymphocytes into the central nervous</p>Formule :C27H27F2NO6Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :499.5116-9e
CAS :<p>116-9e (MAL2-11B) is an Hsp70 chaperone DNAJA1 inhibitor with antiviral properties, inhibits SV40 replication, and can be used to study cancer drug resistance.</p>Formule :C31H32N2O5Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :512.6D-I03
CAS :<p>D-I03 is a selective RAD52 inhibitor with a Kd of 25.8 µM.</p>Formule :C23H36N6SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :428.64CF-1743
CAS :<p>CF-1743 is an anti-varicella zoster virus nucleoside and inhibits VZV replication.</p>Formule :C22H26N2O5Degré de pureté :99.6% - 99.79%Couleur et forme :SolidMasse moléculaire :398.45Abemaciclib metabolite M20
CAS :<p>Abemaciclib metabolite M20 (CDK4/6-IN-4) 是 Abemaciclib 的活性代谢物。 Abemaciclib metabolite M20 是一种特异性 CDK4/6 抑制剂,可用于癌症治疗的相关研究。</p>Formule :C27H32F2N8ODegré de pureté :98.1% - 99.08%Couleur et forme :SolidMasse moléculaire :522.59hDHODH-IN-7
CAS :<p>hDHODH-IN-7 (DHODH-IN-9) is a nitrogen-containing analog and is a human dihydrorotatory dehydrogenase inhibitor.</p>Formule :C21H23FN4ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :366.43DS18561882
CAS :<p>DS18561882: Potent MTHFD2 inhibitor (IC50=0.0063), inhibits MTHFD1 (IC50=0.57), good oral kinetics.</p>Formule :C28H31F3N4O6SDegré de pureté :98.19% - >99.99%Couleur et forme :SolidMasse moléculaire :608.63CD532
CAS :<p>CD532: Potent Aurora A inhibitor, IC50=45 nM, blocks kinase activity, degrades MYCN, interacts with AURKA, studies cancer.</p>Formule :C26H25F3N8ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :522.52GKI-1
CAS :<p>GKI-1, a GWL kinase inhibitor: IC50 - 4.9 µM for hGWLFL, 2.5 µM for hGWL-KinDom, 11 µM for ROCK1; weak on PKA.</p>Formule :C15H12ClN3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :269.73Elarofiban
CAS :<p>Elarofiban(RWJ-53308) is a novel and orally active GPIIb/IIIa antagonist.</p>Formule :C22H32N4O4Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :416.51CDK9-IN-10
CAS :<p>CDK9-IN-10 is a potent CDK9 inhibitor and the ligand for the PROTAC CDK9 degrader-2.</p>Formule :C22H16O5Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :360.36Galocitabine
CAS :<p>Galocitabine (Neofrutulon), a thymidylate synthase inhibitor, is used potentially for the treatment of cancer.</p>Formule :C19H22FN3O8Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :439.39Caracemide
CAS :<p>Caracemide (NSC-253272) inhibits the enzyme ribonucleotide reductase of Escherichia coli. Caracemide can be used in anticancer studies.</p>Formule :C6H11N3O4Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :189.176RK73
CAS :<p>6RK73 is a covalent irreversible and specific UCHL1 inhibitor (IC50: 0.23 µM). 6RK73 shows almost no inhibition of UCHL3 (IC50: 236 µM).</p>Formule :C13H17N5O2SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :307.37GS-6620 PM
CAS :<p>GS-6620 PM, oral Hep C polymerase inhibitor prodrug, is a potent GS-6620 derivative with limited activity against other viruses.</p>Formule :C13H15N5O4Degré de pureté :98.52% - 98.7%Couleur et forme :SolidMasse moléculaire :305.29CHK1-IN-3
CAS :<p>CHK1-IN-3 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM).</p>Formule :C20H23N9ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :405.46
