
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(115 produits)
- CDK(547 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(46 produits)
- Dynamine(27 produits)
- Ferroptose(227 produits)
- HSP(180 produits)
- Intégrine(275 produits)
- Kinésine(87 produits)
- LIM Kinase(21 produits)
- Microtubules associés(273 produits)
- PKC(127 produits)
- PLK(25 produits)
- ROCK(61 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(77 produits)
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3920 produits trouvés pour "Cycle cellulaire/point de contrôle"
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Laromustine
CAS :Laromustine (VNP40101M) is a sulfonyl hydrolysis alkylation prodrug for cancer treatment with significant anticancer activity, inhibiting thioredoxin reductase.Formule :C6H14ClN3O5S2Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :307.78WF-536 Hydrochloride
CAS :WF-536 Hydrochloride, a novel inhibitor of ROCK, inhibits tumour metastasis in some animal models.Formule :C14H16ClN3OCouleur et forme :SolidMasse moléculaire :277.75Beaucage reagent
CAS :Beaucage reagent, which is found to be effective in causing DNA cleavage.Formule :C7H4O3S2Degré de pureté :98.50%Couleur et forme :White To Off-White PowderMasse moléculaire :200.23CBL 0100 free base
CAS :CBL0100 is an inhibitor of viral transcriptional elongation, blocking both HIV-1 replication and reactivation.Formule :C24H26N2O2Degré de pureté :98.18% - 98.86%Couleur et forme :SolidMasse moléculaire :374.48APC 366
CAS :APC 366: Mast cell tryptase inhibitor, Ki 7.1 μM. Reduces EAR, LAR, BHR in allergic asthma (sheep model).Formule :C22H28N6O4Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :440.5PF-2771
CAS :PF-2771: potent CENP-E inhibitor, IC50 of 16.1 nM, used in cancer treatment.Formule :C29H36ClN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :554.08GW8510
CAS :GW8510 is a CDK2 and RRM2 inhibitor that affects DNA synthesis and antiproliferation in tumor cells. In mammalian aging models, GW851 prolongs lifespan.Formule :C21H15N5O3S2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :449.51Werner syndrome RecQ helicase-IN-4
CAS :Werner syndrome RecQ helicase-IN-4 is a WRN inhibitor with anticancer and anti-proliferative activity, used in colorectal and gastric cancer research.Formule :C32H33F3N8O5Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :666.65IRE1α kinase-IN-7
CAS :IRE1α kinase-IN-7 is a chemical compound functioning as an inhibitor of IRE1α kinase, primarily utilized in the research of diseases related to endoplasmicFormule :C28H25F3N6OCouleur et forme :SolidMasse moléculaire :518.53CH-1504
CAS :CH-1504, dihydrofolate reductase (DHFR) inhibitor, is used potentially for the treatment of rheumatoid arthritis.Formule :C23H23N5O5Couleur et forme :SolidMasse moléculaire :449.46IDD388
CAS :IDD388 is a selective and potent aldose reductase (ALR2) inhibitor with antitumor activity that inhibits the ALR1 receptor.Formule :C16H12BrClFNO4Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :416.63MMV688844
CAS :MMV688844 inhibits M. abscessus DNA cyclooxygenase (IC50: 2μM) and has MIC50 of 12μM on strain bamboo; useful in antimicrobial studies.Formule :C23H25ClN4O2Couleur et forme :SolidMasse moléculaire :424.92CDK7-IN-10
CAS :CDK7-IN-10: CDK7 inhibitor, IC50<100 nM, may hinder cell growth, induce apoptosis. (Patent WO2021016388A1, I-1)Formule :C29H35N7O3Couleur et forme :SolidMasse moléculaire :529.63Binucleine 2
CAS :Binucleine 2: Drosophila Aurora B kinase inhibitor (Ki=0.36μM), dose-dependent, minimal effect on human/X. laevis kinases, disrupts mitosis in fly cells.Formule :C13H11ClFN5Couleur et forme :SolidMasse moléculaire :291.71CDK7-IN-16
CAS :CDK7-IN-16, a potent CDK7 inhibitor (IC50: 1-10 nM), is used in cancer research with transcription defects.Formule :C19H21F3N6O2SCouleur et forme :SolidMasse moléculaire :454.47DHX9-IN-1
CAS :DHX9-IN-1 is a potent ATP-dependent RNA helicase A (DHX9) inhibitor, exhibiting an IC50 of 9.45 nM and demonstrating antitumor activity [1].Formule :C21H21F2N5O3SCouleur et forme :SolidMasse moléculaire :461.49Ref: TM-T82569
1mg205,00€5mg528,00€1mL*10mM (DMSO)537,00€10mg782,00€25mg1.161,00€50mg1.558,00€100mg2.322,00€CAY10746
CAS :CAY10746 selectively inhibits ROCK I/II with IC50s: 0.014/0.003 μM, useful for diabetic retinopathy research.Formule :C26H23N3O5Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :457.48Ref: TM-T36196
2mg34,00€5mg54,00€1mL*10mM (DMSO)54,00€10mg86,00€25mg172,00€50mg260,00€100mg411,00€200mg552,00€RHI002-Me
CAS :RHI002-Me is a methylated derivative of RHI002, a selective inhibitor of human RNaseH2.Formule :C18H19N3O2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :373.49Synucleozid
CAS :Synucleozid is a potent the SNCA mRNA inhibitor that encodes α-synuclein protein (IC50=1.5 μM), has the potential for the investigation of Parkinson’s disease.Formule :C22H20N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.43WNK1-IN-1
CAS :WNK1-IN-1, a WNK1 inhibitor (IC50: 1.6 μM), also inhibits OSR1 phosphorylation (IC50: 4.3 μM), used in blood pressure and cancer research.Formule :C13H15BrCl2N2O4SDegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :446.14Ref: TM-T73295
1mg71,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg236,00€25mg485,00€50mg782,00€100mg1.305,00€DENV-IN-4
CAS :DENV-IN-4: Effective DENV inhibitor (EC50=4.79 μM), low toxicity (CC50>100 μM), and strong selectivity (SI>20.9); suppresses DENV2 and RdRp.Formule :C28H32N4O4SiCouleur et forme :SolidMasse moléculaire :516.66Valategrast hydrochloride
CAS :Valategrast hydrochloride (R411), a dual antagonist of integrin α4β1 (VLA-4), is used for the potential treatment of asthma.Formule :C30H33Cl4N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.41CDK9-IN-14
CAS :CDK9-IN-14: Potent CDK9 inhibitor, IC50=6.92 nM, effective on MV-4-11 cells and in vivo tumors, low toxicity, minimal side effects.Formule :C21H23F2N3O4Couleur et forme :SolidMasse moléculaire :419.42PF-4950834
CAS :PF-4950834, a ATP-competitive, selective Rho kinase inhibitor, provides therapeutic benefits in chronic inflammatory diseases.Formule :C21H19N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.39PV-1115
CAS :PV-1115 is an effective and highly selective inhibitor of the Chk2.Formule :C20H19N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.41ROCK-IN-D2
CAS :ROCK-IN-D2 is an effective and selective inhibitor of ROCK.Formule :C22H28N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.5HIV-1 inhibitor-43
CAS :HIV-1 Inhibitor-43 suppresses HIV-1, with EC50: 21.3 nM (Y188L), 6.2 nM (K103N-Y181C), <0.7 nM (K103N/Y181C), and lowers HIV RNA/p24 protein.Formule :C24H21ClN2O4SCouleur et forme :SolidMasse moléculaire :468.95Cylindrospermopsin
CAS :Cylindrospermopsin: a toxic cyanobacterial uracil derivative, disrupts protein/glutathione synthesis in hepatocytes, and is genotoxic.Formule :C15H21N5O7SCouleur et forme :SolidMasse moléculaire :415.42(Rac)-Managlinat dialanetil
CAS :Managlinat dialanetil, an orally available and potent inhibitor of fructose 1,6-bisphosphatase (FBPase) used in research 2 type diabetes.Formule :C21H33N4O6PSDegré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :500.55DHODH-IN-12
CAS :DHODH-IN-12 is a leflunomide derivative and a weak dihydrorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.07.Formule :C10H9N3O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :203.2Ref: TM-T11021
1mg73,00€1mL*10mM (DMSO)122,00€5mg149,00€10mg213,00€25mg319,00€50mg447,00€100mg610,00€200mg823,00€FAK/aurora kinase-IN-1
CAS :FAK/aurora kinase-IN-1, a dual inhibitor of FAK and aurora kinase, has IC50 values of 6.61 nM and 0.91 nM respectively, and demonstrates anticancer effects (WO2018019252A1; compound 11) [1].Formule :C23H24ClN7O3Couleur et forme :SolidMasse moléculaire :481.93CGP 53353
CAS :CGP 53353 (DAPH-7) is a PKC inhibitor with inhibitory effects on PKCβII and PKCβI and can be used to study atherosclerosis.Formule :C20H13F2N3O2Degré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :365.33MDK6204
CAS :MDK6204 is a selective inhibitor of CLK1 and CLK2.Formule :C20H20N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.41P18IN003
CAS :P18IN003 is a selective and effective p18(INK4C) inhibitor that inhibits the activity of p18 protein and can be used to study in vitro expansion ofFormule :C17H16N2O3Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :296.32JFN05510
CAS :Compound: 3'-O-tert-BDMS-5'-O-DMT-N2-IBG 2'-CE phosphoramidite; has anticancer properties and activates enzymes.Formule :C50H68N7O9PSiCouleur et forme :SolidMasse moléculaire :970.18Zalunfiban
CAS :RUC-4 is an aIIb 3 antagonist. It is also used for prehospital therapy of myocardial infarction.Formule :C16H18N8O2SCouleur et forme :SolidMasse moléculaire :386.435-Aminouridine
CAS :5-Aminouridine (4-Chloro-2-isopropyl-5-methylphenol(chlorothymol)) modifies nucleobases and is incorporated into the target DNA.Formule :C9H13N3O6Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :259.22Zelpolib
CAS :Zelpolib is a specific inhibitor of DNA polymerase δ (Pol δ), inhibiting DNA replication. antiproliferative.Formule :C22H21N3O5S2Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :471.55Enocitabine
CAS :Enocitabine is a nucleoside analog.Formule :C31H55N3O6Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :565.78Fosteabine
CAS :Fosteabine is an oral and prodrug analog of cytarabine. It is resistant to deoxycytidine deaminase.Formule :C27H50N3O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :575.67Apricitabine
CAS :Apricitabine (SPD754) is a highly selective and orally active HIV-1 reverse transcriptase inhibitor (Ki=0.08 μM), the (-) enantiomer of 2′-deoxy-3′-oxy-4′-Formule :C8H11N3O3SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :229.26Ref: TM-T14313
1mg283,00€5mg507,00€1mL*10mM (DMSO)592,00€10mg628,00€25mg962,00€50mg1.601,00€100mg2.682,00€PD 130883
CAS :PD 130883 is a potent lipophilic quinazoline antifolate.Formule :C18H15N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.34Aurora Kinases-IN-2
CAS :Aurora Kinases-IN-2 (12Aj) hinders Aurora A/B kinases (IC50: 90/152 nM), used in cancer studies.Formule :C22H18ClN5O3Couleur et forme :SolidMasse moléculaire :435.86Syntelin
CAS :Syntelin: a selective CENP-E inhibitor with an IC50 of 160 nM; distinct from GSK923295, effective on resistant mutants.Formule :C21H20N6O2S3Couleur et forme :SolidMasse moléculaire :484.62DNA Gyrase-IN-5
CAS :DNA Gyrase-IN-5 is a potent inhibitor of DNA gyrase (IC50: 0.10 μM) and has an antibacterial effect on both wild-type and drug-resistant strains.Formule :C25H15BrClN5Couleur et forme :SolidMasse moléculaire :500.78LSN 3213128
CAS :LSN 3213128: a potent oral antifolate targeting AICARFT with IC50s of 16 nM (enzyme) and 19 nM (cells), offers anti-tumor effects.Formule :C17H16FN3O4S2Couleur et forme :SolidMasse moléculaire :409.45Myt1-IN-1
CAS :Myt1-IN-1 has anticancer effects that is a potent inhibitor of Myt1 with an IC 50 of <10 nM [1].Formule :C16H15ClN4O2Couleur et forme :SolidMasse moléculaire :330.77PFM03
CAS :PFM03 is a endonuclease inhibitor that specifically blocks Mre11,reduce MRN endonuclease activity, blocking hMRN-mediated endonucleotomy and nuclear exocytosis.Formule :C14H15NO2S2Degré de pureté :99.81% - 99.98%Couleur et forme :SolidMasse moléculaire :293.4Atuveciclib S-Enantiomer
CAS :Atuveciclib S-Enantiomer is a (S)-form of BAY-1143572; a potent, selective CDK9 inhibitor with an IC50 of 16 nM.Formule :C18H18FN5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.43RP-106
CAS :RP-106 is an ATP-competitive inhibitor of CDK5/p25, CDK1/cyclin B, and GSK-3.Formule :C17H19N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :281.35A 65282
CAS :A 65282: antibacterial isothiazoloquinolone, inhibits P4-unknotting, causes DNA breaks via topoisomerase II.Formule :C17H16F2N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.4CDK8-IN-10
CAS :CDK8-IN-10 is a selective and potent inhibitor of cell cycle protein-dependent kinase (CDK8) (IC50: 8.25 nM) that can be used to study cancer.Formule :C25H15ClF3N5O3Couleur et forme :SolidMasse moléculaire :525.87CLT-28643
CAS :CLT-28643 is a specific α5β1-Integrin inhibitor that prevents fibrosis in GFS, inhibits tumor growth and angiogenesis, suppresses fibrosis and inflammation.Formule :C19H17N3O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :351.36BSJ-01-175
CAS :BSJ-01-175: Selective, potent covalent inhibitor of CDK12/13, targets cancer cells, inhibits phosphorylated RNA polymerase II, downregulates CDK12 genes.Formule :C30H33ClN6O2Couleur et forme :SolidMasse moléculaire :545.08DHODH-IN-24
CAS :DHODH-IN-24 (compound 16) serves as a powerful inhibitor of human dihydroorotate dehydrogenase (DHODH), exhibiting an IC50 value of 91 nM [1].Formule :C26H26N4Couleur et forme :SolidMasse moléculaire :394.51DENV-IN-7
CAS :DENV-IN-7, a flavone analog, inhibits dengue virus at 70 nM EC50 with low toxicity to normal cells.Formule :C24H22O8Couleur et forme :SolidMasse moléculaire :438.43AZD7762 HCl
CAS :AZD7762 HCl is a checkpoint kinase inhibitor, driving checkpoint abrogation and enhancing DNA-targeted treatment.Formule :C17H20ClFN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.88VPC-70619
CAS :VPC-70619: Oral, selective N-Myc inhibitor; blocks cancer growth by hindering N-Myc-Max/DNA binding; well-absorbed.Formule :C16H8ClF3N4OCouleur et forme :SolidMasse moléculaire :364.71P1788
CAS :P1788 is a dihydroorotate dehydrogenase (DHODH) inhibitor that can induce DNA damage [1].Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3Antibacterial agent 89
CAS :Antibacterial agent 89 blocks bacterial transcription and clostridial cytotoxins, inhibiting β'CH-σ interactions.Formule :C21H10Cl2F3NO5SCouleur et forme :SolidMasse moléculaire :516.27CID 5951923
CAS :CID 5951923 is an inhibitor of KLF5 transcription factor with an IC50 of 603 nM.Formule :C16H18N2O7SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :382.39BAY-958
CAS :BAY-958 is a potent and selective inhibitor of PTEFb/CDK9.Formule :C17H16FN5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.4Eg5 Inhibitor V, trans-24
CAS :Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.Formule :C26H21N3O3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :423.46Ref: TM-T11155
1mg96,00€5mg193,00€1mL*10mM (DMSO)215,00€10mg289,00€25mg469,00€50mg642,00€100mg858,00€200mg1.153,00€AS-136A
CAS :AS-136A is an orally active MV RdRp inhibitor with antiviral activity that inhibits measles virus and blocks viral RNA synthesis.Formule :C17H19F3N4O3SDegré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :416.42Ref: TM-T62160
1mg215,00€5mg537,00€1mL*10mM (DMSO)590,00€10mg802,00€25mg1.369,00€50mg1.783,00€100mg2.395,00€CDK5 inhibitor 20-223
CAS :CDK5 inhibitor 20-223 is a potent CDK2/CDK5 inhibitor,anti-Colorectal Cancer (CRC), inhibiting cell migration and inducing cell cycle arrest.Formule :C19H19N3OCouleur et forme :SolidMasse moléculaire :305.37AnnH31
CAS :AnnH31 is a potent Dyrk1A inhibitor with an IC50 value of 81 nM.AnnH31 inhibits MAO-A with an IC50 of 3.2 μM.AnnH31 can be used as a probe to confirm theFormule :C15H13N3ODegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :251.28hDHODH-IN-4
CAS :hDHODH-IN-4, a potent DHODH inhibitor, has a pIC50 of 7.8 and blocks measles virus replication with a pMIC50 of 8.8.Formule :C21H24N4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :364.44SC-203885
CAS :SC-203885 is a checkpoint kinase 2 inhibitor.Formule :C15H13N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.3Indirubin-3'-monoxime-5-sulphonic acid
CAS :Indirubin-3'-monoxime-5-sulphonic acid is a potent and selective inhibitor of GSK-3β, CDK5, and CDK1 with IC50s of 80nM,5 nM, and 7 nM, respectively.Formule :C16H11N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.34Kira8 Hydrochloride
CAS :Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formule :C31H30Cl2N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :637.58Datelliptium chloride
CAS :Datelliptium chloride is a DNA-intercalating agent derived from ellipticine. Datelliptium chloride shows anti-tumor activities.Formule :C23H28ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.94CDK7-IN-13
CAS :CDK7-IN-13 (compound 1) is an effective CDK7 inhibitor for investigating cancers associated with transcriptional dysregulation.Formule :C20H23F3N6OSDegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :452.55,10-Dideazafolic acid
CAS :5,10-Dideazafolic acid is an antileukemic drug.Formule :C21H21N5O6Couleur et forme :SolidMasse moléculaire :439.42Pyrazofurin
CAS :Pyrazofurin, a pyrimidine analogue, blocks cell growth and DNA synthesis by targeting UMP synthase & orotate-phosphoribosyltransferase (IC50: 0.06-0.37 μM).Formule :C9H13N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :259.22IPR-803
CAS :IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity.Formule :C27H23N3O4Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :453.49TC-Mps1-12
CAS :TC-Mps1-12 is an effective and selective inhibitor of monopolar spindle 1 (IC50: 6.4 nM) .Formule :C17H20N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.38CFI-400437
CAS :CFI-400437 is an ATP-competitive PLK4 inhibitor (IC50: 0.6 nM) and is an indolequinone derivative.Formule :C29H28N6O2Couleur et forme :SolidMasse moléculaire :492.572-Keto-D-galactose
CAS :2-Keto-D-galactose inhibits DNA synthesis and inhibits the proliferation of in vitro grown Ehrlich ascites tumor cells.Formule :C6H10O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :178.14CAP-53194
CAS :CAP-53194 is a selective Plk1 inhibitor.Formule :C21H14N6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.378RK64
CAS :8RK64 is a covalent UCHL1 inhibitor ( IC 50 : 0.32 μM) .Formule :C14H16N8O2SCouleur et forme :SolidMasse moléculaire :360.4GSK-3008348
CAS :GSK-3008348 is an antagonist of integrin alpha(v)beta6.Formule :C29H37N5O2Degré de pureté :99.547%Couleur et forme :SolidMasse moléculaire :487.64Mivobulin Isethionate
CAS :Mivobulin, a tubulin inhibitor (CI-980), may treat glioma, melanoma, prostate, and ovarian cancer, targeting colchicine-binding site.Formule :C19H25N5O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.5Picoplatin
CAS :Picoplatin, an anti-cancer agent overcoming platinum resistance, alkylates DNA to block replication, transcription, and induce apoptosis.Formule :C6H10Cl2N2PtDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.14HHL-6
CAS :HHL-6 is a c-Fos and BDNF protein expression modulator.Formule :C19H26N2O3Couleur et forme :SolidMasse moléculaire :330.42Metralindole HCl
CAS :Metralindole is a reversible monoamine oxidase A (RIMA) inhibitor, it was investigated as a potential antidepressant.Formule :C15H18ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :291.78HR22C16
CAS :HR22C16 is an effective, selective, and cell-permeable mitotic kinesin Eg5 inhibitor.Formule :C23H23N3O3Couleur et forme :SolidMasse moléculaire :389.45HIPP
CAS :HIPP is a highly selective inhibitor of antineoplastic CtBP.Formule :C9H9NO3Couleur et forme :SolidMasse moléculaire :179.17NPD9948
CAS :NPD9948 is a competitive inhibitor of MTH1.Formule :C13H14N6Couleur et forme :SolidMasse moléculaire :254.29LDN-209929
CAS :LDN-209929 2HCl is a potent and selective inhibitor of haspin kinase.Formule :C17H17ClN2OSCouleur et forme :SolidMasse moléculaire :332.85Chrysotobibenzyl
CAS :Chrysotobibenzyl from Dendrobium pulchellum stems may trigger cell death in detached cells and hinder lung cancer growth.Formule :C19H24O5Couleur et forme :SolidMasse moléculaire :332.39DYRKi
CAS :DYRKi is a nontoxic, DYRK1-selective inhibitor.Formule :C20H13F3N4O2SCouleur et forme :SolidMasse moléculaire :430.4BIPM
CAS :BIPM inhibits ROCK2, alters SH-SY5Y cell migration, actin fibers, neurite length, and reduces cofilin phosphorylation.Formule :C23H22N2O3Couleur et forme :SolidMasse moléculaire :374.43REV7/REV3L-IN-1
CAS :REV7/REV3L-IN-1 is a inhibitor of REV7/REV3L interaction(IC50 of 78 μM),Formule :C19H21N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.45NSC47924
CAS :NSC47924 is a laminin receptor (LR) inhibitor.Formule :C18H17NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.33AB-182
CAS :AB-182 is an aziridine derivative with antitumor activity.Formule :C11H22N3O4PCouleur et forme :SolidMasse moléculaire :291.28Ro 43-5054
CAS :Ro 43-5054 is a small molecular, noncyclic peptidomimetic inhibitor.Formule :C24H27N5O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :497.5ROCK-IN-D1
CAS :ROCK-IN-D1 is an effective and selective inhibitor of ROCK.Formule :C22H27N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.55Integrin modulator 1
CAS :Integrin modulator 1 is a selective α4β1 integrin agonist (IC50 9.8 nM) that enhances adhesion with EC50 12.9 nM, aiding integrin-dependent studies.Formule :C13H14N2O4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :262.26SNX2-1-108
CAS :SNX2-1-108 is a selective CDK8 and CDK19 inhibitor.Formule :C21H16N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.38CDK7-IN-20
CDK7-IN-20: potent, irreversible CDK7 inhibitor, IC50 of 4nM, 206x selectivity vs. other CDKs, potential for ADPKD study.Formule :C30H26N6O3Couleur et forme :SolidMasse moléculaire :518.57
