
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(115 produits)
- CDK(547 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(46 produits)
- Dynamine(27 produits)
- Ferroptose(227 produits)
- HSP(180 produits)
- Intégrine(275 produits)
- Kinésine(87 produits)
- LIM Kinase(21 produits)
- Microtubules associés(273 produits)
- PKC(127 produits)
- PLK(25 produits)
- ROCK(61 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(77 produits)
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3920 produits trouvés pour "Cycle cellulaire/point de contrôle"
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LIMK-IN-14
CAS :LIMK-IN-14 is an effective and selective inhibitor of LIMK.Formule :C22H27N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :437.49Denopterin
CAS :Denopterin is an antineoplastic agent.Formule :C21H23N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.45SR7826
CAS :SR7826 is a selective LIMK inhibitor.Formule :C22H21N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.431-Acetyl-3-o-toluyl-5-fluorouracil
CAS :1-Acetyl-3-o-toluyl-5-fluorouracil is a potent antineoplastic agent.Formule :C14H11FN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :290.25c-Myc inhibitor 9
CAS :c-Myc inhibitor 9 (compound 332) with logEC50 ≥6, suppresses tumors in mice, useful for cancer research.Formule :C27H31N5OSCouleur et forme :SolidMasse moléculaire :473.63Rabacfosadine succinate
CAS :Rabacfosadine succinate is the acyclic nucleoside phosphonate PMEG double prodrug.Formule :C25H41N8O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :644.623Thiamiprine
CAS :Thiamiprine is an agent with the activity of antineoplastic.Formule :C9H8N8O2SCouleur et forme :SolidMasse moléculaire :292.28CDK4/6-IN-12
CAS :CDK4/6-IN-12 inhibits CDK4/6 with IC50s of 592.3 nM & 3090 nM, useful in cancer research.Formule :C12H10N6Couleur et forme :SolidMasse moléculaire :238.25Meturedepa
CAS :Meturedepa is an antineoplastic agent.Formule :C11H22N3O3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.28Digeranyl bisphosphonate
CAS :Digeranyl bisphosphonate (DGBP) is a potent geranylgeranyl pyrophosphate (GGPP) synthase inhibitor that inhibits geranyl pyrophosphorylation of Rac1.DigeranylFormule :C21H34Na4O6P2Degré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :536.4BzDANP
CAS :BzDANP is a modulator of pre-miR-29a maturation by Dicer.Formule :C18H24N6Couleur et forme :SolidMasse moléculaire :324.42L 703014
CAS :L 703014 is an antagonist of the fibrinogen receptor.Formule :C24H34N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.55SEC inhibitor KL-2
CAS :KL-2: potent SEC inhibitor, selectively disrupts AFF4-CCNT1, dose-dependent, Ki: 1.50 μM.Formule :C17H13ClFNO3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :333.74AM-TS23
CAS :AM-TS23 is used as a DNA polymerase lambda and beta inhibitor.Formule :C17H12N2O3S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.48Cdc7-IN-5
CAS :Cdc7-IN-5: potent Cdc7 serine-threonine kinase inhibitor, critical for starting DNA replication.Formule :C25H23N3O5Degré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :445.47Ref: TM-T10727
1mg96,00€5mg227,00€1mL*10mM (DMSO)250,00€10mg376,00€25mg620,00€50mg847,00€100mg1.169,00€ML366
CAS :ML366 is a Vibrio cholerae Quorum Sensing inhibitor Acting via the LuxO response regulator.Formule :C17H19N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.35HBX28258
CAS :HBX28258, a human USP7 inhibitor, binds covalently and selectively deactivates USP7 in colon cancer and kidney cells.Formule :C26H30ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :435.99BMS-587101
CAS :BMS-587101 is a small molecule antagonist of LFA-1, which can reduce inflammation and joint destruction in the mouse model of arthritis.Formule :C26H20Cl2N4O4SCouleur et forme :SolidMasse moléculaire :555.43JNJ-9676
CAS :JNJ-9676 is an orally active inhibitor of the coronavirus membrane protein, thereby blocking viral assembly and release.coronavirus and SARS-CoV.Formule :C28H21F2N5O2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :497.5Ref: TM-T205924
1mg137,00€5mg330,00€1mL*10mM (DMSO)354,00€10mg532,00€25mg1.108,00€50mg1.738,00€100mg2.592,00€CDK4/6-IN-7
CAS :CDK4/6-IN-7 is an oral, potent CDK4/6 inhibitor with IC50s of 1.58/4.09 nM, crucial for breast cancer studies.Formule :C18H18ClN5O3Couleur et forme :SolidMasse moléculaire :387.82OXA-06 Dihydrochloride
CAS :OXA-06 Dihydrochloride is a PANC-1 cell migration and MYPT1 phosphorylation inhibitor.Formule :C21H18FN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.39ML372
CAS :ML372 is a potent and selective SMN Modulator (EC50 = 12 nM, 325% increase inSMN2) with good potency, pharmacokinetics, tolerance, and CNS penetration.Formule :C18H20N2O4SCouleur et forme :SolidMasse moléculaire :360.4310-Deazaaminopterin
CAS :10-Deazaaminopterin is a poly-gamma-glutamyl metabolite of the experimental anticancer drug, a folic acid antagonist, antineoplastic agent enzyme inhibitor.Formule :C20H21N7O5Couleur et forme :SolidMasse moléculaire :439.42LY 207702
CAS :LY 207702, a difluorinated purine nucleoside, exhibits antitumor activity in preclinical models.Formule :C10H12F2N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.24Codon readthrough inducer 1
CAS :Codon readthrough inducer 1 contains pyrimidine bases and shows good readthrough activity.Formule :C15H11N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.26MS0017509
CAS :MS0017509 is a DNA damage repair inhibitor.Formule :C11H10N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :198.22ERCC1-XPF-IN-1
CAS :ERCC1-XPF-IN-1: potent ERCC1-XPF inhibitor (IC50: 0.49 μM), hampers CPD removal, boosts UV toxicity, hinders DNA repair.Formule :C28H32ClN5O2Couleur et forme :SolidMasse moléculaire :506.04Levofloxacin sodium
CAS :Levofloxacin sodium: synthetic antibacterial, stops DNA replication by inhibiting bacterial DNA gyrase.Formule :C18H20FN3NaO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :384.3632'-Fluorothymidine
CAS :2'-Fluorothymidine is a selective substrate for TK2, related to thymidine and methyluridine.Formule :C10H13FN2O5Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :260.22Ref: TM-T19101
1mg50,00€1mL*10mM (DMSO)101,00€5mg105,00€10mg161,00€25mg276,00€50mg416,00€100mg625,00€200mg837,00€DHFR-IN-5
CAS :DHFR-IN-5: potent, oral DHFR inhibitor, Ki 0.54 nM against mutant P. falciparum, anti-malarial.Formule :C18H24N4O4Couleur et forme :SolidMasse moléculaire :360.41Nucleoside-Analog-2
CAS :Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.Formule :C9H11N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.21MtTMPK-IN-6
CAS :MtTMPK-IN-6 inhibits M. tuberculosis thymidylate kinase with IC50 of 29 μM, promising for TB research.Formule :C23H25N3O3Couleur et forme :SolidMasse moléculaire :391.46Tetrahydrouridine
CAS :Tetrahydrouridine (NSC-112907; THU) is a multidrug resistance modulator.Formule :C9H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :248.23Cdc7-IN-4
CAS :Cdc7-IN-4 is a potent inhibitor of Cdc7 kinase.Formule :C22H24F3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.45Valategrast
CAS :Valategrast: potent, oral dual α4β1/α4β7 integrin antagonist, may treat COPD and asthma.Formule :C30H32Cl3N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :604.95Phelorphan
CAS :Phelorphan is an inhibitor of enkephalinase.Formule :C20H22N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.46CFM-1
CAS :CFM-1 is an antagonist of the anaphase-promoting complex (APC)-2. It also is a cell cycle and apoptosis regulatory protein (CARP)-1 interaction antagonist.Formule :C12H7BrN2O2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.23FINDY
CAS :FINDY selectively inhibits DYRK1A at 35 μM IC50, blocking Ser97 autophosphorylation, useful for neurological disorder research.Formule :C16H17NO2S2SiCouleur et forme :SolidMasse moléculaire :347.53IACS-4759
CAS :IACS-4759 is a novel potent and selective MTH1 inhibitor with excellent cell permeability and good metabolic stability in microsomes.Formule :C10H17N3O2Couleur et forme :SolidMasse moléculaire :211.26XL-188
CAS :XL-188: Potent, selective USP7 inhibitor, IC50 = 193 nM (domain), 90 nM (full). Boosts p53, p21; degrades HDM2. Unique among DUB inhibitors.Formule :C32H42N6O4Couleur et forme :SolidMasse moléculaire :574.71RUC-1
CAS :RUC-1 is an αIIbβ3-selective ADP-induced platelet aggregation inhibitor.Formule :C11H15N5OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.33Homocarbonyltopsentin
CAS :Homocarbonyltopsentin: Small molecule, binds TSL2 pentaloops, enhances SMN2 E7 splicing, EC50 16 μM.Formule :C21H14N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :370.36Guanoctine hydrochloride
CAS :Guanoctine hydrochloride has antihypertensive activity.Formule :C9H22ClN3Couleur et forme :SolidMasse moléculaire :207.74Sibrafiban
CAS :Sibrafiban (RO 48-3657), an oral, nonpeptide prodrug, inhibits platelet aggregation as a selective IIb/IIIa antagonist.Formule :C20H28N4O6Couleur et forme :SolidMasse moléculaire :420.46IRE1α kinase-IN-3
CAS :IRE1α kinase-IN-3 is a potent, ATP-competitive inhibitor of IRE1α (Ki: 480 nM).Formule :C29H32N6O3SCouleur et forme :SolidMasse moléculaire :544.67Nucleoside-Analog-1
CAS :Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.Formule :C9H9N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.2HBV-IN-21
CAS :HBV-IN-21 inhibits HBV DNA replication (IC50: 2.2 μM) and binds HBV capsid protein well (KD: 60.0 μM).Formule :C17H17FN4OS2Couleur et forme :SolidMasse moléculaire :376.47L-Fd4A
CAS :L-Fd4A (compound 36) is an adenine derivative with anti-HIV (EC50=1.5μM) and anti-HBV (EC50=1.7μM) effects, low cytotoxicity.Formule :C10H10FN5O2Couleur et forme :SolidMasse moléculaire :251.22I-138
CAS :I-138 is an orally active and reversible inhibitor of USP1-UAF1.I-138 induces mono-ubiquitination of FANCD2 and PCNA and inhibits USP1 auto-cleavage in cells.Formule :C26H23F3N6ODegré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :492.5Ref: TM-T73560
1mg170,00€5mg349,00€1mL*10mM (DMSO)384,00€10mg492,00€25mg707,00€50mg982,00€100mg1.468,00€CB 3717
CAS :CB 3717 is an enzyme inhibitor, antineoplastic agent, folic acid antagonist.Formule :C24H23N5O6Couleur et forme :SolidMasse moléculaire :477.47FT827
CAS :FT827 is a covalent inhibitor of USP7 that targets the catalytic center of the autoinhibitory apolipoprotein form of USP7 for cancer research.Formule :C27H28N6O5SDegré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :548.61USP28-IN-4
CAS :USP28-IN-4 is a USP28 inhibitor with anticancer activity that dose-dependently down-regulates cellular levels of c-Myc via the ubiquitin-proteasome system.Formule :C22H18Cl2N2O3SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :461.36SRPKIN-1
CAS :SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).Formule :C27H21FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.53LIMK1 inhibitor BMS-4
CAS :BMS-4 is a LIMK inhibitor targeting LIMK1/2, reduces cofilin phosphorylation, noncytotoxic to A549 cells.Formule :C23H23N7O2SCouleur et forme :SolidMasse moléculaire :461.54HBV-IN-15
CAS :HBV-IN-15, a flavone derivative, is a potent cccDNA inhibitor, potentially aiding HBV research.Formule :C24H23ClO6Couleur et forme :SolidMasse moléculaire :442.89FD-IN-1
CAS :FD-IN-1 is an orally active Factor D (FD) inhibitor (IC50=12 nM), inhibits Factor XIa and Tryptase β2 with IC50 values of 7.7 and 6.5 μM, respectively.Formule :C23H23NO4Degré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :377.43XU1
CAS :XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation orFormule :C12H8N2ODegré de pureté :97.81% - 99.59%Couleur et forme :SolidMasse moléculaire :196.2USP28-IN-3
CAS :USP28-IN-3 is a USP28 inhibitor with anticancer activity that dose-dependently down-regulates cellular levels of c-Myc via the ubiquitin-proteasome system.Formule :C23H20Cl2N2O3SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :475.39KIF18A-IN-4
CAS :KIF18A-IN-4: Non-competitive KIF18A inhibitor, IC50 6.16 μM, targets mitotic kinesins/kinases, anti-tumor.Formule :C22H27N3O3SCouleur et forme :SolidMasse moléculaire :413.53BI8622
CAS :BI8622 is a HUWE1 antagonist that restores levels of RP2 mutants in retinal cell lines and inhibits cellular activation of NLRP3 and AIM2 inflammatory vesicles.Formule :C25H26N6ODegré de pureté :98.28% - 98.28%Couleur et forme :SolidMasse moléculaire :426.51DHODH-IN-4
CAS :DHODH-IN-4 inhibits human & Plasmodium DHODH; IC50: 4 μM (Pf), 0.18 μM (Hs). It has antimalarial properties.Formule :C17H12Cl2N2O2Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :347.2Ref: TM-T11027
1mg109,00€2mg163,00€5mg243,00€1mL*10mM (DMSO)248,00€10mg355,00€25mg532,00€50mg750,00€100mg1.009,00€500mg2.035,00€Dihydro-5-azacytidine acetate
CAS :Dihydro-5-azacytidine acetate (DHAC), a nucleoside analog, becomes integrated into DNA, thereby inhibiting DNA methylation, and exhibits antitumor activity [1Formule :C10H18N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.27TDRL-551
CAS :TDRL-551 is a novel and potent replication protein A (RPA) inhibitor (IC50=18 µM) with potential anticancer activity.TDRL-551 inhibits RPA-DNA interaction andFormule :C25H23ClIN3O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :591.83Ref: TM-T28935
1mg73,00€5mg160,00€1mL*10mM (DMSO)202,00€10mg250,00€25mg505,00€50mg803,00€100mg1.288,00€IRE1α kinase-IN-8
CAS :IRE1α kinase-IN-8, a benzoheterocyclecarboxaldehyde derivative, serves as a potent inhibitor of IRE-1α.Formule :C23H22N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.43SPC-839
CAS :SPC-839 is an IKK-2 Inhibitor with oral activity.Formule :C18H14N4O3SCouleur et forme :SolidMasse moléculaire :366.39Piposulfan
CAS :Piposulfan, a water-insoluble alkylating agent, is used as an antineoplastic and anti-tumor agent.Formule :C12H22N2O8S2Couleur et forme :SolidMasse moléculaire :386.44ARN22089
CAS :ARN22089 is an oral active CDC42 GTPase interaction inhibitor that blocks tumour growth in BRAF mutant mouse melanoma models and PDXs in vivo.Formule :C23H27N5Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :373.49Ref: TM-T85727
1mg109,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg385,00€25mg647,00€50mg964,00€100mg1.431,00€200mg1.963,00€MTH1-IN-2
CAS :MTH1-IN-2 is an inhibitor of MutT homolog 1 (MTH1), with anti-tumor activity.Formule :C24H27N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.55Valomaciclovir
CAS :Valomaciclovir is a DNA polymerase inhibitor potentially for treatment of acute herpes zoster and EB virus infection.Formule :C15H24N6O4Couleur et forme :SolidMasse moléculaire :352.39Antitumor agent-85
Antitumor agent-85 stabilizes G4-DNA with potent anti-tumor effects.Formule :C24H33N7Couleur et forme :SolidMasse moléculaire :419.57VE-465
CAS :VE-465 is an inhibitor of Aurora kinase, which involves in multiple mitotic events.Formule :C22H28N8OSCouleur et forme :SolidMasse moléculaire :452.58CCT068127
CAS :CCT068127 is a potent CDK2 and CDK9 inhibitor.Formule :C19H27N7OCouleur et forme :SolidMasse moléculaire :369.46Mequindox
CAS :Mequindox is an antimicrobial agent [1]. Mequindox, as an inhibitor of DNA synthesis, induces genotoxicity and carcinogenicity in mice [2].Formule :C11H10N2O3Couleur et forme :SolidMasse moléculaire :218.21hDHODH-IN-5
CAS :hDHODH-IN-5 is an inhibitor of human dihydroorotate dehydrogenase (hDHODH, IC50 = 0.91 μM).Formule :C21H21F3N2O2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :390.4Ref: TM-T11029
1mg80,00€5mg158,00€1mL*10mM (DMSO)172,00€10mg221,00€25mg356,00€50mg530,00€100mg755,00€ATB107
CAS :ATB107 is a potent and novel inhibitor of indole-3-glycerol phosphate synthase (IGPS, KD: 3 μM).Formule :C21H28N8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.5DHODH-IN-13
CAS :DHODH-IN-13 is an inhibitor of DHODH with IC50 of 4.3 μM for rat liver. DHODH-IN-13 can be used in studies about rheumatoid arthritis.Formule :C10H6F3N3O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :273.17Phen-DC3
CAS :Phen-DC3 is a G-quadruplex (G4) specific ligand which can inhibit FANCJ and DinG helicases (IC50s of 65±6 and 50±10 nM, respectively).Formule :C34H26N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61Cdc7-IN-9
CAS :Cdc7-IN-9 can be used for the research of cancer which is a potent inhibitor of Cdc7 [1].Formule :C15H17N5OSCouleur et forme :SolidMasse moléculaire :315.39(S)-CR8
CAS :(S)-CR8 is an effective second-generation cyclin-dependent kinase inhibitor.Formule :C24H29N7OCouleur et forme :SolidMasse moléculaire :431.53Mycro2
CAS :Mycro2 is an inhibitor of the protein-protein interactions between the bHLHZip proteins c-Myc and Max.Formule :C17H11F3N4OS2Couleur et forme :SolidMasse moléculaire :408.42Nitracrine dihydrochloride
CAS :Nitracrine dihydrochloride is an acridine antineoplastic agent used in mammary and ovarian tumors. It inhibits RNA synthesis.Formule :C18H22Cl2N4O2Couleur et forme :SolidMasse moléculaire :397.32'-Deoxy-L-guanosine
CAS :2'-Deoxy-L-guanosine is a nucleoside that shows antibiotic properties by inhibiting protein synthesis, leading to cell death.Formule :C10H13N5O4Couleur et forme :SolidMasse moléculaire :267.24Antitumor agent-84
Antitumor agent-84 stabilizes G-quadruplex DNA, exhibits potent anti-tumor effects.Formule :C24H31N7Couleur et forme :SolidMasse moléculaire :417.55Metralindole
CAS :Metralindole is a reversible inhibitor of monoamine oxidase A (RIMA).Formule :C15H17N3OCouleur et forme :SolidMasse moléculaire :255.32GR 144053 trihydrochloride
CAS :platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonistFormule :C18H30Cl3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.82TCS 2312
CAS :checkpoint kinase 1 (chk1) inhibitorFormule :C25H24N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.48Trimetrexate
CAS :Trimetrexate is an effective competitive inhibitor of bacterial, protozoan, and mammalian dihydrofolate reductase.Formule :C19H23N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.42hDHODH-IN-3
CAS :hDHODH-IN-3 is an inhibitor of human dihydroorotate dehydrogenase with a pMIC50 value of 8.6. hDHODH-IN-3 can inhibit measles virus replication.Formule :C18H19BrN4O2Degré de pureté :99.871%Couleur et forme :SolidMasse moléculaire :403.27Ref: TM-T11025
500mgÀ demander1mg60,00€2mg88,00€5mg133,00€1mL*10mM (DMSO)142,00€10mg203,00€25mg335,00€50mg474,00€100mg623,00€Laflunimus
CAS :Laflunimus (HR325) is a DHODH inhibitor that inhibits immunoglobulin secretion in vitro and in vivo,by interfering with pyrimidine metabolism,neuralgia.Formule :C15H13F3N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :310.27Tripolin A
CAS :Tripolin A is a specific non-ATP competitive inhibitor of Aurora A kinase(Aurora A and Aurora B with IC50 values of 1.5 μM and 7 μM, respectively)Formule :C15H11NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :253.25Integrin-IN-2
CAS :Integrin-IN-2, an oral αv integrin blocker, enhances αvβ6/3/5/8 affinities with pIC50s: 7.8/8.4/8.4/7.4.Formule :C27H30N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.55Remdesivir maleate
CAS :Remdesivir (GS-5734) is a broad-spectrum antiviral prodrug effective against SARS-CoV-2 and Ebola, used for research, not human treatment.Formule :C31H39N6O12PCouleur et forme :SolidMasse moléculaire :718.656CDK7-IN-8
CAS :CDK7-IN-8 is a potent inhibitor of CDK7 (IC50: 54.29 nM) and exhibits inhibitory activity against several cancer cells and in vivo tumor models.Formule :C25H38N8O3Couleur et forme :SolidMasse moléculaire :498.62Olomoucine II
CAS :Olomoucine II, a CDK inhibitor effective on Cdk1/2/4/7/9, also inhibits ERK2, ABCB1, and various virus replications, not effective on measles/influenza.Formule :C19H26N6O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :370.45360A iodide
CAS :360A iodide is a selective stabilizer of G-quadruplex and inhibits telomerase activity (IC50: 300 nM in TRAP-G4 assay).Formule :C27H23I2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :703.31BMVC
CAS :BMVC is a potent G-quadruplex (G4) stabilizer and a selective telomerase inhibitor (IC50: ~0.2 μM) with anticancer activities.Formule :C28H25I2N3Couleur et forme :SolidMasse moléculaire :657.33MK-0668 Mesylate
CAS :MK-0668 Mesylate is the mesylate form of MK-0668 that is a very potent and orally active very late antigen-4 antagonist.Formule :C32H34Cl2N6O9S2Couleur et forme :SolidMasse moléculaire :781.68NSC 625987
CAS :NSC 625987, Selective CDK4 inhibitor (IC50=0.2 μM), >500-fold selectivity over CDK2, used for p16-associated tumor studies.Formule :C15H13NO2SDegré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :271.33Ref: TM-T23092
10mgÀ demander25mgÀ demander1mL*10mM (DMSO)À demander1mg63,00€5mg137,00€50mg595,00€100mg893,00€Mps1-IN-4
CAS :Mps1-IN-4 is a compound that selectively inhibits Monopolar spindle 1 (Mps1), exhibiting antiproliferative properties useful in cancer research.Formule :C26H31F3N6O2Couleur et forme :SolidMasse moléculaire :516.56SLM6
CAS :SLM6, an inhibitor of cyclin-dependent kinase-9 (CDK9), exhibits potent anti-multiple myeloma activity.Formule :C12H17N7O4Couleur et forme :SolidMasse moléculaire :323.31
