Enzyme
Les inhibiteurs d'enzymes sont des molécules qui se lient aux enzymes et diminuent leur activité. Ces inhibiteurs sont largement utilisés en recherche pour étudier la cinétique enzymatique, la régulation et le rôle spécifique des enzymes dans les voies métaboliques. Les inhibiteurs d'enzymes sont également cruciaux dans le développement de médicaments, car de nombreux agents thérapeutiques agissent en inhibant les enzymes impliquées dans les processus pathologiques. En ciblant les enzymes, ces inhibiteurs peuvent moduler les voies biochimiques et offrir des traitements potentiels pour diverses maladies. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs d'enzymes de haute qualité pour soutenir vos recherches en biochimie, pharmacologie et découverte de médicaments.
Sous-catégories appartenant à la catégorie "Enzyme"
- Anhydrase carbonique(177 produits)
- Hydroxylase(30 produits)
- MPO(2 produits)
- Réductase(52 produits)
- Tyrosinase(67 produits)
3586 produits trouvés pour "Enzyme"
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ACT-678689
CAS :<p>ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].</p>Formule :C23H22ClFN6O4S2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :565.04Brinzolamide
CAS :<p>Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.</p>Formule :C12H21N3O5S3Degré de pureté :99.84% - >99.99%Couleur et forme :Crystalline SolidMasse moléculaire :383.51KW-2450 Formate
<p>KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.</p>Formule :C29H31N5O5SDegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :561.65Methazolamide
CAS :<p>Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.</p>Formule :C5H8N4O3S2Degré de pureté :99.31% - 99.77%Couleur et forme :Crystals From Water SolidMasse moléculaire :236.27Actarit
CAS :<p>Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug.</p>Formule :C10H11NO3Degré de pureté :99.64% - 99.74%Couleur et forme :White Or Off-White Crystal Or Crystalline SolidMasse moléculaire :193.2pNNP
CAS :<p>pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.</p>Formule :C6H6NO6PDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :219.09Methocarbamol
CAS :<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Formule :C11H15NO5Degré de pureté :99.96%Couleur et forme :Crystals From Benzene SolidMasse moléculaire :241.24Topiramate
CAS :<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36Benzthiazide
CAS :<p>Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.</p>Formule :C15H14ClN3O4S3Degré de pureté :99.34% - 99.79%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :431.94p-Ethynylphenylalanine hydrochloride
CAS :<p>p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].</p>Formule :C11H12ClNO2Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :225.67Arbutin
CAS :<p>Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.</p>Formule :C12H16O7Degré de pureté :99.58% - 99.93%Couleur et forme :Colorless Elongated Prisms From Moist Ethyl Acetate White PowderMasse moléculaire :272.25Telotristat ethyl
CAS :<p>Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.</p>Formule :C27H26ClF3N6O3Degré de pureté :98% - 99.89%Couleur et forme :White SolidMasse moléculaire :574.98Flanvotumab
CAS :<p>Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.</p>Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :145.42 kDa4-Chlorosalicylic acid
CAS :<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Formule :C7H5ClO3Degré de pureté :98.59%Couleur et forme :Off-White To Light Beige PowderMasse moléculaire :172.57Acipimox
CAS :<p>Acipimox (K-9321), a niacin derivative, treats hyperlipidemia in type 2 diabetics.</p>Formule :C6H6N2O3Degré de pureté :98.98%Couleur et forme :Low Yellow Liquid Or CrystallineMasse moléculaire :154.12Fenclonine
CAS :<p>Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.</p>Formule :C9H10ClNO2Degré de pureté :98.81% - >99.99%Couleur et forme :Crystals From Methanol White SolidMasse moléculaire :199.635-Feruloylquinic acid
CAS :<p>5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.</p>Formule :C17H20O9Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :368.34Zonisamide
CAS :<p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>Formule :C8H8N2O3SDegré de pureté :99.05% - 99.9%Couleur et forme :Off-White PowderMasse moléculaire :212.23Tioxolone
CAS :<p>Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.</p>Formule :C7H4O3SDegré de pureté :97.79%Couleur et forme :Light Yellow To Beige PowderMasse moléculaire :168.17Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Couleur et forme :Odour SolidCAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Couleur et forme :Odour SolidCAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formule :C23H21N5O3SCouleur et forme :SolidMasse moléculaire :447.51Pyrocatechol
CAS :<p>Pyrocatechol, often known as catechol or benzene-1,2-diol, is a benzenediol, Pyrocatechol was produced at a large scale industrially, mainly as precursors to pesticides, flavors, and fragrances. Its sulfonic acid is often present in the urine of many mammals.</p>Formule :C6H6O2Couleur et forme :SolidMasse moléculaire :110.11Chlorothiazide
CAS :<p>Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.</p>Formule :C7H6ClN3O4S2Degré de pureté :98.46% - 98.91%Couleur et forme :Crystals Physical Description Crystals; White Powder (Ntp 1992)Masse moléculaire :295.72CAIX Inhibitor S4
CAS :<p>CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.</p>Formule :C15H17N3O4SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :335.38hCAIX-IN-19
<p>hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/</p>Couleur et forme :Odour Solid2-Methoxy-4-propylphenol
CAS :<p>2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.</p>Formule :C10H14O2Couleur et forme :SolidMasse moléculaire :166.22Carbonic anhydrase inhibitor 30
<p>Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].</p>Formule :C23H22FN3O5SCouleur et forme :SolidMasse moléculaire :471.12642Xanthine Oxidase, ammonium sulfate suspension
CAS :Couleur et forme :Faint brown to dark brown suspensionAnhydrotetracycline hydrochloride
CAS :<p>Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.</p>Formule :C22H23ClN2O7Degré de pureté :98.90%Couleur et forme :SolidMasse moléculaire :462.88Tyrosinase-IN-34
<p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>Formule :C19H14BrClN4OCouleur et forme :SolidMasse moléculaire :429.7Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Formule :C15H19NO3Couleur et forme :SolidMasse moléculaire :261.32Calmodulin-dependent Protein Kinase II fragment 290-309
CAS :Formule :C103H185N31O24SMasse moléculaire :2273.83(E)-Dehydrodiconiferyl alcohol
CAS :<p>(E)-Dehydrodiconiferyl alcohol inhibits hCA IX/XII enzymes and blocks NF-κB nuclear translocation in healing tissues.</p>Formule :C20H22O6Couleur et forme :SolidMasse moléculaire :358.395,6-Dihydro-2H-pyran-2-one
CAS :<p>5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.</p>Formule :C5H6O2Couleur et forme :SolidMasse moléculaire :98.1Peroxidase
CAS :Degré de pureté :≥ 85units/mg (dry basis)Couleur et forme :Beige to light-brown, reddish brown or dark brown lyophilised powderMasse moléculaire :-
