Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(100 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(66 produits)
- Récepteur CGRP(54 produits)
- Canal calcique(544 produits)
- Canal chlorure(53 produits)
- Récepteur GABA(369 produits)
- Transporteur de monoamine(30 produits)
- Transporteur de monocarboxylate(18 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(10 produits)
- OAT(32 produits)
- OCT(7 produits)
- P-gp(55 produits)
- Canal potassique(283 produits)
- Pompe à protons(41 produits)
- SGLT(31 produits)
- Canal sodique(217 produits)
- Canal TRP/TRPV(96 produits)
Affichez 13 plus de sous-catégories
2575 produits trouvés pour "Transporteur membranaire/Canal ionique"
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Fosphenytoin disodium
CAS :Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blockerFormule :C16H13N2Na2O6PDegré de pureté :99.97%Couleur et forme :White Crystalline PowderMasse moléculaire :406.24Chloroprocaine hydrochloride
CAS :Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.Formule :C13H20Cl2N2O2Degré de pureté :99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :307.22YM90K
CAS :YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.Formule :C11H8ClN5O4Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :309.66Ref: TM-T8435
1mg78,00€5mg169,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)178,00€Esomeprazole Magnesium
CAS :Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.Formule :C34H36MgN6O6S2Degré de pureté :98.76% - 99.73%Couleur et forme :SolidMasse moléculaire :713.12U93631
CAS :GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formule :C17H21N3O2Degré de pureté :99.65% - 99.76%Couleur et forme :SolidMasse moléculaire :299.37Levolansoprazole
CAS :Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).Formule :C16H14F3N3O2SDegré de pureté :98.629%Couleur et forme :SolidMasse moléculaire :369.36Ref: TM-T20714
1mg111,00€5mg246,00€10mg344,00€25mg522,00€50mg692,00€100mg929,00€200mg1.225,00€1mL*10mM (DMSO)255,00€Tenatoprazole sodium
CAS :Tenatoprazole sodium is a potent proton pump inhibitor with an IC50 of 6.2 μM against hog gastric H+/K+-ATPase.Formule :C16H17N4NaO3SCouleur et forme :SolidMasse moléculaire :368.39Homocarnosine acetate
Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.Formule :C12H20N4O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :300.31Ref: TM-T32098L
1mg57,00€2mg79,00€5mg109,00€10mg167,00€25mg334,00€50mg467,00€100mg662,00€200mg892,00€1mL*10mM (DMSO)138,00€DS-1971a
CAS :DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.Formule :C20H21ClFN5O3SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :465.93Temgicoluril
CAS :Temgicoluril (mebikar) acts on GABA Receptor.Formule :C8H14N4O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :198.22(E)-KPT330
CAS :<p>(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.</p>Formule :C17H11F6N7ODegré de pureté :98.69% - 99.49%Couleur et forme :SolidMasse moléculaire :443.31Gaboxadol hydrochloride
CAS :Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formule :C6H9ClN2O2Degré de pureté :99.39%Masse moléculaire :176.601Lomerizine
CAS :<p>Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.</p>Formule :C27H30F2N2O3Couleur et forme :SolidMasse moléculaire :468.54O4I2
CAS :O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.Formule :C12H11ClN2O2SDegré de pureté :97.97% - 99.84%Couleur et forme :SolidMasse moléculaire :282.75HC-056456
CAS :HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.Formule :C12H6N2O4S2Degré de pureté :99.62% - 99.65%Couleur et forme :SolidMasse moléculaire :306.32Ref: TM-T4604
1mg35,00€2mg48,00€5mg70,00€10mg96,00€25mg170,00€50mg274,00€100mg454,00€1mL*10mM (DMSO)77,00€(-)-Dizocilpine maleate
CAS :(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.Formule :C20H19NO4Degré de pureté :>99.99%Couleur et forme :White SolidMasse moléculaire :337.37Tirofiban hydrochloride monohydrate
CAS :<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Formule :C22H39ClN2O6SDegré de pureté :98.81% - >99.99%Couleur et forme :White SolidMasse moléculaire :495.07AMG9810
CAS :AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.Formule :C21H23NO3Degré de pureté :99.79% - 99.95%Couleur et forme :SolidMasse moléculaire :337.41Ref: TM-T7189
2mg34,00€5mg48,00€10mg58,00€25mg110,00€50mg177,00€100mg286,00€200mg425,00€1mL*10mM (DMSO)50,00€HM-30181 mesylate monohydrate
CAS :HM-30181 mesylate monohydrate is an oral P-glycoprotein (P-gp) inhibitor, used to enhance the oral bioavailability of P-gp substrate drugs.Formule :C39H42N6O11SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :802.85Ref: TM-T9173
1mg65,00€2mg94,00€5mg119,00€10mg185,00€25mg309,00€50mg442,00€100mg643,00€200mg835,00€500mg1.251,00€1mL*10mM (DMSO)177,00€Valbenazine
CAS :Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.Formule :C24H38N2O4Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :418.57Ref: TM-T7147
1mg48,00€2mg62,00€5mg106,00€10mg170,00€25mg329,00€50mg512,00€100mg747,00€200mg1.017,00€1mL*10mM (DMSO)119,00€Eliprodil
CAS :Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50>100 uM), explored for Parkinson's and movement issues.Formule :C20H23ClFNODegré de pureté :99.53% - 99.77%Couleur et forme :SolidMasse moléculaire :347.85Chloroprocaine
CAS :Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.Formule :C13H19ClN2O2Couleur et forme :SolidMasse moléculaire :270.76Lorediplon
CAS :Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formule :C20H15FN4O2SDegré de pureté :99.12% - 99.19%Couleur et forme :SolidMasse moléculaire :394.42NS 11021
CAS :NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channelsFormule :C16H9BrF6N6SDegré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :511.24Ref: TM-T4294
1mg42,00€5mg88,00€10mg128,00€25mg263,00€50mg447,00€100mg760,00€200mg1.018,00€1mL*10mM (DMSO)89,00€Azimilide Dihydrochloride
CAS :Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.Formule :C23H30Cl3N5O3Degré de pureté :97.59% - ≥95%Couleur et forme :SolidMasse moléculaire :530.88QX-222 chloride
CAS :QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.Formule :C13H21ClN2ODegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :256.77Tariquidar dihydrochloride
CAS :Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).Formule :C38H40Cl2N4O6Couleur et forme :SolidMasse moléculaire :719.65L-701324
CAS :L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.Formule :C21H14ClNO3Degré de pureté :98.63% - >99.99%Couleur et forme :SolidMasse moléculaire :363.79Acamprosate
CAS :Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can TrustFormule :C5H11NO4SDegré de pureté :98.30%Couleur et forme :SolidMasse moléculaire :181.21Revaprazan hydrochloride
CAS :Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Formule :C22H24ClFN4Degré de pureté :99.62% - 99.91%Couleur et forme :SolidMasse moléculaire :398.9Z944
CAS :Z944 is a T-type calcium channel blocker.Formule :C19H27ClFN3O2Degré de pureté :99.8% - 99.80%Couleur et forme :SolidMasse moléculaire :383.89Ref: TM-T29201
1mg52,00€5mg111,00€10mg180,00€25mg359,00€50mg530,00€100mg758,00€200mg1.035,00€1mL*10mM (DMSO)124,00€SB-705498
CAS :SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.Formule :C17H16BrF3N4ODegré de pureté :99.57% - ≥95%Couleur et forme :SolidMasse moléculaire :429.23Tariquidar
CAS :Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.Formule :C38H38N4O6Degré de pureté :98.07% - 99.45%Couleur et forme :SolidMasse moléculaire :646.73TCN 213
CAS :TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2BFormule :C18H24N4OS2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :376.54Traxoprodil
CAS :Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).Formule :C20H25NO3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :327.42Flecainide acetate
CAS :Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).Formule :C19H24F6N2O5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :474.39L-DABA
CAS :L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formule :C4H10N2O2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :118.13ICA 110381
CAS :ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsyFormule :C12H8Cl2N2ODegré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :267.11Disopyramide phosphate
CAS :Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.Formule :C21H32N3O5PCouleur et forme :SolidMasse moléculaire :437.47ZL006
CAS :ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Formule :C14H11Cl2NO4Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :328.15Ref: TM-T17293
5mg48,00€10mg63,00€25mg111,00€50mg170,00€100mg290,00€200mg420,00€1mL*10mM (DMSO)50,00€VK-II-36
CAS :VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.Formule :C26H26N2O5Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :446.49DNQX disodium salt
CAS :DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptorFormule :C8H2N4Na2O6Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :296.1Ref: TM-T8459
1mg62,00€5mg123,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)123,00€Budipine
CAS :Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.Formule :C21H27NDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :293.45Selamectin
CAS :Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening inFormule :C43H63NO11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :769.96ICA-069673
CAS :ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).Formule :C11H6ClF2N3ODegré de pureté :99.04% - 99.68%Couleur et forme :SolidMasse moléculaire :269.63GS967
CAS :<p>GS967 is a potent, and selective inhibitor of cardiac late sodium current (late INa ).</p>Formule :C14H7F6N3ODegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :347.22Ref: TM-T2049
2mg35,00€5mg52,00€10mg79,00€25mg159,00€50mg284,00€100mg495,00€200mg718,00€500mg1.111,00€TKIM
CAS :TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.Formule :C18H14ClN3O2SDegré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :371.84Ref: TM-T8700
1mg42,00€5mg94,00€10mg131,00€25mg225,00€50mg314,00€100mg420,00€200mg567,00€1mL*10mM (DMSO)92,00€2'-O-Methylisoliquiritigenin
CAS :2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28RY785
CAS :RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.Formule :C21H20N4O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :392.47Ref: TM-T12786
1mg51,00€5mg144,00€10mg235,00€25mg399,00€50mg560,00€100mg787,00€200mg1.093,00€1mL*10mM (DMSO)125,00€L-Allylglycine
CAS :L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.Formule :C5H9NO2Degré de pureté :≥98%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :115.134-Acetamidobutanoic acid
CAS :4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16AER-271
CAS :AER-271 is an inhibitor of aquaporin-4.Formule :C15H9ClF6NO5PDegré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :463.65Ropivacaine hydrochloride monohydrate
CAS :Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.Formule :C17H29ClN2O2Degré de pureté :99.94% - 99.95%Couleur et forme :White SolidMasse moléculaire :328.88AMG 333
CAS :<p>AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.</p>Formule :C20H12F5N3O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :453.32Alinidine hydrobromide
CAS :Alinidine hydrobromide, a specific bradycardic agent, diminishes the slope of the diastolic depolarization in sinoatrial tissue and Purkinje fibers [1].Formule :C12H14BrCl2N3Couleur et forme :SolidMasse moléculaire :351.07Ocinaplon
CAS :Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formule :C17H11N5ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :301.3Ilaprazole sodium
CAS :<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formule :C19H17N4NaO2SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :388.42Mitiglinide Calcium
CAS :Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-Formule :(C19H24NO3)2·CaDegré de pureté :99.83%Couleur et forme :White Crystal PosderMasse moléculaire :668.88Lansoprazole sodium
CAS :Lansoprazole sodium is a PPI used to treat acid reflux and peptic ulcers.Formule :C16H13F3N3NaO2SDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :391.34Metaflumizone
CAS :Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.Formule :C24H16F6N4O2Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :506.40Rapastinel Trifluoroacetate
CAS :Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.Formule :C20H32F3N5O8Degré de pureté :99.01% - 99.77%Couleur et forme :SolidMasse moléculaire :527.49Ref: TM-T5819
1mg39,00€5mg97,00€10mg160,00€25mg296,00€50mg416,00€100mg557,00€200mg743,00€1mL*10mM (DMSO)116,00€(-)-Blebbistatin
CAS :(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.Formule :C18H16N2O2Degré de pureté :99.38% - 99.61%Couleur et forme :SolidMasse moléculaire :292.33HC-067047
CAS :HC-067047 is a potent and selective TRPV4 antagonist.Also inhibits the endogenous TRPV4-mediated response to 4α-PDH .Formule :C26H28F3N3O2Degré de pureté :99.45% - 99.97%Couleur et forme :SolidMasse moléculaire :471.51Arecaidine hydrochloride
CAS :Arecaidine hydrochloride may have carcinogenesis.Formule :C7H12ClNO2Degré de pureté :99.69% - ≥95%Couleur et forme :SolidMasse moléculaire :177.63Ref: TM-T5799
2mg35,00€5mg50,00€10mg71,00€25mg105,00€50mg158,00€100mg225,00€200mg334,00€1mL*10mM (DMSO)51,00€NBI-98782
CAS :NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)Formule :C19H29NO3Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :319.44Ref: TM-T7563
1mg46,00€5mg93,00€10mg119,00€25mg207,00€50mg324,00€100mg482,00€200mg637,00€1mL*10mM (DMSO)92,00€Baclofen hydrochloride
CAS :Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formule :C10H13Cl2NO2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :250.122Neboglamine
CAS :<p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>Formule :C13H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.34Propafenone hydrochloride
CAS :Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.Formule :C21H27NO3·HClDegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :377.9Lansoprazole sulfone
CAS :Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.Formule :C16H14F3N3O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :385.36Ref: TM-T20155
1mg52,00€5mg111,00€10mg173,00€25mg296,00€50mg445,00€100mg655,00€200mg924,00€1mL*10mM (DMSO)47,00€Kv2-IN-A1
CAS :Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.Formule :C20H17ClN4OSDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :396.89Ralfinamide mesylate
CAS :Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.Formule :C18H23FN2O5SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :398.45Ref: TM-T7547
1mg55,00€5mg118,00€10mg180,00€25mg296,00€50mg393,00€100mg553,00€200mg743,00€1mL*10mM (DMSO)180,00€MDR-652
CAS :MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM forFormule :C22H23ClFN3O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :447.95Ref: TM-T22360
1mg60,00€2mg87,00€5mg130,00€10mg178,00€25mg331,00€50mg512,00€100mg707,00€200mg973,00€1mL*10mM (DMSO)142,00€Radiprodil
CAS :Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.Formule :C21H20FN3O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :397.4Ref: TM-T5385
1mg48,00€2mg65,00€5mg96,00€10mg153,00€25mg240,00€50mg354,00€100mg532,00€1mL*10mM (DMSO)96,00€Miltirone
CAS :Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formule :C19H22O2Degré de pureté :99.22% - 99.66%Couleur et forme :SolidMasse moléculaire :282.38Adjudin
CAS :Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.Formule :C15H12Cl2N4ODegré de pureté :96.51% - ≥95%Couleur et forme :SolidMasse moléculaire :335.19Pyr6
CAS :Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influxFormule :C17H9F7N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :418.27Raxatrigine hydrochloride
CAS :Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.Formule :C18H20ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.82α-Asarone
CAS :alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formule :C12H16O3Degré de pureté :99.64% - 99.64%Couleur et forme :Monoclinic Needles From Water Monoclinic Needles From WaterMasse moléculaire :208.25Almitrine mesylate
CAS :Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.Formule :C28H37F2N7O6S2Degré de pureté :99.96%Couleur et forme :CoaMasse moléculaire :669.761-Aminocyclobutanecarboxylic acid
CAS :1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].Formule :C5H9NO2Degré de pureté :99.94%Couleur et forme :White To Tan Powder Crystals Crystalline Powder And/Or With ChunksMasse moléculaire :115.13Cyclothiazide
CAS :Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Formule :C14H16ClN3O4S2Degré de pureté :98.23% - 99.49%Couleur et forme :Crystals From Dilute Alcohol SolidMasse moléculaire :389.88Lesinurad
CAS :Lesinurad (RDEA594), a selective uric acid reabsorption inhibitor, is used to treat gout without causing liver damage.Formule :C17H14BrN3O2SDegré de pureté :99.83% - 99.86%Couleur et forme :SolidMasse moléculaire :404.28Ref: TM-T6875
10mg44,00€25mg80,00€50mg126,00€100mg197,00€200mg294,00€500mg494,00€1mL*10mM (DMSO)34,00€Levamlodipine hydrobromide
CAS :Levamlodipine hydrobromide is a medication used to lower blood pressure and prevent chest pain.Formule :C20H26BrClN2O5Couleur et forme :SolidMasse moléculaire :489.79Guanosine 5'-diphosphate disodium salt
CAS :<p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>Formule :C10H13N5Na2O11P2Degré de pureté :99.40%Couleur et forme :White PowderMasse moléculaire :487.16PF-05186462
CAS :PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.Formule :C19H10ClF4N5O3S2Degré de pureté :99.10% - 99.37%Couleur et forme :SolidMasse moléculaire :531.89PF-4840154
CAS :<p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) & 23 nM (human); triggers nociception in mice.</p>Formule :C26H38N6O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :466.62Talniflumate
CAS :<p>Talniflumate (Somalgen) is a calcium-activated chloride channel (hCLCA1/mCLCA3) blocker that reduces mucin synthesis and releases in animal models and cell</p>Formule :C21H13F3N2O4Degré de pureté :98% - 99.81%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :414.33JNJ 303
CAS :JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).Formule :C21H29ClN2O4SDegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :440.98Ref: TM-T7653
1mg48,00€2mg65,00€5mg89,00€10mg147,00€25mg325,00€50mg472,00€100mg705,00€1mL*10mM (DMSO)92,00€SB 452533
CAS :SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).Formule :C18H22BrN3ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :376.29Ref: TM-T23322
2mg39,00€5mg60,00€10mg92,00€25mg173,00€50mg269,00€100mg389,00€200mg555,00€1mL*10mM (DMSO)73,00€Disopyramide HCl
CAS :Disopyramide HCl, a Class 1a antiarrhythmic, treats ventricular tachycardia, blocks sodium channels, and has anticholinergic effects.Formule :C21H30ClN3OCouleur et forme :SolidMasse moléculaire :375.94AZD-6280
CAS :AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formule :C20H22N4O3Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :366.41Ref: TM-T7136
1mg227,00€5mg464,00€10mg677,00€25mg1.074,00€50mg1.501,00€100mg2.043,00€1mL*10mM (DMSO)510,00€Cabotegravir
CAS :Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (Formule :C19H17F2N3O5Degré de pureté :98.55% - 99.92%Couleur et forme :SolidMasse moléculaire :405.35MDK-4025
CAS :MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.Formule :C19H15ClODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :294.77Fluralaner
CAS :Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formule :C22H17Cl2F6N3O3Degré de pureté :99.72% - 99.99%Couleur et forme :Solid PowderMasse moléculaire :556.29Tetraethylammonium chloride
CAS :Tetraethylammonium chloride is a quaternary ammonium compound.Formule :C8H20ClNDegré de pureté :≥95%Couleur et forme :White Solid Solid Particulate/PowderMasse moléculaire :165.7Co 101244 hydrochloride
CAS :Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Formule :C21H28ClNO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :377.9KM11060
CAS :KM11060 is a novel corrector of the F508del-CFTR trafficking defect, Correcting F508del-CFTR trafficking, increasing the amount of functional CFTR at the plasmaFormule :C19H17Cl2N3O2SDegré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :422.33Rimeporide
CAS :Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.Formule :C11H15N3O5S2Degré de pureté :97.66%Couleur et forme :SolidMasse moléculaire :333.38Ref: TM-T5319
1mg46,00€2mg62,00€5mg90,00€10mg166,00€25mg358,00€50mg523,00€100mg747,00€1mL*10mM (DMSO)108,00€Tenapanor
CAS :Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.Formule :C50H66Cl4N8O10S2Degré de pureté :99.49% - 99.85%Couleur et forme :SolidMasse moléculaire :1145.05(R)-Lansoprazole
CAS :(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitorFormule :C16H14F3N3O2SDegré de pureté :98.09% - 98.99%Couleur et forme :Brown SolidMasse moléculaire :369.36
