Transporteur membranaire/Canal ionique
Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont des composés qui bloquent la fonction des protéines responsables du transport des ions, des nutriments et d'autres molécules à travers les membranes cellulaires. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie cellulaire, la transduction des signaux et la neurotransmission. Les inhibiteurs des transporteurs membranaires et des canaux ioniques sont également importants pour développer des traitements contre des troubles tels que l'épilepsie, les maladies cardiovasculaires et les syndromes métaboliques. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité des transporteurs membranaires et des canaux ioniques pour soutenir vos recherches en physiologie, neurosciences et pharmacologie.
Sous-catégories appartenant à la catégorie "Transporteur membranaire/Canal ionique"
- ABC(3 produits)
- ATPase(93 produits)
- Récepteur de l'adiponectine(5 produits)
- CFTR(64 produits)
- Récepteur CGRP(51 produits)
- Canal calcique(493 produits)
- Canal chlorure(49 produits)
- Récepteur GABA(336 produits)
- Transporteur de monoamine(23 produits)
- Transporteur de monocarboxylate(17 produits)
- NKCC(2 produits)
- NPC1L1(3 produits)
- Cotransporteur Na-K-Cl(8 produits)
- OAT(27 produits)
- OCT(7 produits)
- P-gp(53 produits)
- Canal potassique(276 produits)
- Pompe à protons(39 produits)
- SGLT(30 produits)
- Canal sodique(202 produits)
- Canal TRP/TRPV(92 produits)
Affichez 13 plus de sous-catégories
2270 produits trouvés pour "Transporteur membranaire/Canal ionique"
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Pilsicainide
CAS :<p>Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].</p>Formule :C17H24N2OCouleur et forme :SolidMasse moléculaire :272.39Levolansoprazole
CAS :<p>Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).</p>Formule :C16H14F3N3O2SDegré de pureté :98.629%Couleur et forme :SolidMasse moléculaire :369.36Linerixibat
CAS :<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Formule :C28H38N2O7SDegré de pureté :98.5% - 99.98%Couleur et forme :SolidMasse moléculaire :546.68Verinurad
CAS :<p>Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.</p>Formule :C20H16N2O2SDegré de pureté :97.36% - 99.22%Couleur et forme :SolidMasse moléculaire :348.42Imepitoin
CAS :<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formule :C13H14ClN3O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :279.72MONNA
CAS :<p>MONNA is a potent TMEM16A (Anoctamin-1) blocker (IC50 : 80 nM). It induces vasorelaxation of rodent resistance arteries in presence or absence of chloride ions.</p>Formule :C18H14N2O5Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :338.31A-803467
CAS :<p>A-803467 is a selective NaV1.8 channel blocker.</p>Formule :C19H16ClNO4Degré de pureté :96.94% - 98%Couleur et forme :SolidMasse moléculaire :357.79Vanilloid receptor antagonist 1
CAS :<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Formule :C18H15N3O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :305.33Fenamic acid
CAS :<p>Fenamic acid (N-Phenylanthranilic acid) is a chloride channel blocker that causes renal papillary necrosis in rats.</p>Formule :C13H11NO2Degré de pureté :99.6%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :213.2319AM92016
CAS :<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Formule :C26H30Cl2N2O6SCouleur et forme :SolidMasse moléculaire :569.49SB-366791
CAS :<p>SB-366791 is a new and selective cinnamide TRPV1 antagonist.</p>Formule :C16H14ClNO2Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :287.74Tiagabine hydrochloride hydrate
CAS :<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Formule :C20H28ClNO3S2Couleur et forme :SolidMasse moléculaire :430.02PPQ-102
CAS :<p>PPQ-102 (CFTR Inhibitor), an effective CFTR inhibitor, can completely inhibit CFTR chloride current (IC50: 90 nM).</p>Formule :C26H22N4O3Degré de pureté :99.7% - ≥95%Couleur et forme :SolidMasse moléculaire :438.48Optovin
CAS :<p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>Formule :C15H13N3OS2Degré de pureté :99.47% - 99.67%Couleur et forme :SolidMasse moléculaire :315.41VU6036720 hydrochloride
<p>VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.</p>Formule :C20H23Cl2FN4O2SCouleur et forme :SolidMasse moléculaire :473.39U93631
CAS :<p>GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.</p>Formule :C17H21N3O2Degré de pureté :99.65% - 99.76%Couleur et forme :SolidMasse moléculaire :299.37AMTB hydrochloride
CAS :<p>AMTB HCl: Novel TRPM8 blocker, relieves pain, treats urinary issues, moderates bladder reflexes in rats.</p>Formule :C23H27ClN2O2SDegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :430.99ML365
CAS :<p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>Formule :C22H20N2O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :360.41Azumolene sodium anhydrous
CAS :<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Etripamil
CAS :<p>Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.</p>Formule :C27H36N2O4Degré de pureté :99.47% - 99.83%Couleur et forme :SolidMasse moléculaire :452.59N-Me-aminopyrimidinone9
CAS :<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Formule :C16H21N3OSDegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :303.42Vocacapsaicin
CAS :<p>Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.</p>Formule :C26H41N3O4Couleur et forme :SolidMasse moléculaire :459.631Rimeporide hydrochloride
CAS :<p>Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>Formule :C11H16ClN3O5S2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :369.84Zoniporide hydrochloride hydrate
CAS :<p>Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.</p>Formule :C17H19ClN6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.83SKA-31
CAS :<p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>Formule :C11H8N2SDegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :200.26Cariporide
CAS :<p>Cariporide (HOE-642), an NHE1 inhibitor, reduces human platelet degranulation, platelet-leukocyte aggregates, and GPIIb/IIIa activation.</p>Formule :C12H17N3O3SDegré de pureté :95.4% - 99.88%Couleur et forme :SolidMasse moléculaire :283.35Thonzonium Bromide
CAS :<p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>Formule :C32H55BrN4ODegré de pureté :98.48% - 99.94%Couleur et forme :SolidMasse moléculaire :591.71Polyoxyethylene stearate
CAS :<p>Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.</p>Formule :C20H40O3Degré de pureté :n~9-10Couleur et forme :Light Amber SemisolidMasse moléculaire :328.29775Nav1.8-IN-1
CAS :<p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>Formule :C20H15ClF3N3O2Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :421.8Zosuquidar trihydrochloride
CAS :<p>Zosuquidar trihydrochloride (LY-335979 trihydrochloride) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.</p>Formule :C32H31F2N3O2·3HClDegré de pureté :99.49% - >99.99%Couleur et forme :SolidMasse moléculaire :636.996-(4-Methoxyphenyl)-3-pyridazinamine
CAS :<p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>Formule :C11H11N3ODegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :201.22Pirmenol
CAS :<p>Pirmenol is a new antiarrhythmic drug</p>Formule :C22H30N2ODegré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :338.49HBT1
CAS :<p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>Formule :C16H17F3N4O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :386.39Tulrampator
CAS :<p>Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.</p>Formule :C20H17FN4O3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :380.37Acetoxyvalerensre
CAS :<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formule :C17H24O4Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :292.37ML133 hydrochloride
CAS :<p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>Formule :C19H19NO·HClDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :313.82AZD3965
CAS :<p>AZD3965 (AZD-3965) is a selective inhibitor of monocarboxylate transporter 1 (MCT1).</p>Formule :C21H24F3N5O5SDegré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :515.51Chlorothymol
CAS :<p>Chlorothymol (AI3-00120) is a disinfectant used in oral.</p>Formule :C10H13ClODegré de pureté :99.5%Couleur et forme :White Crystals Or PowderMasse moléculaire :184.66Branaplam
CAS :<p>Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.</p>Formule :C22H27N5O2Degré de pureté :98.28% - 99.72%Couleur et forme :SolidMasse moléculaire :393.48(R)-baclofen
CAS :<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Formule :C10H12ClNO2Degré de pureté :97.20% - 98.94%Couleur et forme :SolidMasse moléculaire :213.66CL 218872
CAS :<p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>Formule :C13H9F3N4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :278.23ML-SA1
CAS :<p>ML-SA1 (Mucolipin synthetic agonist 1) is a selective TRPML agonist, inhibits DENV2 and ZIKV by promoting lysosomal acidification and protease activity.</p>Formule :C22H22N2O3Degré de pureté :99.34% - 99.71%Couleur et forme :SolidMasse moléculaire :362.42WS-12
CAS :<p>WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)</p>Formule :C18H27NO2Degré de pureté :99.99%Couleur et forme :Whitish To White Solid CrystallineMasse moléculaire :289.41Revaprazan
CAS :<p>Revaprazan: novel, K⁺-competitive acid blocker; reversibly halts gastric H⁺/K⁺-ATPase; rivals PPIs in acid reduction.</p>Formule :C22H23FN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :362.44TGN-020
CAS :<p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>Formule :C8H6N4OSDegré de pureté :99.54% - 99.99%Couleur et forme :SolidMasse moléculaire :206.22Ko 143
CAS :<p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>Formule :C26H35N3O5Degré de pureté :99.01% - 99.89%Couleur et forme :SolidMasse moléculaire :469.57Tenatoprazole
CAS :<p>Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).</p>Formule :C16H18N4O3SDegré de pureté :99.57%Couleur et forme :White Crystalline PowderMasse moléculaire :346.4(E)-KPT330
CAS :<p>(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.</p>Formule :C17H11F6N7ODegré de pureté :98.69% - 99.49%Couleur et forme :SolidMasse moléculaire :443.31H3B-120
CAS :<p>H3B-120: selective, competitive CPS1 inhibitor with anti-cancer properties. IC50: 1.5 μM, Ki: 1.4 μM.</p>Formule :C19H24N4O2SDegré de pureté :99.03% - 99.2%Couleur et forme :SolidMasse moléculaire :372.48BZAD01
CAS :<p>BZAD01 is a selective NMDA NR1A/2B receptor antagonist.</p>Formule :C16H12F6N2ODegré de pureté :99.61% - 99.70%Couleur et forme :SolidMasse moléculaire :362.27DHQ
CAS :<p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>Formule :C8H6N2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :162.15Valbenazine
CAS :<p>Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.</p>Formule :C24H38N2O4Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :418.57ICA 110381
CAS :<p>ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsy</p>Formule :C12H8Cl2N2ODegré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :267.116-Aminonicotinic acid
CAS :<p>6-Aminonicotinic acid is a natural product.</p>Formule :C6H6N2O2Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :138.1238Guanosine 5'-diphosphate
CAS :<p>Guanosine 5'-diphosphate (GDP) as Potential Iron Mobilizer, Preventing the Hepcidin-Ferroportin Interaction and Modulating the Interleukin-6/Stat-3 Pathway.</p>Formule :C10H15N5O11P2Degré de pureté :98.46% - 99.52%Couleur et forme :SolidMasse moléculaire :443.2M8-B Hydrochloride
CAS :<p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>Formule :C22H25ClN2O3SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :432.96Rufinamide
CAS :<p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>Formule :C10H8F2N4ODegré de pureté :99.77% - >99.99%Couleur et forme :White PowderMasse moléculaire :238.19Fosphenytoin disodium
CAS :<p>Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blocker</p>Formule :C16H13N2Na2O6PDegré de pureté :99.97%Couleur et forme :White Crystalline PowderMasse moléculaire :406.24Phenyl benzoate
CAS :<p>Phenyl benzoate is a benzoate ester obtained by the formal condensation of phenol with benzoic acid.It is an important organic synthesis intermediate.</p>Formule :C13H10O2Degré de pureté :99.63%Couleur et forme :White Crystalline PowderMasse moléculaire :198.22Chloroprocaine hydrochloride
CAS :<p>Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.</p>Formule :C13H20Cl2N2O2Degré de pureté :99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :307.22Vonoprazan fumarate
CAS :<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Formule :C17H16FN3O2S·C4H4O4Degré de pureté :99.16% - 99.98%Couleur et forme :SolidMasse moléculaire :461.46AZD7325
CAS :<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Formule :C19H19FN4O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :354.38Elobixibat hydrate
CAS :<p>Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.</p>Formule :C36H47N3O8S2Couleur et forme :SolidMasse moléculaire :713.9Revaprazan hydrochloride
CAS :<p>Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.</p>Formule :C22H24ClFN4Degré de pureté :99.62% - 99.91%Couleur et forme :SolidMasse moléculaire :398.9NS 11021
CAS :<p>NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channels</p>Formule :C16H9BrF6N6SDegré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :511.24L-Phenylalanine-15N
CAS :<p>L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.</p>Formule :C9H11NO2Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :166.18Ilaprazole
CAS :<p>Ilaprazole (IY-81149) is a proton pump inhibitor used in the treatment of dyspepsia gastroesophageal reflux disease (GORD/GERD) and duodenal ulcer.</p>Formule :C19H18N4O2SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :366.44Elacridar
CAS :<p>Elacridar (GG918) is a potent inhibitor of P-glycoprotein and BCRP.Cost-effective and quality-assured.</p>Formule :C34H33N3O5Degré de pureté :98.12% - >99.99%Couleur et forme :SolidMasse moléculaire :563.64Lansoprazole sodium
CAS :<p>Lansoprazole sodium is a PPI used to treat acid reflux and peptic ulcers.</p>Formule :C16H13F3N3NaO2SDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :391.34DS-1971a
CAS :<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Formule :C20H21ClFN5O3SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :465.93Tenatoprazole sodium
CAS :<p>Tenatoprazole sodium is a potent proton pump inhibitor with an IC50 of 6.2 μM against hog gastric H+/K+-ATPase.</p>Formule :C16H17N4NaO3SCouleur et forme :SolidMasse moléculaire :368.391-Aminocyclobutanecarboxylic acid
CAS :<p>1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].</p>Formule :C5H9NO2Degré de pureté :99.94%Couleur et forme :White To Tan Powder Crystals Crystalline Powder And/Or With ChunksMasse moléculaire :115.13O4I2
CAS :<p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>Formule :C12H11ClN2O2SDegré de pureté :97.97% - 99.84%Couleur et forme :SolidMasse moléculaire :282.75MDK-4025
CAS :<p>MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.</p>Formule :C19H15ClODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :294.77AMG 333
CAS :<p>AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.</p>Formule :C20H12F5N3O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :453.32Efonidipine hydrochloride
CAS :<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Formule :C34H39ClN3O7PCouleur et forme :SolidMasse moléculaire :668.12Lorediplon
CAS :<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Formule :C20H15FN4O2SDegré de pureté :99.12% - 99.19%Couleur et forme :SolidMasse moléculaire :394.42Phenibut (hydrochloride)
CAS :<p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>Formule :C10H14ClNO2Degré de pureté :99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :215.68(S)-(-)-5-Fluorowillardiine
CAS :<p>(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonist</p>Formule :C7H8FN3O4Degré de pureté :99.69%Couleur et forme :Off-White SolidMasse moléculaire :217.15Tirofiban hydrochloride monohydrate
CAS :<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Formule :C22H39ClN2O6SDegré de pureté :98.81% - >99.99%Couleur et forme :White SolidMasse moléculaire :495.07β-Pompilidotoxin Acetate
<p>β-Pompilidotoxin Acetate is a wasp venom peptide.</p>Formule :C73H128N22O19Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :1617.93L-Allylglycine
CAS :<p>L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.</p>Formule :C5H9NO2Degré de pureté :≥98%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :115.13HC-056456
CAS :<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formule :C12H6N2O4S2Degré de pureté :99.62% - 99.65%Couleur et forme :SolidMasse moléculaire :306.32OAC3
CAS :<p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>Formule :C15H11FN2ODegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :254.26Azimilide Dihydrochloride
CAS :<p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>Formule :C23H30Cl3N5O3Degré de pureté :97.59% - ≥95%Couleur et forme :SolidMasse moléculaire :530.88QX-222 chloride
CAS :<p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>Formule :C13H21ClN2ODegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :256.77Tiludronate
CAS :<p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>Formule :C7H9ClO6P2SCouleur et forme :SolidMasse moléculaire :318.61SB-705498
CAS :<p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>Formule :C17H16BrF3N4ODegré de pureté :99.57% - ≥95%Couleur et forme :SolidMasse moléculaire :429.23Felbamate
CAS :<p>Felbamate (W-554) is an Anti-epileptic Agent.</p>Formule :C11H14N2O4Degré de pureté :99% - >99.99%Couleur et forme :White Powder SolidMasse moléculaire :238.24L-DABA
CAS :<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Formule :C4H10N2O2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :118.13AMG9810
CAS :<p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>Formule :C21H23NO3Degré de pureté :99.79% - 99.95%Couleur et forme :SolidMasse moléculaire :337.41ML213
CAS :<p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>Formule :C17H23NODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :257.37TCN 213
CAS :<p>TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2B</p>Formule :C18H24N4OS2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :376.54Sepimostat dimethanesulfonate
CAS :<p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>Formule :C23H27N5O8S2Couleur et forme :SolidMasse moléculaire :565.62Levcromakalim
CAS :<p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>Formule :C16H18N2O3Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :286.33Flecainide acetate
CAS :<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formule :C19H24F6N2O5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :474.39NS6180
CAS :<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Formule :C16H12F3NOSDegré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :323.33Selamectin
CAS :<p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>Formule :C43H63NO11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :769.96O4I1
CAS :<p>O4I1 is an effective Oct3/4 inducer.</p>Formule :C16H15NO2Degré de pureté :96.25% - 99.47%Couleur et forme :SolidMasse moléculaire :253.39-Phenanthrol
CAS :<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Formule :C14H10ODegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :194.23Methyl homoveratrate
CAS :<p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>Formule :C11H14O4Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :210.23MK6-83
CAS :<p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>Formule :C16H20N2O2S2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :336.47VK-II-36
CAS :<p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>Formule :C26H26N2O5Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :446.49ICA-069673
CAS :<p>ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).</p>Formule :C11H6ClF2N3ODegré de pureté :99.04% - 99.68%Couleur et forme :SolidMasse moléculaire :269.63Tricaine methanesulfonate
CAS :<p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>Formule :C10H15NO5SDegré de pureté :99.259% - 99.86%Couleur et forme :White PowderMasse moléculaire :261.30TKIM
CAS :<p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>Formule :C18H14ClN3O2SDegré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :371.84Budipine
CAS :<p>Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.</p>Formule :C21H27NDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :293.45SSD114 HCl
CAS :<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formule :C18H21ClF3N3ODegré de pureté :99.03% - 99.95%Couleur et forme :SolidMasse moléculaire :387.832'-O-Methylisoliquiritigenin
CAS :<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28Saclofen
CAS :<p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>Formule :C9H12ClNO3SDegré de pureté :99.17%Couleur et forme :White Crystalline SolidMasse moléculaire :249.71TRPM4-IN-1
CAS :<p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>Formule :C15H11Cl2NO4Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :340.16BzATP triethylammonium salt
CAS :<p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>Formule :C30H39N6O15P3Degré de pureté :95% - 99.57%Couleur et forme :SolidMasse moléculaire :816.59Bifemelane
CAS :<p>Bifemelane, a nootropic, releases Ca2+ from stores and enables its entry via channels for astrocyte research.</p>Formule :C18H23NOCouleur et forme :SolidMasse moléculaire :269.38YHO-13351
CAS :<p>YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.</p>Formule :C27H37N3O7S2Degré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :579.73AER-271
CAS :<p>AER-271 is an inhibitor of aquaporin-4.</p>Formule :C15H9ClF6NO5PDegré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :463.65Pico145
CAS :<p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>Formule :C23H20ClF3N4O5Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :524.884-Acetamidobutanoic acid
CAS :<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16Esomeprazole potassium salt
CAS :<p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>Formule :C17H18KN3O3SCouleur et forme :SolidMasse moléculaire :383.517-Chlorokynurenic acid sodium salt
CAS :<p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>Formule :C10H6ClNNaO3Couleur et forme :SolidMasse moléculaire :246.6Ilaprazole sodium
CAS :<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formule :C19H17N4NaO2SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :388.42Dotinurad
CAS :<p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>Formule :C14H9Cl2NO4SDegré de pureté :97.43% - 98.04%Couleur et forme :SolidMasse moléculaire :358.2AC1903
CAS :<p>AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.</p>Formule :C19H17N3ODegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :303.36Basmisanil
CAS :<p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>Formule :C21H20FN3O5SDegré de pureté :99.21% - 99.42%Couleur et forme :SolidMasse moléculaire :445.46Ralfinamide
CAS :<p>Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.</p>Formule :C17H19FN2O2Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :302.34Homo-VK-II-36
CAS :<p>Homo-VK-II-36 (Homo-V-II-36) is a carvedilol analogue that acts by inhibiting store- overload-induced calcium release through the RyR2 channel.</p>Formule :C27H28N2O5Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :460.52Acamprosate calcium
CAS :<p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>Formule :C10H20CaN2O8S2Degré de pureté :98% - 99.93%Couleur et forme :White Odorless Or Nearly Odorless PowderMasse moléculaire :400.48Quadrol
CAS :<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formule :C14H32N2O4Degré de pureté :99.91% - 99.92%Couleur et forme :Viscous Liquid Liquid ViscousMasse moléculaire :292.41S107
CAS :<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formule :C11H15NOSDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :209.31Ocinaplon
CAS :<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formule :C17H11N5ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :301.3Quinine hydrobromide
CAS :<p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>Formule :C20H25BrN2O2Couleur et forme :SolidMasse moléculaire :405.336(-)-Blebbistatin
CAS :<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Formule :C18H16N2O2Degré de pureté :99.38% - 99.61%Couleur et forme :SolidMasse moléculaire :292.33Vanillyl butyl ether
CAS :<p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>Formule :C12H18O3Degré de pureté :99.57%Couleur et forme :Yellowish Liquid LiquidMasse moléculaire :210.27Metaflumizone
CAS :<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Formule :C24H16F6N4O2Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :506.40Esomeprazole hemistrontium
CAS :<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Formule :C34H36N6O6S2SrCouleur et forme :SolidMasse moléculaire :776.44LY 303511 hydrochloride
CAS :<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Formule :C19H19ClN2O2Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :342.82NBI-98782
CAS :<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Formule :C19H29NO3Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :319.44ICA-121431
CAS :<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Formule :C23H19N3O3S2Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :449.55Ropivacaine hydrochloride monohydrate
CAS :<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Formule :C17H29ClN2O2Degré de pureté :99.94% - 99.95%Couleur et forme :White SolidMasse moléculaire :328.88Arecaidine hydrochloride
CAS :<p>Arecaidine hydrochloride may have carcinogenesis.</p>Formule :C7H12ClNO2Degré de pureté :99.69% - ≥95%Couleur et forme :SolidMasse moléculaire :177.63Cis-ACBD
CAS :<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formule :C6H9NO4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :159.14Neboglamine
CAS :<p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>Formule :C13H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.34Guan-fu base A hydrochloride(1394-48-5 free base)
CAS :<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formule :C24H32NO6ClDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :465.97Parimifasor
CAS :<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formule :C18H11Cl2F4N5ODegré de pureté :96.77% - 98.97%Couleur et forme :SolidMasse moléculaire :460.21Lansoprazole sulfone
CAS :<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Formule :C16H14F3N3O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :385.36Ralfinamide mesylate
CAS :<p>Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.</p>Formule :C18H23FN2O5SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :398.45A2793
CAS :<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formule :C13H12ClNO3Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :265.69PF-06869206
CAS :<p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>Formule :C15H14ClF3N4O2Degré de pureté :99.79% - 99.88%Couleur et forme :SolidMasse moléculaire :374.75Vonoprazan Fumarate
CAS :<p>Vonoprazan Fumarate (TAK438) , a novel potassium-competitive acid blocker, inhibits gastric acid secretion.</p>Formule :C21H20FN3O6SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :461.46MDR-652
CAS :<p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>Formule :C22H23ClFN3O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :447.95Kv2-IN-A1
CAS :<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Formule :C20H17ClN4OSDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :396.89Adjudin
CAS :<p>Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.</p>Formule :C15H12Cl2N4ODegré de pureté :96.51% - ≥95%Couleur et forme :SolidMasse moléculaire :335.19Almitrine mesylate
CAS :<p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>Formule :C28H37F2N7O6S2Degré de pureté :99.96%Couleur et forme :CoaMasse moléculaire :669.76KB-R7943 mesylate
CAS :<p>KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.</p>Formule :C17H21N3O6S2Degré de pureté :99.88% - ≥95%Couleur et forme :SolidMasse moléculaire :427.5Eperisone hydrochloride
CAS :<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formule :C17H26ClNODegré de pureté :99.80%Couleur et forme :White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMasse moléculaire :295.85Miltirone
CAS :<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Formule :C19H22O2Degré de pureté :99.22% - 99.66%Couleur et forme :SolidMasse moléculaire :282.38α-Asarone
CAS :<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Formule :C12H16O3Degré de pureté :99.64% - 99.64%Couleur et forme :Monoclinic Needles From Water Monoclinic Needles From WaterMasse moléculaire :208.25Levamlodipine hydrochloride
CAS :<p>Levamlodipine hydrochloride is a medication used to lower blood pressure and prevent chest pain.</p>Formule :C20H26Cl2N2O5Couleur et forme :SolidMasse moléculaire :445.34Baclofen hydrochloride
CAS :<p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>Formule :C10H13Cl2NO2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :250.122Raxatrigine hydrochloride
CAS :<p>Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.</p>Formule :C18H20ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.82Ataluren
CAS :<p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>Formule :C15H9FN2O3Degré de pureté :99.16% - 99.84%Couleur et forme :SolidMasse moléculaire :284.24Cyclothiazide
CAS :<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formule :C14H16ClN3O4S2Degré de pureté :98.23% - 99.49%Couleur et forme :Crystals From Dilute Alcohol SolidMasse moléculaire :389.88PF-05186462
CAS :<p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>Formule :C19H10ClF4N5O3S2Degré de pureté :99.10% - 99.37%Couleur et forme :SolidMasse moléculaire :531.89Mitiglinide calcium hydrate
CAS :<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formule :C38H52CaN2O8Degré de pureté :98.97% - 99.96%Couleur et forme :White SolidMasse moléculaire :704.91Guanosine 5'-diphosphate disodium salt
CAS :<p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>Formule :C10H13N5Na2O11P2Degré de pureté :99.40%Couleur et forme :White PowderMasse moléculaire :487.16CLP290
CAS :<p>CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatric</p>Formule :C19H21FN4O3SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :404.46DAAO inhibitor-1
CAS :<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Formule :C7H5FN2ODegré de pureté :97.84%Couleur et forme :SolidMasse moléculaire :152.13TRPM8 antagonist 2
CAS :<p>TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.</p>Formule :C26H26N2O2Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :398.5Amifampridine phosphate
CAS :<p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>Formule :C5H10N3O4PCouleur et forme :SolidMasse moléculaire :207.12Argireline
CAS :<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formule :C34H60N14O12SDegré de pureté :96.79% - 99.65%Couleur et forme :White PowderMasse moléculaire :888.99CFTR corrector 2
CAS :<p>CFTR corrector 2 (FDL169) is a novel and potent CFTR corrector for treating cystic fibrosis (CF) patients who carry the F508del mutation.</p>Formule :C27H23FN4O4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :486.49N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride
CAS :<p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>Formule :C16H17ClN4Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :300.79SG-209
CAS :<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Formule :C10H12N2O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :208.21KM11060
CAS :<p>KM11060 is a novel corrector of the F508del-CFTR trafficking defect, Correcting F508del-CFTR trafficking, increasing the amount of functional CFTR at the plasma</p>Formule :C19H17Cl2N3O2SDegré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :422.33Rimeporide
CAS :<p>Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>Formule :C11H15N3O5S2Degré de pureté :97.66%Couleur et forme :SolidMasse moléculaire :333.38(R)-Lansoprazole
CAS :<p>(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitor</p>Formule :C16H14F3N3O2SDegré de pureté :98.09% - 98.99%Couleur et forme :Brown SolidMasse moléculaire :369.36Cabotegravir
CAS :<p>Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (</p>Formule :C19H17F2N3O5Degré de pureté :98.55% - 99.92%Couleur et forme :SolidMasse moléculaire :405.35γ-Acetylenic GABA
CAS :<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Formule :C6H9NO2Couleur et forme :SolidMasse moléculaire :127.143PF-4840154
CAS :<p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) & 23 nM (human); triggers nociception in mice.</p>Formule :C26H38N6O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :466.62DL-Willardiine
CAS :<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Formule :C7H9N3O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :199.16Co 101244 hydrochloride
CAS :<p>Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.</p>Formule :C21H28ClNO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :377.9Procyclidine hydrochloride
CAS :<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Formule :C19H30ClNODegré de pureté :99.24% - 99.88%Couleur et forme :Crystals From Petroleum Ether White PowderMasse moléculaire :323.9CTP disodium dihydrate
CAS :<p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>Formule :C9H18N3Na2O16P3Degré de pureté :98.51%Couleur et forme :White Crystalline PowderMasse moléculaire :563.15AZ194
CAS :<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Formule :C34H31F2N3O3Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :567.62KPT185
CAS :<p>KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.</p>Formule :C16H16F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.31JNJ 303
CAS :<p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>Formule :C21H29ClN2O4SDegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :440.98Anthracene-9-carboxylic acid
CAS :<p>Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI.</p>Formule :C15H10O2Degré de pureté :99.05%Couleur et forme :Yellow Cystalline PowderMasse moléculaire :222.24FGH10019
CAS :<p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>Formule :C18H19N3O2S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :373.49Evenamide
CAS :<p>Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.</p>Formule :C16H26N2O2Degré de pureté :96.74% - 99.15%Couleur et forme :SolidMasse moléculaire :278.39Trofinetide
CAS :<p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>Formule :C13H21N3O6Degré de pureté :98.70% - 99.50%Couleur et forme :SolidMasse moléculaire :315.32Prilocaine
CAS :<p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>Formule :C13H20N2ODegré de pureté :98.49%Couleur et forme :Needles SolidMasse moléculaire :220.31Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Formule :C42H68N14O18S2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :1121.24-Chlorophenylguanidine hydrochloride
CAS :<p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity. </p>Formule :C7H9Cl2N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :206.07HC067047 Hydrochloride(883031-03-6 free base)
CAS :<p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>Formule :C26H29ClF3N3O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :507.98Esomeprazole
CAS :<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Formule :C17H19N3O3SDegré de pureté :97.3%Couleur et forme :SolidMasse moléculaire :345.42Epaminurad
CAS :<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Formule :C14H10Br2N2O3Couleur et forme :SolidMasse moléculaire :414.05ML335
CAS :<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Formule :C15H14Cl2N2O3SDegré de pureté :99.73% - 99.79%Couleur et forme :SolidMasse moléculaire :373.25Glibenclamide potassium
CAS :<p>Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.</p>Formule :C23H27ClKN3O5SCouleur et forme :SolidMasse moléculaire :532.09JNJ-26990990
CAS :<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formule :C9H10N2O2S2Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :242.32Isoflurane
CAS :<p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>Formule :C3H2ClF5ODegré de pureté :98%Couleur et forme :Clear Colorless Liquid LiquidMasse moléculaire :184.49Bisaramil
CAS :<p>Bisaramil is a new class I antiarrhythmic agent.</p>Formule :C17H23ClN2O2Couleur et forme :SolidMasse moléculaire :322.83
