Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(34 produits)
- Cystéine protéase(96 produits)
- DPP-4(20 produits)
- Glutaminase(40 produits)
- Protéase du VIH(447 produits)
- PAI-1(25 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(54 produits)
- Protéasome(94 produits)
- Sérine protéase(50 produits)
- p97(14 produits)
Affichez 3 plus de sous-catégories
1045 produits trouvés pour "Protéases/Protéasome"
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N-CBZ-Phe-Arg-AMC
CAS :<p>Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.</p>Formule :C33H36N6O6Degré de pureté :98%Couleur et forme :White To Off-White PowderMasse moléculaire :612.68Zetomipzomib maleate
CAS :<p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>Formule :C34H46N4O12Couleur et forme :SolidMasse moléculaire :702.758CRA-2059
CAS :<p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>Formule :C34H46N12O8Degré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :750.818ADAM8-IN-1
CAS :<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Formule :C44H44Br4N6O12S2Couleur et forme :SolidMasse moléculaire :1232.6MMP-3 Inhibitor
CAS :<p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>Formule :C27H46N10O9SDegré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :686.78(-)-Taxifolin
CAS :<p>(-)-Taxifolin, less active enantiomer with anti-tyrosinase, collagenase inhibition (IC50 = 193.3 μM), antifibrotic, antioxidant properties.</p>Formule :C15H12O7Couleur et forme :SolidMasse moléculaire :304.25TP0597850
CAS :<p>TP0597850, a selective MMP2 inhibitor with an IC50 value of 0.22 nM, demonstrates a prolonged dissociation half-life from MMP2 (t1/2 = 265 minutes) [1].</p>Formule :C41H57N9O13SCouleur et forme :SolidMasse moléculaire :916.01TAPI1 acetate
<p>TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .</p>Formule :C28H41N5O7Degré de pureté :98.82% - 99.94%Couleur et forme :SolidMasse moléculaire :559.65Leptosin D
CAS :<p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>Formule :C25H24N4O3S2Couleur et forme :SolidMasse moléculaire :492.61HCVP-IN-1
CAS :<p>HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.</p>Formule :C30H34FN5O3Couleur et forme :SolidMasse moléculaire :531.632Cathepsin K inhibitor 7
<p>Cathepsin K Inhibitor7 (compound 7) is an inhibitor of Cathepsin K, exhibiting a pKi value of 7.3. It is utilized in research on osteoporosis.</p>Couleur et forme :Odour SolidSofosbuvir impurity A
CAS :<p>Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.</p>Formule :C22H29FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.45Imitrodast
CAS :<p>Imitrodast is a small molecule thromboxane A2 synthase (TXA2 synthase) inhibitor for the treatment of immune system disorders, respiratory disorders, and</p>Formule :C13H12N2O2SDegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :260.31Ellipyrone A
<p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>Formule :C25H34O8Couleur et forme :SolidMasse moléculaire :462.53Neutrophil elastase inhibitor 4
<p>Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.</p>Formule :C20H21N3O5Couleur et forme :SolidMasse moléculaire :383.4HCV-IN-4
CAS :<p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>Formule :C52H58FN9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :956.07Chetoseminudin B
CAS :<p>Chetoseminudin B exhibits inhibitory activity against mushroom tyrosinase, with an IC 50 value of 31.7 μM [1].</p>Formule :C17H21N3O3S2Couleur et forme :SolidMasse moléculaire :379.5Sofosbuvir impurity J
CAS :<p>Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formule :C22H30FN4O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.476-Acetylnimbandiol
CAS :<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Formule :C28H34O8Couleur et forme :SolidMasse moléculaire :498.56α 1(I) Collagen (614-639), human
CAS :<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Formule :C134H189N37O39Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2942.16PF 00356231
CAS :<p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>Formule :C25H20N2O3SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :428.5Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2
CAS :<p>Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).</p>Formule :C49H68N14O12SCouleur et forme :SolidMasse moléculaire :1077.22Bictegravir Sodium
CAS :<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Formule :C21H17F3N3NaO5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :471.36HIV-1 inhibitor-6
CAS :<p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>Formule :C14H10N4O4SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :330.32JC-10
CAS :<p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>Formule :C25H29Cl2IN4Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :583.34Enzyme-IN-1
CAS :<p>Enzyme-IN-1（compound 1）为基于肽的N端亲核试剂（Ntn）水解酶抑制剂，特别针对20S蛋白酶体的糜胰蛋白酶样活性（CT-L）进行抑制，可能展现出抗炎特性。</p>Formule :C36H50N4O7Couleur et forme :SolidMasse moléculaire :650.8Cepeginterferon alfa-2b
CAS :<p>Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.</p>Couleur et forme :LiquidCys-TAT(47-57) acetate(583836-55-9 Free base)
<p>Cys-TAT(47-57) acetate is derived from the HIV-1 transactivating protein. Cys-TAT(47-57) acetate is an arginine rich peptide that can penetrate cells.</p>Formule :C69H128N34O16SDegré de pureté :95.1100%Couleur et forme :SolidMasse moléculaire :1722.04RJS308
<p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>Formule :C63H75N13O11SCouleur et forme :SolidMasse moléculaire :1222.42Talabostat isomer mesylate
<p>Talabostat isomer mesylate, a PT100/Val-boroPro variant, is a potent oral DPP-IV inhibitor (Ki: 0.18 nM).</p>Formule :C10H23BN2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.18PPACK II
CAS :<p>PPACK II is an irreversible and specific glandular and plasma kallikreins inhibitor [1] .</p>Formule :C25H33ClN6O3Couleur et forme :SolidMasse moléculaire :501.02Rivulariapeptolides 1121
<p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>Formule :C56H83N9O15Couleur et forme :SolidMasse moléculaire :1122.31Fotagliptin
CAS :<p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>Formule :C17H19FN6OCouleur et forme :SolidMasse moléculaire :342.37N-CBZ-Phe-Arg-AMC TFA
<p>N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.</p>Formule :C35H37F3N6O8Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :726.7CRA-2059 hydrochloride
<p>CRA-2059 hydrochloride is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].</p>Couleur et forme :Solid7-Methoxy obtusifolin
CAS :<p>7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentration</p>Formule :C17H14O6Couleur et forme :SolidMasse moléculaire :314.29Tyrosinase/elastase-IN-1
<p>Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase</p>Formule :C33H52O5Couleur et forme :SolidMasse moléculaire :528.76DPP8/9-IN-1
<p>DPP8/9-IN-1 (Compound 16) is a selective covalent inhibitor of dipeptidyl peptidase 8 and 9 (DPP8/9), with IC50 values of 14 nM and 298 nM, respectively. It irreversibly binds to the active site serine (such as S730 in DPP9) through a phosphate ester warhead, blocking substrate binding and inhibiting DPP8/9-mediated protein processing. DPP8/9-IN-1 holds potential for research in cancer and inflammatory diseases.</p>Couleur et forme :Odour SolidSofigatran
CAS :<p>Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.</p>Formule :C24H44N4O4SCouleur et forme :SolidMasse moléculaire :484.7L 659286
CAS :<p>L 659286 is one kind of cephalosporin derivative.</p>Formule :C17H21N5O7S2Couleur et forme :SolidMasse moléculaire :471.51Nitidanin
<p>Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.</p>Formule :C21H24O8Couleur et forme :SolidMasse moléculaire :404.415Dutogliptin tartrate
CAS :<p>Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>Formule :C14H26BN3O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.18NS5A-IN-1
<p>NS5A-IN-1 is a proagent of the HCV NS5A inhibitor Pibrentasvir (ABT-530).</p>Formule :C72H86F5N10O14PCouleur et forme :SolidMasse moléculaire :1441.48Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS :<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Formule :C47H64N14O10Couleur et forme :SolidMasse moléculaire :985.1Sofosbuvir impurity M
CAS :<p>Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formule :C22H30N3O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.467Cathepsin D and E FRET Substrate
CAS :<p>Mca-GKPILFFRL-Dpa-r-amide, FRET substrate for cathepsin D and E. Also cleaved by napsin A.</p>Formule :C85H122N22O19Couleur et forme :SolidMasse moléculaire :1756.046FFAGLDD TFA
<p>FFAGLDD TFA: MMP9 peptide for controlled DOX delivery to cytoplasm.</p>Formule :C39H50F3N7O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :897.85L-Methionine-DL-sulfoximine
CAS :<p>MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.</p>Formule :C5H12N2O3SDegré de pureté :99.56% - ≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :180.23NS5A-IN-4
CAS :<p>NS5A-IN-4 (Compound 1.12) is a hepatitis C inhibitor effective against multiple genotypes, with IC50 values ranging from 1.2 to 2296 pM.</p>Formule :C47H48N8O6Couleur et forme :SolidMasse moléculaire :820.93GCPII-IN-1
CAS :<p>GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.</p>Formule :C12H21N3O7Couleur et forme :SolidMasse moléculaire :319.314AL-611
CAS :<p>AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).</p>Formule :C25H33F2N6O8PCouleur et forme :SolidMasse moléculaire :614.544Radalbuvir
CAS :<p>Radalbuvir (GS-9669) is an investigational antiviral agent for the treatment of hepatitis C virus (HCV) infection as an NS5B inhibitor.</p>Formule :C30H41NO6SCouleur et forme :SolidMasse moléculaire :543.71Rivulariapeptolides 1155
<p>Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).</p>Formule :C59H81N9O15Couleur et forme :SolidMasse moléculaire :1156.33Recombinant Proteinase K
<p>Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.</p>Couleur et forme :SolidGSK2336805
CAS :<p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>Formule :C42H52N8O8Couleur et forme :SolidMasse moléculaire :796.91Leptosphaerodione
CAS :<p>Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.</p>Formule :C21H22O5Couleur et forme :SolidMasse moléculaire :354.4Histargin
CAS :<p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>Formule :C14H25N7O4Couleur et forme :SolidMasse moléculaire :355.39Proteasome-IN-7
<p>Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.</p>Formule :C48H56N6O10SCouleur et forme :SolidMasse moléculaire :909.06Peptide 74
CAS :<p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>Formule :C62H107N23O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1558.79α 1 Antichymotrypsin, Human Plasma
CAS :<p>Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.</p>Couleur et forme :SolidAPC-6860
CAS :<p>APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.</p>Formule :C9H7IN2SCouleur et forme :SolidMasse moléculaire :302.13PSI-7409
CAS :<p>PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).</p>Formule :C10H16FN2O14P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.16AMG-222
CAS :<p>AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.</p>Formule :C32H39N9O3Couleur et forme :SolidMasse moléculaire :597.71Ac-VDQQD-pNA
CAS :<p>Ac-VDQQD-pNA serves as a substrate for Caspase 2, which cleaves it to yield the yellow compound pNA (p-nitroaniline).</p>Formule :C31H43N9O14Couleur et forme :SolidMasse moléculaire :765.73Sitagliptin fenilalanil hydrochloride
CAS :<p>Sitagliptin phenylalanine hydrochloride, a dipeptidyl peptidase-4 (DPP-4) inhibitor [1], is a chemical compound utilized in medical applications.</p>Formule :C25H25ClF6N6O2Couleur et forme :SolidMasse moléculaire :590.95PS 915
CAS :<p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>Formule :C27H36ClN7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.08Fotagliptin benzoate
CAS :<p>Fotagliptin benzoate, a DPP-4 inhibitor (IC50=2.27 nM), is safe in rats/dogs, useful for Type 2 diabetes research.</p>Formule :C24H25FN6O3Couleur et forme :SolidMasse moléculaire :464.49HCV-IN-41
CAS :<p>HCV-IN-41: potent HCV inhibitor; EC50 - 0.006762 nM (1b), 5.183 nM (2a), 1.365 nM (3a), 142.2 nM (4a); hinders RNA replication.</p>Formule :C48H56N6O8Couleur et forme :SolidMasse moléculaire :844.99Befovacimab
CAS :<p>Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.</p>Couleur et forme :LiquidBerotralstat
CAS :<p>Berotralstat (BCX7353) is an oral, low-toxicity, specific kallikrein inhibitor for hereditary angioedema research, blocking bradykinin release.</p>Formule :C30H26F4N6OCouleur et forme :SolidMasse moléculaire :562.56Tyrosinase-IN-34
<p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>Formule :C19H14BrClN4OCouleur et forme :SolidMasse moléculaire :429.7Histatin 5 (TFA)(115966-68-2,free)
<p>Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM</p>Formule :C135H196F3N51O35Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3150.32NVP-DPP728 dihydrochloride
CAS :<p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>Formule :C15H20Cl2N6OCouleur et forme :SolidMasse moléculaire :371.27Stevia Powder
<p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>Couleur et forme :Odour SolidCP-346086 dihydrate
CAS :<p>CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.</p>Formule :C26H26F3N5O3Couleur et forme :SolidMasse moléculaire :513.521Ecallantide TFA
<p>Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention of</p>Couleur et forme :Odour SolidPseudostellarin G
CAS :<p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>Formule :C42H56N8O9Couleur et forme :SolidMasse moléculaire :816.94MK-6169
CAS :<p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>Formule :C54H62FN9O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1016.2KKI-5
CAS :<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Formule :C35H55N11O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :773.88Dutogliptin
CAS :<p>Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>Formule :C10H20BN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :241.10CL 82198 hydrochloride
CAS :<p>CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.</p>Formule :C17H23ClN2O3Couleur et forme :SolidMasse moléculaire :338.83Acetyl-Calpastatin(184-210)(human)
CAS :<p>Calpain inhibitor, Ki 0.2 nM for calpain I/II, doesn't affect papain/trypsin/cat L. Raises Aβ42, Aβ40 secretion & Aβ42/Aβ40 ratio.</p>Formule :C142H230N36O44SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3177.65Anticancer agent 114
<p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>Formule :C28H33BF6N2O7Couleur et forme :SolidMasse moléculaire :634.37AP-C2
CAS :<p>AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.</p>Formule :C18H16N4SDegré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :320.41C-telopeptide
CAS :<p>C-telopeptide from type I collagen is released during bone resorption; it correlates with bone mineral density.</p>Formule :C34H56N14O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :868.9Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Formule :C15H19NO3Couleur et forme :SolidMasse moléculaire :261.32EP 171
CAS :<p>EP 171 is a potent agonist of TP-receptors.</p>Formule :C23H29FO5Couleur et forme :SolidMasse moléculaire :404.47Elastatinal
CAS :<p>Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.</p>Formule :C21H36N8O7Couleur et forme :Yellowish SolidMasse moléculaire :512.56Ac-DEMEEC-OH
CAS :<p>Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.</p>Formule :C29H44N6O16S2Couleur et forme :SolidMasse moléculaire :796.82HIV-1 TAT (48-60) Acetate
<p>Lilotomab (HH1) is a murine anti-CD37 antibody that can be used to synthesize anti-CD37 antibody-radionuclide couplings.</p>Formule :C72H135N35O18Degré de pureté :99.93%Couleur et forme :SoildMasse moléculaire :1779.07STK33-IN-1
CAS :<p>STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.</p>Formule :C24H27N7O2Couleur et forme :SolidMasse moléculaire :445.527GSK2818713
CAS :<p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>Formule :C46H56N8O8Couleur et forme :SolidMasse moléculaire :849.002FiVe1
CAS :<p>FiVe1 is a vimentin-binding compound that disrupts mitosis in cancer cells, causing cell death, with an IC50 of 234 nM in FOXC2-HMLER.</p>Formule :C18H16Cl2N4Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :359.25BMS-767778
CAS :<p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Formule :C19H20Cl2N4O2Couleur et forme :SolidMasse moléculaire :407.29Linagliptin Methyldimer
CAS :<p>Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.</p>Formule :C50H56N16O4Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :945.08RXP470
CAS :<p>RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).</p>Formule :C35H35BrClN4O10PCouleur et forme :SolidMasse moléculaire :818Plasma kallikrein-IN-1
CAS :<p>Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.</p>Formule :C23H25F2N7OCouleur et forme :SolidMasse moléculaire :453.498Paritaprevir dihydrate
CAS :<p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>Formule :C40H47N7O9SCouleur et forme :SolidMasse moléculaire :801.91CTTHWGFTLC, CYCLIC
CAS :<p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>Formule :C52H71N13O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1166.33midesteine
CAS :<p>Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.</p>Formule :C12H13NO3S3Degré de pureté :99.52% - 99.98%Couleur et forme :SolidMasse moléculaire :315.43
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