Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(38 produits)
- Cystéine protéase(111 produits)
- DPP-4(24 produits)
- Glutaminase(44 produits)
- Protéase du VIH(505 produits)
- PAI-1(26 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(54 produits)
- Protéasome(89 produits)
- Sérine protéase(54 produits)
- p97(15 produits)
Affichez 3 plus de sous-catégories
987 produits trouvés pour "Protéases/Protéasome"
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Berotralstat
CAS :Berotralstat (BCX7353) is an oral, low-toxicity, specific kallikrein inhibitor for hereditary angioedema research, blocking bradykinin release.Formule :C30H26F4N6OCouleur et forme :SolidMasse moléculaire :562.56EP 171
CAS :EP 171 is a potent agonist of TP-receptors.Formule :C23H29FO5Couleur et forme :SolidMasse moléculaire :404.47Fotagliptin benzoate
CAS :Fotagliptin benzoate, a DPP-4 inhibitor (IC50=2.27 nM), is safe in rats/dogs, useful for Type 2 diabetes research.Formule :C24H25FN6O3Couleur et forme :SolidMasse moléculaire :464.49Dansyl-Glu-Gly-Arg-Chloromethylketone
CAS :Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activatedFormule :C26H36ClN7O7SCouleur et forme :SolidMasse moléculaire :626.12Iso-VQA-ACC acetate
Iso-VQA-ACC acetate serves as a substrate for the constitutive proteasome.Couleur et forme :Odour SolidRJS308
RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)Formule :C63H75N13O11SCouleur et forme :SolidMasse moléculaire :1222.42Lonodelestat TFA
Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.Formule :C73H112F3N15O21Couleur et forme :SolidMasse moléculaire :1592.75Dazcapistat
CAS :Dazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively.Formule :C21H18FN3O4Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :395.38Ref: TM-T9710
1mg92,00€5mg192,00€10mg289,00€25mg522,00€50mg732,00€100mg1.018,00€1mL*10mM (DMSO)212,00€Z-Leu-Tyr-Chloromethylketone
CAS :Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].Formule :C24H29ClN2O5Couleur et forme :SolidMasse moléculaire :460.95Obtusifolin-2-O-glucoside
CAS :Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].Formule :C22H22O10Couleur et forme :SolidMasse moléculaire :446.4Histatin 5 TFA
Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μMFormule :C135H196N51F3O35Couleur et forme :SolidMasse moléculaire :3150.31Sitagliptin fenilalanil hydrochloride
CAS :Sitagliptin phenylalanine hydrochloride, a dipeptidyl peptidase-4 (DPP-4) inhibitor [1], is a chemical compound utilized in medical applications.Formule :C25H25ClF6N6O2Couleur et forme :SolidMasse moléculaire :590.95Sadopeptins A
Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].Formule :C49H71N9O13SCouleur et forme :SolidMasse moléculaire :1026.21Cathepsin L-IN-3
CAS :Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.Formule :C41H49N7O4SCouleur et forme :SolidMasse moléculaire :735.94Carboxypeptidase C
CAS :Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.Couleur et forme :SolidN-CBZ-Phe-Arg-AMC TFA
N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.Formule :C35H37F3N6O8Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :726.7JC-10
CAS :JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.Formule :C25H29Cl2IN4Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :583.34CRA-2059 TFA
CRA-2059 is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].Couleur et forme :SolidSulodexide
CAS :Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.Couleur et forme :Solid[Asp371]-Tyrosinase (369-377), human
CAS :Tyrosinase (369-377,YMDGTMSQV) originates from tyrosinase and needs TAP and proteosome for cell presentation.Formule :C42H66N10O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1031.16Tyrosinase-IN-21
Tyrosinase-IN-21 (compound 3g) is a tyrosinase inhibitor with an IC50 value of 80.93 μM.Formule :C23H20N4O3S2Masse moléculaire :464.09768TR-107
CAS :TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.Formule :C22H19ClN4OCouleur et forme :SoildMasse moléculaire :390.87MMP-3 Inhibitor acetate
MMP-3 Inhibitor acetate is a cell-permeable and potent inhibitor of human MMP-3.Formule :C29H50N10O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :746.83Ref: TM-T37048L
1mg175,00€5mg394,00€10mg590,00€25mg1.060,00€50mg1.591,00€100mg2.387,00€200mg3.580,00€BI-1230
CAS :BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.Formule :C42H52N6O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :816.96ADAM8-IN-1
CAS :ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.
Formule :C44H44Br4N6O12S2Couleur et forme :SolidMasse moléculaire :1232.6Tyrosinase-IN-36
Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.Couleur et forme :Odour SolidLinagliptin Methyldimer
CAS :Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.Formule :C50H56N16O4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :945.08HCVP-IN-1
CAS :HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.Formule :C30H34FN5O3Couleur et forme :SolidMasse moléculaire :531.632HCV-IN-4
CAS :HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.Formule :C52H58FN9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :956.07MMP-3 Inhibitor
CAS :MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.Formule :C27H46N10O9SDegré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :686.78Ref: TM-T37048
1mg77,00€5mg197,00€10mg294,00€25mg497,00€50mg717,00€100mg982,00€500mg1.998,00€1mL*10mM (DMSO)210,00€Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS :Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effectFormule :C47H64N14O10Couleur et forme :SolidMasse moléculaire :985.1LM11
LM11 is a transglutaminase 2 (TG2) inhibitor that exhibits activity against glioblastoma cells by maintaining TG2 in a cytotoxic conformational state.
Formule :C26H18Cl2N4O5Masse moléculaire :536.06543Leptosin D
CAS :Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)Formule :C25H24N4O3S2Couleur et forme :SolidMasse moléculaire :492.61Pirmitegravir
CAS :Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.
Formule :C27H31ClN4O3Degré de pureté :99.79% - 99.79%Couleur et forme :SolidMasse moléculaire :495.01GPLGLAGGWGERDGS
CAS :GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.Formule :C61H93N19O21Couleur et forme :SolidMasse moléculaire :1428.51HCV-IN-7 hydrochloride
CAS :HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.Formule :C40H50Cl2N8O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :841.85Ichorcumab
CAS :Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.
Couleur et forme :Liquid15,16-Dihydrotanshindiol C
15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.Formule :C18H18O5Couleur et forme :SolidMasse moléculaire :314.337Grazoprevir potassium salt
CAS :Grazoprevir, a drug for hepatitis C, is a second-gen NS3/4a protease inhibitor.
Formule :C38H49KN6O9SCouleur et forme :SolidMasse moléculaire :805Relacatib
CAS :Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.Formule :C27H32N4O6SCouleur et forme :SolidMasse moléculaire :540.646,6′-Dihydroxythiobinupharidine
CAS :6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-foldFormule :C30H42N2O4SCouleur et forme :SolidMasse moléculaire :526.73Ac-PAL-AMC
CAS :Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.Formule :C26H34N4O6Couleur et forme :SolidMasse moléculaire :498.57TWH106
TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.Couleur et forme :Odour SolidTyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Formule :C19H14BrClN4OCouleur et forme :SolidMasse moléculaire :429.7PROTAC CG167
PROTAC CG167 is a potent and selective PROTAC degrader of CypA. It degrades CypA in a dose-dependent manner in Jurkat cells, with a DC50 of 123 nM. Additionally, PROTAC CG167 exhibits antiviral activity by inhibiting HIV-1 and HCV. (Pink: CypA Ligand; Black: Linker; Blue: E3LigaseLigand)Formule :C65H79N13O11SCouleur et forme :SolidMasse moléculaire :1250.47Recombinant Trypsin
Recombinant Trypsin is a serine protease that hydrolyzes proteins at the carboxyl side of lysine or arginine.C-telopeptide
CAS :C-telopeptide from type I collagen is released during bone resorption; it correlates with bone mineral density.Formule :C34H56N14O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :868.9VD2173
CAS :VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.Formule :C31H45N9O6SCouleur et forme :SolidMasse moléculaire :671.81(R)-BAY-85-8501
(R)-BAY-85-8501 is the less active enantiomer of BAY-85-8501. BAY-85-8501 is a selective and potent Human Neutrophil Elastase (HNE)inhibitor(IC50 of 65 pM).Formule :C22H17F3N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.46NIM811
CAS :NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.Formule :C62H111N11O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1202.635Histatin 5 (TFA)(115966-68-2,free)
Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μMFormule :C135H196F3N51O35Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3150.32GSK2336805
CAS :GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.Formule :C42H52N8O8Couleur et forme :SolidMasse moléculaire :796.91PM 102
CAS :Peptide that reverses the anticoagulant effect of heparin. Potently binds heparin (Kd = 36 nM in vitro).Formule :C235H425N111O64Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5830Acetyl-Calpastatin(184-210)(human) TFA
Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.Formule :C144H231F3N36O46SCouleur et forme :SolidMasse moléculaire :3291.65LMP7/LMP2-IN-1
CAS :LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.Formule :C16H27BN4O3Couleur et forme :SoildMasse moléculaire :334.22Micropeptin 478A
CAS :Micropeptin 478A is a plasmin inhibitor from the Cyanobacterium Microcystis aeruginosa.Formule :C40H62ClN9O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :976.49Activated Protein C (390-404), human
CAS :Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.Formule :C91H130N22O23Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1900.14S62798
CAS :S62798 is a highly potent and selective compound that inhibits activated thrombin activatable fibrinolysis inhibitor (TAFIa) with an IC50 value of 6 mM.Formule :C20H28FN4O4PCouleur et forme :SolidMasse moléculaire :438.44Ledipasvir D-tartrate
CAS :Ledipasvir D-tartrate (GS-5885 D-tartrate) is an HCV NS5A inhibitor that suppresses viral overphosphorylation and replicationFormule :C53H60F2N8O12Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :1039.09Ref: TM-T11832
1mg34,00€5mg71,00€10mg92,00€25mg146,00€50mg222,00€100mg401,00€200mg675,00€1mL*10mM (DMSO)94,00€Sofosbuvir impurity K
CAS :Sofosbuvir impurity K is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formule :C22H29ClN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :545.91Isoleucylvaline
CAS :Isoleucylvaline is a dipeptide.Formule :C11H22N2O3Couleur et forme :SolidMasse moléculaire :230.30MMP-12 Inhibitor
CAS :MMP-12 Inhibitor is a selective inhibitor of MMP-12 with IC50s of 2, 160, 320, and 22.3 nM for human, mouse, rat, and sheep MMP-12.
Formule :C19H20N2O7SDegré de pureté :97.51% - 99.96%Couleur et forme :SoildMasse moléculaire :420.44Dutogliptin
CAS :Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.Formule :C10H20BN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :241.10Sofigatran
CAS :Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.Formule :C24H44N4O4SCouleur et forme :SolidMasse moléculaire :484.7Cajaninstilbene acid
CAS :Cajaninstilbene acid is a useful organic compound for research related to life sciences. The catalog number is T124035 and the CAS number is 87402-84-4.Formule :C21H22O4Couleur et forme :SolidMasse moléculaire :338.403Sofosbuvir impurity I
Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formule :C21H27FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.43Talabostat isomer mesylate
Talabostat isomer mesylate, a PT100/Val-boroPro variant, is a potent oral DPP-IV inhibitor (Ki: 0.18 nM).Formule :C10H23BN2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.187-Methoxy obtusifolin
CAS :7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentrationFormule :C17H14O6Couleur et forme :SolidMasse moléculaire :314.29Chetoseminudin B
CAS :Chetoseminudin B exhibits inhibitory activity against mushroom tyrosinase, with an IC 50 value of 31.7 μM [1].Formule :C17H21N3O3S2Couleur et forme :SolidMasse moléculaire :379.5Ac-Phe-Gly-pNA
CAS :Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .Formule :C19H20N4O5Couleur et forme :SolidMasse moléculaire :384.39Nostosin G
Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).Formule :C25H33N5O6Couleur et forme :SolidMasse moléculaire :499.56Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2
CAS :Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).Formule :C49H68N14O12SCouleur et forme :SolidMasse moléculaire :1077.22AL-611
CAS :AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).
Formule :C25H33F2N6O8PCouleur et forme :SolidMasse moléculaire :614.544L 659286
CAS :L 659286 is one kind of cephalosporin derivative.Formule :C17H21N5O7S2Couleur et forme :SolidMasse moléculaire :471.51Nostopeptin B
CAS :Nostopeptin B is an inhibitor of elastase.Formule :C46H70N8O12Couleur et forme :SolidMasse moléculaire :927.11Fotagliptin
CAS :Fotagliptin is a dipeptidyl peptidase IV inhibitor.Formule :C17H19FN6OCouleur et forme :SolidMasse moléculaire :342.37Tyrosinase-IN-32
Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.Formule :C15H19NO3Couleur et forme :SolidMasse moléculaire :261.32NS5A-IN-1
NS5A-IN-1 is a proagent of the HCV NS5A inhibitor Pibrentasvir (ABT-530).Formule :C72H86F5N10O14PCouleur et forme :SolidMasse moléculaire :1441.48Ac-DEMEEC-OH
CAS :Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.Formule :C29H44N6O16S2Couleur et forme :SolidMasse moléculaire :796.82GCPII-IN-1
CAS :GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.
Formule :C12H21N3O7Couleur et forme :SolidMasse moléculaire :319.314Fibrinopeptide B, human
CAS :Fibrinopeptide B (FPB) is produced during the cleavage of fibrinogen, by thrombin, to fibrin monomer.Formule :C66H93N19O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1552.56N-CBZ-Phe-Arg-AMC
CAS :Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.Formule :C33H36N6O6Degré de pureté :98%Couleur et forme :White To Off-White PowderMasse moléculaire :612.68MMP-9-IN-6
CAS :MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.Formule :C25H19NO2Degré de pureté :98.96%Couleur et forme :SoildMasse moléculaire :365.42TP0597850
CAS :TP0597850, a selective MMP2 inhibitor with an IC50 value of 0.22 nM, demonstrates a prolonged dissociation half-life from MMP2 (t1/2 = 265 minutes) [1].Formule :C41H57N9O13SCouleur et forme :SolidMasse moléculaire :916.01Acetyl-Calpastatin(184-210)(human)
CAS :Calpain inhibitor, Ki 0.2 nM for calpain I/II, doesn't affect papain/trypsin/cat L. Raises Aβ42, Aβ40 secretion & Aβ42/Aβ40 ratio.Formule :C142H230N36O44SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3177.65(-)-Taxifolin
CAS :(-)-Taxifolin, less active enantiomer with anti-tyrosinase, collagenase inhibition (IC50 = 193.3 μM), antifibrotic, antioxidant properties.Formule :C15H12O7Couleur et forme :SolidMasse moléculaire :304.25Acetyl-Calpastatin (184-210)(human) acetate
Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.
Formule :C144H234N36O46SDegré de pureté :97.84% - 98.16%Couleur et forme :SolidMasse moléculaire :3237.68Alisporivir
CAS :Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.Formule :C63H113N11O12Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :1216.64AP-C2
CAS :AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.Formule :C18H16N4SDegré de pureté :99.99%Couleur et forme :SoildMasse moléculaire :320.41Aristololactam IIIa
CAS :Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.Formule :C16H9NO4Couleur et forme :SolidMasse moléculaire :279.25Histargin
CAS :Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.Formule :C14H25N7O4Couleur et forme :SolidMasse moléculaire :355.39AR-H067637
CAS :AR-H067637 is a fast-acting, reversible thrombin inhibitor with K(i) 2-4 nM; it also reduces clot-bound thrombin and platelet activation/aggregation.Formule :C21H21ClF2N4O4Couleur et forme :SolidMasse moléculaire :466.87Zetomipzomib maleate
CAS :Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.Formule :C34H46N4O12Couleur et forme :SolidMasse moléculaire :702.758KKI-5
CAS :KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.
Formule :C35H55N11O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :773.88NVP-DPP728 dihydrochloride
CAS :NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.Formule :C15H20Cl2N6OCouleur et forme :SolidMasse moléculaire :371.27Ellipyrone A
Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).Formule :C25H34O8Couleur et forme :SolidMasse moléculaire :462.53ZG36
ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrialCouleur et forme :Odour SolidRXP470
CAS :RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).Formule :C35H35BrClN4O10PCouleur et forme :SolidMasse moléculaire :818Dutogliptin tartrate
CAS :Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.Formule :C14H26BN3O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.18PS 915
CAS :PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.Formule :C27H36ClN7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.08
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