Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(34 produits)
- Cystéine protéase(96 produits)
- DPP-4(20 produits)
- Glutaminase(40 produits)
- Protéase du VIH(447 produits)
- PAI-1(25 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(54 produits)
- Protéasome(94 produits)
- Sérine protéase(50 produits)
- p97(14 produits)
Affichez 3 plus de sous-catégories
1045 produits trouvés pour "Protéases/Protéasome"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Sucunamostat
CAS :<p>Sucunamostat is an L-aspartic acid enteropeptidase inhibitor.</p>Formule :C22H22N4O8Couleur et forme :SolidMasse moléculaire :470.438KKI-5
CAS :<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Formule :C35H55N11O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :773.88Sofosbuvir impurity H
<p>Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.</p>Formule :C29H33FN3O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :633.56Fibrinopeptide B, human
CAS :<p>Fibrinopeptide B (FPB) is produced during the cleavage of fibrinogen, by thrombin, to fibrin monomer.</p>Formule :C66H93N19O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1552.56CRA-2059
CAS :<p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>Formule :C34H46N12O8Degré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :750.818ZG36
<p>ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrial</p>Couleur et forme :Odour SolidPSI-7409
CAS :<p>PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).</p>Formule :C10H16FN2O14P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.16Cys-TAT(47-57) acetate(583836-55-9 Free base)
<p>Cys-TAT(47-57) acetate is derived from the HIV-1 transactivating protein. Cys-TAT(47-57) acetate is an arginine rich peptide that can penetrate cells.</p>Formule :C69H128N34O16SDegré de pureté :95.1100%Couleur et forme :SolidMasse moléculaire :1722.047-Methoxy obtusifolin
CAS :<p>7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentration</p>Formule :C17H14O6Couleur et forme :SolidMasse moléculaire :314.29MK-6169
CAS :<p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>Formule :C54H62FN9O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1016.2Recombinant Trypsin
<p>Recombinant Trypsin is a serine protease that hydrolyzes proteins at the carboxyl side of lysine or arginine.</p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS :<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Formule :C47H64N14O10Couleur et forme :SolidMasse moléculaire :985.1Emtricitabine S-oxide
CAS :<p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>Formule :C8H10FN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :263.25JC-10
CAS :<p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>Formule :C25H29Cl2IN4Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :583.34AE-3763
CAS :<p>AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).</p>Formule :C23H34F3N5O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :549.54Sadopeptins B
<p>Sadopeptins B, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].</p>Formule :C48H69N9O13SCouleur et forme :SolidMasse moléculaire :1012.18Relacatib
CAS :<p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>Formule :C27H32N4O6SCouleur et forme :SolidMasse moléculaire :540.64L-Methionine-DL-sulfoximine
CAS :<p>MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.</p>Formule :C5H12N2O3SDegré de pureté :99.56% - ≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :180.23Nostosin G
<p>Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).</p>Formule :C25H33N5O6Couleur et forme :SolidMasse moléculaire :499.56Ichorcumab
CAS :<p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Couleur et forme :LiquidSofosbuvir impurity A
CAS :<p>Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.</p>Formule :C22H29FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.45CRA-2059 TFA
<p>CRA-2059 is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].</p>Couleur et forme :SolidHCV-IN-7 hydrochloride
CAS :<p>HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>Formule :C40H50Cl2N8O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :841.85Rivulariapeptolides 1121
<p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>Formule :C56H83N9O15Couleur et forme :SolidMasse moléculaire :1122.31Sofosbuvir impurity N
CAS :<p>Sofosbuvir impurity N is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formule :C20H25FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :501.404TAPI1 acetate
<p>TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .</p>Formule :C28H41N5O7Degré de pureté :98.82% - 99.94%Couleur et forme :SolidMasse moléculaire :559.65RJS308
<p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>Formule :C63H75N13O11SCouleur et forme :SolidMasse moléculaire :1222.42TMC647055 Choline salt
<p>TMC647055 choline salt is a selective and cell-permeating inhibitor of HCV NS5B (IC50: 34 nM).</p>Formule :C37H53N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :727.91Cathepsin C-IN-6
<p>Cathepsin C-IN-6 (compound 2), an E-64c-hydrazideas-derived inhibitor of cathepsin C, possesses anti-inflammatory properties and impedes neutrophil elastase</p>Formule :C24H35N5O4·xC2HF3O2Couleur et forme :SolidTWH106
<p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>Couleur et forme :Odour SolidPSI-353661
CAS :<p>PSI-353661 (GS-558093), inhibits HCV's NS5B polymerase; EC90: 8nM (wild-type), 11nM (S282T); active in human hepatocytes.</p>Formule :C24H32FN6O8PCouleur et forme :SolidMasse moléculaire :582.52Thrombin (MW 37kDa)
CAS :<p>Thrombin (MW 37kDa) is a trypsin-like allosteric serine protease.</p>Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :37kDaHepcidin-1 (mouse)
CAS :<p>Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.</p>Formule :C111H169N31O35S8Couleur et forme :SolidMasse moléculaire :2754.24Procizumab
<p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Couleur et forme :Odour LiquidHistatin 5
CAS :<p>Histatin 5, a human saliva peptide, blocks MMP-2 and MMP-9 at IC50s of 0.57/0.25 μM and kills fungi.</p>Formule :C133H195N51O33Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3036.29Alisporivir
CAS :<p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>Formule :C63H113N11O12Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :1216.64Ellipyrone B
<p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>Formule :C25H38O7Couleur et forme :SolidMasse moléculaire :450.57Dutogliptin tartrate
CAS :<p>Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>Formule :C14H26BN3O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.18Tyrosinase-IN-36
<p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>Couleur et forme :Odour SolidPS 915
CAS :<p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>Formule :C27H36ClN7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.08Befovacimab
CAS :<p>Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.</p>Couleur et forme :Liquidα 1 Antichymotrypsin, Human Plasma
CAS :<p>Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.</p>Couleur et forme :SolidTR-107
CAS :<p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>Formule :C22H19ClN4OCouleur et forme :SoildMasse moléculaire :390.87PF 00356231
CAS :<p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>Formule :C25H20N2O3SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :428.5Leptosphaerodione
CAS :<p>Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.</p>Formule :C21H22O5Couleur et forme :SolidMasse moléculaire :354.4EP 171
CAS :<p>EP 171 is a potent agonist of TP-receptors.</p>Formule :C23H29FO5Couleur et forme :SolidMasse moléculaire :404.47Histatin 5 TFA
<p>Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μM</p>Formule :C135H196N51F3O35Couleur et forme :SolidMasse moléculaire :3150.31(Iso)-Fosdevirine
CAS :<p>(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.</p>Formule :C20H17ClN3O3PDegré de pureté :99.93%Couleur et forme :SoildMasse moléculaire :413.79HIV-1 inhibitor-6
CAS :<p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>Formule :C14H10N4O4SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :330.32Ala-Phe-Pro-pNA TFA
<p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>Couleur et forme :Odour SolidAPC-6860
CAS :<p>APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.</p>Formule :C9H7IN2SCouleur et forme :SolidMasse moléculaire :302.13Sofosbuvir impurity M
CAS :<p>Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formule :C22H30N3O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.467BPHA
CAS :<p>BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.</p>Formule :C21H20N2O4SDegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :396.46Obtusifolin-2-O-glucoside
CAS :<p>Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].</p>Formule :C22H22O10Couleur et forme :SolidMasse moléculaire :446.4Z-Leu-Tyr-Chloromethylketone
CAS :<p>Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].</p>Formule :C24H29ClN2O5Couleur et forme :SolidMasse moléculaire :460.95NS5A-IN-4
CAS :<p>NS5A-IN-4 (Compound 1.12) is a hepatitis C inhibitor effective against multiple genotypes, with IC50 values ranging from 1.2 to 2296 pM.</p>Formule :C47H48N8O6Couleur et forme :SolidMasse moléculaire :820.93HIV-1 Rev (34-50)
CAS :<p>HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.</p>Formule :C97H173N51O24Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :2437.74Talabostat
CAS :<p>Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.</p>Formule :C9H19BN2O3Couleur et forme :SolidMasse moléculaire :214.07Nitidanin
<p>Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.</p>Formule :C21H24O8Couleur et forme :SolidMasse moléculaire :404.415Tyrosinase/elastase-IN-1
<p>Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase</p>Formule :C33H52O5Couleur et forme :SolidMasse moléculaire :528.76Clathrin-IN-1
CAS :<p>Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.</p>Formule :C20H13BrN2O3S2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :473.36GSK2336805
CAS :<p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>Formule :C42H52N8O8Couleur et forme :SolidMasse moléculaire :796.91CL 82198 hydrochloride
CAS :<p>CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.</p>Formule :C17H23ClN2O3Couleur et forme :SolidMasse moléculaire :338.83Dansyl-Glu-Gly-Arg-Chloromethylketone
CAS :<p>Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activated</p>Formule :C26H36ClN7O7SCouleur et forme :SolidMasse moléculaire :626.12VPLSLYSG
CAS :<p>VPLSLYSG, an octapeptide, degraded by MMP-9, MMP-1, MMP-2; potential MMP substrate uses.</p>Formule :C39H62N8O12Couleur et forme :SolidMasse moléculaire :834.96Recombinant Proteinase K
<p>Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.</p>Couleur et forme :SolidZ-Arg-Arg-βNA acetate
CAS :<p>Z-Arg-Arg-βNA acetate serves as a sensitive dipeptide substrate for Cathepsin B protease, while demonstrating resistance to proteases H and L. This compound is crucial for differentiating non-Cathepsin B type proteins.</p>Formule :C32H43N9O6Couleur et forme :SolidMasse moléculaire :649.74MMP-3 Inhibitor acetate
<p>MMP-3 Inhibitor acetate is a cell-permeable and potent inhibitor of human MMP-3.</p>Formule :C29H50N10O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :746.83Peptide 74
CAS :<p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>Formule :C62H107N23O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1558.79Sitagliptin fenilalanil hydrochloride
CAS :<p>Sitagliptin phenylalanine hydrochloride, a dipeptidyl peptidase-4 (DPP-4) inhibitor [1], is a chemical compound utilized in medical applications.</p>Formule :C25H25ClF6N6O2Couleur et forme :SolidMasse moléculaire :590.95PROTAC 20S proteasome subunit β5 degrader 2
<p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>Couleur et forme :Odour SolidAMG-222
CAS :<p>AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.</p>Formule :C32H39N9O3Couleur et forme :SolidMasse moléculaire :597.71PPACK II
CAS :<p>PPACK II is an irreversible and specific glandular and plasma kallikreins inhibitor [1] .</p>Formule :C25H33ClN6O3Couleur et forme :SolidMasse moléculaire :501.02MMP-3 Inhibitor
CAS :<p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>Formule :C27H46N10O9SDegré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :686.78HCV-IN-4
CAS :<p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>Formule :C52H58FN9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :956.07HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Couleur et forme :Odour SolidLeptosin D
CAS :<p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>Formule :C25H24N4O3S2Couleur et forme :SolidMasse moléculaire :492.61LXE408 fumarate
<p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>Formule :C27H22FN7O6Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :559.51Iso-VQA-ACC acetate
<p>Iso-VQA-ACC acetate serves as a substrate for the constitutive proteasome.</p>Couleur et forme :Odour SolidHCV-IN-41
CAS :<p>HCV-IN-41: potent HCV inhibitor; EC50 - 0.006762 nM (1b), 5.183 nM (2a), 1.365 nM (3a), 142.2 nM (4a); hinders RNA replication.</p>Formule :C48H56N6O8Couleur et forme :SolidMasse moléculaire :844.99MMP-9/MMP-13 Inhibitor I
CAS :<p>MMP-9/MMP-13 Inhibitor I is a dual inhibitor of MMP-9 and MMP-13 with IC50 of both 0.9 nM.</p>Formule :C25H25N3O6SCouleur et forme :SolidMasse moléculaire :495.5515,16-Dihydrotanshindiol C
<p>15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.</p>Formule :C18H18O5Couleur et forme :SolidMasse moléculaire :314.337Grazoprevir potassium salt
CAS :<p>Grazoprevir, a drug for hepatitis C, is a second-gen NS3/4a protease inhibitor.</p>Formule :C38H49KN6O9SCouleur et forme :SolidMasse moléculaire :805RXP470
CAS :<p>RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).</p>Formule :C35H35BrClN4O10PCouleur et forme :SolidMasse moléculaire :8186,6′-Dihydroxythiobinupharidine
CAS :<p>6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-fold</p>Formule :C30H42N2O4SCouleur et forme :SolidMasse moléculaire :526.73Ac-PAL-AMC
CAS :<p>Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.</p>Formule :C26H34N4O6Couleur et forme :SolidMasse moléculaire :498.57Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Couleur et forme :Odour SolidSFTI-1
CAS :<p>SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.</p>Formule :C67H104N18O18S2Couleur et forme :SolidMasse moléculaire :1513.78PROTAC CG167
<p>PROTAC CG167 is a potent and selective PROTAC degrader of CypA. It degrades CypA in a dose-dependent manner in Jurkat cells, with a DC50 of 123 nM. Additionally, PROTAC CG167 exhibits antiviral activity by inhibiting HIV-1 and HCV. (Pink: CypA Ligand; Black: Linker; Blue: E3LigaseLigand)</p>Formule :C65H79N13O11SCouleur et forme :SolidMasse moléculaire :1250.47FFAGLDD TFA
<p>FFAGLDD TFA: MMP9 peptide for controlled DOX delivery to cytoplasm.</p>Formule :C39H50F3N7O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :897.855-epi-Arvestonate A
CAS :<p>5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.</p>Formule :C16H26O5Couleur et forme :SolidMasse moléculaire :298.37VD2173
CAS :<p>VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.</p>Formule :C31H45N9O6SCouleur et forme :SolidMasse moléculaire :671.81Bortezomib analog
<p>Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.</p>Couleur et forme :Odour SolidNIM811
CAS :<p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>Formule :C62H111N11O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1202.635Pentosan Polysulfate
CAS :<p>Pentosan Polysulfate: anti-HIV, anti-inflammatory, supports cartilage, treats interstitial cystitis.</p>Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/ARivulariapeptolides 1155
<p>Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).</p>Formule :C59H81N9O15Couleur et forme :SolidMasse moléculaire :1156.33CP-346086 dihydrate
CAS :<p>CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.</p>Formule :C26H26F3N5O3Couleur et forme :SolidMasse moléculaire :513.521Cathepsin L-IN-3
CAS :<p>Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.</p>Formule :C41H49N7O4SCouleur et forme :SolidMasse moléculaire :735.94Anticancer agent 114
<p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>Formule :C28H33BF6N2O7Couleur et forme :SolidMasse moléculaire :634.37ADAM8-IN-1
CAS :<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Formule :C44H44Br4N6O12S2Couleur et forme :SolidMasse moléculaire :1232.6
![Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76347.webp&w=3840&q=75)
