Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(34 produits)
- Cystéine protéase(96 produits)
- DPP-4(20 produits)
- Glutaminase(40 produits)
- Protéase du VIH(447 produits)
- PAI-1(25 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(54 produits)
- Protéasome(94 produits)
- Sérine protéase(50 produits)
- p97(14 produits)
Affichez 3 plus de sous-catégories
1045 produits trouvés pour "Protéases/Protéasome"
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PROTAC 20S proteasome subunit β5 degrader 2
<p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>Couleur et forme :Odour SolidGSK2818713
CAS :<p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>Formule :C46H56N8O8Couleur et forme :SolidMasse moléculaire :849.002Procizumab
<p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Couleur et forme :Odour LiquidBI-1230
CAS :<p>BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.</p>Formule :C42H52N6O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :816.96Ellipyrone B
<p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>Formule :C25H38O7Couleur et forme :SolidMasse moléculaire :450.57MMP-3 Inhibitor
CAS :<p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>Formule :C27H46N10O9SDegré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :686.78HCV-IN-4
CAS :<p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>Formule :C52H58FN9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :956.07DPP-4-IN-14
<p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>Formule :C33H27N7O3Couleur et forme :SolidMasse moléculaire :569.613HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Couleur et forme :Odour SolidBictegravir Sodium
CAS :<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Formule :C21H17F3N3NaO5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :471.36LXE408 fumarate
<p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>Formule :C27H22FN7O6Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :559.51PS 915
CAS :<p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>Formule :C27H36ClN7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.08Ichorcumab
CAS :<p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Couleur et forme :LiquidKKI-5
CAS :<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Formule :C35H55N11O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :773.88Histargin
CAS :<p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>Formule :C14H25N7O4Couleur et forme :SolidMasse moléculaire :355.39Relacatib
CAS :<p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>Formule :C27H32N4O6SCouleur et forme :SolidMasse moléculaire :540.64Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Couleur et forme :Odour SolidAristololactam IIIa
CAS :<p>Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.</p>Formule :C16H9NO4Couleur et forme :SolidMasse moléculaire :279.25Tiprelestat
CAS :<p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>Formule :C254H416N72O75S10Couleur et forme :SolidMasse moléculaire :5999.09Lonodelestat TFA
<p>Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.</p>Formule :C73H112F3N15O21Couleur et forme :SolidMasse moléculaire :1592.75Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)
<p>Fluorogenic substrate for cathepsins D & E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.</p>Couleur et forme :Odour SolidParitaprevir dihydrate
CAS :<p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>Formule :C40H47N7O9SCouleur et forme :SolidMasse moléculaire :801.91ADAM8-IN-1
CAS :<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Formule :C44H44Br4N6O12S2Couleur et forme :SolidMasse moléculaire :1232.6Ac-Phe-Gly-pNA
CAS :<p>Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .</p>Formule :C19H20N4O5Couleur et forme :SolidMasse moléculaire :384.39Sulodexide
CAS :<p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>Couleur et forme :SolidCerpegin
CAS :<p>Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.</p>Formule :C10H11NO3Couleur et forme :SolidMasse moléculaire :193.2Carboxypeptidase C
CAS :<p>Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.</p>Couleur et forme :SolidMMP-9-IN-6
CAS :<p>MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.</p>Formule :C25H19NO2Degré de pureté :99.75%Couleur et forme :SoildMasse moléculaire :365.42VAMP
<p>VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.</p>Formule :C18H32N4O5SCouleur et forme :SolidMasse moléculaire :416.535Ala-Phe-Pro-pNA TFA
<p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>Couleur et forme :Odour SolidChymotrypsinogen
CAS :<p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>Couleur et forme :SolidCTTHWGFTLC, CYCLIC
CAS :<p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>Formule :C52H71N13O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1166.33Alisporivir
CAS :<p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>Formule :C63H113N11O12Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :1216.64Histatin 5 TFA
<p>Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μM</p>Formule :C135H196N51F3O35Couleur et forme :SolidMasse moléculaire :3150.31Acetyl-Calpastatin(184-210)(human) TFA
<p>Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.</p>Formule :C144H231F3N36O46SCouleur et forme :SolidMasse moléculaire :3291.65Gly-Pro-pNA hydrochloride
CAS :<p>Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase</p>Formule :C13H17ClN4O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :328.75Suc-AAP-Abu-pNA
CAS :<p>Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,</p>Formule :C25H34N6O9Couleur et forme :SolidMasse moléculaire :562.57TR-107
CAS :<p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>Formule :C22H19ClN4OCouleur et forme :SoildMasse moléculaire :390.87LMP7/LMP2-IN-1
CAS :<p>LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.</p>Formule :C16H27BN4O3Couleur et forme :SoildMasse moléculaire :334.22Anticancer agent 114
<p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>Formule :C28H33BF6N2O7Couleur et forme :SolidMasse moléculaire :634.37Phepropeptin C
CAS :<p>Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.</p>Formule :C38H60N6O6Couleur et forme :SolidMasse moléculaire :696.92PD150606
CAS :<p>PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.</p>Formule :C9H7IO2SDegré de pureté :98.19%Couleur et forme :SolidMasse moléculaire :306.12TWH106
<p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>Couleur et forme :Odour SolidBMS-767778
CAS :<p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Formule :C19H20Cl2N4O2Couleur et forme :SolidMasse moléculaire :407.29Roseltide rT1
CAS :<p>Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.</p>Formule :C110H177N31O31S6Couleur et forme :SolidMasse moléculaire :2622.16α 1(I) Collagen (614-639), human
CAS :<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Formule :C134H189N37O39Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2942.16MMP-2 Inhibitor-4
<p>MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).</p>Formule :C19H23N3O5SCouleur et forme :SolidMasse moléculaire :405.468NVP-DPP728 dihydrochloride
CAS :<p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>Formule :C15H20Cl2N6OCouleur et forme :SolidMasse moléculaire :371.27RJS308
<p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>Formule :C63H75N13O11SCouleur et forme :SolidMasse moléculaire :1222.42Stevia Powder
<p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>Couleur et forme :Odour SolidPR 39 (porcine) acetate
<p>PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.</p>Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :N/A6-Acetylnimbandiol
CAS :<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Formule :C28H34O8Couleur et forme :SolidMasse moléculaire :498.56Zetomipzomib maleate
CAS :<p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>Formule :C34H46N4O12Couleur et forme :SolidMasse moléculaire :702.758Rivulariapeptolides 988
<p>Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).</p>Formule :C50H68N8O13Couleur et forme :SolidMasse moléculaire :989.12L 659286
CAS :<p>L 659286 is one kind of cephalosporin derivative.</p>Formule :C17H21N5O7S2Couleur et forme :SolidMasse moléculaire :471.51Pseudostellarin G
CAS :<p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>Formule :C42H56N8O9Couleur et forme :SolidMasse moléculaire :816.94CRA-2059
CAS :<p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>Formule :C34H46N12O8Degré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :750.818Ellipyrone A
<p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>Formule :C25H34O8Couleur et forme :SolidMasse moléculaire :462.53Leptosin D
CAS :<p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>Formule :C25H24N4O3S2Couleur et forme :SolidMasse moléculaire :492.61Emtricitabine S-oxide
CAS :<p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>Formule :C8H10FN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :263.25Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS :<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Formule :C47H64N14O10Couleur et forme :SolidMasse moléculaire :985.1Peptide 74
CAS :<p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>Formule :C62H107N23O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1558.79Fotagliptin
CAS :<p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>Formule :C17H19FN6OCouleur et forme :SolidMasse moléculaire :342.37Rivulariapeptolides 1121
<p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>Formule :C56H83N9O15Couleur et forme :SolidMasse moléculaire :1122.31E-64d [for Biochemical Research]
CAS :Formule :C17H30N2O5Degré de pureté :>95.0%(HPLC)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :342.44CTS-1027
CAS :<p>CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has > 1,000 fold selectivity over MMP1.</p>Formule :C19H20ClNO6SCouleur et forme :SolidMasse moléculaire :425.88Tenofovir hydrate
CAS :<p>Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.</p>Formule :C9H16N5O5PDegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :305.23Ilomastat
CAS :Formule :C20H28N4O4Degré de pureté :>95.0%(HPLC)(qNMR)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :388.47S-Methylglutathione
CAS :<p>S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.</p>Formule :C11H19N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.35Retagliptin
CAS :<p>Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.</p>Formule :C19H18F6N4O3Couleur et forme :SolidMasse moléculaire :464.36PSI-6206 13C,d3
CAS :<p>PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.</p>Formule :C10H13FN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :264.23Tripeptide-32
CAS :<p>Tripeptide-32 is a bioactive peptide recognized for its anti-aging properties, commonly utilized as an ingredient in cosmetics [1].</p>Formule :C12H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.33Glutaminase-IN-3
CAS :<p>Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.</p>Formule :C19H19F3N6O2SDegré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :452.45MMP-8 Inhibitor I
CAS :<p>MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.</p>Formule :C17H18N2O5SCouleur et forme :SolidMasse moléculaire :362.4Tilpisertib
CAS :<p>Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).</p>Formule :C33H33ClN8OCouleur et forme :SolidMasse moléculaire :593.13Teneligliptin hydrobromide hydrate
CAS :<p>Teneligliptin hydrobromide hydrate: potent, long-lasting DPP-4 inhibitor with ~1 nM IC50.</p>Formule :C22H33BrN6O2SCouleur et forme :SolidMasse moléculaire :525.51Sitagliptin fenilalanil
CAS :<p>Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.</p>Formule :C25H24F6N6O2Couleur et forme :SolidMasse moléculaire :554.49PKSI-527
CAS :<p>PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.</p>Formule :C25H32ClN3O4Couleur et forme :SolidMasse moléculaire :473.99H-Arg-4MβNA
CAS :<p>H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.</p>Formule :C17H23N5O2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :329.4BAY-677
CAS :<p>BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.</p>Formule :C20H15F3N4O2Couleur et forme :SolidMasse moléculaire :400.355-Amino-8-hydroxyquinoline
CAS :<p>5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.</p>Formule :C9H8N2ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :160.176-Chloro-7-deazapurine-2F-β-D-arabinofuranose
CAS :<p>6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.</p>Formule :C11H11ClFN3O3Couleur et forme :SolidMasse moléculaire :287.67(Arg)9
CAS :<p>(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).</p>Formule :C54H110N36O10Couleur et forme :SolidMasse moléculaire :1423.69Ubenimex Hydrochloride [for Biochemical Research]
CAS :Formule :C16H24N2O4·HClDegré de pureté :>97.0%(HPLC)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :344.84Dabigatran ethyl ester
CAS :<p>Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.</p>Formule :C27H29N7O3Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :499.56Saquinavir mesylate
CAS :<p>Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy</p>Formule :C39H54N6O8SDegré de pureté :99.19%Couleur et forme :White Or Pale Yellow PowderMasse moléculaire :766.9Teneligliptin D8
CAS :<p>Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.</p>Formule :C22H30N6OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.63PD-166793
CAS :<p>PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.</p>Formule :C17H18BrNO4SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :412.3Tomeglovir
CAS :<p>Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).</p>Formule :C23H27N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.54DMP 777
CAS :<p>DMP 777 is an orally active inhibitor of human leukocyte elastase.</p>Formule :C31H40N4O6Couleur et forme :SolidMasse moléculaire :564.67Thrombin inhibitor 5
CAS :<p>Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.</p>Formule :C11H9FN4O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :264.21H-Pro-Lys-OH TFA
<p>H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.</p>Formule :C13H22F3N3O5Couleur et forme :SolidMasse moléculaire :357.332'-β-C-Ethynyladenosine
CAS :<p>2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.</p>Formule :C12H13N5O4Couleur et forme :SolidMasse moléculaire :291.26Sivelestat Sodium Tetrahydrate
CAS :Formule :C20H21N2NaO7S·4H2ODegré de pureté :>95.0%(T)(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :528.50Urokinase
CAS :<p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>Couleur et forme :SolidPentosan Polysulfate Sodium (W/W 43%)
CAS :<p>Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.</p>Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/AAnguizole
CAS :<p>Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.</p>Formule :C17H11ClF2N4O2SCouleur et forme :SolidMasse moléculaire :408.81Pepstatin A
CAS :Formule :C34H63N5O9Degré de pureté :>90.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :685.90(-)-Gallocatechin Gallate
CAS :Formule :C22H18O11Degré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :458.38Tanaproget
CAS :<p>Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.</p>Formule :C16H15N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.38
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