Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(38 produits)
- Cystéine protéase(111 produits)
- DPP-4(27 produits)
- Glutaminase(46 produits)
- Protéase du VIH(506 produits)
- PAI-1(26 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(55 produits)
- Protéasome(85 produits)
- Sérine protéase(54 produits)
- p97(15 produits)
Affichez 3 plus de sous-catégories
984 produits trouvés pour "Protéases/Protéasome"
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(R)-ND-336
CAS :(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.Formule :C16H18ClNO3S2Couleur et forme :SolidMasse moléculaire :371.89MMP13-IN-4
CAS :MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].Formule :C21H17BrN4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :485.29PF-00356231 hydrochloride
CAS :PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.Formule :C25H21ClN2O3SDegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :464.96MMP-2/9-IN-1
CAS :MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.Formule :C14H16IN7SCouleur et forme :SolidMasse moléculaire :441.29AZD6564
CAS :AZD6564 is a fibrinolysis inhibitor which acts via interference of a protein-protein interaction.Formule :C13H22N2O2Couleur et forme :SolidMasse moléculaire :238.33GLS1 Inhibitor-3
CAS :GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.Formule :C30H32N10O2SCouleur et forme :SolidMasse moléculaire :596.71HCV-IN-36
CAS :HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.Formule :C30H36ClN5Couleur et forme :SolidMasse moléculaire :502.09BC-23
CAS :BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.Formule :C21H14ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.87BRD-8899
CAS :BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].Formule :C17H22N4O3SCouleur et forme :SolidMasse moléculaire :362.45Tyrosinase-IN-5
CAS :Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.Formule :C18H13N3O6Couleur et forme :SolidMasse moléculaire :367.31Efegatran sulfate
CAS :Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.Formule :C21H34N6O7SDegré de pureté :≥98% - ≥98%Couleur et forme :SolidMasse moléculaire :514.6DPP-IV-IN-1
CAS :DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).Formule :C11H18FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :243.28SP-Chymostatin B
CAS :SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.Formule :C30H41N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :595.69Elasnin
CAS :Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.Formule :C24H40O4Couleur et forme :SolidMasse moléculaire :392.57Ono 3307 Free Base
CAS :Ono 3307 Free Base is a new synthetic protease inhibitorFormule :C14H14N4O4SCouleur et forme :SolidMasse moléculaire :334.35Proteasome-IN-1
CAS :Proteasome-IN-1 is an inhibitor of proteasome.Formule :C42H35N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :657.76A-933548
CAS :A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.Formule :C25H21N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.47ASPER-29
CAS :ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.Formule :C31H29BrN2O5SCouleur et forme :SolidMasse moléculaire :621.54CAY10704
CAS :CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.Formule :C18H20Cl2N2Couleur et forme :SolidMasse moléculaire :335.27DPP-4-IN-1
CAS :DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.Formule :C19H19ClN6Couleur et forme :SolidMasse moléculaire :366.85AA10 TG2 inhibitor
CAS :AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).Formule :C32H36N4O5Couleur et forme :SolidMasse moléculaire :556.65PK44 phosphate
CAS :PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).Formule :C17H19F5N7O5PCouleur et forme :SolidMasse moléculaire :527.349BAY8040
CAS :BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.Formule :C21H16F3N5O2Couleur et forme :SolidMasse moléculaire :427.38Z-LLF-CHO
CAS :Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.Formule :C29H39N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.64VEL-0230
CAS :VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.Formule :C14H24NNaO5Couleur et forme :SolidMasse moléculaire :309.33NNGH
CAS :NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.Formule :C13H20N2O5SDegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :316.37ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formule :C23H18ClF3N4O2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :538.99Alicapistat
CAS :Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).Formule :C25H27N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.5Tyrosinase-IN-6
CAS :Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.Formule :C24H31N3O2Couleur et forme :SolidMasse moléculaire :393.52Anticancer agent 82
CAS :Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.Formule :C19H18Cl2N4OCouleur et forme :SolidMasse moléculaire :389.28GS-9256
CAS :GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].Formule :C46H56ClF2N6O8PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :957.46Tyrosinase-IN-3
CAS :Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41Gü2602
CAS :Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for matureFormule :C16H22N4O3Couleur et forme :SolidMasse moléculaire :318.37HCV-IN-33
CAS :HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.Formule :C31H36ClN5Couleur et forme :SolidMasse moléculaire :514.1JNJ-10329670
CAS :JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.Formule :C30H34ClF3N6O3SCouleur et forme :SolidMasse moléculaire :651.14AGLME
CAS :AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Formule :C11H21N3O4Couleur et forme :SolidMasse moléculaire :259.3Odalasvir
CAS :Odalasvir is a novel NS5A inhibitor for the treatment of hepatitis C.Formule :C60H72N8O6Couleur et forme :SolidMasse moléculaire :1001.26Cysteine Protease inhibitor hydrochloride
CAS :Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.Formule :C18H15ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :338.79Tec-IN-21
CAS :Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Formule :C16H15ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :362.83Sheng Gelieting
CAS :CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.Formule :C17H16F6N4OCouleur et forme :SolidMasse moléculaire :406.33ZD8321
CAS :ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).Formule :C18H28F3N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.43Atevirdine
CAS :Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).
Formule :C21H25N5O2Degré de pureté :98.20%Couleur et forme :SolidMasse moléculaire :379.46Tyrosinase-IN-2
CAS :Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Formule :C8H8N4O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€PG-116800
CAS :PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Formule :C24H27N3O7SDegré de pureté :98.03% - 99.66%Couleur et forme :SolidMasse moléculaire :501.55TG-2-IN-1
CAS :TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].Formule :C8H13ClN2OSDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :220.72Cathepsin X-IN-1
CAS :Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].
Formule :C15H13N3O3SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :315.35CPA inhibitor
CAS :CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.Formule :C18H19NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :313.35Ref: TM-T10876
1mg54,00€5mg118,00€10mg155,00€25mg263,00€50mg384,00€100mgÀ demander1mL*10mM (DMSO)131,00€TG2-IN-3h
CAS :TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFormule :C21H26N4O4SDegré de pureté :99.34% - 99.76%Couleur et forme :SolidMasse moléculaire :430.522'-C-Methyladenosine
CAS :2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.Formule :C11H15N5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :281.2720S Proteasome activator 1
CAS :20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Formule :C27H19ClF2N2OSDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :492.97Gemigliptin
CAS :Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)Formule :C18H19F8N5O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :489.36Ref: TM-T7369
2mg38,00€5mg57,00€10mg93,00€25mg148,00€50mg245,00€100mg385,00€500mg873,00€1mL*10mM (DMSO)84,00€TY-51469
CAS :TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).Formule :C20H15FN2O6S4Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :526.6VRK-IN-1
CAS :VRK-IN-1 is a potent and selective inhibitor of cowpox-associated kinase 1 (VRK1), which can be used in the study of neurological disorders.Formule :C18H11F4NO2Degré de pureté :99.18% - 99.25%Couleur et forme :SolidMasse moléculaire :349.28Ref: TM-T35863
1mg98,00€5mg225,00€10mg359,00€25mg710,00€50mg1.071,00€100mg1.431,00€200mg1.953,00€1mL*10mM (DMSO)245,00€UK-396082
CAS :UK-396082 is a TAFI inhibitor that inhibits Carboxypeptidase B and can be used in the study of thrombosis, atherosclerosis, cancer and fibrotic conditions.Formule :C12H21N3O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :239.31UPGL00004
CAS :UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Formule :C25H26N8O2S2Degré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :534.66Lenacapavir
CAS :Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formule :C39H32ClF10N7O5S2Degré de pureté :99.61% - 99.87%Couleur et forme :SolidMasse moléculaire :968.28Ref: TM-T11465
1mg187,00€5mg376,00€10mg565,00€25mg998,00€50mg1.388,00€100mg1.882,00€200mg2.622,00€1mL*10mM (DMSO)615,00€BDCRB
BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.Formule :C12H11BrCl2N2O4Degré de pureté :99.41% - 99.85%Couleur et forme :SoildMasse moléculaire :398.04BILB-1941
CAS :BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.Formule :C34H34N4O4Degré de pureté :99.51% - 99.65%Couleur et forme :SolidMasse moléculaire :562.66Ref: TM-T26815
1mg296,00€5mg718,00€10mg982,00€25mg1.485,00€50mg2.008,00€100mg2.637,00€1mL*10mM (DMSO)1.044,00€DB04760
CAS :DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.Formule :C22H20F2N4O2Degré de pureté :99.93% - 99.99%Couleur et forme :SolidMasse moléculaire :410.42Ref: TM-T15055
1mg84,00€5mg205,00€10mg309,00€25mg522,00€50mg747,00€100mg1.035,00€500mg2.052,00€1mL*10mM (DMSO)178,00€JNJ-10311795
CAS :JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.Formule :C40H35N2O6PDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :670.69Setrobuvir
CAS :Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension withFormule :C25H25FN4O6S2Degré de pureté :99.95% - 99.97%Couleur et forme :SolidMasse moléculaire :560.62Ref: TM-T28762
1mg229,00€5mg570,00€10mg812,00€25mg1.216,00€50mg1.663,00€100mg2.242,00€500mg4.494,00€1mL*10mM (DMSO)737,00€Sovaprevir
CAS :Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Formule :C43H53N5O8SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :799.97Ref: TM-T28830
1mg253,00€5mg620,00€10mg884,00€25mg1.314,00€50mg1.773,00€100mg2.385,00€1mL*10mM (DMSO)982,00€Melagatran
CAS :Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.Formule :C22H31N5O4Degré de pureté :98.29% - >99.99%Couleur et forme :SolidMasse moléculaire :429.51Ref: TM-T11994
1mg487,00€5mg1.134,00€10mg1.468,00€25mg2.215,00€50mg2.962,00€100mg4.024,00€1mL*10mM (DMSO)1.071,00€MMP2-IN-3
CAS :MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Formule :C23H21N3ODegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :355.43Ref: TM-T61271
1mg64,00€5mg132,00€10mg195,00€25mg315,00€50mg439,00€100mg590,00€200mg793,00€1mL*10mM (DMSO)140,00€Sirpiglenastat
CAS :Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Formule :C22H27N5O5Degré de pureté :98.01% - 98.37%Couleur et forme :SolidMasse moléculaire :441.48Isatoribine
CAS :Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.Formule :C10H12N4O6SDegré de pureté :98.99% - 99.75%Couleur et forme :SolidMasse moléculaire :316.29AGPS-IN-2i
CAS :AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Formule :C18H17F2N3O2Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :345.34Ref: TM-T69685
1mg74,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€1mL*10mM (DMSO)154,00€HIV-1 integrase inhibitor 8
CAS :HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].
Formule :C21H24O2Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :308.41MMP-2/MMP-9 Inhibitor I
CAS :MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.Formule :C21H19NO4SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :381.44Ref: TM-T21512
1mg56,00€5mg119,00€10mg177,00€25mg356,00€50mg590,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)133,00€MK-8325
CAS :MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailabilityFormule :C43H54Cl2F2N8O6SiDegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :915.93BAY-43-9695
CAS :BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.Formule :C22H25N3O4SDegré de pureté :99.50% - 99.98%Couleur et forme :SolidMasse moléculaire :427.52BMS-929075
CAS :BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokineticFormule :C31H24F2N4O3Degré de pureté :99.81% - 99.94%Couleur et forme :SolidMasse moléculaire :538.54Ref: TM-T26863
1mg172,00€5mg432,00€10mg618,00€25mg973,00€50mg1.333,00€100mg1.791,00€500mg3.529,00€1mL*10mM (DMSO)538,00€(2RS)-FPMPA
CAS :(2RS)-FPMPA（FPMPA） has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).Formule :C9H13FN5O4PDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :305.2P32/98 hemifumarate
CAS :P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.Formule :C22H40N4O6S2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :520.71CP-544439
CAS :CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.Formule :C18H19FN2O6SDegré de pureté :95.02% - 98.66%Couleur et forme :SolidMasse moléculaire :410.42Uprifosbuvir
CAS :Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.Formule :C22H29ClN3O9PDegré de pureté :99.73% - >99.99%Couleur et forme :SolidMasse moléculaire :545.91TS-021
CAS :TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.Formule :C17H24FN3O5SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :401.45Etarotene
CAS :Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is aFormule :C25H32O2SDegré de pureté :99.58% - 99.98%Couleur et forme :SolidMasse moléculaire :396.59BMS-538305 HCl
CAS :BMS-538305 is a potent, selective inhibitor of dipeptidyl peptidase IV (DPP-IV).Formule :C17H27ClN2O2Couleur et forme :SolidMasse moléculaire :326.86AZD-9819
CAS :AZD-9819 is a neutrophil elastase (HNE) inhibitor applicable for research into chronic obstructive pulmonary disease (COPD).Formule :C25H19F3N6O2Degré de pureté :100% - 99.18%Couleur et forme :SolidMasse moléculaire :492.45(Rac)-Neurodegenerative Disorder-Targeting Compound 1
CAS :(Rac)-Neurodegenerative Disorder-Targeting Compound 1 is a calpain inhibitor.Formule :C28H28N4O4Couleur et forme :SolidMasse moléculaire :484.55Ro 31-9790
CAS :Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).Formule :C15H29N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.41Thrombin inhibitor 1
CAS :Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).Formule :C22H20Cl2F2N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :497.32AA74-1
CAS :AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].Formule :C16H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.42JW 480
CAS :JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.Formule :C22H23NO2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :333.42Ref: TM-T22883
2mg35,00€5mg49,00€10mg79,00€25mg160,00€50mg259,00€100mg416,00€200mg587,00€1mL*10mM (DMSO)57,00€Flovagatran sodium
CAS :Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.Formule :C27H36BN3NaO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :548.4BAY-320
CAS :BAY-320 is a Bub1 inhibitor. With an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.Formule :C26H26F2N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :492.52SQ 32056
CAS :SQ 32056 is a cathepsin E inhibitor.Formule :C37H56N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :636.86BMS-189664 HCl
CAS :BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Formule :C22H35ClN6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.07Tyropeptin A-4
CAS :Tyropeptin A-4 is used as a proteasome inhibitor.Formule :C31H41N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :551.67NS5A-IN-3
CAS :NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formule :C44H44N6O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :784.86NS5A-IN-2
CAS :NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.Formule :C46H45N7O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :807.89TP0556351
CAS :TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.Formule :C50H70N10O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1067.15LM-030
CAS :LM-030, also known as BPR277, is a novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2).Formule :C46H72N8O12Couleur et forme :SolidMasse moléculaire :929.11HCV-IN-44
CAS :HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].Formule :C24H26FN3O5SCouleur et forme :SolidMasse moléculaire :487.54MMP3 inhibitor 1
CAS :MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).Formule :C23H31N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.57(1R,4S)-Yimitasvir diphosphate
CAS :Yimitasvir diphosphate, also known as Emitasvir, is an orally-administered inhibitor of the hepatitis C virus (HCV) nonstructural protein 5A (NS5A).Formule :C49H64N8O14P2Couleur et forme :SolidMasse moléculaire :1051.03MMP13-IN-3
CAS :MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.Formule :C24H22N4O5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :446.46Ref: TM-T16124
1mg93,00€5mg205,00€10mg334,00€25mg587,00€50mg802,00€100mg1.108,00€1mL*10mM (DMSO)227,00€MeOSuc-AAPV-CMK
CAS :MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediatedFormule :C22H35ClN4O7Couleur et forme :SolidMasse moléculaire :502.99Ecallantide
CAS :Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.Formule :C305H448N88O91S8Couleur et forme :SolidMasse moléculaire :7059.88
