Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(34 produits)
- Cystéine protéase(96 produits)
- DPP-4(20 produits)
- Glutaminase(40 produits)
- Protéase du VIH(447 produits)
- PAI-1(25 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(54 produits)
- Protéasome(94 produits)
- Sérine protéase(50 produits)
- p97(14 produits)
Affichez 3 plus de sous-catégories
1045 produits trouvés pour "Protéases/Protéasome"
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Lenacapavir
CAS :<p>Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.</p>Formule :C39H32ClF10N7O5S2Degré de pureté :99.61% - 99.87%Couleur et forme :SolidMasse moléculaire :968.28Etarotene
CAS :<p>Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a</p>Formule :C25H32O2SDegré de pureté :99.58% - 99.93%Couleur et forme :SolidMasse moléculaire :396.59BDCRB
<p>BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.</p>Formule :C12H11BrCl2N2O4Degré de pureté :99.41% - 99.43%Couleur et forme :SoildMasse moléculaire :398.04BILB-1941
CAS :<p>BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.</p>Formule :C34H34N4O4Degré de pureté :99.51% - 99.65%Couleur et forme :SolidMasse moléculaire :562.662'-C-Methyladenosine
CAS :<p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>Formule :C11H15N5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :281.27CPA inhibitor
CAS :<p>CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.</p>Formule :C18H19NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :313.35Cathepsin X-IN-1
CAS :<p>Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].</p>Formule :C15H13N3O3SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :315.35P32/98 hemifumarate
CAS :<p>P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.</p>Formule :C22H40N4O6S2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :520.71Atevirdine
CAS :<p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>Formule :C21H25N5O2Degré de pureté :98.20%Couleur et forme :SolidMasse moléculaire :379.46DB04760
CAS :<p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>Formule :C22H20F2N4O2Degré de pureté :99.93% - 99.99%Couleur et forme :SolidMasse moléculaire :410.42JNJ-10311795
CAS :<p>JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.</p>Formule :C40H35N2O6PDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :670.69TG-2-IN-1
CAS :<p>TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].</p>Formule :C8H13ClN2OSDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :220.72CP-544439
CAS :<p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>Formule :C18H19FN2O6SDegré de pureté :95.02% - 98.66%Couleur et forme :SolidMasse moléculaire :410.42Setrobuvir
CAS :<p>Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension with</p>Formule :C25H25FN4O6S2Degré de pureté :98.92% - >99.99%Couleur et forme :SolidMasse moléculaire :560.62Granotapide
CAS :<p>Granotapide is a microsomal triglyceride transfer protein (MTP) inhibitor that treats and rather prevents atherosclerosis, coronary artery disease, metabolic</p>Formule :C39H37F3N2O8Degré de pureté :99.70% - 99.79%Couleur et forme :SolidMasse moléculaire :718.71PG-116800
CAS :<p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>Formule :C24H27N3O7SDegré de pureté :98.03% - 99.66%Couleur et forme :SolidMasse moléculaire :501.55Sovaprevir
CAS :<p>Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.</p>Formule :C43H53N5O8SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :799.97Melagatran
CAS :<p>Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.</p>Formule :C22H31N5O4Degré de pureté :98.29% - >99.99%Couleur et forme :SolidMasse moléculaire :429.51Opaviraline
CAS :<p>Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.</p>Formule :C14H17FN2O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :280.29MMP2-IN-3
CAS :<p>MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).</p>Formule :C23H21N3ODegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :355.43Uprifosbuvir
CAS :<p>Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.</p>Formule :C22H29ClN3O9PDegré de pureté :99.73% - >99.99%Couleur et forme :SolidMasse moléculaire :545.91Sirpiglenastat
CAS :<p>Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.</p>Formule :C22H27N5O5Degré de pureté :98.01% - 98.37%Couleur et forme :SolidMasse moléculaire :441.48Emivirine
CAS :<p>Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.</p>Formule :C17H22N2O3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :302.37Tyrosinase-IN-2
CAS :<p>Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.</p>Formule :C8H8N4O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :224.24Isatoribine
CAS :<p>Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.</p>Formule :C10H12N4O6SDegré de pureté :98.99% - 99.75%Couleur et forme :SolidMasse moléculaire :316.29AGPS-IN-2i
CAS :<p>AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.</p>Formule :C18H17F2N3O2Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :345.34HIV-1 integrase inhibitor 8
CAS :<p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>Formule :C21H24O2Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :308.41TS-021
CAS :<p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>Formule :C17H24FN3O5SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :401.45MMP-2/MMP-9 Inhibitor I
CAS :<p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>Formule :C21H19NO4SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :381.44KM-023
CAS :<p>KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.</p>Formule :C18H19N3O3Degré de pureté :99.47% - >99.99%Couleur et forme :SolidMasse moléculaire :325.36L 756423
CAS :<p>L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.</p>Formule :C39H48N4O5Degré de pureté :99.34% - 99.88%Couleur et forme :SolidMasse moléculaire :652.8220S Proteasome activator 1
CAS :<p>20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.</p>Formule :C27H19ClF2N2OSDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :492.97Gemigliptin
CAS :<p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>Formule :C18H19F8N5O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :489.36MK-8325
CAS :<p>MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailability</p>Formule :C43H54Cl2F2N8O6SiDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :915.93Thrombin inhibitor 1
CAS :<p>Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).</p>Formule :C22H20Cl2F2N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :497.32GS-6620
CAS :<p>GS-6620 is a HCV nonstructural protein 5B (NS5B) inhibitor.</p>Formule :C29H37N6O9PCouleur et forme :SolidMasse moléculaire :644.61SSR 69071
CAS :<p>SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.</p>Formule :C27H32N4O7SCouleur et forme :SolidMasse moléculaire :556.63NS5A-IN-2
CAS :<p>NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.</p>Formule :C46H45N7O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :807.89XL-784
CAS :<p>XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.</p>Formule :C42H42Cl2F4MgN6O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1122.15Ravidasvir HCl
CAS :<p>Ravidasvir, also known as PPI-668 and ASC16, is a second-generation, orally active, potent and selective HCV NS5A protein inhibitor.</p>Formule :C42H52Cl2N8O6Couleur et forme :SolidMasse moléculaire :835.828Inogatran
CAS :<p>Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.</p>Formule :C21H38N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.56Paltimatrectinib
CAS :<p>Paltimatrectinib (PBI-200) is a tyrosine kinase inhibitor with anticancer activity, and is used in the study of bladder, breast, and colorectal cancers.</p>Formule :C20H15F5N6Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :434.37ABP 25
CAS :<p>ABP 25 is a highly potent and selective activity-based probe (ABP) for cathepsin K imaging.</p>Formule :C55H66ClN5O3Couleur et forme :SolidMasse moléculaire :880.6Beclabuvir HCl
CAS :<p>Beclabuvir (BMS-791325) is an HCV inhibitor targeting NS5B polymerase with sub-28 nM potency for genotypes 1, 3, 4, 5.</p>Formule :C36H46ClN5O5SCouleur et forme :SolidMasse moléculaire :696.3BAY-678
CAS :<p>BAY-678: Oral selective human neutrophil elastase inhibitor; IC50: 20 nM; SGC-approved chemical probe.</p>Formule :C20H15F3N4O2Degré de pureté :97.89%Couleur et forme :SolidMasse moléculaire :400.35Proteasome-IN-5
CAS :<p>Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].</p>Formule :C20H30BN5O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.29Collagen proline hydroxylase inhibitor
CAS :<p>Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.</p>Formule :C18H18N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :354.36Ro 31-9790
CAS :<p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>Formule :C15H29N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.41ONO 4817
CAS :<p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>Formule :C22H28N2O6Couleur et forme :SolidMasse moléculaire :416.47MMP-7-IN-3
CAS :<p>MMP-7-IN-3 (compound 15) is a potent and selective MMP-7 inhibitor, inhibiting renal fibrosis in a unilateral ureteral obstruction mouse model.</p>Formule :C34H43ClF3N7O9SDegré de pureté :99.915%Couleur et forme :SolidMasse moléculaire :818.26KB-R7785
CAS :<p>KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.</p>Formule :C18H27N3O4Couleur et forme :SolidMasse moléculaire :349.42Cipemastat
CAS :<p>Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).</p>Formule :C22H36N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.55Azt-pmap
CAS :<p>AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].</p>Formule :C20H25N6O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.42XL-784 free base
CAS :<p>XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).</p>Formule :C21H22ClF2N3O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :549.93MDL 27324
CAS :<p>MDL 27324 is an inhibitor of human neutrophil elastase.</p>Formule :C29H38F3N5O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.7AA74-1
CAS :<p>AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].</p>Formule :C16H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.42Ro 32-7315
CAS :<p>Ro 32-7315 is a selective inhibitor of ADAM17.</p>Formule :C22H35N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.6MK-3281
CAS :<p>MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.</p>Formule :C29H37N3O3Couleur et forme :SolidMasse moléculaire :475.62MDL 101146
CAS :<p>MDL 101146 is an orally active neutrophil elastase inhibitor.</p>Formule :C29H37F5N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.62JW 480
CAS :<p>JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.</p>Formule :C22H23NO2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :333.42MMP-7-IN-2
CAS :<p>MMP-7-IN-2 acts as a selective and potent MMP7 inhibitor and can be used to study inflammatory responses and vascular-related diseases.</p>Formule :C28H40ClF3N6O9SDegré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :729.17Proteasome β2c/i-IN-1
CAS :<p>Proteasome β2c/i-IN-1 (compound 37) serves as a selective inhibitor targeting the β2c and β2i subunits of the human proteasome [1].</p>Formule :C32H48N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :600.75ND-378
CAS :<p>ND-378 is a potent and selective inhibitor of MMP-2 with no inhibition on MMP-9 and MMP-14.</p>Formule :C18H19NO4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48AZD-7295
CAS :<p>AZD-7295 (A-689) is an NS5A inhibitor that may be used to treat HCV infection.</p>Formule :C32H35F3N4O5SCouleur et forme :SolidMasse moléculaire :644.7PTC725
CAS :<p>PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.</p>Formule :C23H18F4N6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.49EP1013
CAS :<p>EP1013 is a broad-spectrum selective inhibitor of Caspase used in the study of type 1 diabetes.</p>Formule :C18H23FN2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.38HIV-1 protease-IN-12
CAS :<p>HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-</p>Formule :C25H35N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.63GSK-2485852
CAS :<p>GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.</p>Formule :C27H25BF2N2O6SCouleur et forme :SolidMasse moléculaire :554.37MMP13-IN-3
CAS :<p>MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.</p>Formule :C24H22N4O5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :446.46TP0556351
CAS :<p>TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.</p>Formule :C50H70N10O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1067.15Apratastat
CAS :<p>Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs)</p>Formule :C17H22N2O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.5MDL-101146, (R)-
CAS :<p>MDL-101146, (R)- is an effective orally active inhibitor of human neutrophil elastase.</p>Formule :C29H37F5N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.62LU-002i
CAS :<p>LU-002i is a selective inhibitor targeting the human proteasome subunits β2c and β2i, demonstrating an inhibitory concentration (IC50) of 220 nM for β2i [1].</p>Formule :C35H52N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :640.81Phe-Pro-Ala-pNA
CAS :<p>Phe-Pro-Ala-pNA is a chromogenic substrate utilized for assessing tripeptidyl peptidase activity.</p>Formule :C23H27N5O5Couleur et forme :SolidMasse moléculaire :453.49Flovagatran sodium
CAS :<p>Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.</p>Formule :C27H36BN3NaO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :548.4Z-FG-NHO-BzOME
CAS :<p>Z-FG-NHO-BzOME is a chemical compound functioning as a cysteine protease inhibitor, selectively targeting and inhibiting cathepsin B, cathepsin L, cathepsin S,</p>Formule :C27H27N3O7Couleur et forme :SolidMasse moléculaire :505.52HIV-1 protease-IN-7
CAS :<p>HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].</p>Formule :C68H104N10O12SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1285.68BAY-320
CAS :<p>BAY-320 is a Bub1 inhibitor. With an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.</p>Formule :C26H26F2N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :492.52Cyclotheonellazole A
CAS :<p>Cyclotheonellazole A inhibits elastase (IC50=0.034nM) & chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.</p>Formule :C44H54N9NaO14S2Couleur et forme :SolidMasse moléculaire :1020.07JTK-853
CAS :<p>JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).</p>Formule :C28H23F7N6O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :704.64Z-PDLDA-NHOH
CAS :<p>Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].</p>Formule :C22H32N4O6Couleur et forme :SolidMasse moléculaire :448.51HIV-1 protease-IN-9
CAS :<p>HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a</p>Formule :C37H41N7O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :679.83DCLK1-IN-2
CAS :<p>DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cell</p>Formule :C26H32N8O3SCouleur et forme :SolidMasse moléculaire :536.65Berotralstat HCl
CAS :<p>Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.</p>Formule :C30H28Cl2F4N6OCouleur et forme :SolidMasse moléculaire :635.4886Z-DEVD-CMK
CAS :<p>Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].</p>Formule :C27H35ClN4O12Couleur et forme :SolidMasse moléculaire :643.04I-XW-053
CAS :<p>I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-</p>Formule :C22H16N2O2Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :340.37O-Benzoylhydroxylamine
CAS :<p>O-Benzoyl hydroxylamine exhibits properties as a dipeptidyl peptidase-IV (DPP-IV) inhibitor and demonstrates antidiabetic effects[1].</p>Formule :C7H7NO2Couleur et forme :SolidMasse moléculaire :137.14Kallikrein-IN-2
CAS :<p>Kallikrein-IN-2 (compound 1) is an inhibitor of the kinin-releasing enzyme Kallikrein.</p>Formule :C28H25F3N4O4Couleur et forme :SolidMasse moléculaire :538.52Neurodegenerative Disorder-Targeting Compound 1
CAS :<p>Neurodegenerative Disorder-Targeting Compound 1 is an inhibitor of calpain [1].</p>Formule :C28H28N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :484.55NCI-B16
CAS :<p>NCI-B16 is a small-molecule RNA binder that inhibits HCV (hepatitis C virus) replication [1].</p>Formule :C27H26N8O4Couleur et forme :SolidMasse moléculaire :526.55KCC009
CAS :<p>KCC009 is a potent and selective Transglutaminase 2 Inhibitor.</p>Formule :C21H22BrN3O5Couleur et forme :SolidMasse moléculaire :476.32SQ 32056
CAS :<p>SQ 32056 is a cathepsin E inhibitor.</p>Formule :C37H56N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :636.86BMS-189664 HCl
CAS :<p>BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.</p>Formule :C22H35ClN6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.07Ecallantide
CAS :<p>Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.</p>Formule :C305H448N88O91S8Couleur et forme :SolidMasse moléculaire :7059.88Proteasome-IN-4
<p>Proteasome-IN-4, a potent non-covalent inhibitor (IC50=8.39nM), halts cancer cell growth, useful for oncology studies.</p>Formule :C44H58N6O5Couleur et forme :SolidMasse moléculaire :750.97MMP-145
CAS :<p>MMP-145 is used as a protease inhibitor.</p>Formule :C20H20N2O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.45HIV-1 protease-IN-8
CAS :<p>HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.</p>Formule :C25H35N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.63Human enteropeptidase-IN-1
CAS :<p>Enteropeptidase-IN-1: orally active, potent inhibitor, low systemic exposure, for anti-obesity research.</p>Formule :C20H18N4O7Couleur et forme :SolidMasse moléculaire :426.38MeOSuc-AAPV-CMK
CAS :<p>MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediated</p>Formule :C22H35ClN4O7Couleur et forme :SolidMasse moléculaire :502.99NK3201
CAS :<p>NK3201, a specific chymase inhibitor, suppresses bleomycin-induced pulmonary fibrosis in hamsters.</p>Formule :C31H29N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.59
