GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.030 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(159 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(22 produits)
- Récepteur du glucagon(196 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(325 produits)
- PAFR(14 produits)
- PKA(55 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5985 produits trouvés pour "GPCR/G-Protéine"
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α-CGRP, rat
CAS :Endogenous neuropeptide, potent vasodilatorFormule :C162H262N50O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3806.25VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.Formule :C27H35FN6O4Couleur et forme :SolidMasse moléculaire :526.603DOTA-JR11
CAS :DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Formule :C74H98ClN19O21S2Couleur et forme :SolidMasse moléculaire :1689.27GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].Couleur et forme :Odour Solid(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formule :C44H69N13O13S2Couleur et forme :SolidMasse moléculaire :1052.23INCB 3284 dimesylate
CAS :INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Formule :C28H39F3N4O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :712.76Imelciment
CAS :Imelciment (REGN-9035) is a humanised monoclonal antibody targeting NPR1, which can be used for research into heart failure.Degré de pureté :95%Couleur et forme :Soild[D-Phe12]-Bombesin
CAS :<p>Bombesin receptor antagonist</p>Formule :C74H112N22O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1629.88Cannabidiolic acid methyl ester
CAS :Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Formule :C23H32O4Couleur et forme :SolidMasse moléculaire :372.5Fenoldopam
CAS :Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).Formule :C16H16ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.7612(S)-HpEPE
CAS :<p>12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.</p>Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.456Poly-D-lysine hydrobromide (MW 1000-5000)
Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.Couleur et forme :Odour SolidAcmopatide
CAS :Acmopatide (Compound E-153) is a dual agonist of GIP and GLP-1 receptors and can be utilized in diabetes research.Couleur et forme :SolidD5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Couleur et forme :Odour SolidEfranarelaxin alfa
CAS :Efranarelaxin alfa is an agonist of the relaxin receptor. It shows potential for research in cardiovascular diseases and tissue repair.Couleur et forme :LiquidCCG258208 hydrochloride
<p>GRKs-IN-1 HCl (14as) strongly inhibits GRK2 (IC50=130nM) & GRK5 (IC50=7.1μM), is a paroxetine derivative with 100x cardiac boost.</p>Couleur et forme :SolidPoly-D-lysine hydrobromide (MW 150000-300000)
Poly-D-lysine hydrobromide (MW 150000-300000) enhances neural cell adhesion in culture and acts as a calcium-sensing receptor agonist peptide in research.Couleur et forme :Odour SolidFR 113680
CAS :FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.Formule :C35H39N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.726NN1213
NN1213 (Peptide 21) is a long-acting human amylin peptide analogue that functions as a selective amylin receptor agonist. It has an EC50 of 0.177 nM for hAMY3R and 0.262 nM for rAMY3R. In both rat and dog models, NN1213 significantly reduces appetite and is utilized in anti-obesity research.Couleur et forme :Odour SolidAmisulpride hydrochloride
CAS :Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formule :C17H28ClN3O4SCouleur et forme :SolidMasse moléculaire :405.94Zenagamtide sodium
Zenagamtide is an agonist for both glucagon-like peptide-1 (GLP-1) and amylin receptors.Couleur et forme :Odour SolidGS-2278
CAS :GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).Formule :C22H16F5N9O3Couleur et forme :SolidMasse moléculaire :549.412,3-dinor Thromboxane B1
CAS :TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formule :C18H32O6Couleur et forme :SolidMasse moléculaire :344.448AZP-531
CAS :Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.Formule :C40H63N15O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :962.025-OMe-UDP trisodium salt
CAS :Potent P2Y6 agonistFormule :C10H16N2O13P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.19NTRC-824
CAS :NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.Formule :C25H26F3N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :553.55Labradimil
CAS :Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formule :C49H75N15O12SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1098.29L-803087 TFA
CAS :L-803087 TFA: potent sst4 agonist, Ki=0.7 nM, >280x selective vs other somatostatin receptors; boosts AMPA, heightens seizures.Formule :C27H30F5N5O5Couleur et forme :SolidMasse moléculaire :599.554-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine
CAS :4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine is an enantiomericFormule :C27H28ClFN2OSDegré de pureté :99.02%Couleur et forme :SoildMasse moléculaire :483.04Ref: TM-T60126
1mg109,00€2mg163,00€5mg241,00€10mg355,00€25mg532,00€50mg745,00€100mg1.018,00€500mgÀ demander1mL*10mM (DMSO)289,00€Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS :Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formule :C47H66N12O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :975.11LE 300
CAS :LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formule :C20H22N2Degré de pureté :97.91% - 98.79%Couleur et forme :SolidMasse moléculaire :290.4TRPV1/CB2 agonist 1
<p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>Couleur et forme :Odour Solid[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS :High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.Formule :C189H284N54O56SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4241LY83583
CAS :<p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>Formule :C15H10N2O2Degré de pureté :99.54% - 99.80%Couleur et forme :SolidMasse moléculaire :250.25Anti-TSHR Antibody (M22)
Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.Couleur et forme :Odour LiquidFabesetron
CAS :<p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>Formule :C18H19N3OCouleur et forme :SolidMasse moléculaire :293.37Dipivefrin
CAS :Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.Formule :C19H29NO5Couleur et forme :SolidMasse moléculaire :351.44Pellotine
CAS :Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.Formule :C13H19NO3Couleur et forme :SolidMasse moléculaire :237.2955-MeO-pyr-T
CAS :5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.Formule :C15H20N2OCouleur et forme :SolidMasse moléculaire :244.33Cortagine
Potent CRF1 agonist, EC50 = 0.18 nM in rats. Exhibits in vivo anxiolytic and antidepressant effects; reduces mouse defensive behavior.Formule :C192H323N55O63SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4442.06Nafetolol
CAS :Nafetolol (K 5407) is a biochemical reagent that can be used to synthesize other compounds.Formule :C19H29NO3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :319.44α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFormule :C165H268F3N51O51S2Couleur et forme :SolidMasse moléculaire :3903.33IRL-1038
CAS :ETB endothelin receptor antagonistFormule :C68H92N14O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1409.67Galantide
CAS :Galantide is a reversible and non-specific antagonist of galanin receptor.Formule :C104H151N25O26SDegré de pureté :98%Couleur et forme :White Lyophilised SolidMasse moléculaire :2199.53TRV045
CAS :<p>TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.</p>Formule :C18H18N4O3Couleur et forme :SolidMasse moléculaire :338.36ABT 724 trihydrochloride
CAS :ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formule :C17H22Cl3N5Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€GR231118
CAS :Potent NPY Y1 antagonist & Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).Formule :C110H170N34O24Degré de pureté :98%Couleur et forme :Lyophilized PowderMasse moléculaire :2352.77[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
CAS :Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.Formule :C183H281N57O54S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4207.6717-phenyl trinor Prostaglandin E2 ethyl amide
CAS :17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.Formule :C25H35NO4Couleur et forme :SolidMasse moléculaire :413.55(Rac)-Norcisapride
CAS :Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.Formule :C14H20ClN3O3Degré de pureté :99.32%Couleur et forme :SoildMasse moléculaire :313.78Luseogliflozin hydrate
CAS :Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.Formule :C23H32O7SCouleur et forme :SolidMasse moléculaire :452.56Bay 55-9837 TFA
Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.Formule :C150H240F3ClN44O44Couleur et forme :SolidMasse moléculaire :3456.22(Ala13)-Apelin-13
CAS :(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.Formule :C63H107N23O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1474.75ALEPH hydrochloride
CAS :ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Formule :C12H20ClNO2SCouleur et forme :SolidMasse moléculaire :277.81Cinnamtannin A2
CAS :<p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>Formule :C60H50O24Couleur et forme :SolidMasse moléculaire :1155.02IRL-1038 acetate
IRL-1038 acetate is a potent ETB endothelin receptor antagonist.Formule :C70H96N14O17S2Degré de pureté :97.51%Couleur et forme :SoildMasse moléculaire :1469.73Ki16198
CAS :Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).Formule :C24H25ClN2O5SDegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :488.98Glucagon receptor antagonists-1
CAS :Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Formule :C29H34FNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.58Endothelin 1 (swine, human), Alexa Fluor 488-labeled
Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.Couleur et forme :SolidMasse moléculaire :2848.4Urocortin III (human)
CAS :Urocortin III, a human peptide, binds CRF-R2, affecting insulin via somatostatin feedback with K i values 13.5-100+ nM.Formule :C185H307N53O50S2Couleur et forme :SolidMasse moléculaire :4137.93Tiaprost
CAS :Tiaprost is a analog of prostaglandin F2α .Formule :C20H28O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.5DOAM
CAS :DOAM is an antagonist of the 5-HT2 receptor.Formule :C16H27NO2Couleur et forme :SolidMasse moléculaire :265.39RXFP3/4 agonist 1
CAS :RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).Formule :C20H22ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.88Prazobind
CAS :Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Formule :C23H27N5O3Couleur et forme :SolidMasse moléculaire :421.501(+)-Oxypeucedanin methanolate
CAS :(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].Formule :C17H18O6Couleur et forme :SolidMasse moléculaire :318.32VU0453379
CAS :VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).Formule :C26H34N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.57Eledoisin Related Peptide
CAS :Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.Formule :C34H58N8O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :706.94Blue FPG-A trisodium
CAS :Blue FPG-A trisodium is a P2X1 & P2Y1 receptor antagonist, IC50: 35.5 μM & 2.6 μM, related to RB2.Formule :C29H17ClN7Na3O11S3Couleur et forme :SolidMasse moléculaire :840.1PAR 4 (1-6)
CAS :PAR 4 (1-6) can be used for relevant research in the life sciences. Its product number is T36293 and CAS number is 225779-44-2.Formule :C28H41N7O9Couleur et forme :SolidMasse moléculaire :619.676Brexpiprazole S-oxide
CAS :Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Formule :C25H27N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.57Ethylpropyltryptamine
CAS :Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35Pexopiprant
CAS :Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.Formule :C21H17Cl2F2NO4Couleur et forme :SolidMasse moléculaire :456.27M1145
CAS :Potent GAL2 agonist with EC50 = 38 nM; Ki: 6.55 nM (GAL2), 497 nM (GAL3), 587 nM (GAL1); enhances galanin signaling.Formule :C128H205N37O32Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2774.26Neurokinin A(4-10) TFA
Neurokinin A (4-10) TFA is a tachykinin NK 2 receptor agonist [1] .Formule :C36H55F3N8O12SCouleur et forme :SolidMasse moléculaire :880.93HAEGTFTSDVS acetate
HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.Formule :C50H75N13O22Degré de pureté :97.47%Couleur et forme :SolidMasse moléculaire :1210.2LUF6096
CAS :LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormule :C22H21Cl2N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :414.33Mini Gastrin I, human
CAS :Mini Gastrin I, human, is a truncated form of the human gastrin peptide, encompassing amino acids 5-17 of the original sequence.Formule :C74H99N15O26SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1646.73UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38Orexin A (human, rat, mouse) (TFA)
Endogenous orexin receptor agonist with Ki of 20 nM (OX1) and 38 nM (OX2), promotes feeding, may regulate sleep-wake cycle.Formule :C154H244N47F3O46S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3675.12Urocortin III, mouse
CAS :Mouse UcnIII, linked to stress behaviors, mainly occurs in the brain and rises in the hypothalamus post-restraint.Formule :C186H312N52O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4172.97EP4 receptor antagonist 3
CAS :EP4 receptor antagonist 3 from patent WO2010019796 A1 targets EP4 for research on pain, arthritis, and cancer.Formule :C26H21F3N2O3SCouleur et forme :SolidMasse moléculaire :498.52IRL-1620
CAS :IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).Formule :C86H117N17O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1820.9744-Hydroxy MET
CAS :4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formule :C13H18N2OCouleur et forme :SolidMasse moléculaire :218.3INCB3344 R-isomer
INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.Formule :C29H34F3N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :577.59GR 94800
CAS :Potent and selective tachykinin NK2 receptor antagonistFormule :C49H61N9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :904.082Eloralintide sodium
Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.Formule :C201H319N49O65S2·xNaDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :4526.1 (free base)Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Formule :C22H30N2O7SDegré de pureté :97.05% - 98.53%Couleur et forme :SoildMasse moléculaire :466.55des-Gln14-Ghrelin
CAS :Endogenous rat ghrelin gene variant binds GHS-R1a; strong Ca2+ release (EC50=2.4 nM); boosts GH secretion in vivo.Formule :C142H237N43O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3186.7PF-232798
CAS :PF-232798 is a second generation oral CCR5 antagonist with potent broad-spectrum anti-HIV-1 activity.Formule :C29H40FN5O2Couleur et forme :SolidMasse moléculaire :509.6619(S)-HETE
CAS :19-HETE, a CYP450 arachidonic acid metabolite from kidneys, consists of 70% (S) and 30% (R) isomers and dilates renal vessels.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473NSC380324
NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.Formule :C31H24N4O4Couleur et forme :SolidMasse moléculaire :516.55Methapyrilene hydrochloride
CAS :Methapyrilene hydrochloride is a biochemical.Formule :C14H20ClN3SCouleur et forme :Liquid Solution) 5 5 (Ntp 1992)Masse moléculaire :297.85SSTR4 agonist-1
CAS :SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.Formule :C16H23N3O2Couleur et forme :SolidMasse moléculaire :289.37[D-Phe12,Leu14]-Bombesin
CAS :Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.Formule :C77H113F3N22O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1724.9Calcitonin Gene Related Peptide (CGRP) II, rat
CAS :CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Formule :C163H267N51O50S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3805.3117-phenoxy trinor Prostaglandin F2α ethyl amide
CAS :Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.Formule :C25H37NO5Couleur et forme :SolidMasse moléculaire :431.573Neuropeptide Y (human)
CAS :Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.Formule :C189H285N55O57SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4271.68Somatostatin-28 (1-14)
CAS :Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.Formule :C61H105N23O21SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1528.71LY 344864 racemate
CAS :LY 344864 racemate is a 5-HT1F receptor agonist.Formule :C21H22FN3ODegré de pureté :99.75%Couleur et forme :SoildMasse moléculaire :351.42(R)-(+)-Atenolol
CAS :(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formule :C14H22N2O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :266.34
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