GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5986 produits trouvés pour "GPCR/G-Protéine"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
MCL0129
CAS :MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.Formule :C34H47FN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :546.76Succinate/succinate receptor antagonist 1
CAS :Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.
Formule :C17H15N3ODegré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :277.32PZ-128
CAS :PZ-128, a PAR1 antagonist, is used potentially for the treatment of thrombosis.Formule :C55H99N13O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1086.46Dulaglutide
CAS :Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).Couleur et forme :SolidP2Y6R antagonist 1
P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.Couleur et forme :Odour SolidSpns2-IN-2
Spns2-IN-2 (compound 3a) is an inhibitor of SPNS2.Formule :C22H30ClN3O2Couleur et forme :SolidMasse moléculaire :403.95HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Couleur et forme :Odour SolidAdrenocorticotropic Hormone (ACTH) (1-39), rat
CAS :ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.Formule :C210H315N57O57SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4582.23RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.Formule :C28H42N6O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :542.67Ref: TM-T16738L
1mg65,00€5mg125,00€1mL*10mM (DMSO)167,00€10mg182,00€25mg325,00€50mg467,00€100mg645,00€200mg868,00€Dehydro Aripiprazole (hydrochloride)
CAS :Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.Formule :C23H26Cl3N3O2Couleur et forme :SolidMasse moléculaire :482.83Ethylnorepinephrine hydrochloride
CAS :Ethylnorepinephrine hydrochloride is a unique bronchodilator.
Formule :C10H16ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.69CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.Formule :C20H18F3N3O3SCouleur et forme :SolidMasse moléculaire :437.435GLP-1 receptor agonist 4
CAS :GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.Formule :C51H44Cl2N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :879.82TGR5 agonist 7
TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.Formule :C37H59N2NaO9SCouleur et forme :SolidMasse moléculaire :730.93Desmethyl Mirtazapine (hydrochloride)
CAS :Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formule :C16H18ClN3Couleur et forme :SolidMasse moléculaire :287.79Agaridoxin
CAS :Agaridoxin is a mushroom metabolite.
Formule :C11H14N2O5Couleur et forme :SolidMasse moléculaire :254.242Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFormule :C80H112N18O19S2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :1693.98VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.Formule :C27H35FN6O4Couleur et forme :SolidMasse moléculaire :526.603Metaraminol
CAS :Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.Formule :C9H13NO2Couleur et forme :SolidMasse moléculaire :167.21P2Y14R antagonist 3
P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.Formule :C26H25N5O5Couleur et forme :SolidMasse moléculaire :487.51GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].Couleur et forme :Odour SolidHistamine H4 receptor antagonist-1
CAS :Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Formule :C30H38N8O2Couleur et forme :SolidMasse moléculaire :542.68Jmv 167
CAS :Jmv 167 is an antagonist of the Cholecystokinin receptor.Formule :C51H68N8O14SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1049.21INCB 3284 dimesylate
CAS :INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Formule :C28H39F3N4O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :712.76Khusimol
CAS :Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Formule :C15H24ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :220.35Pexopiprant
CAS :Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.Formule :C21H17Cl2F2NO4Couleur et forme :SolidMasse moléculaire :456.274-fluoro MBZP
CAS :4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.Formule :C12H17FN2Couleur et forme :SolidMasse moléculaire :208.28Vapreotide diacetate
CAS :Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.Formule :C61H78N12O13S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1251.47CAY10734
CAS :CAY10734 has a wide range of applications in life science related research.Formule :C23H25N3O3Couleur et forme :SolidMasse moléculaire :391.471D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Couleur et forme :Odour SolidPoly-D-lysine hydrobromide (MW 1000-5000)
Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.Couleur et forme :Odour SolidCannabidiolic acid methyl ester
CAS :Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Formule :C23H32O4Couleur et forme :SolidMasse moléculaire :372.5LHRH, Ala(6)-
CAS :LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formule :C56H77N17O13Couleur et forme :SolidMasse moléculaire :1196.32NSC380324
NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.Formule :C31H24N4O4Couleur et forme :SolidMasse moléculaire :516.55Motilin, canine
CAS :Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.Formule :C120H194N36O34Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2685.05Poly-D-lysine hydrobromide (MW 150000-300000)
Poly-D-lysine hydrobromide (MW 150000-300000) enhances neural cell adhesion in culture and acts as a calcium-sensing receptor agonist peptide in research.Couleur et forme :Odour SolidFR190997
CAS :FR190997 is an agonist of bradykinin B2 receptor.Formule :C37H33Cl2N5O5Couleur et forme :SolidMasse moléculaire :698.59Peptide 401
CAS :Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.Formule :C110H192N40O24S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2587.22FR252384
CAS :FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).Formule :C18H17N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.35Adrenomedullin (11-50), rat
CAS :Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Formule :C194H304N58O59S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4521.175-Bromoimidazo[1,2-A]Pyrazine
CAS :5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.Formule :C6H4BrN3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :198.02Zevaquenabant
CAS :Zevaquenabant (S-MRI-1867): oral CB1/iNOS antagonist combatting obesity-induced CKD.Formule :C25H21ClF3N5O2SCouleur et forme :SolidMasse moléculaire :547.98TGR5 agonist 6
CAS :Compound 22b, also known as TGR5 agonist 6, is a non-systemic, intestine-targeted TGR5 agonist that demonstrates significant and sustained blood glucose-lowering effects with an acceptable safety profile.Formule :C42H48Cl2N6O6Couleur et forme :SolidMasse moléculaire :803.77Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and isFormule :C102H163N31O26Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :2239.58GS-2278
CAS :GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).Formule :C22H16F5N9O3Couleur et forme :SolidMasse moléculaire :549.41WS 9326A
CAS :WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.Formule :C54H68N8O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1037.181LGnRH-III, lamprey
CAS :GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Formule :C59H74N18O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1259.33PAR-4 Agonist Peptide, amide acetate
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).Formule :C36H52N8O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :740.864-Chloromethamphetamine hydrochloride
CAS :4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.Formule :C10H15Cl2NCouleur et forme :SolidMasse moléculaire :220.14[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS :High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.Formule :C189H284N54O56SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4241SB234551
CAS :SB234551 is a selective antagonist of endothelin ETA receptor.Formule :C34H34N2O9Couleur et forme :SolidMasse moléculaire :614.64Anthramycin
CAS :Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.Formule :C16H17N3O4Couleur et forme :SolidMasse moléculaire :315.32Fabesetron
CAS :Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.
Formule :C18H19N3OCouleur et forme :SolidMasse moléculaire :293.37Dipivefrin
CAS :Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.Formule :C19H29NO5Couleur et forme :SolidMasse moléculaire :351.44Pellotine
CAS :Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.Formule :C13H19NO3Couleur et forme :SolidMasse moléculaire :237.295LY83583
CAS :LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.
Formule :C15H10N2O2Degré de pureté :99.54% - 99.80%Couleur et forme :SolidMasse moléculaire :250.25Phenylethanolamine A
CAS :Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formule :C19H24N2O4Couleur et forme :SolidMasse moléculaire :344.40Halometasone
CAS :Halometasone: synthetic corticosteroid for psoriasis and eczema treatment.Formule :C22H27ClF2O5Couleur et forme :SolidMasse moléculaire :444.95-MeO-pyr-T
CAS :5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.Formule :C15H20N2OCouleur et forme :SolidMasse moléculaire :244.33TT-OAD2
CAS :TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.
Formule :C50H49Cl4N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :929.75Clomipramine D3
CAS :Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formule :C19H23ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :317.87LY-426965 hydrochloride
CAS :LY-426965 hydrochloride is a bioactive chemical.Formule :C28H39ClN2O2Couleur et forme :SolidMasse moléculaire :471.07ABT 724 trihydrochloride
CAS :ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formule :C17H22Cl3N5Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :402.75Ref: TM-T22019
5mg40,00€1mL*10mM (DMSO)44,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€GR231118
CAS :Potent NPY Y1 antagonist & Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).Formule :C110H170N34O24Degré de pureté :98%Couleur et forme :Lyophilized PowderMasse moléculaire :2352.77γ-2-MSH (41-58), amide
CAS :Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Formule :C74H100N22O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1569.79Galantide acetate
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.Formule :C106H155N25O28SDegré de pureté :97.8% - 97.91%Couleur et forme :SolidMasse moléculaire :2259.58H4R antagonist 3
CAS :H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFormule :C19H21ClN4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :372.92L 366811
CAS :L 366811 is a potent oxytocin antagonist.Formule :C43H56N8O6Couleur et forme :SolidMasse moléculaire :780.95MDL 19301
CAS :MDL 19301 is a nonsteroidal, anti-inflammatory agent.Formule :C15H21NS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.46OXA(17-33)
CAS :Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formule :C79H125N23O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1749Ki16198
CAS :Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).Formule :C24H25ClN2O5SDegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :488.98IRL-1038 acetate
IRL-1038 acetate is a potent ETB endothelin receptor antagonist.Formule :C70H96N14O17S2Degré de pureté :97.51%Couleur et forme :SoildMasse moléculaire :1469.73(Rac)-Norcisapride
CAS :Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.Formule :C14H20ClN3O3Degré de pureté :99.32%Couleur et forme :SoildMasse moléculaire :313.7811-deoxy Prostaglandin F1α
CAS :11-deoxy PGF1α is a synthetic analog of PGF1α.Formule :C20H36O4Couleur et forme :SolidMasse moléculaire :340.504ALEPH hydrochloride
CAS :ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Formule :C12H20ClNO2SCouleur et forme :SolidMasse moléculaire :277.81(+)-Cloprostenol sodium
CAS :Cloprostenol sodium is a water-soluble PGF2α analog and FP receptor agonist, promoting luteolysis in rats and hamsters.Formule :C22H28ClNaO6Couleur et forme :SolidMasse moléculaire :446.9(S)-Azelastine hydrochloride
CAS :(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formule :C22H25Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.36[bAla8]-Neurokinin A(4-10)
CAS :[bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.Formule :C35H56N8O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :780.94Abediterol napadisylate
CAS :Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formule :C60H68F4N4O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1209.32Zalospirone
CAS :Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Formule :C24H29N5O2Degré de pureté :98.24% - 99.82%Couleur et forme :SolidMasse moléculaire :419.52Iloperidone metabolite P95
CAS :Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formule :C23H25FN2O5Couleur et forme :SolidMasse moléculaire :428.46Luprostiol
CAS :Luprostiol is a prostaglandin analog.Formule :C21H29ClO6SCouleur et forme :SolidMasse moléculaire :444.97Vapiprost
CAS :Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.Formule :C30H39NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.64ECPLA
CAS :ECPLA is an LSD analog and a potent 5-HT2A agonist (EC50 of 14.6 nM), capable of stimulating Gq-mediated calcium flux. It exhibits high affinity for most serotonin receptors, α2-adrenergic receptors, and D2-like dopamine receptors.Formule :C21H25N3OCouleur et forme :SolidMasse moléculaire :335.44Ici 216140
CAS :ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.Formule :C45H65N13O8Couleur et forme :SolidMasse moléculaire :916.08NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Formule :C25H26ClN3O2SDegré de pureté :99.84%Couleur et forme :SoildMasse moléculaire :468.01Ref: TM-T12262L1
1mg38,00€5mg84,00€1mL*10mM (DMSO)92,00€10mg113,00€25mg188,00€50mg273,00€100mg371,00€200mg494,00€(Iso)-RJW100
CAS :Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).Formule :C28H34ODegré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :386.57Ref: TM-T64363
1mg109,00€5mg241,00€1mL*10mM (DMSO)259,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€MRS 4062 triethylammonium salt
CAS :MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).Formule :C42H86N7O15P3Couleur et forme :SolidMasse moléculaire :1022.105Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS
Couleur et forme :Odour SolidM1145
CAS :Potent GAL2 agonist with EC50 = 38 nM; Ki: 6.55 nM (GAL2), 497 nM (GAL3), 587 nM (GAL1); enhances galanin signaling.Formule :C128H205N37O32Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2774.26Ethylpropyltryptamine
CAS :Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35tBPC
CAS :Enhances Y4R response to PP, NPY & PYY with EC50 of 0.03, 0.4, 0.5 nM; selective for Y4R over Y1R, Y2R, Y5R.Formule :C16H24O2Couleur et forme :SolidMasse moléculaire :248.36PF-9184
CAS :PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.Formule :C21H14Cl2N2O4SDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :461.32Mini Gastrin I, human
CAS :Mini Gastrin I, human, is a truncated form of the human gastrin peptide, encompassing amino acids 5-17 of the original sequence.Formule :C74H99N15O26SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1646.73Nebokitug
Nebokitug is a humanized IgG1κ antibody targeting CCL24, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidOrexin A (human, rat, mouse) (TFA)
Endogenous orexin receptor agonist with Ki of 20 nM (OX1) and 38 nM (OX2), promotes feeding, may regulate sleep-wake cycle.Formule :C154H244N47F3O46S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3675.12Urocortin III, mouse
CAS :Mouse UcnIII, linked to stress behaviors, mainly occurs in the brain and rises in the hypothalamus post-restraint.Formule :C186H312N52O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4172.97Glucagon-like peptide 1 (1-37), human
CAS :Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.Formule :C186H275N51O59Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4169.48UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
CAS :Broad-spectrum inverse agonist; potent at ghrelin receptor (EC50=5.2 nM); blocks other neuropeptide receptors; induces apoptosis; inhibits tumor growth.Formule :C79H109N19O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1516.85
![5-Bromoimidazo[1,2-A]Pyrazine](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT77641.webp&w=3840&q=75)
![[Leu31,Pro34]-Neuropeptide Y(human,rat)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1985.webp&w=3840&q=75)
![[bAla8]-Neurokinin A(4-10)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1100.webp&w=3840&q=75)
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931.webp&w=3840&q=75)