GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
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5986 produits trouvés pour "GPCR/G-Protéine"
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Albiglutide fragment TFA
Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as aFormule :C148H224N40O45·xC2HF3O2Couleur et forme :SolidGLP-1R Agonist DMB
CAS :GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).Formule :C13H15Cl2N3O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :348.25Urocortin III, mouse
CAS :Mouse UcnIII, linked to stress behaviors, mainly occurs in the brain and rises in the hypothalamus post-restraint.Formule :C186H312N52O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4172.97SB236057
CAS :SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.Formule :C33H34N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.65TRAP-6 amide TFA
CAS :TRAP-6 amide TFA is a PAR-1 thrombin receptor agonist peptide.Formule :C36H58F3N11O10Couleur et forme :SolidMasse moléculaire :861.922CI-988 hemihydrate
CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.Formule :C35H42N4O6H2OMasse moléculaire :632.321Retrobradykinin
CAS :Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Formule :C50H73N15O11Couleur et forme :SolidMasse moléculaire :1060.228Orexin A (human, rat, mouse) (TFA)
Endogenous orexin receptor agonist with Ki of 20 nM (OX1) and 38 nM (OX2), promotes feeding, may regulate sleep-wake cycle.Formule :C154H244N47F3O46S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3675.12Hydroxybupropion
CAS :Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formule :C13H18ClNO2Degré de pureté :99.73%Couleur et forme :Off-White SolidMasse moléculaire :255.74Ref: TM-T11588
1mg89,00€5mg204,00€1mL*10mM (DMSO)232,00€10mg331,00€25mg545,00€50mg777,00€100mg1.063,00€Neuropeptide FF
CAS :Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).Formule :C54H76N14O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1081.27WAY-639418
CAS :WAY-639418 has potential anti-inflammatory and anti-HIV activity and can be used to study CCR5-mediated inflammatory and immunomodulatory diseases.Formule :C17H16ClN5Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :325.8Neuropeptide Y (2-36) (porcine)
CAS :Porcine Neuropeptide Y (2-36) is 97.14% similar to rat/human, an agonist for Y5, Y2, Y1 receptors, used in obesity research.Formule :C181H278N54O55Couleur et forme :SolidMasse moléculaire :4090.47Lys-[Des-Arg9]Bradykinin TFA
CAS :Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Formule :C54H75F6N13O15Couleur et forme :SolidMasse moléculaire :1260.24Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Formule :C77H112N20O15Degré de pureté :98.9200%Couleur et forme :SolidMasse moléculaire :1557.84Prostaglandin F2α isopropyl ester
CAS :PGF2α isopropyl ester is an ester prodrug of PGF2α with enhanced lipid solubility.Formule :C23H40O5Couleur et forme :SolidMasse moléculaire :396.568Rp-UTP-α-S tetrasodium
Rp-UTP-α-S (tetrasodium) is a nucleotide agonist of the purinergic P2Y2 and P2Y4 receptors. It can induce the accumulation of inositol phosphate in 1321N1 cells expressing P2Y2 or P2Y4, with EC50 values of 5.4 and 27 μM, respectively.Couleur et forme :Odour SolidSch 202596
CAS :Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formule :C25H22Cl2O12Couleur et forme :SolidMasse moléculaire :585.34Teprotumumab
CAS :Teprotumumab: human antibody, inhibits IGF-1R, used for thyroid eye diseases.
Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:99.6%Couleur et forme :LiquidMasse moléculaire :145.62 kDaGalanin (2-29) (rat)
CAS :Peptide agonist for galanin receptorsFormule :C139H208N42O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3107.4M40
CAS :Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in ratFormule :C94H145N23O24Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1981.33Clozapine N-oxide dihydrochloride
CAS :Clozapine N-oxide dihydrochloride is a derivative of Clozapine and an agonist of DREADDs.Formule :C18H21Cl3N4ODegré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :415.74Neuropeptide Y (3-36) (human, rat)
CAS :Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.Formule :C175H269N53O54SCouleur et forme :SolidMasse moléculaire :4011.5K-(D-1-Nal)-FwLL-NH2
CAS :Potent ghrelin receptor inverse agonist with Ki of 4.9/31 nM in COS7/HEK293T; blocks Gq/G13 signaling.Formule :C51H67N9O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :902.13Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.Formule :C212H316F3N57O59SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4696.18Bromchlorbuterol hydrochloride
CAS :Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.Formule :C12H19BrCl2N2OCouleur et forme :SolidMasse moléculaire :358.1Cetirizine D8 dihydrochloride
CAS :Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Formule :C21H26Cl2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.4Minesapride
CAS :Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.
Formule :C21H31ClN4O5Degré de pureté :99.85% - 99.88%Couleur et forme :SolidMasse moléculaire :454.95[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS :'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.Formule :C39H64N8O10Couleur et forme :SolidMasse moléculaire :804.97PACAP (6-38), human, ovine, rat
CAS :PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.Formule :C182H300N56O45SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4024.74BIMU 8
CAS :BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Formule :C19H27ClN4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :378.9Ref: TM-T21946
1mg85,00€5mg168,00€1mL*10mM (DMSO)175,00€10mg235,00€25mg394,00€50mg582,00€100mg827,00€500mg1.674,00€Mabuterol free base
CAS :Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.Formule :C13H18ClF3N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.74ANXA3 degrader 1
ANXA3 degrader 1 (Compound 18a5) is a highly selective ANXA3 degrader with activity against cancer cells. It demonstrates significant inhibitory effects in a triple-negative breast cancer (TNBC) tumor xenograft model, with a tumor growth inhibition (TGI) rate of 96%.Formule :C30H32N6O2S2Couleur et forme :SolidMasse moléculaire :572.74Protease-Activated Receptor-1, PAR-1 Agonist
CAS :Selective peptide agonist that mimics thrombin to activate PAR-1 receptor, enabling targeted receptor activation.Formule :C35H58N10O9Couleur et forme :SolidMasse moléculaire :762.91(2R,2R)-PF-07258669
CAS :(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.
Formule :C25H27FN6O2Couleur et forme :SolidMasse moléculaire :462.52O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS :O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Formule :C11H11NO3Couleur et forme :SolidMasse moléculaire :205.213Xanthine amine congener trihydrochloride
CAS :Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formule :C21H29ClN6O4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :464.9520-hydroxy Prostaglandin F2α
CAS :20-hydroxy Prostaglandin F2α (20-hydroxy PGF2α) is the ω-oxidation product of PGF2α.
Formule :C20H34O6Couleur et forme :SolidMasse moléculaire :370.486Obestatin(rat)
CAS :Endogenous peptide that suppresses food intake and body weight-gainFormule :C114H174N34O31Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2516.81[Asu1,6-Arg8]Vasopressin
CAS :[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formule :C48H68N14O12Couleur et forme :SolidMasse moléculaire :1033.14Bradykinin (1-7)
CAS :Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formule :C35H52N10O9Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :756.85Ilatreotide
CAS :Ilatreotide is a Amadori compound of octreotide.Formule :C61H86N10O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1343.53d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.Formule :C49H71N11O13S2Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :1086.28CRL-42872 free base
CAS :CRL-42872 free base is a bioactive chemical.Formule :C22H26N6O6SCouleur et forme :SolidMasse moléculaire :502.54Urocortin II, human TFA
hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.Formule :C196H340F3N63O56SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4564.3Human growth hormone-releasing factor
CAS :GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.Formule :C215H358N72O66SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :5039.65Luprostiol
CAS :Luprostiol is a prostaglandin analog.Formule :C21H29ClO6SCouleur et forme :SolidMasse moléculaire :444.97Lanepitant
CAS :Lanepitant (LY303870) is a non-peptide neurokinin-1 (NK-1) antagonist with analgesic activity for the prevention of migraine.Formule :C33H45N5O3Degré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :559.74(Iso)-WAY-260022
CAS :(Iso)-WAY-260022 ((Iso)-NRI-022) is a stereoisomer of WAY-260022, a norepinephrine reuptake inhibitor and selective inhibitor of 5-hydroxytryptamine and dopamine transport proteins.Formule :C21H31F3N2O2Degré de pureté :97.68% - 99.36%Couleur et forme :SoildMasse moléculaire :400.48NESS 0327
CAS :NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formule :C24H23Cl3N4ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :489.82CCK (26-30) (sulfated)
CAS :CCK (26-30) is a digestive and satiety-related peptide fragment inhibiting [125I]CCK-33 binding by 10% at 0.1 mM.Formule :C33H41N7O12S2Couleur et forme :SolidMasse moléculaire :791.85Neuropeptide Y (3-36) (porcine)
CAS :Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.Formule :C176H271N53O54Couleur et forme :SolidMasse moléculaire :3993.36MD01-67
CAS :MD01-67 is a macrocyclic compound selectively targeting the neurotensin 2 receptor (NTS2), with a Ki of 2.9 nM. It exhibits analgesic activity and reduces tactile hypersensitivity in rat models of acute, sustained, and chronic inflammatory pain.Formule :C37H58N8O8Couleur et forme :SolidMasse moléculaire :742.91Selepressin acetate
Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.Formule :C48H77N13O13S2Couleur et forme :SolidMasse moléculaire :1108.33Guanylin TFA (mouse,rat)
Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.Formule :C60H90N16O22S4·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1515.71 (free base)Clomipramine D3
CAS :Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formule :C19H23ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :317.87Albenatide
CAS :Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.
Formule :C26H47N7O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :633.7615-keto-17-phenyl trinor Prostaglandin F2α
CAS :Bimatoprost is an F-series prostaglandin (PG) analog which has been approved for use as an ocular hypotensive drug.Formule :C23H30O5Couleur et forme :SolidMasse moléculaire :386.488Vapitadine
CAS :Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formule :C17H20N4ODegré de pureté :99.77% - 99.86%Couleur et forme :SoildMasse moléculaire :296.37[Ala2] Endothelin-3, human
CAS :[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.Formule :C120H166N26O32S4Couleur et forme :SolidMasse moléculaire :2613.02Lys-γ3-MSH(human)
CAS :Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysisFormule :C128H193N45O39SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3018.25BMY-14802
CAS :BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.Formule :C18H22F2N4ODegré de pureté :99.84%Couleur et forme :SoildMasse moléculaire :348.39Ref: TM-T67739
2mg35,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg90,00€25mg164,00€50mg259,00€100mg383,00€200mg545,00€KwFwLL-NH2
CAS :KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).Formule :C49H66N10O6Couleur et forme :SolidMasse moléculaire :891.11AdTx1
Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.Formule :C310H481N87O100S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7283.22Taspoglutide
CAS :Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetesFormule :C152H232N40O45Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3339.763PACAP (6-38), human, ovine, rat TFA
PACAP (6-38) is a PACAP receptor blocker with IC50s of 30, 600, 40 nM for type I, VIP1, and VIP2 receptors.Formule :C184H301N56FO47SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4138.76ANQ-11125 TFA
ANQ-11125 TFA is a motilin antagonist with a pKd of 8.24, inhibiting motilide contractions in rabbits.Formule :C88H126F3N19O23Couleur et forme :SolidMasse moléculaire :1875.05ARC 239 dihydrochloride
CAS :ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).Formule :C24H31Cl2N3O3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :480.43Amitraz
CAS :Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.Formule :C19H23N3Degré de pureté :99.88%Couleur et forme :White/Pale Yellow Crystalline SolidMasse moléculaire :293.41Mosapride citrate dihydrate
CAS :Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.Formule :C27H35ClFN3O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.04Prostaglandin J2
CAS :PGJ2, a PGD2 metabolite, is a DP agonist (Ki: 0.9 nM hDP, 6.6 nM hCRTH2), induces cAMP (EC50: 1.2 nM), oxidative stress, neuronal apoptosis, and neurotoxicity.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.45Pasireotide (diaspartate)
CAS :Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formule :C66H80N12O17Couleur et forme :SolidMasse moléculaire :1313.41Y1 receptor antagonist 1 formic
H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.Formule :C29H35N5O5Couleur et forme :SolidMasse moléculaire :533.62LH-RH (4-10)
CAS :LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formule :C33H53N11O9Couleur et forme :SolidMasse moléculaire :747.841,8-Cineole
CAS :Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formule :C10H18ODegré de pureté :97.44% - 97.44%Couleur et forme :SolidMasse moléculaire :154.25Adrenomedullin (1-50), rat
CAS :Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Formule :C248H381N77O75S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5729.5Prostaglandin B1
CAS :Prostaglandin B1 (PGB1), a metabolite of Prostaglandin E1, acts as a prostanoid receptor ligand [1] [2].Formule :C20H32O4Masse moléculaire :336.47Neuropeptide Y (18-36) (porcine)
CAS :"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."Formule :C112H174N36O27Couleur et forme :SolidMasse moléculaire :2456.8LSN3160440
CAS :LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.Formule :C27H27Cl2N3OCouleur et forme :SolidMasse moléculaire :480.43N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS :N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formule :C10H16ClNCouleur et forme :SolidMasse moléculaire :185.69[Tyr1]-Somatostatin-14
CAS :[Tyr1]-Somatostatin-14 could binds to SSTR2.Formule :C82H108N18O20S2Masse moléculaire :1729.99MR 409
CAS :MR 409, a selective growth hormone-releasing hormone (GHRH) agonist, exhibits notable neuroprotective properties by augmenting endogenous neurogenesis inFormule :C153H252N44O43Couleur et forme :SolidMasse moléculaire :3395.91cAC 253 acetate
cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.
Formule :C128H206N42O42S2Degré de pureté :98.16% - 99.99%Couleur et forme :SoildMasse moléculaire :3069.39[18F]-Labeled L-dopa precursor
CAS :[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formule :C35H36N2O7Couleur et forme :SolidMasse moléculaire :596.67TGR5 agonist 4
TGR5 agonist 4 (compound 19), a derivative of cholic acid, selectively activates the TGR5 receptor with an effective concentration (EC50) of 4 μM [1].Formule :C24H38F2O5Couleur et forme :SolidMasse moléculaire :444.55Septide
CAS :Septide is an NK1 receptor agonist acting at a site distinct from substance P.Formule :C39H53N7O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :763.95GRPP (human)
CAS :GRPP (human), a 30-amino-acid peptide derived from Gcg, modestly elevates plasma insulin levels while reducing plasma glucagon concentrations.Formule :C136H215N41O58SCouleur et forme :SolidMasse moléculaire :3384.47Motilin, canine
CAS :Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.Formule :C120H194N36O34Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2685.05Nastorazepide hemicalcium
CAS :Nastorazepide (Z-360) hemicalcium is a selective, orally-administered 1,5-benzodiazepine derivative that functions as a receptor antagonist for gastrin/cholecystokinin 2 (CCK-2), exhibiting potential antitumor activity.Formule :C29H36N4O5CaCouleur et forme :SolidMasse moléculaire :540.66CB2R/FAAH modulator-1
CAS :CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formule :C24H27NO2Degré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :361.48Ref: TM-T67896
1mg50,00€5mg105,00€1mL*10mM (DMSO)108,00€10mg154,00€25mg224,00€50mg314,00€100mg427,00€200mg575,00€V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
Formule :C20H26ClF3N4O2Degré de pureté :99.97%Couleur et forme :SoildMasse moléculaire :446.89Neuropeptide W-30 (human)
CAS :Neuropeptide W-30 (human) serves as a crucial stress mediator within the central nervous system, influencing the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. It acts as an endogenous ligand for the two related orphan G-protein-coupled receptors (GPCRs), GPR7 and GPR8, binding and activating them at comparable effective doses [1] [2] [3].Formule :C165H249N49O37SCouleur et forme :SolidMasse moléculaire :3543.11rac Desmethyl Citalopram Hydrochloride
CAS :rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.Formule :C19H20ClFN2ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :346.83d[Cha4]-AVP
CAS :Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Formule :C50H71N13O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1094.31BAM(8-22) TFA
BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.Formule :C93H128F3N25O25SCouleur et forme :SolidMasse moléculaire :2085.22Aldioxa
CAS :Aldioxa is a Gastrointestinal Agent.Formule :C4H7AlN4O5Couleur et forme :SolidMasse moléculaire :218.10Scyliorhinin II
CAS :Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.Formule :C77H119N21O26S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1851.09Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formule :C75H110N18O20·xC2HF3O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :1583.78 (free base)Mosliciguat
CAS :Mosliciguat is a guanylate cyclase activator.Formule :C41H36ClF3N2O5Couleur et forme :SolidMasse moléculaire :729.19GIP/GLP-1 dual receptor agonist-1
CAS :Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Couleur et forme :SolidLCKLSL
CAS :LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.Formule :C30H57N7O8SMasse moléculaire :675.89
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