GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.024 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5990 produits trouvés pour "GPCR/G-Protéine"
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Cortistatin 29
Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.Formule :C161H242N46O41S2Couleur et forme :SolidMasse moléculaire :3539.77Calcitonin Gene Related Peptide (CGRP) II, rat TFA
Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.Formule :C165H268F3N51O52S2Couleur et forme :SolidMasse moléculaire :3919.33Neuropeptide S(Mouse) TFA
Neuropeptide S(Mouse) TFA: Endogenous NPSR agonist, EC50 3 nM, boosts Ca2+, activity, wakefulness, and lowers mouse anxiety.
Formule :C92H157F3N34O29Couleur et forme :SolidMasse moléculaire :2296.49Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS :Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFormule :C45H63N15O11S2Couleur et forme :SolidMasse moléculaire :1054.21Dapiglutide
CAS :Dapiglutide (ZP7570) is a long-acting GLP-1R & GLP-2R dual agonist for SBS research.Couleur et forme :SolidBA 1 TFA
BA1 TFA agonizes BB receptors; binds BRS3, GRPR, NMBR with IC50s of 6, 0.4, 2.5 nM.Formule :C59H77F3N14O13Couleur et forme :SolidMasse moléculaire :1247.32ELA-11(human) TFA
ELA-11(human) TFA: apelin receptor agonist, K i =14 nM, inhibits cAMP, stimulates β-arrestin, from ELA-32 fragment.Formule :C60H91F3N16O15S2Couleur et forme :SolidMasse moléculaire :1397.58Cagrilintide
CAS :Cagrilintide is a long-acting amylin analogue acting as a dual agonist of the amylin receptor and calcitonin receptor, reducing body weight and food intake.Formule :C194H312N54O59S2Couleur et forme :SolidMasse moléculaire :4409.01Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe andFormule :C58H77N14O21S2Degré de pureté :98.47% - 98.54%Couleur et forme :SoildMasse moléculaire :1370.44Ref: TM-T14932L1
1mL*10mM (DMSO)34,00€1mg93,00€5mg313,00€10mg465,00€25mg742,00€50mg982,00€100mg1.333,00€500mg2.637,00€Imipramine N-oxide
CAS :Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.Formule :C19H24N2ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :296.41Ref: TM-T74205
1mg72,00€5mg157,00€1mL*10mM (DMSO)167,00€10mg241,00€25mg409,00€50mg565,00€100mg794,00€JKC363 TFA
JKC363 TFA is an MC4 receptor antagonist with 90x more affinity than MC3 (IC50: 0.5 nM vs 44.9 nM), blocks α-MSH's effect on TRH, and is anti-hyperalgesic.Formule :C71H93F3N19O18S2Couleur et forme :SolidMasse moléculaire :1620.73Tezusomant
CAS :Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Formule :C120H171N23O32SCouleur et forme :SolidMasse moléculaire :2479.84FLLRN
CAS :FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.Formule :C31H51N9O7Couleur et forme :SolidMasse moléculaire :661.79Tau conotoxin CnVA
CAS :Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Formule :C72H116N24O17S4Couleur et forme :SolidMasse moléculaire :1718.1HL2-m5
CAS :HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formule :C70H101N15O24S3Couleur et forme :SolidMasse moléculaire :1632.83Xenopus orexin B
CAS :Xenopus orexin B, a neuropeptide identified as an endogenous ligand for an orphan G-protein-coupled receptor, acts as a potent agonist of OX2R [1].Formule :C130H219N45O40S2Couleur et forme :SolidMasse moléculaire :3116.54TRAP-5 amide
CAS :TRAP-5 amide is a peptide agonist for protease-activated receptor 1 (PAR 1) [1].Formule :C30H51N9O6Couleur et forme :SolidMasse moléculaire :633.78Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Degré de pureté :99.22%Couleur et forme :SoildAntibacterial agent 189
Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.Formule :C37H28N4OMasse moléculaire :544.22631Palmitoyl tetrapeptide-20 TFA
Palmitoyl tetrapeptide-20 (PTP20) TFA is a biomimetic peptide and acts as an agonist of α-MSH. It protects follicular melanocytes by boosting catalase expression and activating melanogenesis.Formule :C38H70N6O8·xC2HF3O2Peptide C105Y TFA
Peptide C105Y TFA is a cell-penetrating peptide synthesized based on the amino acid sequence of residues 359-374 of α1-antitrypsin. It enhances the gene expression of DNA nanoparticles.Formule :C97H148N20O23S·xC2HF3O2Endolide F
Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.Formule :C25H32N4O6Masse moléculaire :484.23218Relaxin H3 (human) TFA
Relaxin H3 (human) (TFA) is a relaxin peptide that exerts antifibrotic effects through the RXFP1 receptor.Formule :C237H374N70O69S6·xC2HF3O2GLP-1R agonist 20
GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.Formule :C31H30Cl2F2N4O5Masse moléculaire :646.15613palm11-PrRP31
Palm11-PrRP31 is a lipid-modified analog of the endogenous appetite-suppressing neuropeptide (PrRP). It functions as a potent dual agonist for GPR10 (EC50 = 39 pM) and NPFF-R2. By mimicking the natural activity of PrRP, palm11-PrRP31 binds to these receptors to reduce food intake. It has potential applications as an anti-obesity agent and is useful in studying neuropeptide and receptor interactions.Formule :C181H289N55O46SMasse moléculaire :4001.16865Neuropeptide Y (human) free acid
CAS :Neuropeptide Y (human) free acid is the deamidated form of Neuropeptide Y (human, rat, mouse). The amidation of the C-terminal tyrosine in Neuropeptide Y is essential for its function, while the non-amidated form cannot initiate G-protein signaling.Formule :C189H284N54O58SMasse moléculaire :4270.06542Wy 43657
CAS :Wy 43657 is a gonadorelin antagonist.Formule :C71H86N14O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1343.554APTAA-LHRH
CAS :APTAA-LHRH is a gonadorelin antagonist.Formule :C69H91Cl2N17O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1453.47U 67827E
CAS :U 67827E is a long-lasting cholecystokinin agonist. It acts by decreases food intake.Formule :C53H68N10O17SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1149.24AA 497 HCl
CAS :AA 497, a beta-2 agonist, suppresses Ca spikes.Formule :C14H22ClNO3Couleur et forme :SolidMasse moléculaire :287.78Anticancer agent 258
CAS :Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.Formule :C17H12F2N4Couleur et forme :SolidMasse moléculaire :310.3Azaline
CAS :Azaline is a gonadorelin antagonist.Formule :C74H106ClN23O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1545.26Clopidogrel-related Compound B hydrochloride
CAS :Clopidogrel Related Compound B is a useful organic compound for research related to life sciences.Formule :C16H17Cl2NO2SCouleur et forme :SolidMasse moléculaire :358.28L 366811
CAS :L 366811 is a potent oxytocin antagonist.Formule :C43H56N8O6Couleur et forme :SolidMasse moléculaire :780.95AC-178335
CAS :AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.Formule :C49H63N13O7Couleur et forme :SolidMasse moléculaire :946.11Acrinor
CAS :Acrinor is a adrenergic beta receptor agonist.Formule :C35H46Cl2N10O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :805.72ADTN
CAS :ADTN is an agonist of the dopamine receptor.Formule :C10H13NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.22Ono 3708
CAS :Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.Formule :C23H37NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.54LHRH, Ala(6)-
CAS :LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formule :C56H77N17O13Couleur et forme :SolidMasse moléculaire :1196.32Rubraxanthone
CAS :Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.Formule :C24H26O6Couleur et forme :SolidMasse moléculaire :410.466Alverine hydrochloride
CAS :Alverine hydrochloride is a parasympatholytic.Formule :C20H28ClNCouleur et forme :SolidMasse moléculaire :317.9GRL093-22
GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.Formule :C33H29FN6O3Couleur et forme :SolidMasse moléculaire :576.62Jmv 167
CAS :Jmv 167 is an antagonist of the Cholecystokinin receptor.Formule :C51H68N8O14SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1049.21Vapreotide diacetate
CAS :Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.Formule :C61H78N12O13S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1251.47Ethylnorepinephrine hydrochloride
CAS :Ethylnorepinephrine hydrochloride is a unique bronchodilator.
Formule :C10H16ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.69MCL0129
CAS :MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.Formule :C34H47FN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :546.76TGR5 agonist 7
TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.Formule :C37H59N2NaO9SCouleur et forme :SolidMasse moléculaire :730.935-hydroxy Propranolol
CAS :5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Formule :C16H21NO3Couleur et forme :SolidMasse moléculaire :275.348Alprostadil ethyl ester
CAS :Alprostadil ethyl ester is a biochemical used in the treatment of scleroderma.
Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.53Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47CAY10597
CAS :PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).
Formule :C20H14ClFN2O5Couleur et forme :SolidMasse moléculaire :416.79Gemeprost
CAS :Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.Formule :C23H38O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.545-methoxy-α-Ethyltryptamine
CAS :5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formule :C13H18N2ODegré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :218.29CAY10734
CAS :CAY10734 has a wide range of applications in life science related research.Formule :C23H25N3O3Couleur et forme :SolidMasse moléculaire :391.471Leukotriene B5
CAS :LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.4561,2,3-Trilinoelaidoyl-rac-glycerol
CAS :1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.Formule :C57H98O6Couleur et forme :SolidMasse moléculaire :879.405Prosaptide TX14(A)
CAS :GPR37L1/GPR37 agonist with EC50 of 5/7 nM, activates G proteins, enhances ERK, myelin synthesis, neuro/glioprotection.Formule :C69H110N16O26Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1579.72Nocistatin(human)
CAS :Blocker of nociceptin-induced allodynia and hyperalgesiaFormule :C149H238N42O53S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3561.936α-Prostaglandin I1
CAS :6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487Xylamidine
CAS :Xylamidine is a biochemical.Formule :C19H24N2O2Couleur et forme :SolidMasse moléculaire :312.4126Rfa, Hypothalamic Peptide, human
CAS :26RFa, a human neuropeptide, stimulates appetite and possibly regulates feeding and the gonadotropic axis, with ≈80% identity across human, rat, and frog.Formule :C127H195N37O37Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2832.13(+)-5-trans Cloprostenol
CAS :Cloprostenol, a synthetic PGF2α derivative, induces estrus and treats reproductive issues in livestock; its minor impurity, (+)-5-trans, is less effective.Formule :C22H29ClO6Couleur et forme :SolidMasse moléculaire :424.92Secretoneurin, rat
CAS :Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formule :C159H252N40O58Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3651.95ORG 2766
CAS :ORG 2766 is an ACTH 4-9 (H-Met(O)-Glu-His-Phe-D-Lys-Phe-OH) analog and neurotrophic peptide.Formule :C40H55N9O11SCouleur et forme :SolidMasse moléculaire :869.99Endothelin-3, human, mouse, rabbit, rat
CAS :Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.Formule :C121H168N26O33S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2643.04(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS :'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM forFormule :C107H162N30O30Couleur et forme :SolidMasse moléculaire :2348.61[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Formule :C58H82N16O12Couleur et forme :SolidMasse moléculaire :1195.37Acetyl neurotensin (8-13)
CAS :Acetyl neurotensin (8-13), the most concise analog of neurotensin, retains complete binding and pharmacological properties [1].Formule :C40H66N12O9Couleur et forme :SolidMasse moléculaire :859.03KISS1-305
CAS :KISS1-305: Metastin analog, prototype peptide, resists protease degradation, suboptimal KISS1R agonist.Formule :C56H76N16O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1165.3Nemifitide diTFA
CAS :Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain barrier.Formule :C37H45F7N10O10Degré de pureté :99.78% - 99.84%Couleur et forme :SolidMasse moléculaire :922.8(Iso)-Landipirdine
CAS :(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formule :C18H19FN2O3SDegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :362.42AL 34662
CAS :AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFormule :C10H13N3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :191.23CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formule :C97H131F3I2N20O25S2Couleur et forme :SolidMasse moléculaire :2352.13β-MSH, human
CAS :beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).Formule :C118H174N34O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2660.92LY-426965 hydrochloride
CAS :LY-426965 hydrochloride is a bioactive chemical.Formule :C28H39ClN2O2Couleur et forme :SolidMasse moléculaire :471.074-P-PDOT
CAS :4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.Formule :C19H21NODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :279.38PAMP-12(human, porcine)
CAS :Potent endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 57.2 nM). Corresponds to amino acids 9 to 20 of proadrenomedullin.Formule :C77H119N25O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1618.95rGHRH(1-29)NH2
RGHRH (1-29)NH2 is a synthetic peptide that stimulates the secretion of growth hormone (GH).Formule :C155H251N49O40SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3473.02Petrelintide acetate
Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.Formule :C185H305N49O61·xC2H4O2Couleur et forme :SolidMasse moléculaire :4191.69 (free base)Crustacean Cardioactive Peptide (CCAP)
CAS :Crustacean Cardioactive Peptide (CCAP) is a conserved modified cyclic nonapeptide primary structure of PFCNAFTGC-NH2, a disulfide bridge between Cys3 and Cys9.Formule :C42H58N10O12S2Degré de pureté :95.40%Couleur et forme :SolidMasse moléculaire :959.1CRSP-1
CAS :Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.Formule :C175H294N54O49S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4098.88γ-2-MSH (41-58), amide
CAS :Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Formule :C74H100N22O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1569.79WAY-313170
CAS :WAY-313170 Inhibits hedgehog signaling and phosphodiesterase.Formule :C19H17ClN2O2S2Degré de pureté :97.92%Couleur et forme :SolidMasse moléculaire :404.93SDV-Exendin-3/4
SDV-Exendin-3/4 is a 32-amino acid peptide.Formule :NADegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3443.87Prepro VIP (81-122), human
CAS :Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Formule :C202H325N53O64SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4552.13Ornipressin
CAS :Ornipressin is a vasoconstrictor, haemostatic and renal agent.Formule :C45H63N13O12S2Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1042.195-HT5AR/5-HT6R ligand-1
5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.Formule :C25H30N4O2SCouleur et forme :SolidMasse moléculaire :450.6PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formule :C61H89N15O13Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :1240.4519(R)-HETE
CAS :19(R)-HETE is a renal artery vasodilator and can be used to study angiotensin II-induced cardiac hypertrophy.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47Beraprost
CAS :Beraprost is a stable prostacyclin analog.Formule :C24H30O5Couleur et forme :SolidMasse moléculaire :398.495-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55BE-24566B
CAS :BE-24566B, a polyketide from S. violaceusniger, inhibits various bacteria and blocks ET receptors (ETA IC50=11 μM, ETB=3.9 μM).Formule :C27H24O7Couleur et forme :SolidMasse moléculaire :460.48211-deoxy Prostaglandin F1α
CAS :11-deoxy PGF1α is a synthetic analog of PGF1α.Formule :C20H36O4Couleur et forme :SolidMasse moléculaire :340.504GRP (porcine)
CAS :GRP: agonist for GRPR, stimulates amygdala GABA release reducing fear in mice, aids mitogenesis, GI function, and appetite control.Formule :C126H198N38O31S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2805.31Amylin (1-37), human acetate
Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.Degré de pureté :96.21%Couleur et forme :Odour SolidDesglymidodrine
CAS :Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Formule :C10H15NO3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :197.23CCR6 antagonist 2
CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.Formule :C19H24N4O4Couleur et forme :SolidMasse moléculaire :372.42PSEM 308 hydrochloride
PSAM agonist targeting PSAML141F-GlyR and related ion channels in mice; ideal concentration ≤5 mg/kg; plasmids at Addgene.Couleur et forme :SolidGIP/GLP-1 dual receptor agonist-1 sodium
GIP/GLP-1 dual receptor agonist-1 (Compound 4) (sodium) functions as a GIP/GLP-1 receptor agonist. This compound is applicable for research into metabolic disorders and liver diseases, including non-alcoholic steatohepatitis (NASH) and non-alcoholic fatty liver disease (NAFLD).Couleur et forme :Odour SolidIloperidone metabolite P95
CAS :Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formule :C23H25FN2O5Couleur et forme :SolidMasse moléculaire :428.46
