GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.022 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5985 produits trouvés pour "GPCR/G-Protéine"
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PAR-4 Agonist Peptide, amide TFA
CAS :PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.Formule :C36H49F3N8O9Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :794.82Ref: TM-TP1065
1mg34,00€5mg92,00€1mL*10mM (DMSO)131,00€10mg138,00€25mg225,00€50mg323,00€100mg467,00€200mg643,00€4F 4PP oxalate
CAS :4F 4PP oxalate is a 5-HT2A antagonist.Formule :C22H26FNO·C2H2O4Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :429.49Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formule :C46H60F3N13O12SDegré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :1076.12Ref: TM-T7627L
1mg54,00€2mg71,00€5mg92,00€10mg152,00€1mL*10mM (DMSO)202,00€25mg324,00€50mg485,00€100mg620,00€200mg897,00€Pramlintide acetate(151126-32-8 free base)
CAS :Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.Formule :C173H271N51O55S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :4009Tasimelteon
CAS :Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formule :C15H19NO2Degré de pureté :98.93% - 99.93%Couleur et forme :SolidMasse moléculaire :245.32Terazosin hydrochloride dihydrate
CAS :Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formule :C19H25N5O4·HCl·2H2ODegré de pureté :99.81%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :459.92Relenopride hydrochloride
CAS :Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formule :C24H31Cl2FN4O4Couleur et forme :SolidMasse moléculaire :529.43Nafarelin acetate(76932-56-4 free base)
CAS :Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formule :C68H87N17O15Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :1382.55BQ-788 sodium salt
CAS :BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formule :C34H51N5NaO7Couleur et forme :SolidMasse moléculaire :664.8Naluzotan
CAS :Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formule :C23H38N4O3SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :450.64Antazoline
CAS :Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formule :C17H19N3Degré de pureté :≥95%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :265.35ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.Formule :C60H94N16O15S2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :1343.61CB1 antagonist 4
CAS :TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formule :C30H25Cl2F3N4OSDegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :617.51Ref: TM-T8511
2mg46,00€5mg92,00€10mg152,00€1mL*10mM (DMSO)155,00€25mg259,00€50mg405,00€100mg597,00€200mg848,00€Fenspiride
CAS :Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.Formule :C15H20N2O2Couleur et forme :SolidMasse moléculaire :260.33Bupranolol
CAS :Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.Formule :C14H22ClNO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :271.78Ref: TM-T8580
1mg52,00€1mL*10mM (DMSO)96,00€5mg105,00€10mg159,00€25mg309,00€50mg440,00€100mg583,00€200mg785,00€Fluorogestone acetate
CAS :FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formule :C23H31FO5Degré de pureté :99.47%Couleur et forme :CoaMasse moléculaire :406.49Ref: TM-T21335
2mg39,00€5mg58,00€1mL*10mM (DMSO)74,00€10mg93,00€25mg167,00€50mg245,00€100mg371,00€200mg494,00€Dobutamine tartrate
CAS :Dobutamine tartrate is a cardiotonic.Formule :C22H29NO9Couleur et forme :SolidMasse moléculaire :451.472RTICBM-189
CAS :RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formule :C15H14Cl2N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :309.19Ref: TM-T9466
2mg34,00€5mg52,00€1mL*10mM (DMSO)67,00€10mg84,00€25mg161,00€50mg250,00€100mg369,00€200mg522,00€Afamelanotide acetate
CAS :Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.
Formule :C80H115N21O21Degré de pureté :98% - 99.494%Couleur et forme :SolidMasse moléculaire :1706.9Naftopidil hydrochloride
CAS :Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formule :C24H29ClN2O3Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :428.95Ref: TM-T9220
1mg42,00€5mg82,00€1mL*10mM (DMSO)92,00€10mg111,00€25mg192,00€50mg289,00€100mg414,00€200mg580,00€Darusentan
CAS :Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteriesFormule :C22H22N2O6Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :410.43Ref: TM-T5458
2mg43,00€5mg65,00€1mL*10mM (DMSO)67,00€10mg100,00€25mg173,00€50mg288,00€100mg414,00€200mg583,00€GRK5-IN-2
CAS :GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.Formule :C20H20N4O4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :380.4Ref: TM-T9609
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg75,00€25mg138,00€50mg215,00€100mg318,00€200mg444,00€NPS2390
CAS :NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)Formule :C19H21N3ODegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :307.39LY310762
CAS :LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formule :C24H27FN2O2·HClDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :430.94Liraglutide
CAS :Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.Formule :C172H265N43O51Degré de pureté :97.65% - 99.04%Couleur et forme :SolidMasse moléculaire :3751.25Ref: TM-T6876
1mg111,00€2mg197,00€5mg447,00€10mg527,00€25mg843,00€50mg1.144,00€100mg1.521,00€200mg2.052,00€[Des-Arg9]-Bradykinin TFA
CAS :[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formule :C46H62F3N11O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1018.05MK-3697
CAS :MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).Formule :C23H21N5O3SDegré de pureté :97.69% - 98.15%Couleur et forme :SolidMasse moléculaire :447.51Ref: TM-T1913
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)100,00€10mg113,00€25mg200,00€50mg333,00€100mg477,00€Orexin 2 Receptor Agonist
CAS :Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formule :C32H34N4O5SDegré de pureté :98.26% - 99.43%Couleur et forme :SolidMasse moléculaire :586.7Ref: TM-T3177
2mg39,00€5mg60,00€10mg75,00€1mL*10mM (DMSO)77,00€25mg130,00€50mg220,00€100mg323,00€200mg447,00€Metadoxine
CAS :Metadoxine (Metadoxil) is a neurotransmitter stimulant.Formule :C8H11NO3·C5H7NO3Degré de pureté :99.19%Couleur et forme :Off-White PowderMasse moléculaire :298.29Talnetant hydrochloride
CAS :Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.Formule :C25H23ClN2O2Couleur et forme :SolidMasse moléculaire :418.92PD 117519
CAS :PD 117519 (CI947) is an agonist of adenosine receptorFormule :C19H21N5O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :383.4Poloxamer 407
CAS :Poloxamer 407 is a nonionic surfactant.Degré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :12000 (Average)Decynium 22
CAS :Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormule :C23H23IN2Degré de pureté :99.92%Couleur et forme :Dark Red CrystalsMasse moléculaire :454.35Aripiprazole monohydrate
CAS :Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formule :C23H29Cl2N3O3Couleur et forme :SolidMasse moléculaire :466.4Tandospirone hydrochloride
CAS :Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.Formule :C21H30ClN5O2Couleur et forme :SolidMasse moléculaire :419.95Clozapine HCl
CAS :Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.Formule :C18H20Cl2N4Couleur et forme :SolidMasse moléculaire :363.29ML-191
CAS :ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formule :C24H25N3O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :403.47Bavisant dihydrochloride hydrate
CAS :Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.Formule :C19H31Cl2N3O3Couleur et forme :SolidMasse moléculaire :420.38Quipazine
CAS :Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.Formule :C13H15N3Couleur et forme :SolidMasse moléculaire :213.28Brefonalol
CAS :Brefonalol is a vasodilating beta-adrenergic receptor blocker.Formule :C22H28N2O2Couleur et forme :SolidMasse moléculaire :352.47Raclopride tartrate
CAS :Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).Formule :C19H26Cl2N2O9Couleur et forme :SolidMasse moléculaire :497.32Midaglizole
CAS :Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.Formule :C16H17N3Couleur et forme :SolidMasse moléculaire :251.33Cangrelor free acid
CAS :Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.Formule :C17H25Cl2F3N5O12P3S2Couleur et forme :SolidMasse moléculaire :776.36Eltoprazine dihydrochloride
CAS :Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Formule :C12H18Cl2N2O2Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :293.194-Methylhistamine hydrochloride
CAS :Compound with imidazole ring & amine group; inhibits copper enzymes, affects gene expression.Formule :C6H12ClN3Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :161.633Ref: TM-T50049
1mg74,00€2mg96,00€1mL*10mM (DMSO)126,00€5mg156,00€10mg225,00€25mg379,00€50mg568,00€100mg810,00€500mg1.644,00€Butyrophenone
CAS :Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.Formule :C10H12ODegré de pureté :99.84%Couleur et forme :Colourless To Yellow LiquidMasse moléculaire :148.2BCTC
CAS :BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formule :C20H25ClN4ODegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :372.89Ibutamoren
CAS :Ibutamoren (MK-677) is a drug which acts as a potent, orally active growth hormone secretagogue, mimicking the GH stimulating action of the endogenous hormone ghrelin. It also alters the metabolism of body fat and so may have an application in the treatment of obesity.Formule :C27H36N4O5SDegré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :528.66GBR 12935
CAS :GBR-12935: selective dopamine inhibitor, used in Parkinson's research.Formule :C28H34N2OCouleur et forme :SolidMasse moléculaire :414.58M 1145 acetate
M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; >90x affinity vs GAL1, 76x vs GalR3. Enhances galanin signal.Formule :C130H209N37O34Degré de pureté :99.1%Couleur et forme :SolidMasse moléculaire :2834.28Ref: TM-TP1991L
1mg248,00€5mg532,00€10mg712,00€25mg1.054,00€50mg1.425,00€100mg1.928,00€200mg2.593,00€Loxapine hydrochloride
CAS :Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Formule :C18H19Cl2N3OCouleur et forme :SolidMasse moléculaire :364.27Brompheniramine
CAS :Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formule :C16H19BrN2Couleur et forme :SolidMasse moléculaire :319.24GSK 789472 hydrochloride
CAS :GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Formule :C15H22ClN3ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :295.81Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Formule :C65H102N16O25Degré de pureté :95.55%Couleur et forme :SolidMasse moléculaire :1507.6CYM 50358 hydrochloride (1314212-39-9 free base)
CAS :CYM50358 HCl is an S1P4 antagonist.Formule :C20H19Cl3N2O2Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :425.73N-ACETYLTRYPTAMINE
CAS :N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Formule :C12H14N2ODegré de pureté :98.79%Couleur et forme :PowderMasse moléculaire :202.25GR 125743
CAS :GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Formule :C25H28N4O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :416.52Ref: TM-T8737
1mg40,00€2mg52,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg113,00€25mg222,00€50mg333,00€100mg495,00€Enavogliflozin
CAS :Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.Formule :C24H27ClO6Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :446.92Ref: TM-T38843
1mg147,00€5mg358,00€1mL*10mM (DMSO)394,00€10mg560,00€25mg973,00€50mg1.333,00€100mg1.765,00€Intepirdine
CAS :Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Formule :C19H19N3O2SDegré de pureté :98% - 98.63%Couleur et forme :SolidMasse moléculaire :353.44ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS :ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)Formule :C14H15NO2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :261.34Olodaterol hydrochloride
CAS :Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.Formule :C21H27ClN2O5Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :422.9Mosapride Citrate
CAS :Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formule :C21H25ClFN3O3·C6H8O7Degré de pureté :99.70%Couleur et forme :White PowderMasse moléculaire :614.02Blarcamesine
CAS :Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
Formule :C19H23NODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :281.39Nomifensine maleate
CAS :Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
Formule :C20H22N2O4Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :354.4Mecamylamine hydrochloride
CAS :Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formule :C11H22ClNDegré de pureté :99.76% - >99.99%Couleur et forme :White SolidMasse moléculaire :203.75Buserelin Acetate (57982-77-1 free base)
CAS :Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Formule :C62H90N16O15Degré de pureté :99.31% - 99.78%Couleur et forme :SolidMasse moléculaire :1299.48SB 242084 dihydrochloride
CAS :SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formule :C21H21Cl3N4O2Couleur et forme :SolidMasse moléculaire :467.781-(1-Naphthyl) piperazine hydrochloride
CAS :1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multipleFormule :C14H17ClN2Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :248.75HAEGTFTSDVSSYLE
HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.Formule :C71H103N17O28Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1642.71Alimemazine hemitartrate
CAS :Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formule :C18H22N2SC4H6O6Degré de pureté :98.16% - 99.69%Couleur et forme :SolidMasse moléculaire :448.53CCR2 antagonist 4 hydrochloride
CAS :CCR2 antagonist 4 hydrochloride is a specific CCR2 antagonist (IC50s: 180 nM for CCR2b). It potently inhibits MCP-1-induced chemotaxis (IC50: 24 nM).Formule :C21H22Cl2F3N3O2Couleur et forme :SolidMasse moléculaire :476.32CAY10444
CAS :CAY10444 is an S1P3 specific antagonist.Formule :C15H29NO2SDegré de pureté :99.15% - 99.61%Couleur et forme :SolidMasse moléculaire :287.46Ref: TM-T23860
5mg44,00€1mL*10mM (DMSO)48,00€10mg71,00€25mg137,00€50mg222,00€100mg371,00€200mg505,00€500mg795,00€CYM-5520
CAS :CYM-5520 is a noncompetitive allosteric agonist of S1P2Formule :C21H19N3O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :345.39Ref: TM-T22703
1mg46,00€2mg60,00€5mg88,00€1mL*10mM (DMSO)98,00€10mg135,00€25mg236,00€50mg354,00€100mg528,00€ML 10302
CAS :ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formule :C15H21ClN2O3Couleur et forme :SolidMasse moléculaire :312.79N-Cbz-DL-tryptophan
CAS :N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formule :C19H18N2O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :338.36Samelisant dihydrochloride
CAS :SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.Formule :C21H33Cl2N3O3Couleur et forme :SolidMasse moléculaire :446.41Galnon TFA
CAS :Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).Formule :C42H47F3N4O8Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :792.84Ref: TM-T8559
1mg58,00€1mL*10mM (DMSO)86,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€CRT0273750
CAS :CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formule :C25H22ClF3N4O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :502.92Picotamide
CAS :Picotamide has anticoagulant and fibrinolytic properties.Formule :C21H20N4O3Degré de pureté :98.90%Couleur et forme :SolidMasse moléculaire :376.41Ref: TM-T9153
1mg38,00€5mg92,00€1mL*10mM (DMSO)94,00€10mg147,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€Bevantolol
CAS :Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formule :C20H27NO4Couleur et forme :SolidMasse moléculaire :345.43Lodoxamide
CAS :Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formule :C11H6ClN3O6Degré de pureté :99.13% - 99.96%Couleur et forme :SolidMasse moléculaire :311.63Benorilate
CAS :Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formule :C17H15NO5Degré de pureté :98.39% - 99.85%Couleur et forme :SolidMasse moléculaire :313.3NPS ALX Compound 4a
CAS :NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formule :C25H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.55Carbazochrome
CAS :Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.Formule :C10H12N4O3Degré de pureté :98.36%Couleur et forme :Nacarat Crystalline PowderMasse moléculaire :236.23Quipazine maleate
CAS :Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formule :C17H19N3O4Couleur et forme :SolidMasse moléculaire :329.356Olcegepant
CAS :Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formule :C38H47Br2N9O5Degré de pureté :96.08% - 97.24%Couleur et forme :SolidMasse moléculaire :869.65Sigma-LIGAND-1 hydrochloride
CAS :Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formule :C27H34ClNO4Couleur et forme :SolidMasse moléculaire :472.02Volinanserin
CAS :Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formule :C22H28FNO3Degré de pureté :98.94% - 99.95%Couleur et forme :SolidMasse moléculaire :373.46Ref: TM-T5389
1mg39,00€5mg84,00€1mL*10mM (DMSO)92,00€10mg117,00€25mg220,00€50mg285,00€100mg371,00€200mg530,00€Enprofylline
CAS :Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Ref: TM-T21389
2mg42,00€1mL*10mM (DMSO)59,00€5mg62,00€10mg88,00€25mg141,00€50mg215,00€100mg318,00€200mg442,00€Niaprazine
CAS :Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44Rimcazole dihydrochloride
CAS :Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.Formule :C21H28ClN3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :357.92Ref: TM-T23234
1mg43,00€2mg56,00€5mg93,00€10mg137,00€25mg289,00€50mg470,00€100mg683,00€500mg1.423,00€γ-L-Glutamyl-L-alanine
CAS :γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).Formule :C8H14N2O5Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :218.21Tavapadon
CAS :Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formule :C19H16F3N3O3Degré de pureté :99.33% - 99.8%Couleur et forme :SolidMasse moléculaire :391.34Ref: TM-T16999
1mg77,00€5mg166,00€1mL*10mM (DMSO)178,00€10mg260,00€25mg475,00€50mg668,00€100mg888,00€Piboserod hydrochloride
CAS :Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formule :C22H32ClN3O2Couleur et forme :SolidMasse moléculaire :405.96YIL781 hydrochloride
CAS :YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).Formule :C24H29ClFN3O2Couleur et forme :SolidMasse moléculaire :445.96Cyclopiazonic acid
CAS :Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Formule :C20H20N2O3Degré de pureté :99.27% - 99.80%Couleur et forme :SolidMasse moléculaire :336.38SB756050
CAS :SB756050 is a specific TGR5 agonist.Formule :C21H28N2O8S2Degré de pureté :98.78% - >99.99%Couleur et forme :SolidMasse moléculaire :500.59ML-193
CAS :ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formule :C28H25N5O4SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :527.59Dolasetron Mesylate hydrate
CAS :Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Formule :C20H26N2O7SDegré de pureté :99.86% - 99.99%Couleur et forme :SolidMasse moléculaire :438.49BMY-25368
CAS :BMY-25368 is a long-acting antagonist of the H2-receptor.Formule :C19H25N3O3Couleur et forme :SolidMasse moléculaire :343.42
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