GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5986 produits trouvés pour "GPCR/G-Protéine"
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SR2640
CAS :SR2640 is a potent and highly selective LTD4/LTE4 antagonist, specifically inhibiting LTD4-induced contractions in guinea pig ileum and tracheal smooth muscle in a concentration-dependent manner, without affecting histamine-induced contractions. It blocks the binding of 0.4 nM [3H]LTD4 to guinea pig lung membrane receptors with an IC50 of 23 nM. SR2640 also causes a parallel rightward shift in the dose-response curve for LTD4-induced bronchoconstriction in guinea pigs when administered intravenously, with the degree of shift correlating positively with its dosage. SR2640 is applicable for asthma research.Formule :C23H18N2O3Couleur et forme :SolidMasse moléculaire :370.401LPA5 antagonist 2
LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.Formule :C26H25FN2O4SCouleur et forme :SolidMasse moléculaire :480.55Nedemelteon
CAS :Nedemelteon is an agonist of the melatonin receptor (melatonin receptor).Formule :C15H18N2O2Couleur et forme :SolidMasse moléculaire :258.32Monlunabant
CAS :Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor [1].Formule :C26H22ClF3N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :591.0016(R)-Iloprost
CAS :Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49SGLT1/2-IN-1
CAS :SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.488-iso Prostaglandin F3α
CAS :8-iso PGF3α is an isoprostane produced from the free-radical peroxidation of EPA.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47Becondogrel
CAS :Becondogrel (2-Oxoclopidogrel) is a metabolite of Clopidogrel. It irreversibly inhibits the P2Y12 receptor, thereby preventing platelet aggregation and thrombosis.Formule :C16H16ClNO3SCouleur et forme :SolidMasse moléculaire :337.821BIIE-0246 HCl
CAS :BIIE-0246: A potent, non-peptide Y2 receptor antagonist; >650-fold more selective than Y1, Y4, Y5.Formule :C49H59Cl2N11O6Couleur et forme :SolidMasse moléculaire :968.97NK1 receptor antagonist 2
CAS :NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.Formule :C31H35F7N4O2Couleur et forme :SolidMasse moléculaire :628.62NPR-C activator 1
CAS :NPR-C activator 1 is an activator of the natriuretic peptide receptor C (NPR-C), which can be used to study cardiovascular diseases.Formule :C18H24N6O3Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :372.42Vibegron
CAS :Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Formule :C26H28N4O3Couleur et forme :SolidMasse moléculaire :444.53SB 258741 hydrochloride
SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].Formule :C19H31ClN2O2SCouleur et forme :SolidMasse moléculaire :386.98VA012
CAS :VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. It has been shown to reduce food intake and prevent weight gain during subchronic administration without causing central nervous system-related discomfort. VA012 is applicable in obesity research.Formule :C21H19N3Couleur et forme :SolidMasse moléculaire :313.40MRS2905 trisodium
CAS :MRS2905 (α,β-Methylene-2-thio-UDP) trisodium is a selective P2Y14R agonist with an EC50 of 0.92 nM. It shows no activity on UDP-activated P2Y6 receptors or other P2Y receptors.Formule :C10H13N2Na3O10P2SCouleur et forme :SolidMasse moléculaire :484.199Elsovaptan
CAS :Elsovaptan is an antagonist of the vasopressin receptor and is applicable for research in Alzheimer's disease.Formule :C19H20ClN5O2Couleur et forme :SolidMasse moléculaire :385.847YNT-3708
CAS :YNT-3708 is an orexin receptor (OXR) agonist, exhibiting EC50 values of 14.6 nM for OX1R and 277 nM for OX2R.Formule :C35H36N4O6SCouleur et forme :SolidMasse moléculaire :640.749Neflumozide
CAS :Neflumozide (HRP 913) is an orally effective derivative of benzisoxazole, characterized by its potent dopamine antagonist properties and antipsychotic activity. It is utilized in research related to psychiatric disorders.Formule :C22H23FN4O2Couleur et forme :SolidMasse moléculaire :394.44hA3AR agonist 1
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .Formule :C10H14N6OSCouleur et forme :SolidMasse moléculaire :266.32Befiradol hydrochloride
CAS :Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.Formule :C20H23Cl2F2N3ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :430.32Dersimelagon
CAS :Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.Formule :C36H45F4N3O5Degré de pureté :97.35% - 98.23%Couleur et forme :SolidMasse moléculaire :675.75Vofopitant
CAS :Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).Formule :C21H23F3N6ODegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :432.44LSN3318839
CAS :LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and canFormule :C26H23Cl2N3O2Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :480.39AZD-5672
CAS :AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.Formule :C32H38F2N2O5S2Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :632.78Ref: TM-T30260
1mg192,00€5mg434,00€1mL*10mM (DMSO)530,00€10mg610,00€25mg888,00€50mg1.243,00€100mg1.693,00€Treprostinil diethanolamine
CAS :Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,Formule :C27H45NO7Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :495.65SB-423562
CAS :SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.Formule :C26H32N2O4Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :436.54Ref: TM-T12846
1mg37,00€5mg80,00€1mL*10mM (DMSO)89,00€10mg119,00€25mg210,00€50mg319,00€100mg442,00€200mg605,00€BMS-986141
CAS :BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614Formule :C27H23N5O5S2Degré de pureté :98.43% - 99.26%Couleur et forme :SolidMasse moléculaire :561.63AZD5462
CAS :AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.Formule :C30H41FN2O6Degré de pureté :98.32% - 99.63%Couleur et forme :SolidMasse moléculaire :544.65SB-224289 hydrochloride
CAS :SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formule :C32H33ClN4O3Degré de pureté :98.99% - 99.96%Couleur et forme :SolidMasse moléculaire :557.08Vofopitant dihydrochloride
CAS :Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.Formule :C21H25Cl2F3N6ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :505.36Ref: TM-T13329L
1mg94,00€5mg222,00€1mL*10mM (DMSO)248,00€10mg356,00€25mg675,00€50mg1.009,00€100mg1.378,00€500mg2.673,00€BQ-788
CAS :BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.Formule :C34H51N5O7Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :641.8Ref: TM-T10595
1mg130,00€2mg178,00€5mg313,00€1mL*10mM (DMSO)341,00€10mg447,00€25mg713,00€50mg964,00€100mg1.305,00€500mg2.592,00€PF-07258669
CAS :PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.Formule :C25H27FN6O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :462.52Rolapitant hydrochloride
CAS :Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Formule :C25H27ClF6N2O2Degré de pureté :98.35% - 99.79%Couleur et forme :SolidMasse moléculaire :536.94Ref: TM-T3724
1mg153,00€5mg365,00€1mL*10mM (DMSO)439,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€200mg1.882,00€CYM 9484
CAS :CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with an IC50 value of 19 nM.Formule :C27H31N3O3S2Couleur et forme :SolidMasse moléculaire :509.68ML-290
CAS :ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.Formule :C24H21F3N2O5SCouleur et forme :SolidMasse moléculaire :506.49HOKU-81
CAS :HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.Formule :C12H18ClNO2Couleur et forme :SolidMasse moléculaire :243.73Beraprost sodium
CAS :Beraprost sodium is a stable and orally active prodrug of PGI2.Formule :C24H29NaO5Couleur et forme :SolidMasse moléculaire :420.4817-Desmethyl-agomelatine
CAS :7-Desmethyl-agomelatine, a metabolite of Agomelatine, exhibits lower activity than Agomelatine, which functions as a melatonergic (MT1 and MT2) agonist and 5-HT2C antagonist.Formule :C14H15NO2Couleur et forme :SolidMasse moléculaire :229.27BIBP3226 TFA
CAS :BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).Formule :C29H32F3N5O5Couleur et forme :SolidMasse moléculaire :587.59ML-00253764 hydrochloride
CAS :ML-00253764 hydrochloride is an antagonist of nonpeptidic melanocortin receptor 4 (MC4R) (Ki and IC50 of 0.16 µM and 0.103 µM, respectively).Formule :C18H19BrClFN2OCouleur et forme :SolidMasse moléculaire :413.71JMV 2959
CAS :JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).Formule :C30H32N6O2Couleur et forme :SolidMasse moléculaire :508.61SR 146131
CAS :SR 146131 is a potent and selective agonist of the nonpeptide receptor.Formule :C32H36ClN3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :610.16Pumosetrag Hydrochloride
CAS :Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.Formule :C15H18ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :339.84Arotinolol
CAS :Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand [125I-ICYP] to [5HT1B-serotonergic] receptor sites. It is an antihypertensive agent.Formule :C15H21N3O2S3Couleur et forme :White SolidMasse moléculaire :371.54SB-399885 hydrochloride
CAS :SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.Formule :C18H22Cl3N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.81Protease-Activated Receptor-4
CAS :Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.Formule :C33H46N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :666.77Picumeterol
CAS :Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth muscle relaxation. Picumeterol is a pure R enantiomer that can be used to improve lung function and reduce airway hyperreactivity in patients with asthma.Formule :C21H29Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.38TAK-683
CAS :TAK-683: a full KISS1R agonist, IC50=170 pM; a nonapeptide metastin analog with human EC50=0.96 nM, rat EC50=1.6 nM.Formule :C64H83N17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1298.45Sarizotan
CAS :Sarizotan (EMD 128130) is an orally active compound that acts as an agonist for serotonin 5-HT 1A receptors and dopamine receptors, with IC50 values of 6.5 nM for rat 5-HT 1A, 0.1 nM for human 5-HT 1A, 15.1 nM for rat D 2, 17 nM for human D 2, 6.8 nM for human D 3, and 2.4 nM for human D 4.2.Formule :C22H21FN2OCouleur et forme :SolidMasse moléculaire :348.421Vornorexant
CAS :Vornorexant (ORN-0829; TS-142) is a potent dual OX1R and OX2R antagonist with IC50 values of 1.05 nM and 1.27 nM, respectively. It exhibits potent sleep-promoting effects in vivo and can be used for insomnia treatment research.Formule :C23H22FN7O2Couleur et forme :SolidMasse moléculaire :447.4744-Hydroxyatomoxetine
CAS :4-Hydroxyatomoxetine, an active metabolite of Atomoxetine, is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.Formule :C17H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :271.35SKF 89748
CAS :SKF 89748 is an agonists of alpha 1-adrenoceptor.Formule :C12H17NOSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :223.33CRTh2 antagonist 3
CAS :CRTh2 antagonist 3, a potent molecule, activates PDK1 (EC50=2μM, Kd=8.4μM) and may cause cardiovascular inflammation.Formule :C19H20N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.44BRL 15572
CAS :BRL 15572 is a useful organic compound for research related to life sciences. The catalog number is T64501 and the CAS number is 734517-40-9.Formule :C25H27ClN2OCouleur et forme :SolidMasse moléculaire :406.95BX471 hydrochloride
CAS :BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist with a Ki of 1 nM for human CCR1, exhibiting 250-fold selectivity over CCR2, CCR5, and CXCR4.Formule :C21H25Cl2FN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :471.351-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol
CAS :1-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol is a useful organic compound for research related to life sciences. The catalog number is T65156 and the CAS number is 24155-42-8.Formule :C11H10Cl2N2OCouleur et forme :SolidMasse moléculaire :257.11Anti-GLP1R Antibody
Anti-GLP1R Antibody is a human antibody expressed in CHO cells, targeting GLP1R. For isotype controls, refer to Human IgG1 kappa, Isotype Control.
Couleur et forme :Odour LiquidGoserelin acetate(65807-02-5 Free base)
Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.
Degré de pureté :99.77%Couleur et forme :Odour SolidAmelubant
CAS :Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315 with anti-inflammatory activity[1]. It is a potent, oral, long-acting LTB4 receptor antagonist that negligibly binds to the LTB4 receptor, exhibiting Kis of 221 nM and 230 nM in vital cells and membranes.Formule :C33H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :538.63TAK-448
CAS :TAK-448 (MVT-602), a potent KISS1R agonist, IC50: 460 pM, EC50: 632 pM, trialed for Prostate Cancer and Hypogonadism.Formule :C58H80N16O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1225.36GSK-3050002
GSK-3050002 (HGS-1035) is a humanized IgG1 antibody that targets and binds to CCL20. It holds potential for inflammation research. For isotype control, refer to Human IgG1 kappa, Isotype Control.
Couleur et forme :Odour Liquid(R)-(-)-α-Methylhistamine dihydrochloride
CAS :R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.Formule :C6H13Cl2N3Couleur et forme :SolidMasse moléculaire :198.094-Hydroxypropranolol hydrochloride
CAS :4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).Formule :C16H22ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :311.80dapitant
CAS :Dapitant, a non-peptide, selective antagonist of human NKI receptors, is representative of the 7,7,4-triarylperhydroisoindol-4-ols.Formule :C37H39NO4Couleur et forme :SolidMasse moléculaire :561.711-Oleoyl Lysophosphatidic Acid
CAS :1-Oleoyl Lysophosphatidic Acid (1-Oleoyl LPA) is a biologically active phospholipid that can be used to study cancer and atherosclerosis.
Formule :C21H41O7PCouleur et forme :SolidMasse moléculaire :436.526-Chloro-5-(2-chloroethyl)indolin-2-one
CAS :6-Chloro-5-(2-chloroethyl)indolin-2-one is a useful organic compound for research related to life sciences. The catalog number is T64862 and the CAS number is 118289-55-7.Formule :C10H9Cl2NOCouleur et forme :SolidMasse moléculaire :230.09(Rac)-Zevaquenabant
CAS :(Rac)-Zevaquenabant ((Rac)-MRI-1867, compound 6b) is a potent and selective antagonist of cannabinoid receptor type 1 (CB1R) and inducible nitric oxide synthase (iNOS), with a binding affinity (Ki) of 5.7 nM for CB1R. It holds promise as an investigative tool in liver fibrosis research due to these characteristics.Formule :C25H21ClF3N5O2SCouleur et forme :SolidMasse moléculaire :547.98Propiram fumarate HCl
CAS :Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
Formule :C16H25N3O·xClHDegré de pureté :99.25%Couleur et forme :SoildDesmethyl cariprazine
CAS :Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).Formule :C20H30Cl2N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.38Patecibart
CAS :Patecibart is a humanized immunoglobulin G4-kappa monoclonal antibody that functions as an antagonist to the endothelin receptor A (EDNRA).
Degré de pureté :98%Couleur et forme :LiquidN-methyl-2-AI (hydrochloride)
CAS :N-methyl-2-AI (hydrochloride) is a useful organic compound for research related to life sciences. The catalog number is T66396 and the CAS number is 10408-85-2.Formule :C10H14ClNCouleur et forme :SolidMasse moléculaire :183.683-Hydroxybenzylamine
CAS :3-Hydroxybenzylamine is a useful organic compound for research related to life sciences. The catalog number is T124305 and the CAS number is 73604-31-6.Formule :C7H9NOCouleur et forme :SolidMasse moléculaire :123.155Canagliflozin-d4
CAS :Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.
Formule :C24H25FO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.542-Methyl-5-HT hydrochloride
CAS :2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Formule :C11H15ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.7RU 24969 succinate
CAS :RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.
Formule :C18H22N2O5Couleur et forme :SolidMasse moléculaire :346.38Pamoic acid
CAS :Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.
Formule :C23H16O6Degré de pureté :99.99%Couleur et forme :Fine Yellow PowderMasse moléculaire :388.37MEN11467
CAS :MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75Neurokinin antagonist 1
CAS :Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75Flumexadol
CAS :Flumexadol is a selective 5-HT2C receptor agonist with an affinity (Ki) of 25 nM for the (+)-enantiomer and exhibits 40-fold selectivity over the 5-HT2A receptor. It is an orally active, non-narcotic analgesic.Formule :C11H12F3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.21SB251023
CAS :SB251023 is an agonist of β3-adrenoceptor.Formule :C28H34NO6PCouleur et forme :SolidMasse moléculaire :511.55GR 218,231
CAS :GR 218,231 is a selective antagonist of D3 dopamine receptor.Formule :C24H33NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.59Imetit dihydrobromide
CAS :Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).Formule :C6H12Br2N4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.06AEF0117
CAS :AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.
Formule :C29H40O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :436.63Ref: TM-T79909
Produit arrêtéS1P1 agonist 6
CAS :Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive
Formule :C25H26F3NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.47Dimethandrolone Undecanoate
CAS :Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Formule :C31H50O3Degré de pureté :99.65% - >99.99%Couleur et forme :SolidMasse moléculaire :470.732-MNG
CAS :2-MNG (2-Mercaptonicotinoyl glycine) is a novel melanogenesis inhibitor. 2-MNG inhibits two mechanisms of UV-induced skin pigmentation in vivo.
Formule :C8H8N2O3SCouleur et forme :LiquidMasse moléculaire :212.23Ref: TM-T89029
Produit arrêté
